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Wyszukujesz frazę ""Almehizia, Abdulrahman A."" wg kryterium: Autor


Wyświetlanie 1-16 z 16
Tytuł:
Nanoparticles of a Pyrazolo-Pyridazine Derivative as Potential EGFR and CDK-2 Inhibitors: Design, Structure Determination, Anticancer Evaluation and In Silico Studies.
Autorzy:
Hashem HE; Department of Chemistry, Faculty of Women, Ain Shams University, Cairo 11757, Egypt.
Amr AEE; Applied Organic Chemistry Department, National Research Center, Cairo 12622, Egypt.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Naglah AM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Kariuki BM; School of Chemistry, Cardiff University, Main Building, Park Place, Cardiff CF10 3AT, UK.
Eassa HA; Department of Pharmaceutics and Pharmaceutical Technology, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo 11754, Egypt.; Department of Pharmaceutical Sciences, School of Pharmacy and Physician Assistant Studies, University of Saint Joseph, West Hartford, CT 06117, USA.
Nossier ES; Department of Pharmaceutical Medicinal Chemistry and Drug Design, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo 11754, Egypt.; The National Committee of Drugs, Academy of Scientific Research and Technology, Cairo 11516, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Oct 25; Vol. 28 (21). Date of Electronic Publication: 2023 Oct 25.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents*/chemistry
Pyridazines*/pharmacology
Nanoparticles*
Humans ; Structure-Activity Relationship ; Cell Proliferation ; Cell Line, Tumor ; ErbB Receptors/metabolism ; Amines/pharmacology ; Molecular Structure ; Molecular Docking Simulation ; Drug Screening Assays, Antitumor ; Protein Kinase Inhibitors/chemistry
Czasopismo naukowe
Tytuł:
In Vitro Evaluation and Bioinformatics Analysis of Schiff Bases Bearing Pyrazole Scaffold as Bioactive Agents: Antioxidant, Anti-Diabetic, Anti-Alzheimer, and Anti-Arthritic.
Autorzy:
Alkahtani HM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Al-Omar MA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Obaidullah AJ; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Zen AA; Chemistry & Forensics Department, Clifton Campus, Nottingham Trent University, Nottingham Ng11 8NS, UK.
Hassan AS; Organometallic and Organometalloid Chemistry Department, National Research Centre, Cairo 12622, Egypt.
Aboulthana WM; Biochemistry Department, Biotechnology Research Institute, National Research Centre, Cairo 12622, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Oct 17; Vol. 28 (20). Date of Electronic Publication: 2023 Oct 17.
Typ publikacji:
Journal Article
MeSH Terms:
Antioxidants*/pharmacology
Antioxidants*/chemistry
Schiff Bases*/chemistry
Acetylcholinesterase/metabolism ; Pyrazoles ; alpha-Amylases ; Molecular Structure ; Molecular Docking Simulation
Czasopismo naukowe
Tytuł:
Investigations of Electronic, Structural, and In Silico Anticancer Potential of Persuasive Phytoestrogenic Isoflavene-Based Mannich Bases.
Autorzy:
Mutahir S; School of Chemistry and Chemical Engineering, Linyi University, Linyi 276000, China.; Department of Chemistry, University of Sialkot, Sialkot 51300, Pakistan.
Khan MA; School of Chemistry and Chemical Engineering, Linyi University, Linyi 276000, China.; Department of Chemistry, University of Sialkot, Sialkot 51300, Pakistan.
Mushtaq M; Department of Chemistry, University of Sialkot, Sialkot 51300, Pakistan.
Deng H; School of Pharmacy, Nanjing University of Chinese Medicine, Nanjing 210023, China.
Naglah AM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Al-Omar MA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Alrayes FI; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Kalmouch A; Peptide Chemistry Department, Chemical Industries Research Institute, National Research Centre, Cairo 12622, Egypt.
El-Mowafi SA; Peptide Chemistry Department, Chemical Industries Research Institute, National Research Centre, Cairo 12622, Egypt.
Refat MS; Department of Chemistry, Faculty of Science, Port Said University, Port Said 42526, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Aug 06; Vol. 28 (15). Date of Electronic Publication: 2023 Aug 06.
Typ publikacji:
Journal Article
MeSH Terms:
Phytoestrogens*/pharmacology
Mannich Bases*/pharmacology
Mannich Bases*/chemistry
Molecular Docking Simulation ; Ligands
Czasopismo naukowe
Tytuł:
Targeting Transcriptional CDKs 7, 8, and 9 with Anilinopyrimidine Derivatives as Anticancer Agents: Design, Synthesis, Biological Evaluation and In Silico Studies.
