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Wyszukujesz frazę ""Adrenergic alpha-1 Receptor Agonists"" wg kryterium: Temat


Tytuł:
Comparison of the electromechanical responsiveness of alpha-1-adrenoceptor stimulation in ventricles of normal and cardiomyopathic hamsters.
Autorzy:
Chen WP; Pharmacological Institute, College of Medicine, National Taiwan University, Taipei, Taiwan, ROC.
Su MJ
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Źródło:
Journal of biomedical science [J Biomed Sci] 2001 Nov-Dec; Vol. 8 (6), pp. 453-61.
Typ publikacji:
Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Cardiomyopathies/*physiopathology
Heart Ventricles/*physiopathology
Receptors, Adrenergic, alpha-1/*physiology
Action Potentials/drug effects ; Action Potentials/physiology ; Adrenergic Agents/pharmacology ; Adrenergic alpha-1 Receptor Agonists ; Animals ; Biomechanical Phenomena ; Calcium/metabolism ; Cricetinae ; Drug Interactions ; Electrophysiology ; Heart Ventricles/drug effects ; In Vitro Techniques ; Male ; Mesocricetus ; Models, Animal ; Phenylephrine/pharmacology ; Phorbol 12,13-Dibutyrate/pharmacology ; Propranolol/pharmacology ; Staurosporine/pharmacology
Czasopismo naukowe
Tytuł:
Activation of alpha 1-adrenoceptors is not essential for the mediation of ischaemic preconditioning in rat heart.
Autorzy:
Vasara E; Laboratory of Animal Physiology, Department of Zoology, School of Biology, Aristotle University of Thessaloniki, Thessaloniki, Greece.
Seraskeris S
Lazou A
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Źródło:
Clinical and experimental pharmacology & physiology [Clin Exp Pharmacol Physiol] 2002 Jan-Feb; Vol. 29 (1-2), pp. 11-7.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Heart/*physiology
Ischemic Preconditioning, Myocardial/*methods
Receptors, Adrenergic, alpha-1/*metabolism
Adrenergic Antagonists/pharmacology ; Adrenergic Antagonists/therapeutic use ; Adrenergic alpha-1 Receptor Agonists ; Adrenergic alpha-1 Receptor Antagonists ; Adrenergic alpha-Agonists/pharmacology ; Adrenergic alpha-Agonists/therapeutic use ; Animals ; Heart/drug effects ; In Vitro Techniques ; Male ; Myocardial Ischemia/metabolism ; Myocardial Ischemia/prevention & control ; Rats ; Rats, Wistar ; Ventricular Function, Left/drug effects ; Ventricular Function, Left/physiology
Czasopismo naukowe
Tytuł:
Uneven changes in circulating blood cell counts with adrenergic stimulation to the canine spleen.
Autorzy:
Ojiri Y; Department of Pharmacology, School of Medicine, Faculty of Medicine, University of the Ryukyus, Okinawa, Japan. />Noguchi K
Shiroma N
Matsuzaki T
Sakanashi M
Sakanashi M
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Źródło:
Clinical and experimental pharmacology & physiology [Clin Exp Pharmacol Physiol] 2002 Jan-Feb; Vol. 29 (1-2), pp. 53-9.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Adrenergic Agonists/*pharmacology
Blood Platelets/*drug effects
Erythrocytes/*drug effects
Leukocytes/*drug effects
Spleen/*drug effects
Adrenergic alpha-1 Receptor Agonists ; Animals ; Blood Cell Count/methods ; Blood Cell Count/statistics & numerical data ; Blood Platelets/cytology ; Blood Platelets/physiology ; Dogs ; Erythrocytes/cytology ; Erythrocytes/physiology ; Female ; Leukocytes/cytology ; Leukocytes/physiology ; Male ; Receptors, Adrenergic, alpha-1/physiology ; Spleen/physiology
Czasopismo naukowe
Tytuł:
Salivary glands and noradrenergic transmission in diabetic rats.
Autorzy:
Vatta MS; Catedra de Fisiologia, Facultad de Farmacia y Bioquimica, Universidad de Buenos Aires, Junin 956-7mo piso, 1113 Buenos Aires, Argentina.
