Informacja

Drogi użytkowniku, aplikacja do prawidłowego działania wymaga obsługi JavaScript. Proszę włącz obsługę JavaScript w Twojej przeglądarce.

Wyszukujesz frazę ""Chloroquine"" wg kryterium: Temat


Tytuł:
N-Substituted Phenylhydrazones Kill the Ring Stage of Plasmodium falciparum .
Autorzy:
Amengor CDK; Department of Pharmaceutical Chemistry, School of Pharmacy, University of Health and Allied Sciences, Ho, Ghana.
Biniyam PD; Department of Pharmaceutical Chemistry, School of Pharmacy, University of Health and Allied Sciences, Ho, Ghana.
Brobbey AA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Pharmaceutical Sciences, Kwame Nkrumah University of Science and Technology, Kumasi, Ghana.
Kekessie FK; Department of Chemistry and Biochemistry, The University of Southern Mississippi, Hattiesburg Campus, 118 College Drive, Hattiesburg, USA.
Zoiku FK; Department of Epidemiology, Noguchi Memorial Institute for Medical Research, College of Health Sciences, University of Ghana, P.O. Box LG 581, Legon, Accra, Ghana.
Hamidu S; Department of Clinical Pathology, Noguchi Memorial Institute for Medical Research, College of Health Sciences, University of Ghana, P.O. Box LG 581, Legon, Accra, Ghana.
Gyan P; Department of Pharmaceutical Chemistry, School of Pharmacy, University of Health and Allied Sciences, Ho, Ghana.
Abudey BM; Department of Pharmaceutical Chemistry, School of Pharmacy, University of Health and Allied Sciences, Ho, Ghana.
Pokaż więcej
Źródło:
BioMed research international [Biomed Res Int] 2024 Feb 13; Vol. 2024, pp. 6697728. Date of Electronic Publication: 2024 Feb 13 (Print Publication: 2024).
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/therapeutic use
Malaria*/parasitology
Hydrazones*
Humans ; Plasmodium falciparum ; Chloroquine/therapeutic use
Czasopismo naukowe
Tytuł:
Molecular surveillance of chloroquine resistance in Plasmodium vivax isolates from malaria cases in Yunnan Province of China using pvcrt-o gene polymorphisms.
Autorzy:
Ding H; Faculty of Life Science and Technology, Kunming University of Science and Technology, Kunming, 650500, China.; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Dong Y; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China. .
Deng Y; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Xu Y; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Liu Y; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Wu J; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Chen M; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Zhang C; Yunnan Provincial Key Laboratory of Vector-borne Diseases Control and Research, Yunnan International Joint Laboratory of Tropical Infectious Diseases, Yunnan Institute of Parasitic Diseases Control, Pu'er, 665000, China.
Liu L; Faculty of Life Science and Technology, Kunming University of Science and Technology, Kunming, 650500, China. .
Lin Y; Center for Disease Control and Prevention, Dehong, 678499, China. .
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Nov 08; Vol. 22 (1), pp. 338. Date of Electronic Publication: 2023 Nov 08.
Typ publikacji:
Journal Article
MeSH Terms:
Malaria, Vivax*/epidemiology
Antimalarials*/pharmacology
Antimalarials*/therapeutic use
Malaria*/drug therapy
Humans ; Chloroquine/pharmacology ; Chloroquine/therapeutic use ; Plasmodium vivax/genetics ; Plasmodium vivax/metabolism ; Cohort Studies ; Drug Resistance/genetics ; Membrane Transport Proteins/genetics ; Membrane Transport Proteins/metabolism ; China ; Polymorphism, Single Nucleotide ; Protozoan Proteins/metabolism
Czasopismo naukowe
Tytuł:
Mechanism of DNA Intercalation by Chloroquine Provides Insights into Toxicity.
Autorzy:
Joshi J; Department of Physics, Northeastern University, Boston, MA 02115, USA.
McCauley MJ; Department of Physics, Northeastern University, Boston, MA 02115, USA.
