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Wyszukujesz frazę ""Benzothiazoles"" wg kryterium: Temat


Tytuł :
The amoebicidal activity of three substances derived from benzothiazole on Acanthamoeba castellanii cysts and trophozoites and its cytotoxic potentials.
Autorzy :
Ozpinar N; Department of Emergency Aid and Disaster Management, Faculty of Health Sciences, Mustafa Kemal University, Hatay, Antakya 31060, Turkey. Electronic address: .
Culha G; Department of Parasitology, Faculty of Medicine, Mustafa Kemal University, Hatay, Antakya 31060, Turkey.
Kaya T; Department of Parasitology, Faculty of Medicine, Mustafa Kemal University, Hatay, Antakya 31060, Turkey.
Yucel H; Department of Emergency Aid and Disaster Management, Faculty of Health Sciences, Mustafa Kemal University, Hatay, Antakya 31060, Turkey.
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Źródło :
Acta tropica [Acta Trop] 2021 Aug; Vol. 220, pp. 105981. Date of Electronic Publication: 2021 May 25.
Typ publikacji :
Journal Article
MeSH Terms :
Acanthamoeba castellanii/*drug effects
Acanthamoeba castellanii/*growth & development
Amebiasis/*drug therapy
Benzothiazoles/*chemistry
Benzothiazoles/*pharmacology
Cysts/*drug therapy
Trophozoites/*drug effects
Amebicides/chemistry ; Amebicides/pharmacology ; Amebicides/therapeutic use ; Animals ; Benzothiazoles/therapeutic use
Czasopismo naukowe
Tytuł :
Discovery of Novel Benzothiazepinones as Irreversible Covalent Glycogen Synthase Kinase 3β Inhibitors for the Treatment of Acute Promyelocytic Leukemia.
Autorzy :
Zhang P; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.; State Key Lab of New Drug & Pharmaceutical Process, Shanghai Key Lab of Anti-Infectives, Shanghai Institute of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry, Shanghai 201203, China.
Min Z; Institute of Clinical Science, Zhongshan Hospital, Fudan University, Shanghai 200032, China.
Gao Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
Bian J; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
Lin X; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
He J; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
Ye D; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
Li Y; National Facility for Protein Science in Shanghai, Zhangjiang Lab, Shanghai Advanced Research Institute, Chinese Academy of Science, Shanghai 201210, China.
Peng C; National Facility for Protein Science in Shanghai, Zhangjiang Lab, Shanghai Advanced Research Institute, Chinese Academy of Science, Shanghai 201210, China.
Cheng Y; Institute of Clinical Science, Zhongshan Hospital, Fudan University, Shanghai 200032, China.
Chu Y; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai 201203, China.
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Źródło :
Journal of medicinal chemistry [J Med Chem] 2021 Jun 10; Vol. 64 (11), pp. 7341-7358. Date of Electronic Publication: 2021 May 24.
Typ publikacji :
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms :
Benzothiazoles/*chemistry
Glycogen Synthase Kinase 3 beta/*antagonists & inhibitors
Protein Kinase Inhibitors/*chemistry
Animals ; Apoptosis/drug effects ; Benzothiazoles/metabolism ; Benzothiazoles/pharmacology ; Benzothiazoles/therapeutic use ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Female ; Glycogen Synthase Kinase 3 beta/metabolism ; Half-Life ; Humans ; Isoenzymes/antagonists & inhibitors ; Isoenzymes/metabolism ; Kinetics ; Leukemia, Promyelocytic, Acute/drug therapy ; Male ; Mice ; Mice, Inbred ICR ; Mice, Nude ; Protein Kinase Inhibitors/metabolism ; Protein Kinase Inhibitors/pharmacology ; Protein Kinase Inhibitors/therapeutic use ; Structure-Activity Relationship ; Xenograft Model Antitumor Assays
Czasopismo naukowe
Tytuł :
Exploratory Assessment of K-means Clustering to Classify 18F-Flutemetamol Brain PET as Positive or Negative.
Autorzy :
Zukotynski K; From the Department of Medicine and Radiology, McMaster University, Hamilton.
Black SE
Kuo PH; Departments of Medical Imaging, Medicine, and Biomedical Engineering, University of Arizona Cancer Center, University of Arizona, Tucson, AZ.
