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Tytuł:
Transfer of rhodamine-123 into the brain and cerebrospinal fluid of fetal, neonatal and adult rats.
Autorzy:
Koehn LM; Department of Pharmacology & Therapeutics, University of Melbourne, Parkville, Victoria, 3010, Australia. liam_.
Dziegielewska KM; Department of Pharmacology & Therapeutics, University of Melbourne, Parkville, Victoria, 3010, Australia.
Habgood MD; Department of Pharmacology & Therapeutics, University of Melbourne, Parkville, Victoria, 3010, Australia.
Huang Y; Department of Pharmacology & Therapeutics, University of Melbourne, Parkville, Victoria, 3010, Australia.
Saunders NR; Department of Pharmacology & Therapeutics, University of Melbourne, Parkville, Victoria, 3010, Australia.
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Źródło:
Fluids and barriers of the CNS [Fluids Barriers CNS] 2021 Feb 08; Vol. 18 (1), pp. 6. Date of Electronic Publication: 2021 Feb 08.
Typ publikacji:
Journal Article
MeSH Terms:
Brain*
Cerebrospinal Fluid*
ATP Binding Cassette Transporter, Subfamily B, Member 1/*pharmacokinetics
Fluorescent Dyes/*pharmacokinetics
Rhodamine 123/*pharmacokinetics
ATP Binding Cassette Transporter, Subfamily B, Member 1/administration & dosage ; Age Factors ; Animals ; Animals, Newborn ; Biological Transport/physiology ; Embryo, Mammalian ; Female ; Fluorescent Dyes/administration & dosage ; Male ; Pregnancy ; Rats ; Rats, Sprague-Dawley ; Rhodamine 123/administration & dosage ; Spectrometry, Fluorescence
Czasopismo naukowe
Tytuł:
In Vitro Evaluation of the Interaction of Seven Biologically Active Components in Anemarrhenae rhizoma with P-gp.
Autorzy:
Dai J; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
He Y; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
Fang J; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
Wang H; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
Chao L; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
Zhao L; Department of Pharmacy, Shanghai Baoshan Luodian Hospital, Shanghai 201908, China.
Hong Z; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
Chai Y; School of Pharmacy, Naval Medical University, Shanghai 200433, China.; Shanghai Key Laboratory for Pharmaceutical Metabolite Research, Shanghai 200433, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Dec 05; Vol. 27 (23). Date of Electronic Publication: 2022 Dec 05.
Typ publikacji:
Journal Article
MeSH Terms:
Anemarrhena*
Rhizome ; ATP Binding Cassette Transporter, Subfamily B, Member 1 ; ATP Binding Cassette Transporter, Subfamily B ; Rhodamine 123
Czasopismo naukowe
Tytuł:
Carnosine Potentiates Doxorubicin-Induced Cytotoxicity in Resistant NCI/ADR-RES Cells by Inhibiting P-Glycoprotein-In Silico and In Vitro Evidence.
Autorzy:
Morsy MA; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt.
Kandeel M; Department of Biomedical Sciences, College of Veterinary Medicine, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Veterinary Medicine, Kafrelsheikh University, Kafr El-Sheikh 33516, Egypt.
Ibrahim ARN; Clinical Pharmacy Department, College of Pharmacy, King Khalid University, Abha 61441, Saudi Arabia.; Department of Biochemistry, Faculty of Pharmacy, Minia University, El-Minia 61511, Egypt.
Abdel-Gaber SA; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt.
Jacob S; Department of Pharmaceutical Sciences, College of Pharmacy, Gulf Medical University, Ajman 4184, United Arab Emirates.
Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Biotechnology and Food Science, Faculty of Applied Sciences, Durban University of Technology, Durban 4000, South Africa.
Shinu P; Department of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
El-Daly M; Department of Pharmacology & Toxicology, Faculty of Pharmacy, Minia University, El-Minia 61511, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Oct 30; Vol. 27 (21). Date of Electronic Publication: 2022 Oct 30.
