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Wyszukujesz frazę ""Abou-Seri SM"" wg kryterium: Autor


Wyświetlanie 1-12 z 12
Tytuł:
Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors.
Autorzy:
Elsayed ZM; Scientific Research and Innovation Support Unit, Kafrelsheikh University, Kafrelsheikh, Egypt.
Almahli H; Department of Chemistry, University of Cambridge, Cambridge, UK.
Nocentini A; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy.
Ammara A; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy.
Supuran CT; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy.
Eldehna WM; Department of Pharmaceutical Chemistry, Kafrelsheikh University, Kafrelsheikh, Egypt.; School of Biotechnology, Badr University in Cairo, Badr City, Cairo, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Cairo University, Cairo, Egypt.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2191163.
Typ publikacji:
Journal Article
MeSH Terms:
Carbonic Anhydrases*/metabolism
Neoplasms*/pathology
Humans ; Carbonic Anhydrase IX ; Molecular Structure ; Structure-Activity Relationship ; Carboxylic Acids/pharmacology ; Carbonic Anhydrase Inhibitors ; Quinazolines/pharmacology ; Antigens, Neoplasm/metabolism
Czasopismo naukowe
Tytuł:
New proapoptotic chemotherapeutic agents based on the quinolone-3-carboxamide scaffold acting by VEGFR-2 inhibition.
Autorzy:
El-Fakharany ZS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, October University for Modern Sciences and Arts, Cairo, 12451, Egypt.
Nissan YM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, October University for Modern Sciences and Arts, Cairo, 12451, Egypt.; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, 11562, Egypt.
Sedky NK; Department of Biochemistry, School of Life and Medical Sciences, University of Hertfordshire Hosted By Global Academic Foundation, New Administrative Capital, Cairo, Egypt.
Arafa RK; Biomedical Sciences Program, University of Science and Technology, Zewail City of Science and Technology, October Gardens, 6th of October City, Giza, 12578, Egypt. .; Drug Design and Discovery Lab, Zewail City of Science and Technology, Cairo, 12578, Egypt. .
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, 11562, Egypt. .
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Źródło:
Scientific reports [Sci Rep] 2023 Jul 13; Vol. 13 (1), pp. 11346. Date of Electronic Publication: 2023 Jul 13.
Typ publikacji:
Journal Article
MeSH Terms:
Quinolones*/pharmacology
Antineoplastic Agents*/chemistry
Humans ; Molecular Structure ; Structure-Activity Relationship ; Caspase 7/metabolism ; Sorafenib/pharmacology ; Vascular Endothelial Growth Factor Receptor-2/metabolism ; Molecular Docking Simulation ; bcl-2-Associated X Protein ; Protein Kinase Inhibitors/pharmacology ; Drug Screening Assays, Antitumor ; Cell Proliferation ; Drug Design
Czasopismo naukowe
Tytuł:
Design and synthesis of novel cytotoxic fluoroquinolone analogs through topoisomerase inhibition, cell cycle arrest, and apoptosis.
Autorzy:
Elanany MA; Department of Pharmaceutical Chemistry, School of Pharmacy and Pharmaceutical Industries, Badr University in Cairo (BUC), Badr City, 11829, Cairo, Egypt. .
Osman EEA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, 11562, Egypt.
Gedawy EM; Department of Pharmaceutical Chemistry, School of Pharmacy and Pharmaceutical Industries, Badr University in Cairo (BUC), Badr City, 11829, Cairo, Egypt.; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo, 11562, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, 11562, Egypt. .
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Źródło:
Scientific reports [Sci Rep] 2023 Mar 13; Vol. 13 (1), pp. 4144. Date of Electronic Publication: 2023 Mar 13.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Fluoroquinolones*/pharmacology
Antineoplastic Agents*/chemistry
Humans ; Molecular Structure ; Structure-Activity Relationship ; Moxifloxacin/pharmacology ; Cell Proliferation ; Cell Cycle Checkpoints ; Cell Line, Tumor ; Ciprofloxacin/pharmacology ; Apoptosis ; Ofloxacin/pharmacology ; Drug Screening Assays, Antitumor ; Cell Cycle
Czasopismo naukowe
Tytuł:
Multi-stage structure-based virtual screening approach towards identification of potential SARS-CoV-2 NSP13 helicase inhibitors.