Bhan A; LC Campbell Cognitive Neurology Research Unit, Hurvitz Brain Sciences Research Program, Sunnybrook Research Institute, University of Toronto.
Adamo S; LC Campbell Cognitive Neurology Research Unit, Hurvitz Brain Sciences Research Program, Sunnybrook Research Institute, University of Toronto.
Scott CJM; LC Campbell Cognitive Neurology Research Unit, Hurvitz Brain Sciences Research Program, Sunnybrook Research Institute, University of Toronto.
Lam B
Masellis M
Kumar S
Fischer CE; Keenan Research Centre for Biomedical Science, St Michael's Hospital, University of Toronto.
Tartaglia MC
Lang AE
Tang-Wai DF
Freedman M
Vasdev N
Gaudet V; Department of Electrical and Computer Engineering, University of Waterloo, Waterloo, Ontario, Canada.
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Źródło :
Clinical nuclear medicine [Clin Nucl Med] 2021 Aug 01; Vol. 46 (8), pp. 616-620.
Typ publikacji :
Journal Article; Observational Study
MeSH Terms :
Aniline Compounds*
Benzothiazoles*
Positron-Emission Tomography*
Brain/*diagnostic imaging
Image Processing, Computer-Assisted/*methods
Aged ; Aged, 80 and over ; Amyloid/metabolism ; Brain/metabolism ; Cluster Analysis ; Female ; Humans ; Male ; Middle Aged ; Neurocognitive Disorders/diagnostic imaging ; Neurocognitive Disorders/metabolism ; Retrospective Studies
Czasopismo naukowe
Tytuł :
Ratiometric sensing of Zn with a new benzothiazole-based fluorescent sensor and living cell imaging.
Autorzy :
Wu Q; School of Chemistry and Chemical Engineering, Shanxi University, Taiyuan 030006, PR China. .
Feng L
Chao JB
Wang Y
Shuang S
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Źródło :
The Analyst [Analyst] 2021 Jul 07; Vol. 146 (13), pp. 4348-4356. Date of Electronic Publication: 2021 Jun 11.
Typ publikacji :
Journal Article
MeSH Terms :
Benzothiazoles*
Fluorescent Dyes*
HeLa Cells ; Humans ; Spectrometry, Fluorescence ; Zinc
Czasopismo naukowe
Tytuł :
From High-Throughput Screening to Target Validation: Benzo[ d ]isothiazoles as Potent and Selective Agonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 5 Possessing In Vivo Gastrointestinal Prokinetic Activity in Rodents.
Autorzy :
Barilli A; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Aldegheri L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Bianchi F; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Brault L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Brodbeck D; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Castelletti L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Feriani A; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Lingard I; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Myers R; Takeda Pharmaceuticals, 9625 Towne Centre Drive, San Diego, California 92121, United States.
Nola S; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Piccoli L; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Pompilio D; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Raveglia LF; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Salvagno C; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Tassini S; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Virginio C; Aptuit, an Evotec Company, Via Alessandro Fleming, 4, Verona 37135, Italy.
Sabat M; Takeda Pharmaceuticals, 9625 Towne Centre Drive, San Diego, California 92121, United States.
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Źródło :
Journal of medicinal chemistry [J Med Chem] 2021 May 13; Vol. 64 (9), pp. 5931-5955. Date of Electronic Publication: 2021 Apr 23.
Typ publikacji :
Journal Article
MeSH Terms :
High-Throughput Screening Assays*
Benzothiazoles/*chemistry
Benzothiazoles/*pharmacology
Gastrointestinal Tract/*metabolism
TRPM Cation Channels/*agonists
Animals ; Benzothiazoles/metabolism ; Benzothiazoles/pharmacokinetics ; Drug Design ; Gastrointestinal Tract/drug effects ; Humans ; Male ; Mice ; Molecular Targeted Therapy ; Reproducibility of Results ; Tissue Distribution
Czasopismo naukowe
Tytuł :
Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors.
Autorzy :
Gao D; School of Pharmacy, Fudan University, Shanghai, 201203, China; Innovation Research Institute of Traditional Chinese Medicine (IRI), Shanghai University of Traditional Chinese Medicine, Shanghai, 201203, China.
Jin N; Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
Fu Y; Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China.
Zhu Y; School of Pharmacy, Fudan University, Shanghai, 201203, China.
Wang Y; School of Pharmacy, Fudan University, Shanghai, 201203, China.