Hope SI
Prendes GM
Bianciotti LG
Elverdin JC
Fernandez BE
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Źródło:
Autonomic & autacoid pharmacology [Auton Autacoid Pharmacol] 2002 Apr; Vol. 22 (2), pp. 65-71.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Diabetes Mellitus, Experimental/*metabolism
Norepinephrine/*metabolism
Salivary Glands/*metabolism
Adrenergic Agonists/pharmacology ; Adrenergic alpha-1 Receptor Agonists ; Animals ; Dose-Response Relationship, Drug ; Male ; Rats ; Rats, Wistar ; Receptors, Adrenergic, alpha-1/metabolism ; Receptors, Adrenergic, beta/metabolism ; Salivary Glands/drug effects
Czasopismo naukowe
Tytuł:
Physiological antagonism between ventricular beta 1-adrenoceptors and alpha 1-adrenoceptors but no evidence for beta 2- and beta 3-adrenoceptor function in murine heart.
Autorzy:
Heubach JF; Institut für Pharmakologie und Toxikologie, Medizinische Fakultät Carl Gustav Carus der TU Dresden, D-01307 Dresden, Germany.
Rau T
Eschenhagen T
Ravens U
Kaumann AJ
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2002 May; Vol. 136 (2), pp. 217-29.
Typ publikacji:
Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptors, Adrenergic, alpha-1/*physiology
Receptors, Adrenergic, beta-1/*physiology
Receptors, Adrenergic, beta-2/*physiology
Receptors, Adrenergic, beta-3/*physiology
Adrenergic alpha-1 Receptor Agonists ; Adrenergic alpha-1 Receptor Antagonists ; Adrenergic beta-1 Receptor Agonists ; Adrenergic beta-1 Receptor Antagonists ; Adrenergic beta-2 Receptor Agonists ; Adrenergic beta-2 Receptor Antagonists ; Adrenergic beta-3 Receptor Agonists ; Adrenergic beta-3 Receptor Antagonists ; Animals ; Dose-Response Relationship, Drug ; Heart Ventricles/drug effects ; In Vitro Techniques ; Male ; Mice ; Mice, Inbred C57BL ; Myocardial Contraction/drug effects ; Myocardial Contraction/physiology ; Sinoatrial Node/drug effects ; Sinoatrial Node/physiology ; Ventricular Function
Czasopismo naukowe
Tytuł:
Alpha 1-adrenoceptor effects mediated by protein kinase C alpha in human cultured prostatic stromal cells.
Autorzy:
Preston A; School of Medical Sciences, RMIT University, Bundoora, Victoria 3083, Australia. />Haynes JM
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2003 Jan; Vol. 138 (1), pp. 218-24.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Prostate/*cytology
Prostate/*enzymology
Protein Kinase C/*metabolism
Receptors, Adrenergic, alpha-1/*metabolism
Stromal Cells/*enzymology
Adrenergic alpha-1 Receptor Agonists ; Adrenergic alpha-1 Receptor Antagonists ; Aged ; Cell Size/drug effects ; Cells, Cultured ; Dose-Response Relationship, Drug ; Humans ; Male ; Phenylephrine/pharmacology ; Prostate/drug effects ; Prostate/metabolism ; Protein Kinase C/antagonists & inhibitors ; Protein Kinase C-alpha ; Protein Transport/drug effects ; Protein Transport/physiology ; Stromal Cells/cytology ; Stromal Cells/drug effects
Czasopismo naukowe
Tytuł:
Functional characterization of alpha 1-adrenoceptor subtypes in vascular tissues using different experimental approaches: a comparative study.
Autorzy:
Gisbert R; Departament de Farmacologia, Facultat de Farmacia, Universitat de València, Avda, Vincent Andres Estelles s/n 46100, Burjassot, Valencia, Spain.
Madrero Y
Sabino V
Noguera MA
Ivorra MD
D'Ocon P
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2003 Jan; Vol. 138 (2), pp. 359-68.
Typ publikacji:
Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptors, Adrenergic, alpha-1/*physiology
Vasoconstriction/*physiology
Adrenergic Agonists/pharmacology ; Adrenergic Antagonists/pharmacology ; Adrenergic alpha-1 Receptor Agonists ; Adrenergic alpha-1 Receptor Antagonists ; Animals ; Aorta/drug effects ; Aorta/physiology ; Dose-Response Relationship, Drug ; Endothelium, Vascular/drug effects ; Endothelium, Vascular/physiology ; Female ; In Vitro Techniques ; Rats ; Rats, Wistar ; Tail/blood supply ; Tail/drug effects ; Tail/physiology ; Vasoconstriction/drug effects
Czasopismo naukowe
Tytuł:
Modulation of intracellular Ca2+ via L-type calcium channels in heart cells by the autoantibody directed against the second extracellular loop of the alpha1-adrenoceptors.