Autorzy:
Eskandrani R; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Al-Rasheed LS; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Ansari SA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Bakheit AH; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Almehizia AA; Drug Exploration and Development (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Almutairi M; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Alkahtani HM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 May 23; Vol. 28 (11). Date of Electronic Publication: 2023 May 23.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents*/chemistry
Neoplasms*
Humans ; Molecular Structure ; Structure-Activity Relationship ; Ligands ; Molecular Docking Simulation ; Cyclin-Dependent Kinases ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Drug Design ; Cell Line, Tumor
Czasopismo naukowe
Tytuł:
Exploring Antimicrobial Features for New Imidazo[4,5-b]pyridine Derivatives Based on Experimental and Theoretical Study.
Autorzy:
Hjouji MY; Laboratory of Applied Organic Chemistry, Faculty of Science and Technology Saiss, Sidi Mohammed Ben Abdallah University, Fez 30050, Morocco.
Almehdi AM; Department of Chemistry, College of Sciences, University of Sharjah, Sharjah P.O. Box 27272, United Arab Emirates.
Elmsellem H; Laboratory of Applied Chemistry and Environment (LCAE), Sciences Faculty, Oujda 60000, Morocco.
Seqqat Y; Laboratory of Applied Organic Chemistry, Faculty of Science and Technology Saiss, Sidi Mohammed Ben Abdallah University, Fez 30050, Morocco.
Ouzidan Y; Laboratoire de Chimie-Physique et Biotechnologie des Biomolécules et Matériaux, Faculté des Sciences et Techniques, Université Hassan II, BP 146, Mohammedia 28800, Morocco.
Tebbaa M; Laboratoire de Chimie-Physique et Biotechnologie des Biomolécules et Matériaux, Faculté des Sciences et Techniques, Université Hassan II, BP 146, Mohammedia 28800, Morocco.
Lfakir NA; Laboratoire de Chimie-Physique et Biotechnologie des Biomolécules et Matériaux, Faculté des Sciences et Techniques, Université Hassan II, BP 146, Mohammedia 28800, Morocco.
Kandri Rodi Y; Laboratory of Applied Organic Chemistry, Faculty of Science and Technology Saiss, Sidi Mohammed Ben Abdallah University, Fez 30050, Morocco.
Chahdi FO; Laboratory of Applied Organic Chemistry, Faculty of Science and Technology Saiss, Sidi Mohammed Ben Abdallah University, Fez 30050, Morocco.
Chraibi M; Laboratory of Microbial Biotechnology, Faculty of Science and Technology Saïss, Sidi Mohamed Ben Abdellah University, Fez 30050, Morocco.
Fikri Benbrahim K; Laboratory of Microbial Biotechnology, Faculty of Science and Technology Saïss, Sidi Mohamed Ben Abdellah University, Fez 30050, Morocco.
Al-Omar MA; Drug Exploration & Development Chair (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Almehizia AA; Drug Exploration & Development Chair (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Naglah AM; Drug Exploration & Development Chair (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
El-Mowafi SA; Peptide Chemistry Department, Chemical Industries Research Institute, National Research Centre, Dokki, Cairo 12622, Egypt.
Elhenawy AA; Chemistry Department, Faculty of Science, Al-Azhar University, Cairo 11884, Egypt.; Chemistry Department, Faculty of Science and Art, Albaha University, Albahah 65731, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Apr 04; Vol. 28 (7). Date of Electronic Publication: 2023 Apr 04.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Infective Agents*/pharmacology
Anti-Infective Agents*/chemistry
Molecular Docking Simulation ; Molecular Conformation ; Anti-Bacterial Agents/pharmacology ; Anti-Bacterial Agents/chemistry ; Gram-Positive Bacteria ; Pyridines/pharmacology ; Pyridines/chemistry
Czasopismo naukowe
Tytuł:
Development and In Vitro Characterization of Antibiotic-Loaded Nanocarriers for Dental Delivery.
Autorzy:
Ghazwani M; Department of Pharmaceutics, College of Pharmacy, King Khalid University (KKU), Abha 61421, Saudi Arabia.
Vasudevan R; Department of Pharmacology, College of Pharmacy, King Khalid University (KKU), Abha 61421, Saudi Arabia.
Kandasamy G; Department of Clinical Pharmacy, College of Pharmacy, King Khalid University (KKU), Abha 61421, Saudi Arabia.
