- Tytuł :
-
PET imaging and pharmacological therapy targeting
carbonic anhydrase -IX high-expressing tumors using US2 platform based on bivalent ureidosulfonamide. - Autorzy :
- Źródło :
- PloS one [PLoS One] 2020 Dec 09; Vol. 15 (12), pp. e0243327. Date of Electronic Publication: 2020 Dec 09 (Print Publication: 2020).
- Typ publikacji :
- Journal Article; Research Support, Non-U.S. Gov't
- MeSH Terms :
-
Antigens, Neoplasm*/metabolism
Carbonic Anhydrase IX */antagonists & inhibitorsCarbonic Anhydrase IX */metabolismCarbonic Anhydrase Inhibitors*/chemistryCarbonic Anhydrase Inhibitors*/pharmacokineticsCarbonic Anhydrase Inhibitors*/pharmacology
Neoplasm Proteins*/antagonists & inhibitors
Neoplasm Proteins*/metabolism
Neoplasms, Experimental*/diagnostic imaging
Neoplasms, Experimental*/drug therapy
Neoplasms, Experimental*/enzymology
Positron-Emission Tomography*
Yttrium Radioisotopes*/chemistry
Yttrium Radioisotopes*/pharmacokinetics
Yttrium Radioisotopes*/pharmacology
Animals ; HT29 Cells ; Humans ; Male ; Mice ; Mice, Inbred BALB C ; Mice, Nude ; Xenograft Model Antitumor Assays -
Czasopismo naukowe