Typ publikacji:
Journal Article
MeSH Terms:
Carnosine*/pharmacology
Carnosine*/metabolism
Antineoplastic Agents*/pharmacology
Drug Resistance, Multiple ; ATP Binding Cassette Transporter, Subfamily B, Member 1/metabolism ; Molecular Docking Simulation ; Drug Resistance, Neoplasm ; Doxorubicin/pharmacology ; Rhodamine 123/pharmacology ; Verapamil/pharmacology ; ATP Binding Cassette Transporter, Subfamily B/metabolism
Czasopismo naukowe
Tytuł:
A multi-chamber microfluidic intestinal barrier model using Caco-2 cells for drug transport studies.
Autorzy:
Tan HY; Technical University of Denmark, Department of Micro and Nanotechnology, Ørsteds Plads, Lyngby, Denmark.; Technical University of Denmark, Center for Nanomedicine and Theranostics, Ørsteds Plads, Lyngby, Denmark.; Biomedical Institute for Global Health Research & Technology (BIGHEART), National University of Singapore, Singapore.
Trier S; Global Research, Novo Nordisk A/S, Maaloev, Denmark.
Rahbek UL; Global Research, Novo Nordisk A/S, Maaloev, Denmark.
Dufva M; Technical University of Denmark, Department of Micro and Nanotechnology, Ørsteds Plads, Lyngby, Denmark.
Kutter JP; Department of Pharmacy, University of Copenhagen, Universitetsparken 2, Copenhagen, Denmark.
Andresen TL; Technical University of Denmark, Department of Micro and Nanotechnology, Ørsteds Plads, Lyngby, Denmark.; Technical University of Denmark, Center for Nanomedicine and Theranostics, Ørsteds Plads, Lyngby, Denmark.
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Źródło:
PloS one [PLoS One] 2018 May 10; Vol. 13 (5), pp. e0197101. Date of Electronic Publication: 2018 May 10 (Print Publication: 2018).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Dextrans*/pharmacokinetics
Dextrans*/pharmacology
Insulin*/pharmacokinetics
Insulin*/pharmacology
Lab-On-A-Chip Devices*
Mannitol*/pharmacokinetics
Mannitol*/pharmacology
Microfluidic Analytical Techniques*/instrumentation
Microfluidic Analytical Techniques*/methods
Rhodamine 123*/pharmacokinetics
Rhodamine 123*/pharmacology
Intestinal Absorption/*drug effects
Intestinal Mucosa/*metabolism
Maltose/*analogs & derivatives
ATP Binding Cassette Transporter, Subfamily B/metabolism ; Caco-2 Cells ; Humans ; Intestinal Mucosa/cytology ; Maltose/pharmacokinetics ; Maltose/pharmacology
Czasopismo naukowe
Tytuł:
Is the Mitochondrial Membrane Potential (∆Ψ) Correctly Assessed? Intracellular and Intramitochondrial Modifications of the ∆Ψ Probe, Rhodamine 123.
Autorzy:
Zorova LD; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Demchenko EA; Biological Faculty, Lomonosov Moscow State University, 119992 Moscow, Russia.
Korshunova GA; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Tashlitsky VN; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Zorov SD; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.; Faculty of Bioengineering and Bioinformatics, Lomonosov Moscow State University, 119992 Moscow.
Andrianova NV; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Popkov VA; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Babenko VA; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Pevzner IB; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Silachev DN; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Plotnikov EY; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
Zorov DB; A.N. Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, 119992 Moscow, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Jan 01; Vol. 23 (1). Date of Electronic Publication: 2022 Jan 01.
Typ publikacji:
Journal Article
MeSH Terms:
Membrane Potential, Mitochondrial*
Mitochondria/*metabolism
Molecular Probes/*metabolism
Rhodamine 123/*metabolism
Animals ; Astrocytes/metabolism ; Cell Extracts ; Cell Line, Tumor ; Fluorescence ; Glioma/metabolism ; Rats ; Time Factors
Czasopismo naukowe
Tytuł:
EGFR Transgene Stimulates Spontaneous Formation of MCF7 Breast Cancer Cells Spheroids with Partly Loss of HER3 Receptor.
Autorzy:
Troitskaya O; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.
Novak D; Department of Natural Sciences, Novosibirsk State University, 630090 Novosibirsk, Russia.
Nushtaeva A; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.
Savinkova M; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.; Department of Natural Sciences, Novosibirsk State University, 630090 Novosibirsk, Russia.