Hani U; Department of Pharmaceutics, College of Pharmacy, King Khalid University (KKU), Abha 61421, Saudi Arabia.
Niharika G; Department of Pharmaceutics, St. Peter's Institute of Pharmaceutical Sciences, Hanamkonda 506001, Telangana, India.
Naredla M; Department of Pharmaceutics, St. Peter's Institute of Pharmaceutical Sciences, Hanamkonda 506001, Telangana, India.
Devanandan P; Department of Pharmacy Practice, St. Peter's Institute of Pharmaceutical Sciences, Hanamkonda 506001, Telangana, India.
Puvvada RC; Department of Pharmacy Practice, St. Peter's Institute of Pharmaceutical Sciences, Hanamkonda 506001, Telangana, India.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Hakami AR; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, King Khalid University (KKU), Abha 61481, Saudi Arabia.
Dhurke R; Department of Pharmaceutics, St. Peter's Institute of Pharmaceutical Sciences, Hanamkonda 506001, Telangana, India.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Mar 24; Vol. 28 (7). Date of Electronic Publication: 2023 Mar 24.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Bacterial Agents*/chemistry
Dental Caries*
Humans ; Staphylococcus aureus ; Escherichia coli ; Ciprofloxacin/pharmacology ; Ciprofloxacin/chemistry
Czasopismo naukowe
Tytuł:
Nanomaterials-Based Novel Immune Strategies in Clinical Translation for Cancer Therapy.
Autorzy:
Wahab S; Department of Pharmacognosy, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Ghazwani M; Department of Pharmaceutics, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Hani U; Department of Pharmaceutics, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Hakami AR; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, King Khalid University, Abha 61481, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, Drug Exploration and Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Ahmad W; Department of Pharmacy, Mohammed Al-Mana College for Medical Sciences, Dammam 34222, Saudi Arabia.
Ahmad MZ; Department of Pharmaceutics, College of Pharmacy, Najran University, Najran 11001, Saudi Arabia.
Alam P; Department of Pharmacognosy, College of Pharmacy, Prince Sattam Bin Abdulaziz University, Al-Kharj 11942, Saudi Arabia.
Annadurai S; Department of Pharmacognosy, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Jan 26; Vol. 28 (3). Date of Electronic Publication: 2023 Jan 26.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Nanostructures*/therapeutic use
Antineoplastic Agents*/therapeutic use
Neoplasms*/drug therapy
Humans ; Nanotechnology ; Immunotherapy
Czasopismo naukowe
Tytuł:
Isolation and Bioassay of a New Terminalone A from Terminalia arjuna .
Autorzy:
Bushra; Institute of Chemical Sciences, Gomal University, Dera Ismail Khan 29050, KPK, Pakistan.
Rehman KU; Institute of Chemical Sciences, Gomal University, Dera Ismail Khan 29050, KPK, Pakistan.
Khan D; Institute of Chemical Sciences, Gomal University, Dera Ismail Khan 29050, KPK, Pakistan.
Almehizia AA; Drug Exploration and Development Chair (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Naglah AM; Drug Exploration and Development Chair (DEDC), Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Al-Wasidi AS; Department of Chemistry, College of Science, Princess Nourah bint Abdulrahman University, Riyadh 11671, Saudi Arabia.
Refat MS; Department of Chemistry, College of Science, Taif University, P.O. Box 11099, Taif 21944, Saudi Arabia.
El-Sayed MY; Chemistry Department, College of Science, Jouf University, P.O. Box: 2014, Sakaka, Saudi Arabia.
Ullah H; Department of Chemistry, Balochistan University of Information Technology, Engineering and Management Sciences, Quetta 87300, Pakistan.
Khan S; Institute of Chemical Sciences, Gomal University, Dera Ismail Khan 29050, KPK, Pakistan.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Jan 19; Vol. 28 (3). Date of Electronic Publication: 2023 Jan 19.
Typ publikacji:
Journal Article
MeSH Terms:
Antioxidants*/chemistry
Terminalia*/chemistry
Plant Extracts/chemistry ; Flavonoids/pharmacology ; Anti-Bacterial Agents/pharmacology ; Biological Assay
Czasopismo naukowe
Tytuł:
Synthesis, Cytotoxic Evaluation, and Structure-Activity Relationship of Substituted Quinazolinones as Cyclin-Dependent Kinase 9 Inhibitors.
