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Tytuł:
The Protein Kinase A Inhibitor KT5720 Prevents Endothelial Dysfunctions Induced by High-Dose Irradiation.
Autorzy:
Boittin FX; Unité de Radiobiologie, Département Effets Biologiques des Rayonnements, IRBA-Institut de Recherche Biomédicale des Armées, Place du Général Valérie André, 91223 Brétigny-sur-Orge, France.
Guitard N; Unité de Radiobiologie, Département Effets Biologiques des Rayonnements, IRBA-Institut de Recherche Biomédicale des Armées, Place du Général Valérie André, 91223 Brétigny-sur-Orge, France.
Toth M; Université Paris-Saclay, INSERM, Laboratory of Signalling and Cardiovascular Pathophysiology U1180, 91400 Orsay, France.
Riccobono D; Unité de Radiobiologie, Département Effets Biologiques des Rayonnements, IRBA-Institut de Recherche Biomédicale des Armées, Place du Général Valérie André, 91223 Brétigny-sur-Orge, France.
Théry H; Unité de Radiobiologie, Département Effets Biologiques des Rayonnements, IRBA-Institut de Recherche Biomédicale des Armées, Place du Général Valérie André, 91223 Brétigny-sur-Orge, France.
Bobe R; Université Paris-Saclay, INSERM, Hémostase Inflammation Thrombose HITh U1176, 94276 Le Kremlin-Bicêtre, France.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2024 Feb 14; Vol. 25 (4). Date of Electronic Publication: 2024 Feb 14.
Typ publikacji:
Journal Article
MeSH Terms:
Endothelial Cells*/metabolism
Cyclic AMP-Dependent Protein Kinases*/metabolism
Carbazoles*
Pyrroles*
Intracellular Signaling Peptides and Proteins*
Humans ; Cells, Cultured
Czasopismo naukowe
Tytuł:
Impact of chiglitazar on glycemic control in type 2 diabetic patients with metabolic syndrome and insulin resistance: A pooled data analysis from two phase III trials.
Autorzy:
Ning Z; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Ai G; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Chen B; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Yao H; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Cao H; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Pan D; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
Lu X; Shenzhen Chipscreen Biosciences Co., Ltd., Shenzhen, China.
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Źródło:
Journal of diabetes [J Diabetes] 2024 Feb; Vol. 16 (2), pp. e13484. Date of Electronic Publication: 2023 Oct 18.
Typ publikacji:
Clinical Trial, Phase III; Journal Article
MeSH Terms:
Diabetes Mellitus, Type 2*/complications
Diabetes Mellitus, Type 2*/drug therapy
Metabolic Syndrome*/complications
Metabolic Syndrome*/drug therapy
Insulin Resistance*
Carbazoles*
Propionates*
Adult ; Humans ; Male ; Female ; Glycated Hemoglobin ; Blood Glucose/metabolism ; Glycemic Control ; Hypoglycemic Agents/therapeutic use ; Sitagliptin Phosphate/therapeutic use
Czasopismo naukowe
Tytuł:
First-Line Alectinib vs. Brigatinib in Advanced Non-Small Cell Lung Cancer with ALK Rearrangement: Real-World Data.
Autorzy:
Jeon Y; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Park S; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Jung HA; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Sun JM; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Lee SH; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Ahn JS; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
Ahn MJ; Division of Hematology-Oncology, Department of Medicine, Samsung Medical Center, Sungkyunkwan University School of Medicine, Seoul, Korea.
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Źródło:
Cancer research and treatment [Cancer Res Treat] 2024 Jan; Vol. 56 (1), pp. 61-69. Date of Electronic Publication: 2023 Jul 14.
Typ publikacji:
Observational Study; Journal Article
MeSH Terms:
Carcinoma, Non-Small-Cell Lung*/drug therapy
Carcinoma, Non-Small-Cell Lung*/genetics
Lung Neoplasms*/drug therapy
Lung Neoplasms*/genetics
Carbazoles*
Organophosphorus Compounds*
Pyrimidines*
Humans ; Piperidines/adverse effects ; Protein Kinase Inhibitors/adverse effects
Czasopismo naukowe
Tytuł:
Effect of storage duration on carprofen concentration measurements in dog plasma.
Autorzy:
Shuttleworth JR; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
Behrens KN; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
Biggo MR; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
Horne RL; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
Cox S; University of Tennessee College of Veterinary Medicine, Knoxville, Tennessee, USA.
Lakritz J; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
Tinga S; The Ohio State University College of Veterinary Medicine, Columbus, Ohio, USA.