Autorzy:
El Hassab MA; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, King Salman International University (KSIU), Ras Sudr, Egypt.
Eldehna WM; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Kafrelsheikh University, Kafrelsheikh, Egypt.
Al-Rashood ST; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.
Alharbi A; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.
Eskandrani RO; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.
Alkahtani HM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.
Elkaeed EB; Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh, Saudi Arabia.
Abou-Seri SM; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Cairo University, Cairo, Egypt.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2022 Dec; Vol. 37 (1), pp. 563-572.
Typ publikacji:
Journal Article
MeSH Terms:
Drug Discovery*
Molecular Docking Simulation*
COVID-19 Drug Treatment*
Exoribonucleases/*antagonists & inhibitors
High-Throughput Screening Assays/*methods
SARS-CoV-2/*drug effects
Viral Nonstructural Proteins/*antagonists & inhibitors
COVID-19/virology ; Catalytic Domain ; Humans ; Ligands ; Molecular Dynamics Simulation ; Quantitative Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
New 5-Aryl-1,3,4-Thiadiazole-Based Anticancer Agents: Design, Synthesis, In Vitro Biological Evaluation and In Vivo Radioactive Tracing Studies.
Autorzy:
El-Masry RM; Organic Chemistry Department, Faculty of Pharmacy, October University for Modern Sciences and Arts (MSA), October 6 City 12451, Egypt.
Essa BM; Radioactive Isotopes and Generator Department, Hot Labs Center, Egyptian Atomic Energy Authority, P.O. Box 13759, Cairo 13759, Egypt.
Selim AA; Labeled Compounds Department, Hot Labs Center, Egyptian Atomic Energy Authority, P.O. Box 13759, Cairo 13759, Egypt.
El-Emam SZ; Department of Pharmacology and Toxicology, Faculty of Pharmacy, October 6 University (O6U), October 6 City 12585, Egypt.
Mohamed KO; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11565, Egypt.
Sakr TM; Radioactive Isotopes and Generator Department, Hot Labs Center, Egyptian Atomic Energy Authority, P.O. Box 13759, Cairo 13759, Egypt.
Kadry HH; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11565, Egypt.
Taher AT; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11565, Egypt.; Department of Organic Pharmaceutical Chemistry, Faculty of Pharmacy, October 6 University (O6U), October 6 City 12585, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11565, Egypt.
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Źródło:
Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2022 Nov 27; Vol. 15 (12). Date of Electronic Publication: 2022 Nov 27.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Multi-Step In Silico Discovery of Natural Drugs against COVID-19 Targeting Main Protease.
Autorzy:
Elkaeed EB; Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh 13713, Saudi Arabia.
Youssef FS; Department of Pharmacognosy, Faculty of Pharmacy, Ain-Shams University, Abbasia, Cairo 11566, Egypt.
Eissa IH; Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo 11884, Egypt.
Elkady H; Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo 11884, Egypt.
Alsfouk AA; Department of Pharmaceutical Sciences, College of Pharmacy, Princess Nourah bint Abdulrahman University, P.O. Box 84428, Riyadh 11671, Saudi Arabia.
Ashour ML; Department of Pharmacognosy, Faculty of Pharmacy, Ain-Shams University, Abbasia, Cairo 11566, Egypt.; Department of Pharmaceutical Sciences, Pharmacy Program, Batterjee Medical College, Jeddah 21442, Saudi Arabia.
El Hassab MA; Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), South Sinai 46612, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo P.O. Box 11562, Egypt.
Metwaly AM; Pharmacognosy and Medicinal Plants Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo 11884, Egypt.; Biopharmaceutical Product Research Department, Genetic Engineering and Biotechnology Research Institute, City of Scientific Research and Technological Applications, Alexandria 21934, Egypt.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Jun 21; Vol. 23 (13). Date of Electronic Publication: 2022 Jun 21.