Autorzy:
Alkahtani HM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Zen AA; Chemistry & Forensics Department, Clifton Campus, Nottingham Trent University, Nottingham Ng11 8NS, UK.
Obaidullah AJ; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Alanazi MM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Ansari SA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Aleanizy FS; Department of Pharmaceutics, College of Pharmacy, King Saud University, P.O. Box 22452, Riyadh 11495, Saudi Arabia.
Alqahtani FY; Department of Pharmaceutics, College of Pharmacy, King Saud University, P.O. Box 22452, Riyadh 11495, Saudi Arabia.
Aldossari RM; Department of Pharmacology & Toxicology, College of Pharmacy, 11 Prince Sattam Bin Abdulaziz University, P.O. Box 173, Al-Kharj 11942, Saudi Arabia.
Algamdi RA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Al-Rasheed LS; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Abdel-Hamided SG; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Al-Azhar University, Cairo 11884, Egypt.
Abdel-Aziz AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
El-Azab AS; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Dec 23; Vol. 28 (1). Date of Electronic Publication: 2022 Dec 23.
Typ publikacji:
Journal Article
MeSH Terms:
Cyclin-Dependent Kinase 9*
Antineoplastic Agents*/chemistry
Molecular Docking Simulation ; Quinazolinones/pharmacology ; Protein Kinase Inhibitors/chemistry ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Identification of Antibacterial Metabolites from Endophytic Fungus Aspergillus fumigatus, Isolated from Albizia lucidior Leaves (Fabaceae), Utilizing Metabolomic and Molecular Docking Techniques.
Autorzy:
Hussein ME; Pharmacognosy Department, Faculty of Pharmacy, Cairo University, Kasr el Aini St., Cairo 11562, Egypt.
Mohamed OG; Pharmacognosy Department, Faculty of Pharmacy, Cairo University, Kasr el Aini St., Cairo 11562, Egypt.; Natural Products Discovery Core, Life Sciences Institute, University of Michigan, Ann Arbor, MI 48109, USA.
El-Fishawy AM; Pharmacognosy Department, Faculty of Pharmacy, Cairo University, Kasr el Aini St., Cairo 11562, Egypt.
El-Askary HI; Pharmacognosy Department, Faculty of Pharmacy, Cairo University, Kasr el Aini St., Cairo 11562, Egypt.
El-Senousy AS; Pharmacognosy Department, Faculty of Pharmacy, Cairo University, Kasr el Aini St., Cairo 11562, Egypt.
El-Beih AA; Department of Chemistry of Natural and Microbial Products, National Research Centre, Dokki, Giza 12622, Egypt.
Nossier ES; Department of Pharmaceutical Medicinal Chemistry and Drug Design, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo 11754, Egypt.
Naglah AM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Tripathi A; Natural Products Discovery Core, Life Sciences Institute, University of Michigan, Ann Arbor, MI 48109, USA.; Department of Medicinal Chemistry, College of Pharmacy, University of Michigan, Ann Arbor, MI 48109, USA.
Hamed AA; Microbial Chemistry Department, National Research Centre, 33 El-Buhouth Street, Dokki, Giza 12622, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Feb 08; Vol. 27 (3). Date of Electronic Publication: 2022 Feb 08.
Typ publikacji:
Journal Article
MeSH Terms:
Albizzia/*microbiology
Anti-Bacterial Agents/*metabolism
Aspergillus fumigatus/*metabolism
Anti-Bacterial Agents/chemistry ; Anti-Bacterial Agents/isolation & purification ; Anti-Bacterial Agents/pharmacology ; Aspergillus fumigatus/chemistry ; Humans ; Metabolome ; Molecular Docking Simulation ; Plant Leaves/chemistry ; Staphylococcal Infections/drug therapy ; Staphylococcus aureus/drug effects
Czasopismo naukowe
Tytuł:
Solid-Contact Potentiometric Sensors Based on Main-Tailored Bio-Mimics for Trace Detection of Harmine Hallucinogen in Urine Specimens.
Autorzy:
Amr AEE; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.; Applied Organic Chemistry Department, National Research Center, Dokki, Giza 12622, Egypt.
Kamel AH; Department of Chemistry, Faculty of Science, Ain Shams University, Cairo 11566, Egypt.
Almehizia AA; Applied Organic Chemistry Department, National Research Center, Dokki, Giza 12622, Egypt.
Sayed AYA; Applied Organic Chemistry Department, National Research Center, Dokki, Giza 12622, Egypt.
