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Wyszukujesz frazę ""Aromatase"" wg kryterium: Temat


Tytuł:
Targeting aromatase to restrain oestrogen production and developing efficacious interventions against ER-positive cancer.
Autorzy:
Rani S; Department of Chemistry, Guru Nanak Dev University, Amritsar, 143005, India.
Vermani S; Department of Chemistry, Guru Nanak Dev University, Amritsar, 143005, India.
Kaur V; Department of Chemistry, Guru Nanak Dev University, Amritsar, 143005, India.
Singh P; Department of Chemistry, Guru Nanak Dev University, Amritsar, 143005, India. Electronic address: palwinder_singh_.
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Źródło:
European journal of medicinal chemistry [Eur J Med Chem] 2024 Feb 05; Vol. 265, pp. 116111. Date of Electronic Publication: 2023 Dec 31.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase*/metabolism
Breast Neoplasms*/drug therapy
Female ; Humans ; Aromatase Inhibitors/pharmacology ; Aromatase Inhibitors/therapeutic use ; Estrogens/metabolism ; Kinetics ; Receptors, Estrogen/metabolism ; Tamoxifen/pharmacology
Czasopismo naukowe
Tytuł:
Aromatase enzyme: Paving the way for exploring aromatization for cardio-renal protection.
Autorzy:
Eissa MA; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Merit University, New Sohag, Sohag, Egypt.
Gohar EY; Division of Nephrology and Hypertension, Department of Medicine, Vanderbilt University Medical Center, Nashville, TN, United States. Electronic address: .
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Źródło:
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie [Biomed Pharmacother] 2023 Dec; Vol. 168, pp. 115832. Date of Electronic Publication: 2023 Nov 06.
Typ publikacji:
Meta-Analysis; Journal Article; Review
MeSH Terms:
Aromatase*
Cardiovascular Diseases*/drug therapy
Cardiovascular Diseases*/prevention & control
Male ; Female ; Humans ; Aromatase Inhibitors/pharmacology ; Androgens/pharmacology ; Estrogens/pharmacology ; Receptors, Estrogen
Czasopismo naukowe
Tytuł:
New 1,2,3-Triazole/1,2,4-triazole Hybrids as Aromatase Inhibitors: Design, Synthesis, and Apoptotic Antiproliferative Activity.
Autorzy:
Maghraby MT; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Assiut University, Assiut 71526, Egypt.; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, New Valley University, New Valley 72511, Egypt.
Mazyad Almutairi T; Department of Chemistry, College of Science, King Saud University, Riyadh 11451, Saudi Arabia.
Bräse S; Institute of Biological and Chemical Systems, IBCS-FMS, Karlsruhe Institute of Technology, 76131 Karlsruhe, Germany.
Salem OIA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Assiut University, Assiut 71526, Egypt.
Youssif BGM; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Assiut University, Assiut 71526, Egypt.
Sheha MM; Department of Medicinal Chemistry, Faculty of Pharmacy, Assiut University, Assiut 71526, Egypt.; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Sphinx University, New-Assiut 71684, Egypt.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Oct 14; Vol. 28 (20). Date of Electronic Publication: 2023 Oct 14.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase Inhibitors*/chemistry
Antineoplastic Agents*/chemistry
Aromatase ; Molecular Docking Simulation ; Structure-Activity Relationship ; Erlotinib Hydrochloride/pharmacology ; Cell Line, Tumor ; Triazoles/chemistry ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Molecular Structure
Czasopismo naukowe
Tytuł:
Repurposing of approved drugs for targeting CDK4/6 and aromatase protein using molecular docking and molecular dynamics studies.
Autorzy:
Yousif FA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Gezira, Wad Madani, Sudan.
Alzain AA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Gezira, Wad Madani, Sudan.
Alraih AM; Department of Chemistry, College of Science and Arts, Mohail Aseer, King Khalid University, Abha, Kingdom of Saudi Arabia.
