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Tytuł:
2-Oxoquinoline-based-thiosemicarbazones as multitargeting neurotherapeutics against Alzheimer's disease: In vitro and in silico studies of MAO and ChE inhibitors.
Autorzy:
Basri R; Institute of Chemical Sciences, Bahauddin Zakariya University, Multan, Pakistan.
Fatima S; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
Jalil S; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, Pakistan.
Imran A; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, Pakistan.; Department of Pharmacy, COMSATS University Islamabad, Lahore Campus, Islamabad, Punjab, Pakistan.
Fatima N; Department of Chemistry, Quaid-i-Azam University, Islamabad, Pakistan.
Syed A; Department of Botany and Microbiology, King Saud University, Riyadh, Saudi Arabia.
Bahkali AH; Department of Botany and Microbiology, King Saud University, Riyadh, Saudi Arabia.
Iqbal J; Centre for Advanced Drug Research, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, Pakistan.; Department of Chemistry, COMSATS University Islamabad, Abbottabad Campus, Abbottabad, Pakistan.
Shafiq Z; Institute of Chemical Sciences, Bahauddin Zakariya University, Multan, Pakistan.; Department of Pharmaceutical & Medicinal Chemistry, University of Bonn, Bonn, Germany.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep 17, pp. e2300430. Date of Electronic Publication: 2023 Sep 17.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Potent inhibitors of tumor associated carbonic anhydrases endowed with cathepsin B inhibition.
Autorzy:
Kumar A; Department of Chemistry, Kurukshetra University, Kurukshetra, India.
Arya P; Department of Chemistry, Kurukshetra University, Kurukshetra, India.
Sharma V; Department of Chemistry, Kurukshetra University, Kurukshetra, India.; Department of Chemistry, Pt. Chiranji Lal Sharma Government College, Karnal, India.
Giovannuzzi S; Neurofarba Department, Pharmaceutical and Nutraceutical Section, University of Florence, Florence, Italy.
Raghav N; Department of Chemistry, Kurukshetra University, Kurukshetra, India.
Supuran CT; Neurofarba Department, Pharmaceutical and Nutraceutical Section, University of Florence, Florence, Italy.
Sharma PK; Department of Chemistry, Kurukshetra University, Kurukshetra, India.; Department of Chemistry, Central University of Haryana, Mahendergarh, India.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep 13, pp. e2300349. Date of Electronic Publication: 2023 Sep 13.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Exploration of 3-aryl pyrazole-tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors.
Autorzy:
Ommi O; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Paoletti N; Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.; Laboratory of Molecular Modeling Cheminformatics & QSAR, Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.
Bonardi A; Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.; Laboratory of Molecular Modeling Cheminformatics & QSAR, Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.
Gratteri P; Laboratory of Molecular Modeling Cheminformatics & QSAR, Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.
Bhalerao HA; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Sau S; Department of Biological Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Nanduri S; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Mohammed A; Department of Chemistry, Directorate of Distance Education, Maulana Azad National Urdu University, Hyderabad, India.
Kalia NP; Department of Biological Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Sonti R; Department of Pharmaceutical Analysis, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
Supuran CT; Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.; Laboratory of Molecular Modeling Cheminformatics & QSAR, Department NEUROFARBA, Pharmaceutical and Nutraceutical Section, University of Florence, Sesto Fiorentino (Florence), Italy.
Yaddanapudi VM; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, Telangana, India.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep 10, pp. e2300309. Date of Electronic Publication: 2023 Sep 10.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Design and synthesis of benzofuran- and naphthalene-fused thiazinones as antimycobacterial agents.
Autorzy:
Keiff F; Transfer Group Anti-infectives, Leibniz Institute for Natural Product Research and Infection Biology-Leibniz-HKI, Jena, Germany.
Jacques Dit Lapierre TJW; Transfer Group Anti-infectives, Leibniz Institute for Natural Product Research and Infection Biology-Leibniz-HKI, Jena, Germany.
Bernal FA; Transfer Group Anti-infectives, Leibniz Institute for Natural Product Research and Infection Biology-Leibniz-HKI, Jena, Germany.
Kloss F; Transfer Group Anti-infectives, Leibniz Institute for Natural Product Research and Infection Biology-Leibniz-HKI, Jena, Germany.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep 04, pp. e2300356. Date of Electronic Publication: 2023 Sep 04.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Synthesis of 1,2,4-triazole and 1,3,4-oxadiazole derivatives as inhibitors for STAT3 enzymes of breast cancer.
Autorzy:
Fawzy SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Sinai University, Kantara Branch, Al-Ismailia, Egypt.