Typ publikacji:
Journal Article
MeSH Terms:
COVID-19 Drug Treatment*
Antiviral Agents/chemistry ; Antiviral Agents/pharmacology ; Cysteine Endopeptidases/metabolism ; Humans ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Peptide Hydrolases/metabolism ; Protease Inhibitors/chemistry ; Protease Inhibitors/pharmacology ; SARS-CoV-2 ; Viral Nonstructural Proteins/metabolism
Czasopismo naukowe
Tytuł:
Comparative Study of the Synthetic Approaches and Biological Activities of the Bioisosteres of 1,3,4-Oxadiazoles and 1,3,4-Thiadiazoles over the Past Decade.
Autorzy:
El-Masry RM; Organic Chemistry Department, Faculty of Pharmacy, October University for Modern Sciences and Arts (MSA), 6th of October City 12451, Egypt.
Kadry HH; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt.
Taher AT; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt.; Department of Organic Pharmaceutical Chemistry, Faculty of Pharmacy, October 6 University (O6U), 6th of October City 12585, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Apr 22; Vol. 27 (9). Date of Electronic Publication: 2022 Apr 22.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Thiadiazoles*/pharmacology
Drug Design ; Oxadiazoles/pharmacology ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Dual PI3K/Akt Inhibitors Bearing Coumarin-Thiazolidine Pharmacophores as Potential Apoptosis Inducers in MCF-7 Cells.
Autorzy:
Abdelnaby RM; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Heliopolis University, Cairo 11785, Egypt.
Rateb HS; Pharmaceutical Chemistry Department, Faculty of Pharmaceutical Science and Drug Manufacturing, Misr University for Science and Technology, 6th of October City 12585, Egypt.
Ali O; Egyptian Drug Authority, Cairo 12618, Egypt.
Saad AS; Pharmacology and Toxicology Department, Faculty of Pharmacy, Port Said University, Port Said 42511, Egypt.
Nadeem RI; Pharmacology and Toxicology Department, Faculty of Pharmacy, Heliopolis University, Cairo 11785, Egypt.
Abou-Seri SM; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt.
Amin KM; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt.
Younis NS; Pharmaceutical Sciences Department, Faculty of Clinical Pharmacy, King Faisal University, Al Hofuf 31982, Al-Ahsa, Saudi Arabia.
Abdelhady R; Pharmacology and Toxicology Department, Faculty of Pharmacy, Fayoum University, Fayoum 63514, Egypt.
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Źródło:
Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2022 Mar 31; Vol. 15 (4). Date of Electronic Publication: 2022 Mar 31.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Development of novel isatin-nicotinohydrazide hybrids with potent activity against susceptible/resistant Mycobacterium tuberculosis and bronchitis causing-bacteria.
Autorzy:
Elsayed ZM; Faculty of Pharmacy, Scientific Research and Innovation Support Unit, Kafrelsheikh University, Kafrelsheikh, Egypt.
Eldehna WM; Faculty of Pharmacy, Scientific Research and Innovation Support Unit, Kafrelsheikh University, Kafrelsheikh, Egypt.; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Kafrelsheikh University, Kafrelsheikh, Egypt.
Abdel-Aziz MM; The Regional Center for Mycology & Biotechnology, Al-Azhar University, Cairo, Egypt.
El Hassab MA; Department of Pharmaceutical Chemistry, School of Pharmacy, Badr University in Cairo, Badr City, Egypt.
Elkaeed EB; Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Ad Diriyah, Saudi Arabia.; Faculty of Pharmacy (Boys), Department of Pharmaceutical Organic Chemistry, Al-Azhar University, Cairo, Egypt.
Al-Warhi T; Department of Chemistry, College of Science, Princess Nourah bint Abdulrahman University, Riyadh, Saudi Arabia.
Abdel-Aziz HA; Department of Applied Organic Chemistry, National Research Center, Giza, Egypt.
Abou-Seri SM; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Cairo University, Cairo, Egypt.
Mohammed ER; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Cairo University, Cairo, Egypt.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2021 Dec; Vol. 36 (1), pp. 384-393.