Ibraheem W; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Gezira, Wad Madani, Sudan.
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Źródło:
PloS one [PLoS One] 2023 Sep 08; Vol. 18 (9), pp. e0291256. Date of Electronic Publication: 2023 Sep 08 (Print Publication: 2023).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Aromatase*
Breast Neoplasms*
Female ; Humans ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Apomorphine ; Drug Repositioning ; Estrogens ; Aromatase Inhibitors/pharmacology ; Cyclin-Dependent Kinase 4
Czasopismo naukowe
Tytuł:
A Systematic Review of Systematic Reviews on the Use of Aromatase Inhibitors for the Treatment of Endometriosis: The Evidence to Date.
Autorzy:
Peitsidis P; Department of Obstetrics and Gynecology Helena Venizelou Hospital, Athens, Greece.
Tsikouras P; Department of Obstetrics and Gynecology.The Democritus University of Thrace, Alexandroupolis, Greece.
Laganà AS; Unit of Gynecologic Oncology ARNAS 'Civico-Di Cristina-Benfratelli', Department of Health Promotion, Mother and Child Care, Internal Medicine and Medical Specialties, Palermo, Italy.
Laios A; Department of Gynecological Oncology St James Institute of Oncology, Leeds Teaching Hospitals, Leeds, Uk.
Gkegkes ID; Department of Colorectal Surgery, Royal Devon and Exeter NHS Foundation, Devon, UK.
Iavazzo C; Gynaecological Oncology Department, Metaxa Cancer Hospital, Piraeus, Greece.
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Źródło:
Drug design, development and therapy [Drug Des Devel Ther] 2023 May 04; Vol. 17, pp. 1329-1346. Date of Electronic Publication: 2023 May 04 (Print Publication: 2023).
Typ publikacji:
Journal Article; Review; Systematic Review
MeSH Terms:
Aromatase Inhibitors*/therapeutic use
Aromatase Inhibitors*/pharmacology
Endometriosis*/drug therapy
Endometriosis*/pathology
Female ; Humans ; Aromatase/therapeutic use ; Estrogens ; Systematic Reviews as Topic
Czasopismo naukowe
Tytuł:
Virtual Screening for Identification of Dual Inhibitors against CDK4/6 and Aromatase Enzyme.
Autorzy:
Adon T; Department of Pharmaceutical Chemistry, JSS College of Pharmacy, JSS Academy of Higher Education and Research, Mysuru 570015, Karnataka, India.
Shanmugarajan D; Department of Pharmaceutical Chemistry, JSS College of Pharmacy, JSS Academy of Higher Education and Research, Mysuru 570015, Karnataka, India.
Ather H; Department of Pharmaceutical Chemistry, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Ansari SMA; Department of Clinical Pharmacy, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Hani U; Department of Pharmaceutics, College of Pharmacy, King Khalid University, Abha 62529, Saudi Arabia.
Madhunapantula SV; Department of Biochemistry, JSS Medical College, JSS Academy of Higher Education & Research, Mysore 570015, Karnataka, India.; Special Interest Group in Cancer Biology and Cancer Stem Cells, JSS Academy of Higher Education & Research, Mysore 570015, Karnataka, India.
Honnavalli YK; Department of Pharmaceutical Chemistry, JSS College of Pharmacy, JSS Academy of Higher Education and Research, Mysuru 570015, Karnataka, India.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Mar 08; Vol. 28 (6). Date of Electronic Publication: 2023 Mar 08.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase Inhibitors*/pharmacology
Aromatase Inhibitors*/chemistry
Breast Neoplasms*/drug therapy
Breast Neoplasms*/pathology
Humans ; Female ; Aromatase ; Molecular Docking Simulation ; Anastrozole/therapeutic use ; Molecular Dynamics Simulation ; Enzyme Inhibitors/therapeutic use ; Cyclin-Dependent Kinase 4
Czasopismo naukowe
Tytuł:
Aromatase Inhibitors as a Promising Direction for the Search for New Anticancer Drugs.