Abd-Rabboh HSM; Department of Chemistry, Faculty of Science, Ain Shams University, Cairo 11566, Egypt.; Chemistry Department, Faculty of Science, King Khalid University, P.O. Box 9004, Abha 61413, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2021 Jan 10; Vol. 26 (2). Date of Electronic Publication: 2021 Jan 10.
Typ publikacji:
Journal Article
MeSH Terms:
Biosensing Techniques*
Hallucinogens*/analysis
Hallucinogens*/urine
Harmine*/analysis
Harmine*/urine
Biomimetic Materials/*chemistry
Bridged Bicyclo Compounds, Heterocyclic/chemistry ; Humans ; Methacrylates/chemistry ; Polymers/chemistry ; Potentiometry
Czasopismo naukowe
Tytuł:
Validated Reversed-Phase Liquid Chromatographic Method with Gradient Elution for Simultaneous Determination of the Antiviral Agents: Sofosbuvir, Ledipasvir, Daclatasvir, and Simeprevir in Their Dosage Forms.
Autorzy:
Ezzeldin E; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.; Bioavailability Center, National Organization for Drug Control and Research (NODCAR), Giza P.O. Box 29, Egypt.
Abo-Talib NF; Bioavailability Center, National Organization for Drug Control and Research (NODCAR), Giza P.O. Box 29, Egypt.
Tammam MH; Bioavailability Center, National Organization for Drug Control and Research (NODCAR), Giza P.O. Box 29, Egypt.
Asiri YA; Clinical Pharmacy Department, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Amr AEE; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.; Applied Organic Chemistry Department, National Research Center, Dokki, Cairo 12622, Egypt.
Almehizia AA; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Oct 10; Vol. 25 (20). Date of Electronic Publication: 2020 Oct 10.
Typ publikacji:
Journal Article
MeSH Terms:
Antiviral Agents/*chemistry
Benzimidazoles/*chemistry
Chromatography, Reverse-Phase/*methods
Fluorenes/*chemistry
Hepatitis C, Chronic/*virology
Simeprevir/*chemistry
Sofosbuvir/*chemistry
Chromatography, High Pressure Liquid ; Limit of Detection ; Temperature
Czasopismo naukowe
Tytuł:
Preparation and Characterization of Two Immunogens and Production of Polyclonal Antibody with High Affinity and Specificity for Darunavir.
Autorzy:
Darwish IA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Almehizia AA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
Radwan AA; Kayyali Chair for Pharmaceutical Industries, Department of Pharmaceutics, College of Pharmacy, King Saud University, P.O. Box 2460, Riyadh 11451, Saudi Arabia.
Herqash RN; Medicinal Aromatic and Poisonous Plant Research Centre, College of Pharmacy, King Saud University, P.O. Box 2457, Riyadh 11451, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Sep 07; Vol. 25 (18). Date of Electronic Publication: 2020 Sep 07.
Typ publikacji:
Journal Article
MeSH Terms:
Antibodies/*immunology
Antibody Affinity/*immunology
Antibody Specificity/*immunology
Antigens/*immunology
Darunavir/*adverse effects
HIV Protease Inhibitors/*adverse effects
Animals ; Darunavir/immunology ; Darunavir/pharmacokinetics ; Drug Monitoring ; Enzyme-Linked Immunosorbent Assay ; HIV Protease Inhibitors/immunology ; HIV Protease Inhibitors/pharmacokinetics ; Haptens/chemistry ; Haptens/immunology ; Humans ; Magnetic Resonance Spectroscopy ; Mice ; Molecular Structure
Czasopismo naukowe
Tytuł:
Novel Validated Analytical Method Based on Potentiometric Transduction for the Determination of Citicoline Psychostimulant/Nootropic Agent.
Autorzy:
Kamel AH; Department of Chemistry, Faculty of Science, Ain Shams University, Cairo 11566, Egypt.
Amr AEE; Pharmaceutical Chemistry Department, Drug Exploration & Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.; Applied Organic Chemistry Department, National Research Center, Dokki 12622, Giza, Egypt.
Galal HR; Inorganic Chemistry Department, National Research Center, Dokki 12622, Giza, Egypt.
Almehizia AA; Pharmaceutical Chemistry Department, Drug Exploration & Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Jul 31; Vol. 25 (15). Date of Electronic Publication: 2020 Jul 31.