Wang T; Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
Chen Y; Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
Zhang M; School of Pharmacy, Fudan University, Shanghai, 201203, China.
Xiao Q; School of Pharmacy, Fudan University, Shanghai, 201203, China.
Huang M; Division of Antitumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China.
Li Y; School of Pharmacy, Fudan University, Shanghai, 201203, China. Electronic address: .
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Źródło :
European journal of medicinal chemistry [Eur J Med Chem] 2021 Apr 15; Vol. 216, pp. 113333. Date of Electronic Publication: 2021 Mar 02.
Typ publikacji :
Journal Article
MeSH Terms :
Drug Design*
Antineoplastic Agents/*chemistry
Benzothiazoles/*chemistry
STAT3 Transcription Factor/*antagonists & inhibitors
Antineoplastic Agents/metabolism ; Antineoplastic Agents/pharmacology ; Apoptosis/drug effects ; Benzothiazoles/metabolism ; Benzothiazoles/pharmacology ; Binding Sites ; Cell Line, Tumor ; Cell Proliferation/drug effects ; G2 Phase Cell Cycle Checkpoints/drug effects ; Humans ; Janus Kinase 2/antagonists & inhibitors ; Janus Kinase 2/metabolism ; Molecular Docking Simulation ; Phosphorylation/drug effects ; STAT3 Transcription Factor/genetics ; STAT3 Transcription Factor/metabolism ; Signal Transduction/drug effects ; Structure-Activity Relationship ; Transcription, Genetic/drug effects ; src Homology Domains
Czasopismo naukowe
Tytuł :
Modern Approaches to the Synthesis and Transformations of Practically Valuable Benzothiazole Derivatives.
Autorzy :
Zhilitskaya LV; E. Favorsky Irkutsk Institute of Chemistry, Siberian Branch of the Russian Academy of Sciences, 1 Favorsky Street, 664033 Irkutsk, Russia.
Shainyan BA; E. Favorsky Irkutsk Institute of Chemistry, Siberian Branch of the Russian Academy of Sciences, 1 Favorsky Street, 664033 Irkutsk, Russia.
Yarosh NO; E. Favorsky Irkutsk Institute of Chemistry, Siberian Branch of the Russian Academy of Sciences, 1 Favorsky Street, 664033 Irkutsk, Russia.
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Źródło :
Molecules (Basel, Switzerland) [Molecules] 2021 Apr 10; Vol. 26 (8). Date of Electronic Publication: 2021 Apr 10.
Typ publikacji :
Journal Article; Review
MeSH Terms :
Green Chemistry Technology*
Benzothiazoles/*chemical synthesis
Pharmacology/*trends
Benzothiazoles/chemistry ; Benzothiazoles/therapeutic use ; Humans
Czasopismo naukowe
Tytuł :
Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A 2A receptor ligands.
Autorzy :
Renk DR; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; University of Cologne, Faculty of Medicine and University Hospital Cologne, Institute of Radiochemistry and Experimental Molecular Imaging, Kerpener Straße 62, 50937, Köln, Germany; Forschungszentrum Jülich GmbH, Germany.
Skraban M; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; Forschungszentrum Jülich GmbH, Germany.
Bier D; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; Forschungszentrum Jülich GmbH, Germany.
Schulze A; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; Forschungszentrum Jülich GmbH, Germany.
Wabbals E; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; Forschungszentrum Jülich GmbH, Germany.
Wedekind F; Molecular Organization of the Brain (INM-2), Wilhelm-Johnen-Straße, 52428, Jülich, Germany; Forschungszentrum Jülich GmbH, Germany.
Neumaier F; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; University of Cologne, Faculty of Medicine and University Hospital Cologne, Institute of Radiochemistry and Experimental Molecular Imaging, Kerpener Straße 62, 50937, Köln, Germany; Forschungszentrum Jülich GmbH, Germany.
Neumaier B; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; University of Cologne, Faculty of Medicine and University Hospital Cologne, Institute of Radiochemistry and Experimental Molecular Imaging, Kerpener Straße 62, 50937, Köln, Germany; Forschungszentrum Jülich GmbH, Germany.
Holschbach M; Institute of Neuroscience and Medicine, Nuclear Chemistry (INM-5), Germany; Forschungszentrum Jülich GmbH, Germany. Electronic address: .