Autorzy:
Janowska S; Department of Pathobiochemistry and Interdisciplinary Applications of Ion Chromatography, Biomedical Sciences, Medical University of Lublin, 1 Chodzki Street, 20-093 Lublin, Poland.
Holota S; Department of Pharmaceutical, Organic and Bioorganic Chemistry, Danylo Halytsky Lviv National Medical University, Pekarska 69, 79010 Lviv, Ukraine.
Lesyk R; Department of Pharmaceutical, Organic and Bioorganic Chemistry, Danylo Halytsky Lviv National Medical University, Pekarska 69, 79010 Lviv, Ukraine.
Wujec M; Department of Organic Chemistry, Faculty of Pharmacy, Medical University of Lublin, 4A Chodzki Street, 20-093 Lublin, Poland.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2024 Jan 10; Vol. 29 (2). Date of Electronic Publication: 2024 Jan 10.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Aromatase Inhibitors*/pharmacology
Aromatase Inhibitors*/therapeutic use
Aromatase*
Female ; Male ; Humans ; Estrogens ; Adipose Tissue ; Androgens
Czasopismo naukowe
Tytuł:
Medicinal chemistry aspects and synthetic strategies of coumarin as aromatase inhibitors: an overview.
Autorzy:
Ratre P; Department of Pharmaceutical Sciences and Natural Products, School of Pharmaceutical Sciences, Central University of Punjab, Bathinda, Punjab, 151401, India.
Kulkarni S; Department of Pharmaceutical Sciences and Natural Products, School of Pharmaceutical Sciences, Central University of Punjab, Bathinda, Punjab, 151401, India.
Das S; Department of Pharmaceutical Sciences and Natural Products, School of Pharmaceutical Sciences, Central University of Punjab, Bathinda, Punjab, 151401, India.
Liang C; School of Food and Bioengineering, Shaanxi University of Science & Technology, Xi'an, 710 021, People's Republic of China.
Mishra PK; Department of Molecular Biology, ICMR-National Institute for Research in Environmental Health, Bhopal, Madhya Pradesh, India.
Thareja S; Department of Pharmaceutical Sciences and Natural Products, School of Pharmaceutical Sciences, Central University of Punjab, Bathinda, Punjab, 151401, India. .
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Źródło:
Medical oncology (Northwood, London, England) [Med Oncol] 2022 Dec 05; Vol. 40 (1), pp. 41. Date of Electronic Publication: 2022 Dec 05.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Antineoplastic Agents*/therapeutic use
Aromatase Inhibitors*/pharmacology
Aromatase Inhibitors*/chemistry
Aromatase Inhibitors*/therapeutic use
Breast Neoplasms*/drug therapy
Coumarins*/pharmacology
Coumarins*/chemistry
Coumarins*/therapeutic use
Estrogens*/metabolism
Neoplasms, Hormone-Dependent*/drug therapy
Female ; Humans ; Aromatase/metabolism ; Chemistry, Pharmaceutical
Czasopismo naukowe
Tytuł:
Single-digit nanomolar inhibitors lock the aromatase active site via a dualsteric targeting strategy.
Autorzy:
Caciolla J; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, via Belmeloro 6, 40126, Bologna, Italy.
Martini S; Molecular Pharmacology Unit, Fondazione IRCSS Istituto Nazionale dei Tumori, via Amadeo 42, 20113, Milano, Italy.
Spinello A; Department of Biological, Chemical and Pharmaceutical Sciences and Technologies, University of Palermo, Viale delle Scienze, 90128, Palermo, Italy.
Belluti F; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, via Belmeloro 6, 40126, Bologna, Italy.
Bisi A; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, via Belmeloro 6, 40126, Bologna, Italy.
Zaffaroni N; Molecular Pharmacology Unit, Fondazione IRCSS Istituto Nazionale dei Tumori, via Amadeo 42, 20113, Milano, Italy.