Autorzy:
Bkaily G; Department of Anatomy and Cell Biology, Faculty of Medicine, Université de Sherbrooke, Sherbrooke, QC J1H 5N4, Canada. />El-Bizri N
Bui M
Sukarieh R
Jacques D
Fu ML
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Źródło:
Canadian journal of physiology and pharmacology [Can J Physiol Pharmacol] 2003 Mar; Vol. 81 (3), pp. 234-46.
Typ publikacji:
Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Autoantibodies/*pharmacology
Calcium/*metabolism
Calcium Channels, L-Type/*physiology
Myocytes, Cardiac/*physiology
Receptors, Adrenergic, alpha-1/*physiology
Adrenergic alpha-1 Receptor Agonists ; Aniline Compounds ; Animals ; Calcium Channel Blockers/pharmacology ; Calcium Channels, T-Type/physiology ; Cells, Cultured ; Chick Embryo ; Fetus ; Fluorescent Dyes ; Humans ; Methoxamine/pharmacology ; Myocardial Contraction ; Myocytes, Cardiac/drug effects ; Nifedipine/pharmacology ; Patch-Clamp Techniques ; Potassium Channels/drug effects ; Potassium Channels/physiology ; Receptors, Adrenergic, alpha-1/immunology ; Sodium Channels/drug effects ; Sodium Channels/physiology ; Xanthenes
Czasopismo naukowe
Tytuł:
Myocardial adenosine does not correlate with the protection mediated by ischaemic or pharmacological preconditioning in rat heart.
Autorzy:
Vasara E; Laboratory of Animal Physiology, Department of Zoology, School of Biology, Aristotle University of Thessaloniki, Thessaloniki, Greece.
Katharou I
Lazou A
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Źródło:
Clinical and experimental pharmacology & physiology [Clin Exp Pharmacol Physiol] 2003 May-Jun; Vol. 30 (5-6), pp. 350-6.
Typ publikacji:
Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Adenosine/*metabolism
Cardiotonic Agents/*therapeutic use
Ischemic Preconditioning, Myocardial/*methods
Myocardial Ischemia/*metabolism
Myocardium/*metabolism
Adrenergic alpha-1 Receptor Agonists ; Animals ; Cardiotonic Agents/pharmacology ; Male ; Myocardial Ischemia/drug therapy ; Rats ; Rats, Wistar ; Receptors, Adrenergic, alpha-1/metabolism
Czasopismo naukowe
Tytuł:
Mechanism of the negative inotropic effects of alpha 1-adrenoceptor agonists on mouse myocardium.
Autorzy:
Varma DR; Department of Pharmacology and Theraputics, McGill University, Montréal, QC H3G 1Y6, Canada. />Rindt H
Chemtob S
Mulay S
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Źródło:
Canadian journal of physiology and pharmacology [Can J Physiol Pharmacol] 2003 Aug; Vol. 81 (8), pp. 783-9.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Adrenergic alpha-1 Receptor Agonists*
Adrenergic alpha-Agonists/*pharmacology
Myocardial Contraction/*drug effects
Myocardium/*metabolism
Animals ; Depression, Chemical ; Dose-Response Relationship, Drug ; In Vitro Techniques ; Male ; Mice ; Myocardial Contraction/physiology ; Phenylephrine/pharmacology ; Protein Kinase C/metabolism ; Receptors, Adrenergic, alpha-1/metabolism
Czasopismo naukowe
Tytuł:
Bulk is a determinant of oxymetazoline affinity for the alpha1A-adrenergic receptor.
Autorzy:
McCune D; Department of Molecular Cardiology, Lerner Research Institute, Cleveland Clinic Foundation, Cleveland, Ohio 44195, USA.
Gaivin R
Rorabaugh B
Perez D
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Źródło:
Receptors & channels [Recept Channels] 2004; Vol. 10 (3-4), pp. 109-16.
Typ publikacji:
Journal Article; Research Support, U.S. Gov't, P.H.S.
MeSH Terms:
Oxymetazoline/*metabolism
Receptors, Adrenergic, alpha-1/*metabolism
Adrenergic alpha-1 Receptor Agonists ; Adrenergic alpha-1 Receptor Antagonists ; Amino Acid Sequence ; Animals ; COS Cells ; Chlorocebus aethiops ; Models, Molecular ; Molecular Sequence Data ; Mutation ; Rats ; Receptors, Adrenergic, alpha-1/genetics ; Sequence Alignment
Czasopismo naukowe
Tytuł:
A randomized crossover study to evaluate Ro 115-1240, a selective alpha1A/1L-adrenoceptor partial agonist in women with stress urinary incontinence.