Varlamov M; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.; Department of Natural Sciences, Novosibirsk State University, 630090 Novosibirsk, Russia.
Ermakov M; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.
Richter V; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.
Koval O; Institute of Chemical Biology and Fundamental Medicine SB RAS, 630090 Novosibirsk, Russia.; Department of Natural Sciences, Novosibirsk State University, 630090 Novosibirsk, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2021 Nov 29; Vol. 22 (23). Date of Electronic Publication: 2021 Nov 29.
Typ publikacji:
Evaluation Study; Journal Article
MeSH Terms:
Genes, erbB-1*
MCF-7 Cells*
Spheroids, Cellular*
Receptor, ErbB-3/*metabolism
CD24 Antigen/metabolism ; Cell Culture Techniques, Three Dimensional ; Humans ; Hyaluronan Receptors/metabolism ; Rhodamine 123 ; Transgenes ; Tumor Cells, Cultured
Czasopismo naukowe
Tytuł:
Structure activity relationships and the binding mode of quinolinone-pyrimidine hybrids as reversal agents of multidrug resistance mediated by P-gp.
Autorzy:
Laiolo J; Fine Chemical and Natural Products Laboratory, IRNASUS CONICET-UCC, Universidad Católica de Córdoba, Avda. Armada Argentina 3555, X5016DHK, Córdoba, Argentina.
Lanza PA; Department of Chemistry, College of Exact and Natural Sciences, Universidad Nacional de Mar del Plata - QUIAMM - INBIOTEC CONICET, Funes 3350, Mar del Plata, Argentina.
Parravicini O; Faculty of Chemistry, Biochemistry and Pharmacy, Universidad Nacional de San Luis, IMIBIO-SL, Ejército de los Andes 950, 5700, San Luis, Argentina.
Barbieri C; Department of Chemistry, College of Exact and Natural Sciences, Universidad Nacional de Mar del Plata - QUIAMM - INBIOTEC CONICET, Funes 3350, Mar del Plata, Argentina.
Insuasty D; Department of Chemistry and Biology, Universidad del Norte, Km 5 vía Puerto Colombia, 081007, Barranquilla, Colombia.; Department of Inorganic and Organic Chemistry, Universidad de Jaén, Campus Las Lagunillas s/n, 23071, Jaén, Spain.
Cobo J; Department of Inorganic and Organic Chemistry, Universidad de Jaén, Campus Las Lagunillas s/n, 23071, Jaén, Spain.
Vera DMA; Department of Chemistry, College of Exact and Natural Sciences, Universidad Nacional de Mar del Plata - QUIAMM - INBIOTEC CONICET, Funes 3350, Mar del Plata, Argentina. .
Enriz RD; Faculty of Chemistry, Biochemistry and Pharmacy, Universidad Nacional de San Luis, IMIBIO-SL, Ejército de los Andes 950, 5700, San Luis, Argentina. .
Carpinella MC; Fine Chemical and Natural Products Laboratory, IRNASUS CONICET-UCC, Universidad Católica de Córdoba, Avda. Armada Argentina 3555, X5016DHK, Córdoba, Argentina. .
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Źródło:
Scientific reports [Sci Rep] 2021 Aug 19; Vol. 11 (1), pp. 16856. Date of Electronic Publication: 2021 Aug 19.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
ATP Binding Cassette Transporter, Subfamily B, Member 1/*metabolism
Drug Resistance, Multiple/*drug effects
Pyrimidines/*pharmacology
Quinolones/*pharmacology
Cell Death/drug effects ; Humans ; K562 Cells ; Molecular Dynamics Simulation ; Protein Transport/drug effects ; Pyrimidines/chemistry ; Pyrimidines/toxicity ; Quinolones/chemistry ; Quinolones/toxicity ; Rhodamine 123/metabolism ; Structure-Activity Relationship ; Thermodynamics
Czasopismo naukowe
Tytuł:
Subcellular distribution of ezrin/radixin/moesin and their roles in the cell surface localization and transport function of P-glycoprotein in human colon adenocarcinoma LS180 cells.
Autorzy:
Kobori T; Laboratory of Clinical Pharmaceutics, Faculty of Pharmacy, Osaka Ohtani University, Tondabayashi, Osaka, Japan.