Magistrato A; National Research Council of Italy Institute of Materials (CNR-IOM) c/o SISSA, via Bonomea 265, 34136, Trieste, Italy. Electronic address: .
Gobbi S; Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, via Belmeloro 6, 40126, Bologna, Italy. Electronic address: .
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Źródło:
European journal of medicinal chemistry [Eur J Med Chem] 2022 Dec 15; Vol. 244, pp. 114802. Date of Electronic Publication: 2022 Sep 30.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase*/metabolism
Breast Neoplasms*/pathology
Humans ; Female ; Catalytic Domain ; Aromatase Inhibitors/chemistry ; Receptors, Estrogen/metabolism
Czasopismo naukowe
Tytuł:
4th generation nonsteroidal aromatase inhibitors: An iterative SAR-guided design, synthesis, and biological evaluation towards picomolar dual binding inhibitors.
Autorzy:
Eissa AG; School of Pharmacy and Pharmaceutical Sciences, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, UK.
Barrow D; School of Pharmacy and Pharmaceutical Sciences, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, UK.
Gee J; School of Pharmacy and Pharmaceutical Sciences, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, UK.
Powell LE; Institute of Metabolism and Systems Research, College of Medical and Dental Sciences, University of Birmingham, Birmingham, B15 2TT, UK.
Foster PA; Institute of Metabolism and Systems Research, College of Medical and Dental Sciences, University of Birmingham, Birmingham, B15 2TT, UK; Centre for Endocrinology, Diabetes, and Metabolism, Birmingham Health Partners, Birmingham, B15 2TT, UK.
Simons C; School of Pharmacy and Pharmaceutical Sciences, Cardiff University, King Edward VII Avenue, Cardiff, CF10 3NB, UK. Electronic address: .
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Źródło:
European journal of medicinal chemistry [Eur J Med Chem] 2022 Oct 05; Vol. 240, pp. 114569. Date of Electronic Publication: 2022 Jul 06.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase Inhibitors*/chemistry
Aromatase Inhibitors*/pharmacology
Breast Neoplasms*/metabolism
Aromatase/metabolism ; Female ; Humans ; Receptors, Estrogen ; Triazoles/pharmacology
Czasopismo naukowe
Tytuł:
Aromatase deficiency in transplanted bone marrow cells improves vertebral trabecular bone quantity, connectivity, and mineralization and decreases cortical porosity in murine bone marrow transplant recipients.
Autorzy:
Rubitschung K; Department of Radiology, University of Texas Southwestern Medical Center, Dallas, Texas, United States of America.
Sherwood A; Department of Radiology, University of Texas Southwestern Medical Center, Dallas, Texas, United States of America.
Kapadia R; Scanco USA Incorporated, Wayne, Pennsylvania, United States of America.
Xi Y; Department of Radiology, University of Texas Southwestern Medical Center, Dallas, Texas, United States of America.
Hajibeigi A; Department of Radiology, University of Texas Southwestern Medical Center, Dallas, Texas, United States of America.
Rubinow KB; Division of Metabolism, Endocrinology, and Nutrition, University of Washington Medicine Diabetes Institute, Seattle, Washington, United States of America.
Zerwekh JE; Charles and Jane Pak Center for Mineral Metabolism and Clinical Research, UT Southwestern Medical Center, Dallas, Texas, United States of America.
Öz OK; Department of Radiology, University of Texas Southwestern Medical Center, Dallas, Texas, United States of America.; Charles and Jane Pak Center for Mineral Metabolism and Clinical Research, UT Southwestern Medical Center, Dallas, Texas, United States of America.
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Źródło:
PloS one [PLoS One] 2024 Feb 05; Vol. 19 (2), pp. e0296390. Date of Electronic Publication: 2024 Feb 05 (Print Publication: 2024).