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Źródło:
Veterinary medicine and science [Vet Med Sci] 2023 Sep; Vol. 9 (5), pp. 2022-2025. Date of Electronic Publication: 2023 Jul 20.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Anti-Inflammatory Agents, Non-Steroidal*
Carbazoles*/metabolism
Dogs ; Animals
Czasopismo naukowe
Tytuł:
Multi-Resonant Indolo[3,2,1- jk ]carbazole-Based Host for Blue Phosphorescent Organic Light-Emitting Diodes.
Autorzy:
Li X; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Yuan P; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Song J; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Chang Y; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Jiao X; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Zhao J; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Zhang C; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
Li W; Nanjing Jianuolin Optoelectronics Technology Co., Ltd., 5th Xin Mofan Road, Nanjing 210009, China.
Hang XC; School of Flexible Electronics (Future Technologies), Nanjing Tech University, 30 South Puzhu Road, Nanjing 211816, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Jun 29; Vol. 28 (13). Date of Electronic Publication: 2023 Jun 29.
Typ publikacji:
Journal Article
MeSH Terms:
Carbazoles*
Radiation*
Humans ; Electron Transport ; Tissue Donors ; Vibration
Czasopismo naukowe
Tytuł:
Near-Infrared Light-Excited Quinolinium-Carbazole Small Molecule as Two-Photon Fluorescence Nucleic Acid Probe.
Autorzy:
Sun Y; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.
Wu B; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.
Liu X; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.
Liu L; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.; Heilongjiang Provincial Key Laboratory of New Drug Development and Pharmacotoxicological Evaluation, Jiamusi 154007, China.
Zhou S; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.; Heilongjiang Provincial Key Laboratory of New Drug Development and Pharmacotoxicological Evaluation, Jiamusi 154007, China.
Feng Y; College of Pharmacy, Jiamusi University, Jiamusi 154007, China.; Heilongjiang Provincial Key Laboratory of New Drug Development and Pharmacotoxicological Evaluation, Jiamusi 154007, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2024 Feb 29; Vol. 29 (5). Date of Electronic Publication: 2024 Feb 29.
Typ publikacji:
Journal Article
MeSH Terms:
Iodides*
Photons*
Fluorescence ; Carbazoles ; DNA ; Infrared Rays ; Nucleic Acid Probes ; Fluorescent Dyes
Czasopismo naukowe
Tytuł:
Identifying optimal ALK inhibitors in first- and second-line treatment of patients with advanced ALK-positive non-small-cell lung cancer: a systematic review and network meta-analysis.
Autorzy:
Zhao M; Department of Pharmacoeconomics, School of International Pharmaceutical Business, China Pharmaceutical University, Nanjing, Jiangsu, China.; Center for Pharmacoeconomics and Outcomes Research, China Pharmaceutical University, Nanjing, Jiangsu, China.
Shao T; Department of Pharmacoeconomics, School of International Pharmaceutical Business, China Pharmaceutical University, Nanjing, Jiangsu, China.; Center for Pharmacoeconomics and Outcomes Research, China Pharmaceutical University, Nanjing, Jiangsu, China.
Shao H; Department of Pharmacoeconomics, School of International Pharmaceutical Business, China Pharmaceutical University, Nanjing, Jiangsu, China.; Center for Pharmacoeconomics and Outcomes Research, China Pharmaceutical University, Nanjing, Jiangsu, China.
Zhou C; Shanghai Pulmonary Hospital, Tongji University, Shanghai, China. .
Tang W; Department of Pharmacoeconomics, School of International Pharmaceutical Business, China Pharmaceutical University, Nanjing, Jiangsu, China. .; Center for Pharmacoeconomics and Outcomes Research, China Pharmaceutical University, Nanjing, Jiangsu, China. .
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Źródło:
BMC cancer [BMC Cancer] 2024 Feb 08; Vol. 24 (1), pp. 186. Date of Electronic Publication: 2024 Feb 08.
Typ publikacji:
Meta-Analysis; Systematic Review; Journal Article
MeSH Terms:
Carcinoma, Non-Small-Cell Lung*/drug therapy
Lung Neoplasms*/drug therapy
Lung Neoplasms*/chemically induced
Sulfones*
Aminopyridines*
Lactams*
Pyrimidines*
Pyrazoles*
Organophosphorus Compounds*
Humans ; Crizotinib/therapeutic use ; Network Meta-Analysis ; Bayes Theorem ; Quality of Life ; Anaplastic Lymphoma Kinase ; Protein Kinase Inhibitors/therapeutic use ; Carbazoles/therapeutic use
Czasopismo naukowe
Tytuł:
A case of inflammatory myofibroblastic tumor harboring EML4-ALK fusion with a brain metastasis responding to alectinib.