Tameishi M; Laboratory of Clinical Pharmaceutics, Faculty of Pharmacy, Osaka Ohtani University, Tondabayashi, Osaka, Japan.
Tanaka C; Laboratory of Clinical Pharmaceutics, Faculty of Pharmacy, Osaka Ohtani University, Tondabayashi, Osaka, Japan.
Urashima Y; Laboratory of Clinical Pharmaceutics, Faculty of Pharmacy, Osaka Ohtani University, Tondabayashi, Osaka, Japan.
Obata T; Laboratory of Clinical Pharmaceutics, Faculty of Pharmacy, Osaka Ohtani University, Tondabayashi, Osaka, Japan.
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Źródło:
PloS one [PLoS One] 2021 May 11; Vol. 16 (5), pp. e0250889. Date of Electronic Publication: 2021 May 11 (Print Publication: 2021).
Typ publikacji:
Journal Article
MeSH Terms:
ATP Binding Cassette Transporter, Subfamily B, Member 1/*metabolism
Adenocarcinoma/*metabolism
Cell Membrane/*metabolism
Colonic Neoplasms/*metabolism
Cytoskeletal Proteins/*metabolism
Membrane Proteins/*metabolism
Microfilament Proteins/*metabolism
Biological Transport ; Caco-2 Cells ; Cell Line, Tumor ; Cytoskeletal Proteins/genetics ; Gene Expression Profiling ; Gene Silencing ; Humans ; Membrane Proteins/genetics ; Microfilament Proteins/genetics ; Microscopy, Confocal ; RNA, Messenger/metabolism ; RNA, Small Interfering ; Real-Time Polymerase Chain Reaction ; Rhodamine 123
Czasopismo naukowe
Tytuł:
Shenmai injection suppresses multidrug resistance in MCF-7/ADR cells through the MAPK/NF-κB signalling pathway.
Autorzy:
Yang L; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.; Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals, Zhejiang University of Technology, Hangzhou, China.
Zhang C; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.
Chen J; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.; Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals, Zhejiang University of Technology, Hangzhou, China.
Zhang S; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.
Pan G; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.
Xin Y; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.; Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals, Zhejiang University of Technology, Hangzhou, China.
Lin L; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.
You Z; Zhejiang Academy of Medical Sciences, Hangzhou Medical College, Hangzhou, China.
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Źródło:
Pharmaceutical biology [Pharm Biol] 2020 Dec; Vol. 58 (1), pp. 276-285.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Combined Chemotherapy Protocols/*pharmacology
Breast Neoplasms/*drug therapy
Doxorubicin/*pharmacology
Drugs, Chinese Herbal/*pharmacology
MAP Kinase Signaling System/*drug effects
NF-kappa B/*metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1/antagonists & inhibitors ; ATP Binding Cassette Transporter, Subfamily B, Member 1/metabolism ; Animals ; Antineoplastic Combined Chemotherapy Protocols/metabolism ; Antineoplastic Combined Chemotherapy Protocols/therapeutic use ; Breast Neoplasms/metabolism ; Down-Regulation/drug effects ; Doxorubicin/metabolism ; Doxorubicin/therapeutic use ; Drug Combinations ; Drug Resistance, Multiple/drug effects ; Drug Resistance, Neoplasm/drug effects ; Drugs, Chinese Herbal/administration & dosage ; Drugs, Chinese Herbal/therapeutic use ; Female ; Humans ; MCF-7 Cells ; Male ; Mice ; Mice, Inbred BALB C ; Mice, Nude ; Rhodamine 123/metabolism ; Signal Transduction/drug effects ; Xenograft Model Antitumor Assays
Czasopismo naukowe
Tytuł:
Comparison of Chemotherapeutic Activities of Rhodamine-Based GUMBOS and NanoGUMBOS.
Autorzy:
Bhattarai N; Department of Chemistry, Louisiana State University, Baton Rouge, LA 70803, USA.
Chen M; Department of Chemistry, Louisiana State University, Baton Rouge, LA 70803, USA.
L Pérez R; Department of Chemistry, Louisiana State University, Baton Rouge, LA 70803, USA.