Loksha YM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Sinai University, Al-Arish Branch, North Sinai, Egypt.
El-Sadek M; Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
Ibrahim SM; Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
Beshay BY; Department of Pharmaceutical Chemistry, College of Pharmacy, Arab Academy for Science, Technology and Maritime Transport, Alexandria, Egypt.
Shamaa MM; Department of Biochemistry, Clinical and Biological Sciences Division, College of Pharmacy, Arab Academy for Science, Technology and Maritime Transport, Alexandria, Egypt.
Kothayer H; Department of Medicinal Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep 03, pp. e2300345. Date of Electronic Publication: 2023 Sep 03.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Novel hydrazone-isatin derivatives as potential EGFR inhibitors: Synthesis and in vitro pharmacological profiling.
Autorzy:
Ahmed MF; Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, Taif, Saudi Arabia.
El-Haggar R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.
Almalki AH; Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, Taif, Saudi Arabia.; Addition and Neuroscience Research Unit, College of Pharmacy, Taif University, Taif, Al-Hawiah, Saudi Arabia.
Abdullah O; Pharmaceutical Chemistry Department, College of Pharmacy, Umm Al-Qura University, Makkah, Saudi Arabia.
El Hassab MA; Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), South Sinai, Egypt.
Masurier N; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS, Université de Montpellier, ENSCM, Montpellier, France.
Hammad SF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.; Basic and Applied Science Institute, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Alexandria, Egypt.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300244. Date of Electronic Publication: 2023 Jul 05.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
In silico characterization of ligand-receptor interactions for U-47700, N,N-didesmethyl-U-47700, U-50488 at mu- and kappa-opioid receptors.
Autorzy:
Laus A; Department of Biomedical Sciences, University of Cagliari, Cittadella Universitaria di Monserrato, Cagliari, Italy.
Kumar A; Department of Electrical and Electronic Engineering, University of Cagliari, Cagliari, Italy.
Caboni P; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria di Monserrato, Cagliari, Italy.
De Luca MA; Department of Biomedical Sciences, University of Cagliari, Cittadella Universitaria di Monserrato, Cagliari, Italy.
Baumann MH; Designer Drug Research Unit, Intramural Research Program, National Institute on Drug Abuse, National Institutes of Health, Baltimore, Maryland, USA.
Pieroni E; CRS4, Modelling, Simulation and Data Analysis Program, Pula, Italy.
Tocco G; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria di Monserrato, Cagliari, Italy.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300256. Date of Electronic Publication: 2023 Jul 14.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid, kappa*/chemistry
Receptors, Opioid, kappa*/metabolism
Receptors, Opioid, mu*/metabolism
3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer/pharmacology ; Ligands ; Structure-Activity Relationship ; Analgesics, Opioid/pharmacology ; Analgesics, Opioid/chemistry
Czasopismo naukowe
Tytuł:
Unraveling the chemical profile, antioxidant, enzyme inhibitory, cytotoxic potential of different extracts from Astragalus caraganae.
Autorzy:
Kurt-Celep İ; Faculty of Pharmacy, Department of Pharmacognosy, Ataşehir, Acıbadem Mehmet Ali Aydınlar University, İstanbul, Turkey.
Zengin G; Department of Biology, Science Faculty, Selcuk University, Konya, Turkey.
Uba AI; Department of Molecular Biology and Genetics, Istanbul AREL University, Istanbul, Turkey.
Caprioli G; School of Pharmacy, University of Camerino, Camerino, Italy.
Mustafa AM; School of Pharmacy, University of Camerino, Camerino, Italy.
Angeloni S; School of Pharmacy, University of Camerino, Camerino, Italy.
Cakilcioglu U; Pertek Sakine Genç Vocational School, Munzur University, Pertek, Turkey.
Guler O; Pertek Sakine Genç Vocational School, Munzur University, Pertek, Turkey.
Kaplan A; Sason Vocational School, Batman University, Batman, Turkey.
Sharmeen J; Department of Health Sciences, Faculty of Medicine and Health Sciences, University of Mauritius, Reduit, Mauritius.
Mahomoodally MF; Department of Health Sciences, Faculty of Medicine and Health Sciences, University of Mauritius, Reduit, Mauritius.; Department of Pharmacology, Center for Transdisciplinary Research, Saveetha Dental College, Saveetha Institute of Medical and Technical Science, Saveetha University, Chennai, India.; Centre of Excellence for Pharmaceutical Sciences, North-West University, Potchefstroom, South Africa.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300263. Date of Electronic Publication: 2023 Jul 11.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Novel promising benzoxazole/benzothiazole-derived immunomodulatory agents: Design, synthesis, anticancer evaluation, and in silico ADMET analysis.