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Źródło :
European journal of medicinal chemistry [Eur J Med Chem] 2021 Mar 15; Vol. 214, pp. 113214. Date of Electronic Publication: 2021 Jan 30.
Typ publikacji :
Journal Article
MeSH Terms :
Drug Design*
Adenosine A2 Receptor Antagonists/*pharmacology
Benzothiazoles/*pharmacology
Receptor, Adenosine A2A/*metabolism
Adenosine A2 Receptor Antagonists/chemical synthesis ; Adenosine A2 Receptor Antagonists/chemistry ; Animals ; Benzothiazoles/chemical synthesis ; Benzothiazoles/chemistry ; CHO Cells ; Cells, Cultured ; Cricetulus ; Dose-Response Relationship, Drug ; Humans ; Ligands ; Molecular Structure ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł :
Highly Selective Y 4 Receptor Antagonist Binds in an Allosteric Binding Pocket.
Autorzy :
Schüß C; Institute of Biochemistry, Leipzig University, Leipzig 04103, Germany.
Vu O; Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37235, United States.
Schubert M; Institute of Biochemistry, Leipzig University, Leipzig 04103, Germany.
Du Y; Department of Pharmacology, Vanderbilt University, Nashville, Tennessee 37232, United States.
Mishra NM; Department of Pharmaceutical Sciences, UNT System College of Pharmacy, University of North Texas Health Science Center, Fort Worth, Texas 76107, United States.
Tough IR; King's College London, Wolfson Centre for Age-Related Diseases, Institute of Psychiatry, Psychology & Neuroscience, London SE1 1UL, U.K.
Stichel J; Institute of Biochemistry, Leipzig University, Leipzig 04103, Germany.
Weaver CD; Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37235, United States.; Department of Pharmacology, Vanderbilt University, Nashville, Tennessee 37232, United States.; Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States.
Emmitte KA; Department of Pharmaceutical Sciences, UNT System College of Pharmacy, University of North Texas Health Science Center, Fort Worth, Texas 76107, United States.
Cox HM; King's College London, Wolfson Centre for Age-Related Diseases, Institute of Psychiatry, Psychology & Neuroscience, London SE1 1UL, U.K.
Meiler J; Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37235, United States.; Department of Pharmacology, Vanderbilt University, Nashville, Tennessee 37232, United States.; Institute for Drug Discovery, Leipzig University, Leipzig 04103, Germany.
Beck-Sickinger AG; Institute of Biochemistry, Leipzig University, Leipzig 04103, Germany.
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Źródło :
Journal of medicinal chemistry [J Med Chem] 2021 Mar 11; Vol. 64 (5), pp. 2801-2814. Date of Electronic Publication: 2021 Feb 17.
Typ publikacji :
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms :
Benzothiazoles/*pharmacology
Receptors, Neuropeptide Y/*antagonists & inhibitors
Sulfonamides/*pharmacology
Allosteric Site ; Animals ; Benzothiazoles/chemical synthesis ; Benzothiazoles/metabolism ; Chlorocebus aethiops ; HEK293 Cells ; Humans ; Molecular Docking Simulation ; Mutagenesis ; Mutation ; Protein Binding ; Receptors, Neuropeptide Y/genetics ; Receptors, Neuropeptide Y/metabolism ; Stereoisomerism ; Sulfonamides/chemical synthesis ; Sulfonamides/metabolism
Czasopismo naukowe
Tytuł :
Label-Free Fluorescence Molecular Beacon Probes Based on G-Triplex DNA and Thioflavin T for Protein Detection.
Autorzy :
Xue J; College of Chemistry and Chemical Engineering, Gannan Normal University, Ganzhou 341000, China.
Yi J; College of Chemistry and Chemical Engineering, Gannan Normal University, Ganzhou 341000, China.
Zhou H; College of Chemistry and Chemical Engineering, Gannan Normal University, Ganzhou 341000, China.
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Źródło :
Molecules (Basel, Switzerland) [Molecules] 2021 May 17; Vol. 26 (10). Date of Electronic Publication: 2021 May 17.
Typ publikacji :
Journal Article
MeSH Terms :
Benzothiazoles/*chemistry
Biosensing Techniques/*methods
DNA/*chemistry
Benzothiazoles/metabolism ; Fluorescence ; Fluorescent Dyes/chemistry ; Limit of Detection ; Molecular Probes ; Nucleic Acid Hybridization/methods ; Proteins/chemistry ; Proteins/metabolism ; Spectrometry, Fluorescence/methods
Czasopismo naukowe
Tytuł :
Comparative evaluation and design of a G-triplex/thioflavin T-based molecular beacon.