Autorzy:
Sakoda S; Department of Respiratory Medicine, Graduate School of Medical Sciences, Kyushu University, Fukuoka, Japan.; Department of Respiratory Medicine, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Tanaka K; Department of Respiratory Medicine, Graduate School of Medical Sciences, Kyushu University, Fukuoka, Japan.
Koga Y; Department of Respiratory Medicine, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Mikumo H; Department of Respiratory Medicine, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Tsuchiya-Kawano Y; Department of Respiratory Medicine, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Harada E; Department of Respiratory Medicine, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Tamiya S; Department of Pathology, Kitakyushu Municipal Medical Center, Fukuoka, Japan.
Okamoto I; Department of Respiratory Medicine, Graduate School of Medical Sciences, Kyushu University, Fukuoka, Japan.
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Źródło:
Thoracic cancer [Thorac Cancer] 2024 Feb; Vol. 15 (5), pp. 415-418. Date of Electronic Publication: 2024 Jan 11.
Typ publikacji:
Case Reports
MeSH Terms:
Brain Neoplasms*/drug therapy
Brain Neoplasms*/genetics
Brain Neoplasms*/secondary
Granuloma, Plasma Cell*/pathology
Female ; Humans ; Aged ; Anaplastic Lymphoma Kinase/genetics ; Piperidines/therapeutic use ; Carbazoles/therapeutic use ; Oncogene Proteins, Fusion/genetics
Raport
Tytuł:
Synthesis of a Tetrahedral Metal-Organic Supramolecular Cage with Dendritic Carbazole Arms.
Autorzy:
Lianglu J; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
Hu W; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
Zhu X; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
Zhang HY; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.; School of Basic Medical Science, Zhengzhou University, Zhengzhou 450001, China.
Shi L; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
Hao XQ; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
Song MP; College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Dec 08; Vol. 23 (24). Date of Electronic Publication: 2022 Dec 08.
Typ publikacji:
Journal Article
MeSH Terms:
Carbazoles*
Coloring Agents*
Gases ; Luminescence ; Metals
Czasopismo naukowe
Tytuł:
Carprofen alleviates Alzheimer-like phenotypes of 5XFAD transgenic mice by targeting the pathological hallmarks induced by amyloid-β aggregation.
Autorzy:
Lee D; Department of Pharmacy, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.; Yonsei Institute of Pharmaceutical Sciences, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.
Ryoo JE; Department of Pharmacy, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.; Yonsei Institute of Pharmaceutical Sciences, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.
Hong S; Department of Pharmacy, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.; Yonsei Frontier Lab, Yonsei University, Seoul, 03722, Republic of Korea.; Pharmaceutical Sciences Division, School of Pharmacy, University of Wisconsin-Madison, Madison, WI, USA.; Wisconsin Center for NanoBioSystems, University of Wisconsin-Madison, Madison, WI, USA.
Kim HY; Department of Pharmacy, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.; Yonsei Institute of Pharmaceutical Sciences, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea.
Kim Y; Department of Pharmacy, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea. .; Yonsei Institute of Pharmaceutical Sciences, College of Pharmacy, Yonsei University, Incheon, 21983, Republic of Korea. .; Yonsei Frontier Lab, Yonsei University, Seoul, 03722, Republic of Korea. .; Department of Integrative Biotechnology and Translational Medicine, Yonsei University, Incheon, 21983, Republic of Korea. .
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Źródło:
Scientific reports [Sci Rep] 2023 Jul 05; Vol. 13 (1), pp. 10889. Date of Electronic Publication: 2023 Jul 05.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Alzheimer Disease*/drug therapy
Alzheimer Disease*/genetics
Alzheimer Disease*/metabolism
Mice ; Animals ; Mice, Transgenic ; Amyloid beta-Peptides/metabolism ; Carbazoles/pharmacology ; Carbazoles/therapeutic use ; Memory Disorders/pathology ; Disease Models, Animal
Czasopismo naukowe
Tytuł:
The Aryl Hydrocarbon Receptor Ligand FICZ Improves Left Ventricular Remodeling and Cardiac Function at the Onset of Pressure Overload-Induced Heart Failure in Mice.