Typ publikacji:
Journal Article
MeSH Terms:
Cytidine Diphosphate Choline/*analysis
Nootropic Agents/*analysis
Potentiometry/*methods
Electrodes ; Hydrogen-Ion Concentration ; Limit of Detection ; Membranes, Artificial ; Plasticizers/chemistry ; Polyvinyl Chloride/chemistry ; Reproducibility of Results
Czasopismo naukowe
Tytuł:
Discovery of New Schiff Bases Tethered Pyrazole Moiety: Design, Synthesis, Biological Evaluation, and Molecular Docking Study as Dual Targeting DHFR/DNA Gyrase Inhibitors with Immunomodulatory Activity.
Autorzy:
Hassan AS; Organometallic and Organometalloid Chemistry Department, National Research Centre, Dokki 12622, Cairo, Egypt.
Askar AA; Botany and Microbiology Department, Faculty of Science (Boys), Al-Azhar University, Nasr City, Cairo, Egypt.
Naglah AM; Department of Pharmaceutical Chemistry, Drug Exploration and Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.; Peptide Chemistry Department, National Research Centre, Dokki 12622, Cairo, Egypt.
Almehizia AA; Department of Pharmaceutical Chemistry, Drug Exploration and Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
Ragab A; Chemistry Department, Faculty of Science (Boys), Al-Azhar University, Nasr City, Cairo, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Jun 02; Vol. 25 (11). Date of Electronic Publication: 2020 Jun 02.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Bacterial Agents/*chemical synthesis
DNA Gyrase/*metabolism
Folic Acid Antagonists/*chemical synthesis
Pyrazoles/*chemical synthesis
Tetrahydrofolate Dehydrogenase/*metabolism
Topoisomerase II Inhibitors/*chemical synthesis
Anti-Bacterial Agents/chemistry ; Anti-Bacterial Agents/pharmacology ; Bacillus subtilis/drug effects ; Bacillus subtilis/enzymology ; Bacterial Proteins/chemistry ; Bacterial Proteins/metabolism ; Binding Sites ; Cell Line, Tumor ; Cell Proliferation/drug effects ; DNA Gyrase/chemistry ; Drug Screening Assays, Antitumor ; Escherichia coli/drug effects ; Escherichia coli/enzymology ; Folic Acid Antagonists/chemistry ; Folic Acid Antagonists/pharmacology ; Hep G2 Cells ; Humans ; MCF-7 Cells ; Microbial Sensitivity Tests ; Models, Molecular ; Molecular Docking Simulation ; Molecular Structure ; Protein Conformation ; Pyrazoles/chemistry ; Pyrazoles/pharmacology ; Schiff Bases/chemistry ; Staphylococcus aureus/drug effects ; Staphylococcus aureus/enzymology ; Structure-Activity Relationship ; Tetrahydrofolate Dehydrogenase/chemistry ; Topoisomerase II Inhibitors/chemistry ; Topoisomerase II Inhibitors/pharmacology
Czasopismo naukowe
Tytuł:
Novel Carbon/PEDOT/PSS-Based Screen-Printed Biosensors for Acetylcholine Neurotransmitter and Acetylcholinesterase Detection in Human Serum.
Autorzy:
Ashmawy NH; Chemistry Department, Faculty of Science, Ain Shams University, P.O. Cairo 11566, Egypt. .
Almehizia AA; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia. .
Youssef TA; Chemistry Department, Faculty of Science, Ain Shams University, P.O. Cairo 11566, Egypt. trease_.
El-Galil E Amr A; Pharmaceutical Chemistry Department, Drug Exploration & Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia. .; Applied Organic Chemistry Department, National Research Centre, 12622 Dokki, Giza, Egypt. .
Al-Omar MA; Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia. .; Pharmaceutical Chemistry Department, Drug Exploration & Development Chair (DEDC), College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia. .
Kamel AH; Chemistry Department, Faculty of Science, Ain Shams University, P.O. Cairo 11566, Egypt. .
Pokaż więcej
Źródło:
Molecules (Basel, Switzerland) [Molecules] 2019 Apr 18; Vol. 24 (8). Date of Electronic Publication: 2019 Apr 18.
Typ publikacji:
Journal Article
MeSH Terms:
Printing*
Acetylcholine/*blood
Acetylcholinesterase/*blood
Biosensing Techniques/*methods
Bridged Bicyclo Compounds, Heterocyclic/*chemistry
Carbon/*chemistry
Neurotransmitter Agents/*blood
Polymers/*chemistry
Polystyrenes/*chemistry
Flow Injection Analysis ; Humans ; Hydrodynamics ; Hydrolysis ; Kinetics ; Potentiometry ; Water/chemistry
Czasopismo naukowe
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