Ravula S; Department of Chemistry, Louisiana State University, Baton Rouge, LA 70803, USA.
M Strongin R; Department of Chemistry, Portland State University, Portland, OR 97207, USA.
McDonough K; AgCenter Biotechnology Labs, Louisiana State University, Baton Rouge, LA 70803, USA.
M Warner I; Department of Chemistry, Louisiana State University, Baton Rouge, LA 70803, USA.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Jul 17; Vol. 25 (14). Date of Electronic Publication: 2020 Jul 17.
Typ publikacji:
Journal Article
MeSH Terms:
Nanoparticles/*chemistry
Neoplasms/*drug therapy
Rhodamines/*chemistry
Cell Line, Tumor ; Humans ; Hydrophobic and Hydrophilic Interactions/drug effects ; Neoplasms/pathology ; Organic Chemicals/chemistry ; Organic Chemicals/pharmacology ; Rhodamine 123/chemistry ; Rhodamine 123/pharmacology ; Rhodamines/pharmacology ; Solubility/drug effects ; Water/chemistry
Czasopismo naukowe
Tytuł:
Computational Insights into Allosteric Conformational Modulation of P-Glycoprotein by Substrate and Inhibitor Binding.
Autorzy:
Xing J; College of Basic Medical Science and College of Pharmacy, Southwest Medical University, Luzhou 646000, China.
Huang S; Key Laboratory of Biorheological Science and Technology (Ministry of Education), College of Bioengineering, Chongqing University, Chongqing 400045, China.
Heng Y; Key Laboratory of Biorheological Science and Technology (Ministry of Education), College of Bioengineering, Chongqing University, Chongqing 400045, China.
Mei H; Key Laboratory of Biorheological Science and Technology (Ministry of Education), College of Bioengineering, Chongqing University, Chongqing 400045, China.
Pan X; College of Basic Medical Science and College of Pharmacy, Southwest Medical University, Luzhou 646000, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Dec 18; Vol. 25 (24). Date of Electronic Publication: 2020 Dec 18.
Typ publikacji:
Journal Article
MeSH Terms:
Molecular Dynamics Simulation*
ATP Binding Cassette Transporter, Subfamily B, Member 1/*antagonists & inhibitors
Peptides, Cyclic/*pharmacology
ATP Binding Cassette Transporter, Subfamily B, Member 1/chemistry ; ATP Binding Cassette Transporter, Subfamily B, Member 1/metabolism ; Adenosine Triphosphate/metabolism ; Allosteric Regulation/drug effects ; Fluorescent Dyes/chemistry ; Humans ; Hydrolysis ; Peptides, Cyclic/chemistry ; Protein Conformation ; Rhodamine 123/chemistry
Czasopismo naukowe
Tytuł:
Super-Resolution Fluorescence Imaging of Arabidopsis thaliana Transfer Cell Wall Ingrowths using Pseudo-Schiff Labelling Adapted for the Use of Different Dyes.
Autorzy:
Rae AE; School of Environmental and Life Sciences, University of Newcastle, Callaghan, NSW 2308, Australia.; Research School of Biology, The Australian National University, Canberra, ACT 2601, Australia.
Wei X; School of Environmental and Life Sciences, University of Newcastle, Callaghan, NSW 2308, Australia.
Flores-Rodriguez N; Australian Centre for Microscopy and Microanalysis, University of Sydney, Sydney, NSW 2006, Australia.
McCurdy DW; School of Environmental and Life Sciences, University of Newcastle, Callaghan, NSW 2308, Australia.
Collings DA; School of Environmental and Life Sciences, University of Newcastle, Callaghan, NSW 2308, Australia.
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Źródło:
Plant & cell physiology [Plant Cell Physiol] 2020 Oct 01; Vol. 61 (10), pp. 1775-1787.
Typ publikacji:
Journal Article
MeSH Terms:
Fluorescent Dyes*
Arabidopsis/*ultrastructure
Cell Wall/*ultrastructure
Optical Imaging/*methods
Arabidopsis/growth & development ; Cell Membrane/ultrastructure ; Cellulose/metabolism ; Microscopy, Confocal ; Propidium ; Rhodamine 123
Czasopismo naukowe
Tytuł:
Search for ABCB1 Modulators Among 2-Amine-5-Arylideneimidazolones as a New Perspective to Overcome Cancer Multidrug Resistance.