Typ publikacji:
Journal Article
MeSH Terms:
Alcohol Oxidoreductases/*antagonists & inhibitors
Anti-Bacterial Agents/*chemical synthesis
Bacterial Proteins/*antagonists & inhibitors
Drug Resistance, Bacterial/*drug effects
Hydrazines/*chemistry
Isatin/*chemistry
Mycobacterium tuberculosis/*enzymology
Alcohol Oxidoreductases/chemistry ; Alcohol Oxidoreductases/metabolism ; Anti-Bacterial Agents/pharmacology ; Bacterial Proteins/chemistry ; Bacterial Proteins/metabolism ; Binding Sites ; Bordetella pertussis/chemistry ; Bordetella pertussis/enzymology ; Bordetella pertussis/isolation & purification ; Bronchitis/drug therapy ; Bronchitis/microbiology ; Drug Design ; Drug Resistance, Bacterial/genetics ; Haemophilus influenzae/chemistry ; Haemophilus influenzae/enzymology ; Haemophilus influenzae/isolation & purification ; Isoniazid/pharmacology ; Klebsiella pneumoniae/chemistry ; Klebsiella pneumoniae/enzymology ; Klebsiella pneumoniae/isolation & purification ; Microbial Sensitivity Tests ; Molecular Docking Simulation ; Moraxella catarrhalis/chemistry ; Moraxella catarrhalis/enzymology ; Moraxella catarrhalis/isolation & purification ; Mycobacterium tuberculosis/chemistry ; Mycobacterium tuberculosis/isolation & purification ; Protein Binding ; Protein Conformation ; Protein Interaction Domains and Motifs ; Streptococcus pneumoniae/chemistry ; Streptococcus pneumoniae/enzymology ; Streptococcus pneumoniae/isolation & purification ; Streptomycin/pharmacology ; Structure-Activity Relationship ; Tuberculosis/drug therapy ; Tuberculosis/microbiology
Czasopismo naukowe
Tytuł:
Novel benzofuran-based sulphonamides as selective carbonic anhydrases IX and XII inhibitors: synthesis and in vitro biological evaluation.
Autorzy:
Abdelrahman MA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University, Badr City, Egypt.
Eldehna WM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt.
Nocentini A; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy.
Ibrahim HS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University, Badr City, Egypt.
Almahli H; Chemistry Research Laboratory, Department of Chemistry, University of Oxford, Oxford, UK.
Abdel-Aziz HA; Department of Applied Organic Chemistry, National Research Center, Dokki, Egypt.
Abou-Seri SM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt.
Supuran CT; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Firenze, Italy.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2020 Dec; Vol. 35 (1), pp. 298-305.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents/*pharmacology
Benzofurans/*pharmacology
Carbonic Anhydrase IX/*antagonists & inhibitors
Carbonic Anhydrase Inhibitors/*pharmacology
Carbonic Anhydrases/*metabolism
Sulfonamides/*pharmacology
Antigens, Neoplasm/metabolism ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Benzofurans/chemistry ; Carbonic Anhydrase IX/metabolism ; Carbonic Anhydrase Inhibitors/chemical synthesis ; Carbonic Anhydrase Inhibitors/chemistry ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Humans ; Molecular Docking Simulation ; Molecular Structure ; Structure-Activity Relationship ; Sulfonamides/chemical synthesis ; Sulfonamides/chemistry
Czasopismo naukowe
Tytuł:
Synthesis and bioactivity evaluation of new 6-aryl-5-cyano thiouracils as potential antimicrobial and anticancer agents.
Autorzy:
Taher AT; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cairo University, Kasr El-Aini Street, Cairo, P.O. Box, 11562, Egypt. />Abou-Seri SM
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2012 Aug 17; Vol. 17 (8), pp. 9868-86. Date of Electronic Publication: 2012 Aug 17.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Infective Agents/*chemistry
Anti-Infective Agents/*pharmacology
Antineoplastic Agents/*chemistry
Antineoplastic Agents/*pharmacology
Thiouracil/*chemistry
Thiouracil/*pharmacology
Cell Line, Tumor ; Drug Screening Assays, Antitumor ; Fungi/drug effects ; Gram-Negative Bacteria/drug effects ; Gram-Positive Bacteria/drug effects ; Humans ; Inhibitory Concentration 50 ; Microbial Sensitivity Tests
Czasopismo naukowe
    Wyświetlanie 1-12 z 12

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