- Tytuł :
- Inhibition of 14-3-3/Tau by hybrid small-molecule peptides operating via two different binding modes
- Index Terms :
-
14-3-3
drug discovery
inhibitors
peptide chemistry
protein-protein interactions
tau
Phosphorylation
Magnetic Resonance Spectroscopy
Humans
Crystallography, X-Ray
Drug Discovery
Microtubules/metabolism
Protein Binding
14-3-3 Proteins/chemistry
tau Proteins/chemistryAlzheimer Disease /metabolism
Neurofibrillary Tangles/metabolism
Cognitive Neuroscience
Biochemistry
Physiology
Cell Biology
Research Support, Non-U.S. Gov't
Journal Article
Tijdschriftartikel
Article - Źródło :
- ACS Chemical Neuroscience vol.9 (2018) date: 2018-11-21 nr.11 p.2639–2654 [ISSN 1948-7193]
- URL :
-
https://research.tue.nl/en/publications/inhibition-of-1433tau-by-hybrid-smallmolecule-peptides-operating-via-two-different-binding-modes(7429ef0b-4c10-440d-a801-302f4de9450d).html">https://research.tue.nl/en/publications/inhibition-of-1433tau-by-hybrid-smallmolecule-peptides-operating-via-two-different-binding-modes(7429ef0b-4c10-440d-a801-302f4de9450d).html https://pure.tue.nl/ws/files/116540431/acschemneuro.8b00118.pdf">https://pure.tue.nl/ws/files/116540431/acschemneuro.8b00118.pdf https://pure.tue.nl/ws/files/116540431/acschemneuro.8b00118.pdf">https://pure.tue.nl/ws/files/116540431/acschemneuro.8b00118.pdf -
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