- Tytuł :
- The antibiotic sorangicin A inhibits promoter DNA unwinding in a Mycobacterium tuberculosis rifampicin-resistant RNA polymerase.
- Autorzy :
- Źródło :
- Proceedings of the National Academy of Sciences of the United States of America [Proc Natl Acad Sci U S A] 2020 Dec 01; Vol. 117 (48), pp. 30423-30432. Date of Electronic Publication: 2020 Nov 16.
- Typ publikacji :
- Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
- MeSH Terms :
-
Promoter Regions, Genetic*
Aminoglycosides/*pharmacologyAntibiotics ,Antitubercular /*pharmacology
DNA-Directed RNA Polymerases/*metabolism
Drug Resistance, Bacterial/*drug effects
Mycobacterium tuberculosis/*drug effects
Mycobacterium tuberculosis/*physiology
Aminoglycosides/chemistry ;Antibiotics ,Antitubercular /chemistry ; Binding Sites ; Humans ; Models, Molecular ; Molecular Conformation ; Protein Binding ; Rifampin/pharmacology ; Structure-Activity Relationship ; Tuberculosis/drug therapy ; Tuberculosis/microbiology -
Czasopismo naukowe