Autorzy:
Kaczor A; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
Nové M; Department of Medical Microbiology and Immunobiology, Faculty of Medicine, University of Szeged, Dóm tér 10, H-6720 Szeged, Hungary.
Kincses A; Department of Medical Microbiology and Immunobiology, Faculty of Medicine, University of Szeged, Dóm tér 10, H-6720 Szeged, Hungary.
Spengler G; Department of Medical Microbiology and Immunobiology, Faculty of Medicine, University of Szeged, Dóm tér 10, H-6720 Szeged, Hungary.
Szymańska E; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
Latacz G; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
Handzlik J; Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688 Kraków, Poland.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 May 11; Vol. 25 (9). Date of Electronic Publication: 2020 May 11.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents/*pharmacology
Cell Proliferation/*drug effects
Drug Resistance, Neoplasm/*genetics
Imidazoles/*chemistry
Imidazoles/*pharmacology
Lymphoma, T-Cell/*metabolism
ATP Binding Cassette Transporter, Subfamily B/chemistry ; ATP Binding Cassette Transporter, Subfamily B/genetics ; ATP Binding Cassette Transporter, Subfamily B/metabolism ; Animals ; Antineoplastic Agents/chemistry ; Antineoplastic Agents/toxicity ; Cell Line, Tumor ; Cell Survival/drug effects ; Doxorubicin/pharmacology ; Drug Resistance, Multiple/genetics ; Humans ; Imidazoles/chemical synthesis ; In Vitro Techniques ; Inhibitory Concentration 50 ; Lymphoma, T-Cell/enzymology ; Lymphoma, T-Cell/genetics ; Mice ; Models, Molecular ; Molecular Docking Simulation ; Morpholines/chemistry ; Rhodamine 123/metabolism ; Structure-Activity Relationship ; Verapamil/pharmacology
Czasopismo naukowe
Tytuł:
Active transport of rhodamine 123 by the human multidrug transporter P-glycoprotein involves two independent outer gates.
Autorzy:
Nasim F; Institute of Medical Chemistry, Center for Pathobiochemistry and Genetics, Medical University of Vienna, Vienna, Austria.
Schmid D; Institute of Physiology, Center for Physiology and Pharmacology, Medical University of Vienna, Vienna, Austria.
Szakács G; Institute of Cancer Research, Medical University of Vienna, Vienna, Austria.
Sohail A; Institute of Pharmacology, Center for Physiology and Pharmacology, Medical University of Vienna, Vienna, Austria.
Sitte HH; Institute of Pharmacology, Center for Physiology and Pharmacology, Medical University of Vienna, Vienna, Austria.
Chiba P; Institute of Medical Chemistry, Center for Pathobiochemistry and Genetics, Medical University of Vienna, Vienna, Austria.
Stockner T; Institute of Pharmacology, Center for Physiology and Pharmacology, Medical University of Vienna, Vienna, Austria.
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Źródło:
Pharmacology research & perspectives [Pharmacol Res Perspect] 2020 Apr; Vol. 8 (2), pp. e00572.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
ATP Binding Cassette Transporter, Subfamily B, Member 1/*metabolism
Rhodamine 123/*metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1/chemistry ; Biological Transport, Active ; HEK293 Cells ; Humans
Czasopismo naukowe
Tytuł:
Glucosamine Reverses P-Glycoprotein-Mediated Multidrug Resistance in the Daunorubicin-Resistant Human Gastric Cancer Cells.
Autorzy:
Valinezhad Sani F; Department of Clinical Biochemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Isfahan University of Medical Sciences, Isfahan, Iran.
Mosaffa F; Biotechnology Research Center, Pharmaceutical Technology Institute, Mashhad University of Medical Sciences, Mashhad, Iran.; Department of Pharmaceutical Biotechnology, School of Pharmacy, Mashhad University of Medical Sciences, Mashhad, Iran.
Jamialahmadi K; Biotechnology Research Center, Pharmaceutical Technology Institute, Mashhad University of Medical Sciences, Mashhad, Iran.; Department of Medical Biotechnology and Nanotechnology, Faculty of Medicine, Mashhad University of Medical Sciences, Mashhad, Iran.