Morse M; Department of Physics, Northeastern University, Boston, MA 02115, USA.
Muccio MR; Department of Chemistry and Biochemistry, Center for RNA Biology, Ohio State University, Columbus, OH 43210, USA.
Kanlong JG; Department of Chemistry and Biochemistry, Center for RNA Biology, Ohio State University, Columbus, OH 43210, USA.
Rocha MS; Department of Physics, Universidade Federal de Viçosa, Viçosa CEP 36570-900, MG, Brazil.
Rouzina I; Department of Chemistry and Biochemistry, Center for RNA Biology, Ohio State University, Columbus, OH 43210, USA.
Musier-Forsyth K; Department of Chemistry and Biochemistry, Center for RNA Biology, Ohio State University, Columbus, OH 43210, USA.
Williams MC; Department of Physics, Northeastern University, Boston, MA 02115, USA.
Pokaż więcej
Źródło:
International journal of molecular sciences [Int J Mol Sci] 2024 Jan 24; Vol. 25 (3). Date of Electronic Publication: 2024 Jan 24.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*
Antineoplastic Agents*/toxicity
Chloroquine/toxicity ; DNA/chemistry ; Calorimetry
Czasopismo naukowe
Tytuł:
Parallel Synthesis of Piperazine Tethered Thiazole Compounds with Antiplasmodial Activity.
Autorzy:
Rayala R; Herbert Wertheim College of Medicine, Center for Translational Science, Florida International University, Miami, FL 33199, USA.
Chaudhari P; Herbert Wertheim College of Medicine, Center for Translational Science, Florida International University, Miami, FL 33199, USA.
Bunnell A; Herbert Wertheim College of Medicine, Center for Translational Science, Florida International University, Miami, FL 33199, USA.
Roberts B; Division of Molecular Microbiology, Burnett School of Biomedical Sciences, University of Central Florida, Orlando, FL 32826, USA.
Chakrabarti D; Division of Molecular Microbiology, Burnett School of Biomedical Sciences, University of Central Florida, Orlando, FL 32826, USA.
Nefzi A; Herbert Wertheim College of Medicine, Center for Translational Science, Florida International University, Miami, FL 33199, USA.
Pokaż więcej
Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Dec 12; Vol. 24 (24). Date of Electronic Publication: 2023 Dec 12.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/chemistry
Piperazine ; Thiazoles/chemistry ; Chloroquine/pharmacology ; Chloroquine/chemistry ; Plasmodium falciparum
Czasopismo naukowe
Tytuł:
Rapid profiling of Plasmodium parasites from genome sequences to assist malaria control.
Autorzy:
Phelan JE; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK. .
Turkiewicz A; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.
Manko E; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.
Thorpe J; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.
Vanheer LN; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.
van de Vegte-Bolmer M; Department of Medical Microbiology and Radboud Center for Infectious Diseases, Radboud University Medical Center, University of Nijmegen, Nijmegen, The Netherlands.
Ngoc NTH; Molecular Biology Department, Parasitology and Entomology, Vietnam National Institute of Malariology, Hanoi, Vietnam.
Binh NTH; Molecular Biology Department, Parasitology and Entomology, Vietnam National Institute of Malariology, Hanoi, Vietnam.
Thieu NQ; Molecular Biology Department, Parasitology and Entomology, Vietnam National Institute of Malariology, Hanoi, Vietnam.
Gitaka J; Directorate of Research and Innovation, Mount Kenya University, Gen. Kago Rd, Thika, Kenya.
Nolder D; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.; UK Health Security Agency Malaria Reference Laboratory, LSHTM, London, WC1E 7HT, UK.
Beshir KB; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.
Dombrowski JG; Department of Parasitology, Institute of Biomedical Sciences, Univ. of São Paulo, São Paulo, Brazil.
Di Santi SM; School of Medicine, Instituto de Medicina Tropical, University of São Paulo, São Paulo, Brazil.
Bousema T; Department of Medical Microbiology and Radboud Center for Infectious Diseases, Radboud University Medical Center, University of Nijmegen, Nijmegen, The Netherlands.