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase*/genetics
Aromatase*/metabolism
Bone Marrow Transplantation*
Gynecomastia*
Infertility, Male*
Metabolism, Inborn Errors*
46, XX Disorders of Sex Development*
Mice ; Animals ; Male ; Cancellous Bone/diagnostic imaging ; Cancellous Bone/metabolism ; Porosity ; Mice, Inbred C57BL ; Estrogens ; Estradiol ; Bone Marrow Cells/metabolism ; Spine/metabolism ; Mice, Knockout
SCR Disease Name:
Aromatase deficiency
Czasopismo naukowe
Tytuł:
Charged Amino Acids in the Transmembrane Helix Strongly Affect the Enzyme Activity of Aromatase.
Autorzy:
Günther J; Research Institute for Farm Animal Biology (FBN), 18196 Dummerstorf, Germany.
Schuler G; Veterinary Clinic for Reproductive Medicine and Neonatology, Faculty of Veterinary Medicine, Justus Liebig University, 35392 Giessen, Germany.
Teppa E; Université de Lille, CNRS, UMR 8576-UGDF-Unité de Glycobiologie Structurale et Fonctionnelle, 59000 Lille, France.
Fürbass R; Research Institute for Farm Animal Biology (FBN), 18196 Dummerstorf, Germany.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2024 Jan 24; Vol. 25 (3). Date of Electronic Publication: 2024 Jan 24.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase*/genetics
Aromatase*/metabolism
Animals ; Female ; Humans ; Pregnancy ; Amino Acids ; Androstenedione ; Estrogens/metabolism ; Mammals/metabolism ; Protein Isoforms ; Protein Structure, Tertiary/genetics ; Protein Structure, Secondary/genetics
Czasopismo naukowe
Tytuł:
The effect of aromatase inhibitors against possible testis toxicity in pembrolizumab treated rats.
Autorzy:
Türkmen NB; Faculty of Pharmacy, Department of Pharmaceutical Toxicology, Inonu University, Malatya, Turkey.
Çiftçi O; Faculty of Medicine, Department of Medicinal Pharmacology, Pamukkale University, Denizli, Turkey.
Taşlıdere A; Faculty of Medicine, Histology and Embryology Department, Inonu University, Malatya, Turkey.
Aydın M; Faculty of Veterinary Medicine, Department of Obstetrics and Gynecology, Firat University, Elazig, Turkey.
Eke BC; Faculty of Pharmacy, Department of Pharmaceutical Toxicology, Ankara University, Ankara, Turkey.
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Źródło:
Andrologia [Andrologia] 2022 Nov; Vol. 54 (10), pp. e14557. Date of Electronic Publication: 2022 Aug 14.
Typ publikacji:
Journal Article
MeSH Terms:
Antioxidants*/pharmacology
Aromatase Inhibitors*/pharmacology
Testis*
Anastrozole/pharmacology ; Animals ; Antibodies, Monoclonal, Humanized/toxicity ; Aromatase ; Catalase/pharmacology ; Glutathione ; Glutathione Peroxidase ; Male ; Polyphenols/pharmacology ; Programmed Cell Death 1 Receptor/metabolism ; Rats ; Rats, Sprague-Dawley ; Resveratrol/pharmacology ; Semen ; Sperm Motility ; Superoxide Dismutase/metabolism ; Testosterone ; Thiobarbituric Acid Reactive Substances
Czasopismo naukowe
Tytuł:
Novel F-Labeled PET Tracers Specific to Aromatase: Design, Synthesis, and Biological Evaluation.
Autorzy:
Zheng W; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Cheng X; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Chen H; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Jiang Z; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Sun Y; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Yu Z; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Yang T; School of Pharmaceutical Science, Capital Medical University, Beijing 100069, China.
Zhang L; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
Liu Y; School of Pharmaceutical Science, Capital Medical University, Beijing 100069, China.
Ji X; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.; Institute of Hypoxia Medicine, Xuanwu Hospital, Capital Medical University, Beijing 100053, China.