Palizban A; Department of Clinical Biochemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Isfahan University of Medical Sciences, Isfahan, Iran.
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Źródło:
Nutrition and cancer [Nutr Cancer] 2020; Vol. 72 (3), pp. 522-527. Date of Electronic Publication: 2019 Jul 10.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
ATP Binding Cassette Transporter, Subfamily B/*metabolism
Antineoplastic Agents/*pharmacology
Daunorubicin/*metabolism
Drug Resistance, Multiple/*drug effects
Glucosamine/*pharmacology
Stomach Neoplasms/*pathology
ATP Binding Cassette Transporter, Subfamily B/genetics ; ATP Binding Cassette Transporter, Subfamily B, Member 1/genetics ; ATP Binding Cassette Transporter, Subfamily B, Member 1/metabolism ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Cell Survival/drug effects ; Drug Resistance, Neoplasm/drug effects ; Humans ; RNA, Neoplasm/genetics ; Reverse Transcriptase Polymerase Chain Reaction ; Rhodamine 123/metabolism ; Stomach Neoplasms/metabolism
Czasopismo naukowe
Tytuł:
A Miniaturized Pump Out Method for Characterizing Molecule Interaction with ABC Transporters.
Autorzy:
Sevin E; Laboratoire de la Barrière Hémato-Encéphalique (LBHE), University Artois, EA 2465, F-62300 Lens, France.
Dehouck L; Laboratoire de la Barrière Hémato-Encéphalique (LBHE), University Artois, EA 2465, F-62300 Lens, France.
Versele R; Laboratoire de la Barrière Hémato-Encéphalique (LBHE), University Artois, EA 2465, F-62300 Lens, France.
Culot M; Laboratoire de la Barrière Hémato-Encéphalique (LBHE), University Artois, EA 2465, F-62300 Lens, France.
Gosselet F; Laboratoire de la Barrière Hémato-Encéphalique (LBHE), University Artois, EA 2465, F-62300 Lens, France.; Blood-brain Barrier Laboratory, Jean Perrin Faculty, Rue Jean Souvraz, 62300 Lens, France.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2019 Nov 06; Vol. 20 (22). Date of Electronic Publication: 2019 Nov 06.
Typ publikacji:
Journal Article
MeSH Terms:
Miniaturization*
ATP-Binding Cassette Transporters/*metabolism
Caco-2 Cells ; Cell Membrane Permeability/drug effects ; Fluoresceins/metabolism ; Humans ; Quinidine/pharmacology ; Rhodamine 123/metabolism
Czasopismo naukowe
Tytuł:
Effects of MDR1 1236C > T-2677G > T-3435C > T polymorphisms on the intracellular accumulation of tacrolimus, cyclosporine A, sirolimus and everolimus.
Autorzy:
Wang R; a Nursing Department, Renmin Hospital of Wuhan University , Wuhan , China.
Sun X; a Nursing Department, Renmin Hospital of Wuhan University , Wuhan , China.
Deng YS; b Department of Cardiology, Renmin Hospital of Songzi City , Songzi , China.
Qiu XW; c Renmin Hospital of Songzi City , Songzi , China.
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Źródło:
Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2019 Nov; Vol. 49 (11), pp. 1373-1378. Date of Electronic Publication: 2019 Jun 14.
Typ publikacji:
Journal Article; Video-Audio Media
MeSH Terms:
Cyclosporine/*pharmacokinetics
Everolimus/*pharmacokinetics
Sirolimus/*pharmacokinetics
Tacrolimus/*pharmacokinetics
ATP Binding Cassette Transporter, Subfamily B/genetics ; ATP Binding Cassette Transporter, Subfamily B/metabolism ; ATP Binding Cassette Transporter, Subfamily B, Member 1/metabolism ; Animals ; Drug Resistance ; Humans ; Immunosuppressive Agents/pharmacokinetics ; LLC-PK1 Cells ; Polymorphism, Single Nucleotide ; Recombinant Proteins/genetics ; Recombinant Proteins/metabolism ; Rhodamine 123/pharmacokinetics ; Swine
Czasopismo naukowe
Tytuł:
Reversal effect of FW-04-806, a macrolide dilactone compound, on multidrug resistance mediated by ABCB1 and ABCG2 in vitro and in vivo.