Autorzy :
Gao J; Key Laboratory of Applied Surface and Colloid Chemistry, Ministry of Education; Key Laboratory of Analytical Chemistry for Life Science of Shaanxi Province, School of Chemistry and Chemical Engineering, Shaanxi Normal University, Xi'an 710062, China. .
Liu Q; Key Laboratory of Applied Surface and Colloid Chemistry, Ministry of Education; Key Laboratory of Analytical Chemistry for Life Science of Shaanxi Province, School of Chemistry and Chemical Engineering, Shaanxi Normal University, Xi'an 710062, China. .
Liu W; Key Laboratory of Applied Surface and Colloid Chemistry, Ministry of Education; Key Laboratory of Analytical Chemistry for Life Science of Shaanxi Province, School of Chemistry and Chemical Engineering, Shaanxi Normal University, Xi'an 710062, China. .
Jin Y; Key Laboratory of Applied Surface and Colloid Chemistry, Ministry of Education; Key Laboratory of Analytical Chemistry for Life Science of Shaanxi Province, School of Chemistry and Chemical Engineering, Shaanxi Normal University, Xi'an 710062, China. .
Li B; Key Laboratory of Applied Surface and Colloid Chemistry, Ministry of Education; Key Laboratory of Analytical Chemistry for Life Science of Shaanxi Province, School of Chemistry and Chemical Engineering, Shaanxi Normal University, Xi'an 710062, China. .
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Źródło :
The Analyst [Analyst] 2021 Apr 26; Vol. 146 (8), pp. 2567-2573.
Typ publikacji :
Journal Article
MeSH Terms :
Benzothiazoles*
Biosensing Techniques*
G-Quadruplexes*
Fluorescent Dyes
Czasopismo naukowe
Tytuł :
A benzothiazole-based near-infrared fluorescent probe for sensing SO 2 derivatives and viscosity in HeLa cells.
Autorzy :
Li Y; Department of Obstetrics and Gynecology, Affiliated Shenzhen Maternity & Child Healthcare Hospital, Southern Medical University, Shenzhen 518028, Guangdong, China.
Zhu Y; Key Laboratory of Biomedical Information Engineering of Ministry of Education, Institute of Biomedical Photonics and Sensing, School of Life Science and Technology, Xi'an Jiaotong University, Xi'an 710049, China.
Cai X; Department of Obstetrics and Gynecology, The Third Affiliated Hospital of Southern Medical University, No. 183 West Zhongshan Avenue, Guangzhou, Guangdong, China.
Guo J; Department of Obstetrics and Gynecology, Affiliated Shenzhen Maternity & Child Healthcare Hospital, Southern Medical University, Shenzhen 518028, Guangdong, China.
Yao C; Key Laboratory of Biomedical Information Engineering of Ministry of Education, Institute of Biomedical Photonics and Sensing, School of Life Science and Technology, Xi'an Jiaotong University, Xi'an 710049, China.
Pan Q; Shunde Hospital, Southern Medical University (The First People's Hospital of Shunde), Foshan, China.
Wang X; Department of Obstetrics and Gynecology, The Third Affiliated Hospital of Southern Medical University, No. 183 West Zhongshan Avenue, Guangzhou, Guangdong, China. Electronic address: .
Wang KN; Shunde Hospital, Southern Medical University (The First People's Hospital of Shunde), Foshan, China. Electronic address: .
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Źródło :
Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy [Spectrochim Acta A Mol Biomol Spectrosc] 2021 Apr 15; Vol. 251, pp. 119457. Date of Electronic Publication: 2021 Jan 12.
Typ publikacji :
Journal Article
MeSH Terms :
Benzothiazoles*
Fluorescent Dyes*
HeLa Cells ; Humans ; Microscopy, Fluorescence ; Sulfur Dioxide ; Viscosity
Czasopismo naukowe
Tytuł :
Revelation of Fe(V)/Fe(IV) Involvement in the Fe(VI)-ABTS System: Kinetic Modeling and Product Analysis.
Autorzy :
Luo C; School of Civil and Environmental Engineering, Georgia Institute of Technology, Atlanta, Georgia 30332, United States.