Wu Z; Beijing Institute of Brain Disorders, Laboratory of Brain Disorders, Ministry of Science and Technology, Collaborative Innovation Center for Brain Disorders, Capital Medical University, Beijing 100069, China.
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Źródło:
Molecular pharmaceutics [Mol Pharm] 2022 Jul 04; Vol. 19 (7), pp. 2456-2470. Date of Electronic Publication: 2022 May 27.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Aromatase*/metabolism
Positron-Emission Tomography*/methods
Aromatase Inhibitors/metabolism ; Aromatase Inhibitors/pharmacology ; Fluorine Radioisotopes/chemistry ; Molecular Docking Simulation ; Tissue Distribution
Czasopismo naukowe
Tytuł:
Effect of Aromatase Inhibitor Letrozole on the Placenta of Adult Albino Rats: A Histopathological, Immunohistochemical, and Biochemical Study.
Autorzy:
Alabiad MA; Department of Pathology, Faculty of Medicine, Zagazig University, Zagazig, Egypt.
Elhasadi I; Department of Pathology, Faculty of Medicine, University of Benghazi, Benghazi, Libya.
Alnasser SM; Department of Pharmacology and Toxicology, Unaizah College of Pharmacy, Qassim, University, Buraydah, Saudi Arabia.
Alorini M; Department of Basic Medical Sciences, Unaizah College of Medicine and Medical Sciences, Qassim University, Unaizah, Kingdom of Saudi Arabia.
Alshaikh ABA; Department of Obstetrics and Gynecology, College of Medicine, Jouf University, Sakaka, Kingdom of Saudi Arabia.
Jaber FA; Department of Biology, College of Science, University of Jeddah, Jeddah, Kingdom of Saudi Arabia.
Shalaby AM; Department of Histology and Cell Biology, School of Medicine, Tanta University, Tanta, Egypt.
Samy W; Department of Medical Biochemistry and Molecular Biology Department, Faculty of Medicine, Zagazig University, Zagazig, Egypt.
Heraiz AI; Department of Gynecology and Obstetrics, School of Medicine, Zagazig University, Zagazig, Egypt.
Mohammed Albakoush KM; Department of Anatomy and Embryology, Faculty of Medicine, Alasmarya Islamic University, Zliten, Libya.
Khairy DA; Department of Pathology, School of Medicine, Beni-Suef University, Beni-Suef, Egypt.
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Źródło:
Iranian journal of medical sciences [Iran J Med Sci] 2024 Jan 01; Vol. 49 (1), pp. 46-56. Date of Electronic Publication: 2024 Jan 01 (Print Publication: 2024).
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase Inhibitors*/pharmacology
Letrozole*/pharmacology
Placenta*/drug effects
Animals ; Female ; Pregnancy ; Rats ; Receptors, Estrogen ; Vascular Endothelial Growth Factor A
Czasopismo naukowe
Tytuł:
Estrodiol-17β and aromatase inhibitor treatment induced alternations of genome-wide DNA methylation pattern in Takifugu rubripes gonads.
Autorzy:
Shen X; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Life Sciences, Liaoning Normal University, Dalian, Liaoning 116029, China.
Yan H; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Fisheries and Life Science, Dalian Ocean University, Dalian, Liaoning 116023, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China. Electronic address: .
Li W; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Marine Science and Environment Engineering, Dalian Ocean University, 116023 Dalian, Liaoning, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China.
Zhou H; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Fisheries and Life Science, Dalian Ocean University, Dalian, Liaoning 116023, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China.
Wang J; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Fisheries and Life Science, Dalian Ocean University, Dalian, Liaoning 116023, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China.
Zhang Q; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Fisheries and Life Science, Dalian Ocean University, Dalian, Liaoning 116023, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China.
Zhang L; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Marine Science and Environment Engineering, Dalian Ocean University, 116023 Dalian, Liaoning, China.
Liu Q; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China; College of Marine Science and Environment Engineering, Dalian Ocean University, 116023 Dalian, Liaoning, China; Key Laboratory of Pufferfish Breeding and Culture in Liaoning Province, Dalian Ocean University, 116023 Dalian, Liaoning, China. Electronic address: .