Autorzy:
Tamayo M; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Martín-Nunes L; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Piedras MJ; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.; Facultad de Medicina, Universidad Francisco de Vitoria (UFV), 28223 Madrid, Spain.
Martin-Calvo M; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Martí-Morente D; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Gil-Fernández M; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.; Innate Immune Response Group, IdiPAZ, La Paz University Hospital, 28046 Madrid, Spain.
Gómez-Hurtado N; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Moro MÁ; Centro Nacional de Investigaciones Cardiovasculares (CNIC), Melchor Fernández Almagro 3, 28029 Madrid, Spain.
Bosca L; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
Fernández-Velasco M; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.; Innate Immune Response Group, IdiPAZ, La Paz University Hospital, 28046 Madrid, Spain.
Delgado C; Instituto de Investigaciones Biomédicas 'Alberto Sols' (CSIC-UAM), CIBER de Enfermedades Cardiovasculares (CIBERCV), 28029 Madrid, Spain.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 May 12; Vol. 23 (10). Date of Electronic Publication: 2022 May 12.
Typ publikacji:
Journal Article
MeSH Terms:
Carbazoles*/pharmacology
Heart Failure*/drug therapy
Heart Failure*/etiology
Heart Failure*/metabolism
Receptors, Aryl Hydrocarbon*/genetics
Receptors, Aryl Hydrocarbon*/metabolism
Ventricular Remodeling*
Animals ; Cardiomegaly/metabolism ; Fibrosis ; Ligands ; Mice ; Mice, Inbred C57BL ; Myocytes, Cardiac/metabolism
Czasopismo naukowe
Tytuł:
Alectinib-induced red cell morphological changes in a patient with underlying α-thalassaemia trait.
Autorzy:
Li THS; Department of Pathology, Queen Elizabeth Hospital, Hong Kong, Hong Kong.
Chik YKJ; Department of Clinical Oncology, Queen Elizabeth Hospital, Hong Kong, Hong Kong.
Wong WS; Department of Pathology, Queen Elizabeth Hospital, Hong Kong, Hong Kong.
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Źródło:
International journal of laboratory hematology [Int J Lab Hematol] 2022 Feb; Vol. 44 (1), pp. 65-66. Date of Electronic Publication: 2021 Oct 13.
Typ publikacji:
Case Reports
MeSH Terms:
Adenocarcinoma of Lung*/blood
Adenocarcinoma of Lung*/drug therapy
Carbazoles*/administration & dosage
Carbazoles*/adverse effects
Erythrocytes, Abnormal*/metabolism
Erythrocytes, Abnormal*/pathology
Lung Neoplasms*/blood
Lung Neoplasms*/drug therapy
Piperidines*/administration & dosage
Piperidines*/adverse effects
alpha-Thalassemia*/blood
alpha-Thalassemia*/drug therapy
alpha-Thalassemia*/pathology
Humans ; Male ; Middle Aged
Raport
Tytuł:
Exploring determinants of agonist efficacy at the CB1 cannabinoid receptor: Analogues of the synthetic cannabinoid receptor agonist EG-018.
Autorzy:
Finlay DB; Department of Pharmacology and Toxicology, School of Biomedical Sciences, University of Otago, Dunedin, New Zealand.
Nguyen T; RTI International, Research Triangle Park, North Carolina, USA.
Gamage TF; RTI International, Research Triangle Park, North Carolina, USA.
Chen S; Department of Pharmacology and Toxicology, School of Biomedical Sciences, University of Otago, Dunedin, New Zealand.
Barrus DG; RTI International, Research Triangle Park, North Carolina, USA.
Patel PR; RTI International, Research Triangle Park, North Carolina, USA.
Thomas BF; RTI International, Research Triangle Park, North Carolina, USA.
Wiley JL; RTI International, Research Triangle Park, North Carolina, USA.
Zhang Y; RTI International, Research Triangle Park, North Carolina, USA.
Glass M; Department of Pharmacology and Toxicology, School of Biomedical Sciences, University of Otago, Dunedin, New Zealand.
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Źródło:
Pharmacology research & perspectives [Pharmacol Res Perspect] 2022 Feb; Vol. 10 (1), pp. e00901.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Cannabinoid Receptor Agonists/*pharmacology
Carbazoles/*pharmacology
Naphthalenes/*pharmacology
Receptor, Cannabinoid, CB1/*agonists
Cannabinoid Receptor Agonists/chemical synthesis ; Cannabinoid Receptor Agonists/chemistry ; Carbazoles/chemical synthesis ; Carbazoles/chemistry ; Cyclic AMP/metabolism ; GTP-Binding Proteins/metabolism ; HEK293 Cells ; Humans ; Naphthalenes/chemical synthesis ; Naphthalenes/chemistry ; Signal Transduction/drug effects ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Antimicrobial Activity and Toxicity of Newly Synthesized 4-[4-(benzylamino)butoxy]-9 H -carbazole Derivatives.