Sadhasivan M; School of Civil and Environmental Engineering, Georgia Institute of Technology, Atlanta, Georgia 30332, United States.
Kim J; School of Civil and Environmental Engineering, Georgia Institute of Technology, Atlanta, Georgia 30332, United States.
Sharma VK; Department of Environment and Occupational Health, School of Public Health, Texas A&M University, College Station, Texas 77843, United States.
Huang CH; School of Civil and Environmental Engineering, Georgia Institute of Technology, Atlanta, Georgia 30332, United States.
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Źródło :
Environmental science & technology [Environ Sci Technol] 2021 Mar 16; Vol. 55 (6), pp. 3976-3987. Date of Electronic Publication: 2021 Feb 26.
Typ publikacji :
Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
MeSH Terms :
Benzothiazoles*
Sulfonic Acids*
Kinetics ; Oxidation-Reduction
Czasopismo naukowe
Tytuł :
Inhibition of NUPR1-Karyopherin β1 Binding Increases Anticancer Drug Sensitivity.
Autorzy :
Park C; Center for Metareceptome Research, College of Pharmacy, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.; Institute of Gastroenterology, College of Medicine, Yonsei University, 50-1 Yonsei-ro, Seodaemun, Seoul 03772, Korea.
Oh J; Department of Chemistry, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
Lee WM; Center for Metareceptome Research, College of Pharmacy, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
Koh HR; Department of Chemistry, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
Sohn UD; Center for Metareceptome Research, College of Pharmacy, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
Ham SW; Department of Chemistry, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
Oh K; Center for Metareceptome Research, College of Pharmacy, Chung-Ang University, 84 Heukseok-ro, Dongjak, Seoul 06974, Korea.
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Źródło :
International journal of molecular sciences [Int J Mol Sci] 2021 Mar 10; Vol. 22 (6). Date of Electronic Publication: 2021 Mar 10.
Typ publikacji :
Journal Article
MeSH Terms :
Acrylamides/*pharmacology
Basic Helix-Loop-Helix Transcription Factors/*metabolism
Benzothiazoles/*pharmacology
Doxorubicin/*pharmacology
Neoplasm Proteins/*metabolism
beta Karyopherins/*metabolism
Acrylamides/chemistry ; Active Transport, Cell Nucleus/drug effects ; Antibiotics, Antineoplastic/chemistry ; Antibiotics, Antineoplastic/pharmacology ; Benzothiazoles/chemistry ; Cell Line, Tumor ; Cell Nucleus/drug effects ; Cell Nucleus/metabolism ; Cell Survival/drug effects ; Doxorubicin/chemistry ; Drug Synergism ; Humans ; MCF-7 Cells ; Microscopy, Confocal ; Molecular Structure ; Protein Binding/drug effects
Czasopismo naukowe
Tytuł :
Single-cell DNA sequencing reveals complex mechanisms of resistance to quizartinib.
Autorzy :
Peretz CAC; Department of Medicine, University of California, San Francisco, San Francisco, CA.; Children's Hospital and Research Center Oakland, Oakland, CA.; Department of Pediatrics and.
McGary LHF; Department of Medicine, University of California, San Francisco, San Francisco, CA.
Kumar T; Department of Medicine, University of California, San Francisco, San Francisco, CA.
Jackson H; School of Medicine, University of California, San Francisco, San Francisco, CA.
Jacob J; Mission Bio, Inc, San Francisco, CA.
Durruthy-Durruthy R; Mission Bio, Inc, San Francisco, CA.
Levis MJ; Sidney Kimmel Comprehensive Cancer Center, Johns Hopkins University, Baltimore, MD.
Perl A; Abramson Cancer Center, University of Pennsylvania, Philadelphia, PA; and.
Huang BJ; Department of Pediatrics and.; Helen Diller Family Comprehensive Cancer Center, University of California, San Francisco, San Francisco, CA.
Smith CC; Department of Medicine, University of California, San Francisco, San Francisco, CA.; Helen Diller Family Comprehensive Cancer Center, University of California, San Francisco, San Francisco, CA.
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Źródło :
Blood advances [Blood Adv] 2021 Mar 09; Vol. 5 (5), pp. 1437-1441.