Liu Y; Key Laboratory of Environment Controlled Aquaculture (Dalian Ocean University) Ministry of Education, 116023, China.
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Źródło:
Gene [Gene] 2023 Oct 05; Vol. 882, pp. 147641. Date of Electronic Publication: 2023 Jul 15.
Typ publikacji:
Journal Article
MeSH Terms:
DNA Methylation*
Aromatase Inhibitors*/pharmacology
Aromatase Inhibitors*/metabolism
Animals ; Takifugu/genetics ; Sex Differentiation/genetics ; Gonads/metabolism
Czasopismo naukowe
Tytuł:
Use of aromatase inhibitors in menopausal deep endometriosis: a case report and literature review.
Autorzy:
Rotenberg O; Department of Obstetrics & Gynecology, Albert Einstein College of Medicine/Montefiore Medical Center, Bronx, NY, USA.
Kuo DYS; Department of Obstetrics & Gynecology, Albert Einstein College of Medicine/Montefiore Medical Center, Bronx, NY, USA.
Goldberg GL; Department of Obstetrics & Gynecology, Zucker School of Medicine at Hofstra/Northwell and NorthwellHealth, Hempstead, NY, USA.
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Źródło:
Climacteric : the journal of the International Menopause Society [Climacteric] 2022 Jun; Vol. 25 (3), pp. 235-239. Date of Electronic Publication: 2021 Oct 25.
Typ publikacji:
Case Reports; Journal Article; Review
MeSH Terms:
Aromatase Inhibitors*/therapeutic use
Endometriosis*/drug therapy
Endometriosis*/surgery
Aromatase/therapeutic use ; Female ; Humans ; Letrozole/therapeutic use ; Menopause ; Rectum
Czasopismo naukowe
Tytuł:
Glyceollins Trigger Anti-Proliferative Effects in Hormone-Dependent Aromatase-Inhibitor-Resistant Breast Cancer Cells through the Induction of Apoptosis.
Autorzy:
Walker RR; Division of Basic Sciences, College of Pharmacy and Pharmaceutical Sciences, Florida A&M University, 1415 S. Martin L. King Jr. Blvd., Tallahassee, FL 32307, USA.
Patel JR; Division of Basic Sciences, College of Pharmacy and Pharmaceutical Sciences, Florida A&M University, 1415 S. Martin L. King Jr. Blvd., Tallahassee, FL 32307, USA.
Gupta A; Department of Medicine, University of Arizona, 1500 N. Campbell Ave., Tucson, AZ 85724, USA.
Davidson AM; Division of Basic Sciences, College of Pharmacy and Pharmaceutical Sciences, Florida A&M University, 1415 S. Martin L. King Jr. Blvd., Tallahassee, FL 32307, USA.
Williams CC; Division of Basic Sciences, College of Pharmacy, Xavier University of Louisiana, 1 Drexel Dr., New Orleans, LA 70125, USA.
Payton-Stewart F; Division of Mathematics and Physical Sciences, College of Arts and Sciences, Xavier University of Louisiana, 1 Drexel Dr., New Orleans, LA 70125, USA.
Boué SM; Southern Regional Research Center, United States Department of Agriculture, Agricultural Research Service, 1100 Robert E. Lee Blvd., New Orleans, LA 70124, USA.
Burow ME; Section of Hematology and Medical Oncology, School of Medicine, Tulane University, New Orleans, LA 70112, USA.
Khupse R; College of Pharmacy, The University of Findlay, 1000 N. Main St., Findlay, OH 45840, USA.
Tilghman SL; Division of Basic Sciences, College of Pharmacy and Pharmaceutical Sciences, Florida A&M University, 1415 S. Martin L. King Jr. Blvd., Tallahassee, FL 32307, USA.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Mar 07; Vol. 23 (5). Date of Electronic Publication: 2022 Mar 07.