Autorzy:
Elkady H; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.
El-Adl K; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Heliopolis University for Sustainable Development, Cairo, Egypt.
Sakr H; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.
Abdelraheem AS; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.
Eissa SI; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo, Egypt.
El-Zahabi MA; Pharmaceutical Medicinal Chemistry and Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300097. Date of Electronic Publication: 2023 Jun 28.
Typ publikacji:
Journal Article
MeSH Terms:
Immunomodulating Agents*
Antineoplastic Agents*/pharmacology
Humans ; Molecular Structure ; Structure-Activity Relationship ; Vascular Endothelial Growth Factor A/pharmacology ; Thalidomide/pharmacology ; Benzoxazoles/pharmacology ; NF-kappa B ; Tumor Necrosis Factor-alpha ; Cell Proliferation ; MCF-7 Cells ; Benzothiazoles/pharmacology ; Drug Screening Assays, Antitumor ; Molecular Docking Simulation ; Cell Line, Tumor ; Drug Design
Czasopismo naukowe
Tytuł:
Design, synthesis, and structure-activity studies of new rhodanine derivatives as carbonic anhydrase II, IX inhibitors.
Autorzy:
Chinchilli KK; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Akunuri R; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Ghouse SM; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Soujanya D; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Angeli A; Neurofarba Dept. Sezione di Scienze Farmaceutiche e Nutraceutiche, Sesto Fiorentino, Università degli Studi di Firenze, Florence, Italy.
Parupalli R; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Arifuddin M; Department of Chemistry, Directorate of Distance Education, Maulana Azad National Urdu University, Gachibowli, Hyderabad, India.
Yaddanapudi VM; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
Supuran CT; Neurofarba Dept. Sezione di Scienze Farmaceutiche e Nutraceutiche, Sesto Fiorentino, Università degli Studi di Firenze, Florence, Italy.
Nanduri S; Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Balanagar, Hyderabad, India.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300205. Date of Electronic Publication: 2023 Jun 30.
Typ publikacji:
Journal Article
MeSH Terms:
Carbonic Anhydrases*/metabolism
Rhodanine*/pharmacology
Humans ; Carbonic Anhydrase II ; Structure-Activity Relationship ; Molecular Docking Simulation ; Carbonic Anhydrase Inhibitors/pharmacology ; Molecular Structure
Czasopismo naukowe
Tytuł:
Proapoptotic effects of halogenated bis-phenylthiourea derivatives in cancer cells.
Autorzy:
Strzyga-Łach P; Chair and Department of Biochemistry, Medical University of Warsaw, Warsaw, Poland.
Chrzanowska A; Chair and Department of Biochemistry, Medical University of Warsaw, Warsaw, Poland.
Kiernozek-Kalińska E; Department of Immunology, Faculty of Biology, University of Warsaw, Warsaw, Poland.
Żyżyńska-Granica B; Chair and Department of Biochemistry, Medical University of Warsaw, Warsaw, Poland.
Podsadni K; Chair and Department of Biochemistry, Medical University of Warsaw, Warsaw, Poland.
Podsadni P; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, Warsaw, Poland.
Bielenica A; Chair and Department of Biochemistry, Medical University of Warsaw, Warsaw, Poland.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300105. Date of Electronic Publication: 2023 Jul 04.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents*/pharmacology
Neoplasms*
Caspase 3/metabolism ; Caspase 7/metabolism ; Structure-Activity Relationship ; Phenylthiourea/pharmacology ; Reactive Oxygen Species/metabolism ; Interleukin-6/pharmacology ; Cell Line, Tumor ; Apoptosis ; Cell Proliferation
Czasopismo naukowe
Tytuł:
Ruthenium polypyridine complexes containing prenyl groups as antibacterial agents against Staphylococcus aureus through a membrane-disruption mechanism.
Autorzy:
Wang R; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Zhou X; Shenzhen Second People's Hospital, Shenzhen, China.
Chen J; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Chen Y; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Xiong Y; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Duan X; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Liao X; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
Wang J; School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang, China.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300175. Date of Electronic Publication: 2023 Jul 08.
Typ publikacji:
Journal Article
MeSH Terms:
Staphylococcus aureus*
Ruthenium*/pharmacology
Animals ; Mice ; Anti-Bacterial Agents/pharmacology ; Structure-Activity Relationship ; 2,2'-Dipyridyl/pharmacology ; DNA ; Mammals/metabolism
Czasopismo naukowe
Tytuł:
Melatonin-vorinostat hybrid ligands show higher histone deacetylase and cancer cell growth inhibition than vorinostat.