Typ publikacji :
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms :
Benzothiazoles*
Phenylurea Compounds*
Sequence Analysis, DNA
Czasopismo naukowe
Tytuł :
The Novel Benzothiazole Derivative PB11 Induces Apoptosis via the PI3K/AKT Signaling Pathway in Human Cancer Cell Lines.
Autorzy :
Kim J; Department of Systems Biotechnology, Chung-Ang University, Ansung 17546, Korea.
Hong SH; Division of Radiation Biomedical Research, Korea Institute of Radiological and Medical Sciences, Seoul 139-706, Korea.
Jeon SH; Department of Systems Biotechnology, Chung-Ang University, Ansung 17546, Korea.
Park MH; Department of Systems Biotechnology, Chung-Ang University, Ansung 17546, Korea.
Shin CG; Department of Systems Biotechnology, Chung-Ang University, Ansung 17546, Korea.
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Źródło :
International journal of molecular sciences [Int J Mol Sci] 2021 Mar 08; Vol. 22 (5). Date of Electronic Publication: 2021 Mar 08.
Typ publikacji :
Journal Article
MeSH Terms :
Neoplasms*/drug therapy
Neoplasms*/metabolism
Neoplasms*/pathology
Antineoplastic Agents/*pharmacology
Apoptosis/*drug effects
Benzothiazoles/*pharmacology
Signal Transduction/*drug effects
Antineoplastic Agents/chemistry ; Benzothiazoles/chemistry ; HeLa Cells ; Humans ; Phosphatidylinositol 3-Kinases/metabolism ; Proto-Oncogene Proteins c-akt/metabolism
Czasopismo naukowe
Tytuł :
Proximity-Dependent Switchable ATP Aptasensors Utilizing a High-Performance FRET Reporter.
Autorzy :
Wang Q; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
Fang T; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
Zheng J; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
Shi L; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
Shi L; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
Li T; Department of Chemistry, University of Science and Technology of China, 96 Jinzhai Road, Hefei, Anhui 230026, China.
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Źródło :
ACS applied materials & interfaces [ACS Appl Mater Interfaces] 2021 Mar 03; Vol. 13 (8), pp. 9359-9368. Date of Electronic Publication: 2020 Nov 10.
Typ publikacji :
Journal Article
MeSH Terms :
Adenosine Triphosphate/*analysis
Aptamers, Nucleotide/*chemistry
Benzothiazoles/*chemistry
DNA/*chemistry
Fluorescent Dyes/*chemistry
Adenosine Triphosphate/chemistry ; Benzothiazoles/chemical synthesis ; Biosensing Techniques/methods ; Fluorescence Resonance Energy Transfer ; Fluorescent Dyes/chemical synthesis
Czasopismo naukowe
Tytuł :
Simulating the effect of cerebral blood flow changes on regional quantification of [ F]florbetaben studies.
Autorzy :
Heeman F; Amsterdam UMC, Vrije Universiteit Amsterdam, Radiology and Nuclear Medicine, Amsterdam Neuroscience, Amsterdam, Netherlands.
Yaqub M; Amsterdam UMC, Vrije Universiteit Amsterdam, Radiology and Nuclear Medicine, Amsterdam Neuroscience, Amsterdam, Netherlands.
Lopes Alves I; Amsterdam UMC, Vrije Universiteit Amsterdam, Radiology and Nuclear Medicine, Amsterdam Neuroscience, Amsterdam, Netherlands.
Heurling K; Antaros Medical AB, Mölndal, Sweden.
Bullich S; Life Molecular Imaging GmbH, Berlin, Germany.
Gispert JD; Barcelonaβeta Brain Research Centre, Pasqual Maragall Foundation, Barcelona, Spain.; Centro de Investigación Biomédica en Red de Bioingeniería, Biomateriales y Nanomedicina (CIBER-BBN), Madrid, Spain.; Department of Experimental and Health Sciences, Universitat Pompeu Fabra, Barcelona, Spain.
Boellaard R; Amsterdam UMC, Vrije Universiteit Amsterdam, Radiology and Nuclear Medicine, Amsterdam Neuroscience, Amsterdam, Netherlands.
Lammertsma AA; Amsterdam UMC, Vrije Universiteit Amsterdam, Radiology and Nuclear Medicine, Amsterdam Neuroscience, Amsterdam, Netherlands.
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Corporate Authors :
AMYPAD Consortium
Źródło :
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism [J Cereb Blood Flow Metab] 2021 Mar; Vol. 41 (3), pp. 579-589. Date of Electronic Publication: 2020 Apr 11.
