- Tytuł:
- The antischistosomal potential of GSK-J4, an H3K27 demethylase inhibitor: insights from molecular modeling, transcriptomics and in vitro assays.
- Autorzy:
- Źródło:
- Parasites & vectors [Parasit Vectors] 2020 Mar 17; Vol. 13 (1), pp. 140. Date of Electronic Publication: 2020 Mar 17.
- Typ publikacji:
- Journal Article
- MeSH Terms:
-
Models, Molecular*
Anthelmintics/*pharmacology
Benzazepines/*pharmacology
Drug Discovery/*methods
Jumonji Domain-Containing Histone Demethylases/*antagonists & inhibitors
Pyrimidines/*pharmacology
Schistosoma mansoni/*drug effects
Animals ; Computational Biology ; Epigenesis, Genetic/drug effects ; Female ; Jumonji Domain-Containing Histone Demethylases/genetics ; Male ; Microscopy, Electron, Scanning ; Molecular Docking Simulation ; Schistosoma mansoni/genetics ; Schistosoma mansoni/ultrastructure ; Schistosomiasis mansoni/drug therapy ; Transcriptome
Czasopismo naukowe