Autorzy:
Helmi YY; Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Biotechnology, The German University in Cairo, New Cairo City, Cairo, Egypt.
Papenkordt N; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
Rennar G; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
Gbahou F; Université Paris Cité, Institut Cochin, INSERM, CNRS, Paris, France.
El-Hady AK; Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Biotechnology, The German University in Cairo, New Cairo City, Cairo, Egypt.; Department of Organic and Pharmaceutical Chemistry, School of Life and Medical Sciences, University of Hertfordshire hosted by Global Academic Foundation, New Administrative Capitol, Cairo, Egypt.
Labani N; Université Paris Cité, Institut Cochin, INSERM, CNRS, Paris, France.
Schmidtkunz K; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
Boettcher S; Pharmaceutical and Medicinal Chemistry, Saarland University, Saarbruecken, Germany.
Jockers R; Université Paris Cité, Institut Cochin, INSERM, CNRS, Paris, France.
Abdel-Halim M; Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Biotechnology, The German University in Cairo, New Cairo City, Cairo, Egypt.
Jung M; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
Zlotos DP; Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Biotechnology, The German University in Cairo, New Cairo City, Cairo, Egypt.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300149. Date of Electronic Publication: 2023 Jun 20.
Typ publikacji:
Journal Article
MeSH Terms:
Melatonin*/pharmacology
Antineoplastic Agents*/pharmacology
Antineoplastic Agents*/chemistry
Neoplasms*
Vorinostat/pharmacology ; Histone Deacetylases/metabolism ; Histone Deacetylases/pharmacology ; Ligands ; Structure-Activity Relationship ; Histone Deacetylase Inhibitors/pharmacology ; Histone Deacetylase Inhibitors/chemistry ; Hydroxamic Acids/pharmacology ; Cell Line, Tumor ; Cell Proliferation ; Histone Deacetylase 1/metabolism ; Histone Deacetylase 1/pharmacology ; Histone Deacetylase 6
Czasopismo naukowe
Tytuł:
Synthesis and biological profile of benzoxazolone derivatives.
Autorzy:
Prasher P; Department of Chemistry, University of Petroleum & Energy Studies, Energy Acres, Dehradun, India.
Mall T; Department of Chemistry, University of Petroleum & Energy Studies, Energy Acres, Dehradun, India.
Sharma M; Department of Chemistry, Uttaranchal University, Dehradun, India.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300245. Date of Electronic Publication: 2023 Jun 28.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Analgesics*/pharmacology
Benzoxazoles*/chemistry
Structure-Activity Relationship ; Hydrophobic and Hydrophilic Interactions
Czasopismo naukowe
Tytuł:
Multitargeting in cardioprotection: An example of biaromatic compounds.
Autorzy:
Mokrov GV; FSBI 'Zakusov Institute of Pharmacology', Moscow, Russia.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Sep; Vol. 356 (9), pp. e2300196. Date of Electronic Publication: 2023 Jun 22.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Drug Design*
Cardiovascular Diseases*
Humans ; Structure-Activity Relationship ; Chemistry, Pharmaceutical ; Pharmacophore ; Ligands
Czasopismo naukowe
Tytuł:
The anti-breast cancer potential of indole/isatin hybrids.
Autorzy:
Wang R; Department of General Surgery, Comprehensive Breast Health Center, Ruijin Hospital, Shanghai Jiao Tong University School of Medicine, Shanghai, China.
Huang R; Department of General Surgery, Comprehensive Breast Health Center, Ruijin Hospital, Shanghai Jiao Tong University School of Medicine, Shanghai, China.
Yuan Y; Laboratory of Molecule Synthesis and Function Discovery (Fujian Province University), Department of Chemistry, Fuzhou University, Fuzhou, China.
Wang Z; Department of General Surgery, Comprehensive Breast Health Center, Ruijin Hospital, Shanghai Jiao Tong University School of Medicine, Shanghai, China.
Shen K; Department of General Surgery, Comprehensive Breast Health Center, Ruijin Hospital, Shanghai Jiao Tong University School of Medicine, Shanghai, China.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Aug 31, pp. e2300402. Date of Electronic Publication: 2023 Aug 31.
Typ publikacji:
Journal Article; Review
Czasopismo naukowe
Tytuł:
Neuroprotective effect of Potentilla reptans L. root in the rat brain global ischemia/reperfusion model.