Typ publikacji :
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms :
Aniline Compounds/*chemistry
Benzothiazoles/*chemistry
Cerebrovascular Circulation/*physiology
Radiopharmaceuticals/*chemistry
Stilbenes/*chemistry
Alzheimer Disease/pathology ; Aniline Compounds/pharmacology ; Benzothiazoles/pharmacology ; Case-Control Studies ; Cerebrovascular Circulation/drug effects ; Fluorine Radioisotopes/chemistry ; Humans ; Positron-Emission Tomography/methods ; Radiopharmaceuticals/pharmacology ; Stilbenes/pharmacology
Czasopismo naukowe
Tytuł :
Benzimidazole-based fluorophores for the detection of amyloid fibrils with higher sensitivity than Thioflavin-T.
Autorzy :
Pravin N; Department of Chemistry, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Kumar R; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.; Division of Neurogeriatrics, Department of Neurobiology, Care Sciences and Society, Karolinska Institutet, Stockholm, Sweden.
Tripathi S; Department of Chemistry, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Kumar P; Department of Chemistry, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Mohite GM; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Navalkar A; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Panigrahi R; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Singh N; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Gadhe LG; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Manchanda S; Division of Neurogeriatrics, Department of Neurobiology, Care Sciences and Society, Karolinska Institutet, Stockholm, Sweden.
Shimozawa M; Division of Neurogeriatrics, Department of Neurobiology, Care Sciences and Society, Karolinska Institutet, Stockholm, Sweden.
Nilsson P; Division of Neurogeriatrics, Department of Neurobiology, Care Sciences and Society, Karolinska Institutet, Stockholm, Sweden.
Johansson J; Division of Neurogeriatrics, Department of Neurobiology, Care Sciences and Society, Karolinska Institutet, Stockholm, Sweden.
Kumar A; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Maji SK; Department of Biosciences and Bioengineering, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
Shanmugam M; Department of Chemistry, Indian Institute of Technology Bombay, Mumbai, Maharashtra, India.
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Źródło :
Journal of neurochemistry [J Neurochem] 2021 Mar; Vol. 156 (6), pp. 1003-1019. Date of Electronic Publication: 2020 Sep 09.
Typ publikacji :
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms :
Amyloidosis/*pathology
Benzimidazoles/*chemistry
Benzothiazoles/*chemistry
Fluorescent Dyes/*chemistry
Amyloid beta-Peptides/chemistry ; Animals ; Benzimidazoles/chemical synthesis ; Benzimidazoles/toxicity ; Benzothiazoles/toxicity ; Cell Line ; Circular Dichroism ; Fluorescent Dyes/chemical synthesis ; Fluorescent Dyes/toxicity ; Gene Knock-In Techniques ; Humans ; Magnetic Resonance Spectroscopy ; Mice ; Microscopy, Electron, Transmission ; Peptide Fragments/chemistry ; Quantum Theory ; Reference Standards ; alpha-Synuclein/chemistry
Czasopismo naukowe
Tytuł :
Determination of benzotriazole and benzothiazole derivatives in marketed fish by double-vortex-ultrasonic assisted matrix solid-phase dispersion and ultrahigh-performance liquid chromatography-high resolution mass spectrometry.
Autorzy :
Chen CH; Department of Chemistry, National Central University, Chung-Li 320, Taiwan.
Chung WH; Department of Chemistry, National Central University, Chung-Li 320, Taiwan; Department of Chemical Engineering, Army Academy ROC, Chung-Li 320, Taiwan.
Ding WH; Department of Chemistry, National Central University, Chung-Li 320, Taiwan. Electronic address: .
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Źródło :
Food chemistry [Food Chem] 2020 Dec 15; Vol. 333, pp. 127516. Date of Electronic Publication: 2020 Jul 10.
Typ publikacji :
Journal Article
MeSH Terms :
Benzothiazoles/*chemistry
Fishes/*metabolism
Solid Phase Extraction/*methods
Animals ; Benzothiazoles/analysis ; Benzothiazoles/isolation & purification ; Chromatography, High Pressure Liquid/methods ; Limit of Detection ; Reproducibility of Results ; Spectrometry, Mass, Electrospray Ionization ; Ultrasonics
Czasopismo naukowe

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