Autorzy:
Zhang Z; Department of Pharmacology, School of Pharmacy, Fujian Provincial Key Laboratory of Natural Medicine Pharmacology, Fujian Medical University, Fuzhou, 350122, China.
Ma C; Department of Pharmacology, School of Pharmacy, Fujian Provincial Key Laboratory of Natural Medicine Pharmacology, Fujian Medical University, Fuzhou, 350122, China.; State Key Laboratory of Oncology in South China, Collaborative Innovation Center for Cancer Medicine, Guangdong Esophageal Cancer Institute, Sun Yat-sen University Cancer Center, Guangzhou, 510060, China.
Li P; Department of Pharmacology, School of Pharmacy, Fujian Provincial Key Laboratory of Natural Medicine Pharmacology, Fujian Medical University, Fuzhou, 350122, China.
Wu M; Department of Pharmacology, School of Pharmacy, Fujian Provincial Key Laboratory of Natural Medicine Pharmacology, Fujian Medical University, Fuzhou, 350122, China.
Ye S; The First Affiliated Hospital of Fujian Medical University, Fuzhou, 350004, China. .
Fu L; State Key Laboratory of Oncology in South China, Collaborative Innovation Center for Cancer Medicine, Guangdong Esophageal Cancer Institute, Sun Yat-sen University Cancer Center, Guangzhou, 510060, China. .
Xu J; Department of Pharmacology, School of Pharmacy, Fujian Provincial Key Laboratory of Natural Medicine Pharmacology, Fujian Medical University, Fuzhou, 350122, China. .
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Źródło:
Cell communication and signaling : CCS [Cell Commun Signal] 2019 Sep 01; Vol. 17 (1), pp. 110. Date of Electronic Publication: 2019 Sep 01.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
ATP Binding Cassette Transporter, Subfamily G, Member 2/*metabolism
Antineoplastic Agents/*pharmacology
Drug Resistance, Multiple/*drug effects
Drug Resistance, Neoplasm/*drug effects
Neoplasm Proteins/*metabolism
ATP Binding Cassette Transporter, Subfamily B/metabolism ; Animals ; Antineoplastic Agents/chemistry ; Cell Proliferation/drug effects ; Cells, Cultured ; Dose-Response Relationship, Drug ; Doxorubicin/pharmacology ; Drug Screening Assays, Antitumor ; HEK293 Cells ; Humans ; K562 Cells ; KB Cells ; Mice ; Molecular Docking Simulation ; Molecular Structure ; Neoplasms, Experimental/drug therapy ; Neoplasms, Experimental/metabolism ; Neoplasms, Experimental/pathology ; Oxazoles/chemistry ; Oxazoles/pharmacology ; Rhodamine 123/pharmacology ; Signal Transduction/drug effects ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Elimination of autofluorescence in fluorescence correlation spectroscopy using the AzaDiOxaTriAngulenium (ADOTA) fluorophore in combination with time-correlated single-photon counting (TCSPC).
Autorzy:
Rich RM; Department of Molecular Biology and Immunology, Center for Commercialization of Fluorescence Technologies, University of North Texas Health Science Center, Fort Worth, TX 76107, USA.
Mummert M
Gryczynski Z
Borejdo J
Sørensen TJ
Laursen BW
Foldes-Papp Z
Gryczynski I
Fudala R
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Źródło:
Analytical and bioanalytical chemistry [Anal Bioanal Chem] 2013 May; Vol. 405 (14), pp. 4887-94. Date of Electronic Publication: 2013 Apr 06.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Artifacts*
Heterocyclic Compounds, 4 or More Rings/*chemistry
Hyaluronoglucosaminidase/*analysis
Photometry/*methods
Rhodamine 123/*chemistry
Spectrometry, Fluorescence/*methods
Heterocyclic Compounds, 4 or More Rings/analysis ; Hyaluronoglucosaminidase/chemistry ; Reproducibility of Results ; Rhodamine 123/analysis ; Sensitivity and Specificity
Czasopismo naukowe

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