Informacja

Drogi użytkowniku, aplikacja do prawidłowego działania wymaga obsługi JavaScript. Proszę włącz obsługę JavaScript w Twojej przeglądarce.

Wyszukujesz frazę ""Amoroso R"" wg kryterium: Autor


Wyświetlanie 1-5 z 5
Tytuł:
Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.
Autorzy:
Ammazzalorso A; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Carradori S; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Angeli A; b Laboratorio di Chimica Bioinorganica , Università degli Studi di Firenze , Florence , Italy.
Akdemir A; c Department of Pharmacology, Faculty of Pharmacy, Computer-Aided Drug Discovery Laboratory , Bezmialem Vakif University , Istanbul , Turkey.
De Filippis B; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Fantacuzzi M; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Giampietro L; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Maccallini C; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Amoroso R; a Department of Pharmacy , 'G. d'Annunzio' University of Chieti-Pescara , Chieti , Italy.
Supuran CT; b Laboratorio di Chimica Bioinorganica , Università degli Studi di Firenze , Florence , Italy.; d Neurofarba Department , Section of Pharmaceutical and Nutriceutical Sciences, Università degli Studi di Firenze , Florence , Italy.
Pokaż więcej
Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2019 Dec; Vol. 34 (1), pp. 1051-1061.
Typ publikacji:
Journal Article
MeSH Terms:
Molecular Docking Simulation*
Carbonic Anhydrase Inhibitors/*pharmacology
Carbonic Anhydrases/*metabolism
Sulfonamides/*pharmacology
Carbonic Anhydrase Inhibitors/chemical synthesis ; Carbonic Anhydrase Inhibitors/chemistry ; Catalytic Domain/drug effects ; Dose-Response Relationship, Drug ; Humans ; Molecular Structure ; Structure-Activity Relationship ; Sulfonamides/chemical synthesis ; Sulfonamides/chemistry
Czasopismo naukowe
Tytuł:
N-acylsulfonamides: Synthetic routes and biological potential in medicinal chemistry.
Autorzy:
Ammazzalorso A; Dipartimento di Farmacia, Università G. d'Annunzio, Chieti, Italy.
De Filippis B; Dipartimento di Farmacia, Università G. d'Annunzio, Chieti, Italy.
Giampietro L; Dipartimento di Farmacia, Università G. d'Annunzio, Chieti, Italy.
Amoroso R; Dipartimento di Farmacia, Università G. d'Annunzio, Chieti, Italy.
Pokaż więcej
Źródło:
Chemical biology & drug design [Chem Biol Drug Des] 2017 Dec; Vol. 90 (6), pp. 1094-1105. Date of Electronic Publication: 2017 Jul 11.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Enzyme Inhibitors/*chemical synthesis
Sulfonamides/*chemistry
Carboxylic Acids/chemistry ; Chemistry, Pharmaceutical ; Drug Design ; Enzyme Inhibitors/chemistry ; Enzyme Inhibitors/metabolism ; Peroxisome Proliferator-Activated Receptors/agonists ; Peroxisome Proliferator-Activated Receptors/antagonists & inhibitors ; Peroxisome Proliferator-Activated Receptors/metabolism ; Receptors, Prostaglandin E/metabolism ; Structure-Activity Relationship ; Sulfonamides/chemical synthesis ; Sulfonamides/metabolism ; Viral Nonstructural Proteins/chemistry ; Viral Nonstructural Proteins/metabolism
Czasopismo naukowe
Tytuł:
Cytotoxic effect of a family of peroxisome proliferator-activated receptor antagonists in colorectal and pancreatic cancer cell lines.
Autorzy:
Ammazzalorso A; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
De Lellis L; Unità di Patologia Generale, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.; Aging Research Center (Ce.S.I.), Università 'G. d'Annunzio', Chieti, Italy.
Florio R; Unità di Patologia Generale, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.; Aging Research Center (Ce.S.I.), Università 'G. d'Annunzio', Chieti, Italy.
Bruno I; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
De Filippis B; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
Fantacuzzi M; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
Giampietro L; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
Maccallini C; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
Perconti S; Aging Research Center (Ce.S.I.), Università 'G. d'Annunzio', Chieti, Italy.
Verginelli F; Unità di Patologia Generale, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.; Aging Research Center (Ce.S.I.), Università 'G. d'Annunzio', Chieti, Italy.
Cama A; Unità di Patologia Generale, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.; Aging Research Center (Ce.S.I.), Università 'G. d'Annunzio', Chieti, Italy.
Amoroso R; Unità di Chimica Farmaceutica, Dipartimento di Farmacia, Università 'G. d'Annunzio', Chieti, Italy.
Pokaż więcej
Źródło:
Chemical biology & drug design [Chem Biol Drug Des] 2017 Nov; Vol. 90 (5), pp. 1029-1035. Date of Electronic Publication: 2017 Jul 19.
Typ publikacji:
Letter
MeSH Terms:
Antineoplastic Agents/*pharmacology
Colorectal Neoplasms/*drug therapy
PPAR alpha/*antagonists & inhibitors
PPAR gamma/*antagonists & inhibitors
Pancreatic Neoplasms/*drug therapy
Sulfonamides/*pharmacology
Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Cell Line, Tumor ; Cell Survival/drug effects ; Colorectal Neoplasms/metabolism ; Humans ; PPAR alpha/metabolism ; PPAR gamma/metabolism ; Pancreatic Neoplasms/metabolism ; Sulfonamides/chemical synthesis ; Sulfonamides/chemistry
Opinia redakcyjna
    Wyświetlanie 1-5 z 5

    Ta witryna wykorzystuje pliki cookies do przechowywania informacji na Twoim komputerze. Pliki cookies stosujemy w celu świadczenia usług na najwyższym poziomie, w tym w sposób dostosowany do indywidualnych potrzeb. Korzystanie z witryny bez zmiany ustawień dotyczących cookies oznacza, że będą one zamieszczane w Twoim komputerze. W każdym momencie możesz dokonać zmiany ustawień dotyczących cookies