Autorzy:
Musselman DM; Hoffmann-La Roche, Inc., Nutley, NJ, USA. />Ford AP
Gennevois DJ
Harbison ML
Laurent AL
Mokatrin AS
Stoltz RR
Blue DR
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Źródło:
BJU international [BJU Int] 2004 Jan; Vol. 93 (1), pp. 78-83.
Typ publikacji:
Clinical Trial; Journal Article; Multicenter Study; Randomized Controlled Trial
MeSH Terms:
Adrenergic alpha-1 Receptor Agonists*
Adrenergic alpha-Agonists/*therapeutic use
Urinary Incontinence, Stress/*drug therapy
Adolescent ; Adrenergic alpha-Agonists/adverse effects ; Adult ; Aged ; Cross-Over Studies ; Female ; Humans ; Imidazoles/therapeutic use ; Middle Aged ; Sulfonamides/therapeutic use
Czasopismo naukowe
Tytuł:
Pharmacological characteristics of Ro 115-1240, a selective alpha1A/1L-adrenoceptor partial agonist: a potential therapy for stress urinary incontinence.
Autorzy:
Blue DR; Roche Palo Alto, Palo Alto, CA, USA. />Daniels DV
Gever JR
Jett MF
O'Yang C
Tang HM
Williams TJ
Ford AP
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Źródło:
BJU international [BJU Int] 2004 Jan; Vol. 93 (1), pp. 162-70.
Typ publikacji:
Journal Article
MeSH Terms:
Adrenergic alpha-1 Receptor Agonists*
Adrenergic alpha-Agonists/*therapeutic use
Urinary Incontinence, Stress/*drug therapy
Adrenergic alpha-Agonists/pharmacology ; Animals ; Cricetinae ; Dose-Response Relationship, Drug ; Ethanolamines/pharmacology ; Female ; Heart Rate/drug effects ; Imidazoles/pharmacology ; Imidazoles/therapeutic use ; Male ; Models, Biological ; Prazosin/metabolism ; Rabbits ; Sulfonamides/pharmacology ; Sulfonamides/therapeutic use ; Swine ; Swine, Miniature
Czasopismo naukowe
Tytuł:
Protein kinase Czeta regulates phospholipase D activity in rat-1 fibroblasts expressing the alpha1A adrenergic receptor.
Autorzy:
Parmentier JH; Department of Pharmacology and Center for Connective Tissue Diseases and Vascular Biology, College of Medicine, The University of Tennessee Health Science Center, 874 Union Avenue, Memphis, TN 38163, USA. />Gandhi GK
Wiggins MT
Saeed AE
Bourgoin SG
Malik KU
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Źródło:
BMC cell biology [BMC Cell Biol] 2004 Jan 21; Vol. 5, pp. 4. Date of Electronic Publication: 2004 Jan 21.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
MeSH Terms:
Adrenergic alpha-1 Receptor Agonists*
Fibroblasts/*enzymology
Phospholipase D/*metabolism
Protein Kinase C/*physiology
Adrenergic alpha-Agonists/pharmacology ; Animals ; Cell Line ; Enzyme Inhibitors/pharmacology ; Fibroblasts/drug effects ; Fibroblasts/metabolism ; Gene Expression ; Phenylephrine/pharmacology ; Protein Kinase C/antagonists & inhibitors ; Rats ; Receptors, Adrenergic, alpha-1/genetics ; Receptors, Adrenergic, alpha-1/metabolism ; Tetradecanoylphorbol Acetate/pharmacology
Czasopismo naukowe
Tytuł:
Central nervous alpha1-adrenoceptor stimulation induces duodenal luminal release of melatonin.
Autorzy:
Sjöblom M; Department of Neuroscience, Division of Physiology, Uppsala University, Uppsala, Sweden. />Flemström G
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Źródło:
Journal of pineal research [J Pineal Res] 2004 Mar; Vol. 36 (2), pp. 103-8.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Brain/*metabolism
Duodenum/*metabolism
Melatonin/*metabolism
Receptors, Adrenergic, alpha-1/*metabolism
Adrenergic alpha-1 Receptor Agonists ; Animals ; Bicarbonates/metabolism ; Brain/drug effects ; Chromatography, High Pressure Liquid ; Duodenum/drug effects ; Injections, Intraventricular ; Melatonin/analysis ; Phenylephrine/administration & dosage ; Phenylephrine/pharmacology ; Rats ; Time Factors
Czasopismo naukowe

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