Autorzy:
Noorgaldi S; Neuroscience Research Center, Golestan University of Medical Sciences, Gorgan, Iran.; Department of Anatomy, Faculty of Medicine, Neuroscience Research Center, Golestan University of Medical Sciences, Gorgan, Iran.
Sarkala HB; Department of Anatomy, School of Medicine, Iran University of Medical Sciences, Tehran, Iran.
Enayati A; Ischemic Disorders Research Center, Golestan University of Medical Sciences, Gorgan, Iran.
Khori V; Ischemic Disorders Research Center, Golestan University of Medical Sciences, Gorgan, Iran.
Zengin G; Department of Biology, Science Faculty, Selcuk University, Konya, Turkey.
Jahanshahi M; Department of Anatomy, Faculty of Medicine, Neuroscience Research Center, Golestan University of Medical Sciences, Gorgan, Iran.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Aug 29, pp. e2300363. Date of Electronic Publication: 2023 Aug 29.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
The beneficial effects of l-carnitine and infliximab in methotrexate-induced hepatotoxicity: Emphasis on Notch1/Hes-1 signaling.
Autorzy:
Radwan SM; Biochemistry Department, Faculty of Pharmacy, Ain Shams University, Cairo, Egypt.
Abdel-Latif GA; Pharmacology and Toxicology Department, Faculty of Pharmacy, Misr International University (MIU), Cairo, Egypt.; Translational and Clinical Research Unit, Faculty of Pharmacy, Misr International University (MIU), Cairo, Egypt.
Abbas SS; Pharmacology and Toxicology Department, Faculty of Pharmacy, Misr International University (MIU), Cairo, Egypt.; Translational and Clinical Research Unit, Faculty of Pharmacy, Misr International University (MIU), Cairo, Egypt.
Elmongy NF; Physiology Department, Faculty of Medicine, Al-Azhar University, Damietta, Egypt.
Wasfey EF; Biochemistry Department, Faculty of Pharmacy, Ain Shams University, Cairo, Egypt.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Aug 25, pp. e2300312. Date of Electronic Publication: 2023 Aug 25.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Benzimidazolone-piperazine/triazole/thiadiazole/furan/thiophene conjugates: Synthesis, in vitro urease inhibition, and in silico molecular docking studies.
Autorzy:
Güven O; Department of Chemistry, Art and Science Faculty, Recep Tayyip Erdogan University, Rize, Turkey.
Menteşe E; Department of Chemistry, Art and Science Faculty, Recep Tayyip Erdogan University, Rize, Turkey.
Emirik M; Department of Chemistry, Art and Science Faculty, Recep Tayyip Erdogan University, Rize, Turkey.
Sökmen BB; Department of Chemistry, Faculty of Arts and Sciences, Giresun University, Giresun, Turkey.
Akyüz G; Department of Chemistry, Art and Science Faculty, Recep Tayyip Erdogan University, Rize, Turkey.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Aug 23, pp. e2300336. Date of Electronic Publication: 2023 Aug 23.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Biological evaluation of [4-(4-aminophenyl)-1-(4-fluorophenyl)-1H-pyrrol-3-yl](3,4,5-trimethoxyphenyl)methanone as potential antineoplastic agent in 2D and 3D breast cancer models.
Autorzy:
Mazzoccoli C; Laboratory of Preclinical and Translational Research, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Crispo F; Laboratory of Preclinical and Translational Research, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Laurenzana I; Laboratory of Preclinical and Translational Research, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Pietrafesa M; Clinical Pathology Unit, A.O.R. San Carlo Potenza, Potenza, Italy.
Sisinni L; Clinical Pathology Unit, Azienda Sanitaria Locale, Potenza, Italy.
Lerose R; Hospital Pharmacy, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Telesca D; Hospital Pharmacy, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Milella MR; Hospital Pharmacy, Centro di Riferimento Oncologico della Basilicata (IRCCS-CROB), Rionero in Vulture, Italy.
Liu T; Shanghai Geriatric Institute of Chinese Medicine, Shanghai University of Traditional Chinese Medicine, Shanghai, China.
Della Sala G; Department of Eco-Sustainable Marine Biotechnology, Stazione Zoologica Anton Dohrn, Naples, Italy.
Sebastiani J; Laboratory Affiliated with the Institute Pasteur Italy - Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome, Italy.
Silvestri R; Laboratory Affiliated with the Institute Pasteur Italy - Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome, Italy.
La Regina G; Laboratory Affiliated with the Institute Pasteur Italy - Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome, Italy.
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Źródło:
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2023 Aug 21, pp. e2300354. Date of Electronic Publication: 2023 Aug 21.
Typ publikacji:
Journal Article
Czasopismo naukowe

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