Autorzy:
Niedziałkowska K; Department of Industrial Microbiology and Biotechnology, Faculty of Biology and Environmental Protection, University of Lodz, 90-237 Lodz, Poland.
Felczak A; Department of Industrial Microbiology and Biotechnology, Faculty of Biology and Environmental Protection, University of Lodz, 90-237 Lodz, Poland.
Głowacka IE; Bioorganic Chemistry Laboratory, Faculty of Pharmacy, Medical University of Lodz, 90-151 Lodz, Poland.
Piotrowska DG; Bioorganic Chemistry Laboratory, Faculty of Pharmacy, Medical University of Lodz, 90-151 Lodz, Poland.
Lisowska K; Department of Industrial Microbiology and Biotechnology, Faculty of Biology and Environmental Protection, University of Lodz, 90-237 Lodz, Poland.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Sep 06; Vol. 24 (18). Date of Electronic Publication: 2023 Sep 06.
Typ publikacji:
Journal Article
MeSH Terms:
Escherichia coli*
Staphylococcus aureus*
Humans ; Antifungal Agents/pharmacology ; Candida albicans ; Carbazoles/toxicity ; Pseudomonas aeruginosa
Czasopismo naukowe
Tytuł:
Photophysical Exploration of Alectinib and Rilpivirine: Insights from Theory and Experiment.
Autorzy:
Zhang C; School of Life Sciences and Health Engineering, Jiangnan University, Wuxi 214122, China.
Yang Y; School of Life Sciences and Health Engineering, Jiangnan University, Wuxi 214122, China.
Gan S; School of Life Sciences and Health Engineering, Jiangnan University, Wuxi 214122, China.
Ren A; Institute of Theoretical Chemistry, College of Chemistry, Jilin University, Liutiao Road 2#, Changchun 130061, China.
Zhou YB; National Center for Drug Screening, State key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, SSIP Healthcare and Medicine Demonstration Zone, Zhongshan Tsuihang New District, Zhongshan 528400, China.
Li J; National Center for Drug Screening, State key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China.; Zhongshan Institute for Drug Discovery, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, SSIP Healthcare and Medicine Demonstration Zone, Zhongshan Tsuihang New District, Zhongshan 528400, China.
Xiang DJ; Xishan People's Hospital of Wuxi City, Wuxi 214105, China.
Wang WL; School of Life Sciences and Health Engineering, Jiangnan University, Wuxi 214122, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Aug 21; Vol. 28 (16). Date of Electronic Publication: 2023 Aug 21.
Typ publikacji:
Journal Article
MeSH Terms:
Rilpivirine*
Lung Neoplasms*
Humans ; HeLa Cells ; Carbazoles/pharmacology
Czasopismo naukowe
Tytuł:
A Bayesian network meta-analysis of ALK inhibitor treatments in patients with ALK-positive non-small cell lung cancer.
Autorzy:
Zheng B; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Jiang H; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Yang W; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Li Y; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Liang B; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Zhu J; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Chen N; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Chen M; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
Zhang M; Department of Pharmacy, Tongde Hospital Zhejiang Province, Hangzhou, China.; Department of Pharmacy, Zhejiang Academy of Traditional Chinese Medicine, Hangzhou, China.
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Źródło:
Cancer medicine [Cancer Med] 2023 Aug; Vol. 12 (15), pp. 15983-15997. Date of Electronic Publication: 2023 Jun 19.
Typ publikacji:
Meta-Analysis; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Carcinoma, Non-Small-Cell Lung*/drug therapy
Carcinoma, Non-Small-Cell Lung*/genetics
Lung Neoplasms*/drug therapy
Lung Neoplasms*/genetics
Brain Neoplasms*/secondary
Humans ; Crizotinib/therapeutic use ; Network Meta-Analysis ; Bayes Theorem ; Anaplastic Lymphoma Kinase/genetics ; Protein Kinase Inhibitors/adverse effects ; Carbazoles/therapeutic use
Czasopismo naukowe
Tytuł:
Design, Synthesis and Evaluation of Novel Carbazole-Derived Photocages.
Autorzy:
Wang Z; Department of Chemistry, The University of Texas at Austin, Austin, Texas, 78712, USA.