Typ publikacji:
Journal Article
MeSH Terms:
Aromatase Inhibitors*/pharmacology
Aromatase Inhibitors*/therapeutic use
Breast Neoplasms*/drug therapy
Breast Neoplasms*/pathology
Apoptosis ; Aromatase ; Cell Line, Tumor ; Drug Resistance, Neoplasm ; Estrogens/pharmacology ; Estrogens/therapeutic use ; Female ; Humans ; Lapatinib/pharmacology ; Lapatinib/therapeutic use ; Letrozole/pharmacology ; Neoplasm Recurrence, Local/drug therapy ; Nitriles/therapeutic use ; Pterocarpans ; Triazoles/pharmacology
Czasopismo naukowe
Tytuł:
Aromatase Inhibitor-Related Symptoms Reported by Postmenopausal Women with Nonmetastatic, Estrogen Receptor-Positive Breast Cancer: A Systematic Review.
Autorzy:
Lund-Jacobsen T; BSN, MSc, PhD student, Department of Endocrinology and Metabolism, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark. Electronic address: .
Bentsen L; MD, PhD student, Department of Oncology, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark.
Schwarz P; Professor, MD, DMSc, Department of Endocrinology and Metabolism, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Denmark, and Department of Clinical Medicine, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark.
Knop AS; MD, PhD, Department of Oncology, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark.
Pappot H; Professor, MD, DMSc, Department of Oncology, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark and Department of Clinical Medicine, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen, Denmark.
Piil K; MHScN, associate professor, Department of Oncology, Centre for Cancer and Organ Diseases, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark and Department of Publich Health, Faculty of Health, University of Aarhus, Aarhus C, Denmark.
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Źródło:
Seminars in oncology nursing [Semin Oncol Nurs] 2023 Oct; Vol. 39 (5), pp. 151487. Date of Electronic Publication: 2023 Aug 21.
Typ publikacji:
Systematic Review; Journal Article; Review; Research Support, Non-U.S. Gov't
MeSH Terms:
Aromatase Inhibitors*/adverse effects
Breast Neoplasms*/drug therapy
Female ; Humans ; Receptors, Estrogen ; Postmenopause ; Quality of Life
Czasopismo naukowe
Tytuł:
Influence of cholesterol on kinetic parameters for human aromatase (P450 19A1) in phospholipid nanodiscs.
Autorzy:
Sumangala N; Division of Metabolism, Endocrinology, & Diabetes, Department of Internal Medicine, Ann Arbor, MI 48109, USA; Program in Biophysics, University of Michigan, Ann Arbor, MI 48109, USA.
Im SC; Division of Metabolism, Endocrinology, & Diabetes, Department of Internal Medicine, Ann Arbor, MI 48109, USA; Department of Pharmacology, University of Michigan, Ann Arbor, MI 48109, USA; Veterans Affairs Medical Center, Ann Arbor, MI 48105, United States.
Valentín-Goyco J; Division of Metabolism, Endocrinology, & Diabetes, Department of Internal Medicine, Ann Arbor, MI 48109, USA; Department of Pharmacology, University of Michigan, Ann Arbor, MI 48109, USA.
Auchus RJ; Division of Metabolism, Endocrinology, & Diabetes, Department of Internal Medicine, Ann Arbor, MI 48109, USA; Program in Biophysics, University of Michigan, Ann Arbor, MI 48109, USA; Department of Pharmacology, University of Michigan, Ann Arbor, MI 48109, USA; Veterans Affairs Medical Center, Ann Arbor, MI 48105, United States. Electronic address: .
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Źródło:
Journal of inorganic biochemistry [J Inorg Biochem] 2023 Oct; Vol. 247, pp. 112340. Date of Electronic Publication: 2023 Jul 24.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Aromatase*/metabolism
Phospholipids*
Humans ; Oxidation-Reduction ; Steroids ; Cholesterol
Czasopismo naukowe

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