Tytuł pozycji:
The Discovery of Polo-LikeKinase 4 Inhibitors: Identification of (1R,2S)-2-(3-((E)-4-(((cis)-2,6-Dimethylmorpholino)methyl)styryl)-1H-indazol-6-yl)-5′-methoxyspiro[cyclopropane-1,3′-indolin]-2′-one(CFI-400945) as a Potent, Orally...
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Tytuł:
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The Discovery of Polo-LikeKinase 4 Inhibitors: Identification of (1R,2S)-2-(3-((E)-4-(((cis)-2,6-Dimethylmorpholino)methyl)styryl)-1H-indazol-6-yl)-5′-methoxyspiro[cyclopropane-1,3′-indolin]-2′-one(CFI-400945) as a Potent, Orally...
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Autorzy:
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Sampson, Peter B.
Liu, Yong
Forrest, Bryan
Cumming, Graham
Li, Sze-Wan
Patel, Narendra Kumar
Edwards, Louise
Laufer, Radoslaw
Feher, Miklos
Ban, Fuqiang
Awrey, Donald E.
Mao, Guodong
Plotnikova, Olga
Hodgson, Richard
Beletskaya, Irina
Mason, Jacqueline M.
Luo, Xunyi
Nadeem, Vincent
Wei, Xin
Kiarash, Reza
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Źródło:
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Journal of Medicinal Chemistry; Jan2015, Vol. 58 Issue 1, p147-169, 23p
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