Martin SF; Department of Chemistry, The University of Texas at Austin, Austin, Texas, 78712, USA.
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Źródło:
Chemistry (Weinheim an der Bergstrasse, Germany) [Chemistry] 2022 Mar 28; Vol. 28 (18), pp. e202200311. Date of Electronic Publication: 2022 Feb 25.
Typ publikacji:
Journal Article
MeSH Terms:
Carbazoles*
Solubility
Czasopismo naukowe
Tytuł:
Differential Modulation of Dendritic Cell Biology by Endogenous and Exogenous Aryl Hydrocarbon Receptor Ligands.
Autorzy:
Sadeghi Shermeh A; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Royzman D; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Kuhnt C; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Draßner C; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Stich L; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Steinkasserer A; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Knippertz I; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
Wild AB; Department of Immune Modulation, Universitätsklinikum Erlangen, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91052 Erlangen, Germany.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Apr 25; Vol. 24 (9). Date of Electronic Publication: 2023 Apr 25.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Aryl Hydrocarbon*/genetics
Receptors, Aryl Hydrocarbon*/metabolism
Gene Expression Regulation*
Humans ; Ligands ; Carbazoles/pharmacology ; Carbazoles/metabolism ; Indican/metabolism ; Dendritic Cells ; Biology
Czasopismo naukowe
Tytuł:
Antiviral Activities of Carbazole Derivatives against Porcine Epidemic Diarrhea Virus In Vitro.
Autorzy:
Chen Z; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Chen J; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Wei X; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Hua H; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Hu R; Jiangxi Provincial Key Laboratory for Animal Health, Institute of Animal Population Health, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Ding N; State Key Laboratory for Pig Genetic Improvement and Production Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Zhang J; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Song D; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Ye Y; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Tang Y; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Ding Z; Department of Preventive Veterinary Medicine, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.; Jiangxi Engineering Research Center for Animal Health Products, College of Animal Science and Technology, Jiangxi Agricultural University, Nanchang 330045, China.
Ke S; Hubei Biopesticide Engineering Research Centre, Hubei Academy of Agricultural Sciences, Wuhan 430064, China.
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Źródło:
Viruses [Viruses] 2021 Dec 16; Vol. 13 (12). Date of Electronic Publication: 2021 Dec 16.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antiviral Agents/*pharmacology
Carbazoles/*pharmacology
Porcine epidemic diarrhea virus/*drug effects
Animals ; Antiviral Agents/chemistry ; Carbazoles/chemistry ; Cell Survival/drug effects ; Chlorocebus aethiops ; Dose-Response Relationship, Drug ; Molecular Structure ; Vero Cells ; Virus Attachment/drug effects ; Virus Replication/drug effects
Czasopismo naukowe
Tytuł:
Molecular Mechanisms of Anticancer Activity of N-Glycosides of Indolocarbazoles LCS-1208 and LCS-1269.
Autorzy:
Zenkov RG; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Vlasova OA; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Maksimova VP; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Fetisov TI; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Karpechenko NY; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Ektova LV; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Eremina VA; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Popova VG; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.; Faculty of Biotechnology and Industrial Ecology, Mendeleev University of Chemical Technology of Russia, 9 Miusskaya Ploshchad, 125047 Moscow, Russia.
Usalka OG; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.; International School 'Medicine of the Future', I.M. Sechenov First Moscow State Medical University, 8-2 Trubetskaya St., 119991 Moscow, Russia.
Lesovaya EA; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.; Department of Oncology, I.P. Pavlov Ryazan State Medical University, 9 Vysokovoltnaya St., 390026 Ryazan, Russia.
Belitsky GA; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Yakubovskaya MG; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.
Kirsanov KI; N. N. Blokhin Russian Cancer Research Center, 24 Kashirskoe Shosse, 115478 Moscow, Russia.; Institute of Medicine, RUDN University, 6 Miklukho-Maklaya St., 117198 Moscow, Russia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2021 Dec 02; Vol. 26 (23). Date of Electronic Publication: 2021 Dec 02.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents/*pharmacology
Carbazoles/*pharmacology
Glycosides/*pharmacology
Antineoplastic Agents/chemistry ; Carbazoles/chemistry ; Cell Line, Tumor ; Epigenesis, Genetic/drug effects ; Glycosides/chemistry ; Humans ; Indoles/chemistry ; Indoles/pharmacology ; Neoplasms/drug therapy ; Neoplasms/genetics
Czasopismo naukowe

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