Sutherland CJ; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK.; UK Health Security Agency Malaria Reference Laboratory, LSHTM, London, WC1E 7HT, UK.
Campino S; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK. .
Clark TG; Faculty of Infectious and Tropical Diseases, London School of Hygiene & Tropical Medicine (LSHTM), London, WC1E 7HT, UK. .; Faculty of Epidemiology and Population Health, LSHTM, London, WC1E 7HT, UK. .
Pokaż więcej
Źródło:
Genome medicine [Genome Med] 2023 Nov 10; Vol. 15 (1), pp. 96. Date of Electronic Publication: 2023 Nov 10.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antimalarials*/pharmacology
Antimalarials*/therapeutic use
Parasites*
Coinfection*/drug therapy
Malaria*/drug therapy
Malaria*/parasitology
Plasmodium*/genetics
Malaria, Falciparum*/drug therapy
Malaria, Vivax*
Humans ; Animals ; Chloroquine/therapeutic use ; Drug Resistance/genetics ; Plasmodium falciparum/genetics
Czasopismo naukowe
Tytuł:
Antiplasmodial and Antileishmanial Activities of a New Limonoid and Other Constituents from the Stem Bark of Khaya senegalensis .
Autorzy:
Amang À Ngnoung GA; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.
Nganso Ditchou YO; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.
Leutcha PB; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.; Natural Product and Environmental Chemistry Group (NAPEC), Department of Chemistry, Higher Teachers' Training College, University of Maroua, Maroua P.O. Box 55, Cameroon.
Dize D; Antimicrobial and Biocontrol Agents Unit (AmBcAU), Laboratory for Phytobiochemistry and Medicinal Plants Studies, Department of Biochemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.
Tatsimo SJN; Natural Product and Environmental Chemistry Group (NAPEC), Department of Chemistry, Higher Teachers' Training College, University of Maroua, Maroua P.O. Box 55, Cameroon.
Tchokouaha LRY; Laboratory of Pharmacology, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.
Kowa TK; Laboratory of Phytochemistry, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.
Tembeni B; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Mamoudou H; Department of Biological Sciences, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.
Poka M; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Demana PH; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Siwe Noundou X; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Fekam Boyom F; Antimicrobial and Biocontrol Agents Unit (AmBcAU), Laboratory for Phytobiochemistry and Medicinal Plants Studies, Department of Biochemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.; Laboratory of Pharmacology, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.; Advanced Research and Health Innovation Hub (ARHIH), Yaoundé P.O. Box 20133, Cameroon.
Meli Lannang A; Natural Product and Environmental Chemistry Group (NAPEC), Department of Chemistry, Higher Teachers' Training College, University of Maroua, Maroua P.O. Box 55, Cameroon.; Department of Chemical Engineering, School of Chemical Engineering and Mineral Industries, University of Ngaoundere, Ngaoundere P.O. Box 454, Cameroon.
Pokaż więcej
Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Oct 23; Vol. 28 (20). Date of Electronic Publication: 2023 Oct 23.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/chemistry
Limonins*/pharmacology
Limonins*/analysis
Antiprotozoal Agents*/pharmacology
Antiprotozoal Agents*/analysis
Malaria, Falciparum*
Meliaceae*/chemistry
Humans ; Plant Extracts/chemistry ; Sulfadoxine/analysis ; Plant Bark/chemistry ; Chloroquine ; Plasmodium falciparum
Czasopismo naukowe
Tytuł:
Structure-Activity Relationships and Antiplasmodial Potencies of Novel 3,4-Disubstituted 1,2,5-Oxadiazoles.
Autorzy:
Hochegger P; Institute of Pharmaceutical Sciences, Pharmaceutical Chemistry, University of Graz, Schubertstraße 1, A-8010 Graz, Austria.
Hermann T; Institute of Pharmaceutical Sciences, Pharmaceutical Chemistry, University of Graz, Schubertstraße 1, A-8010 Graz, Austria.
Dolensky J; Institute of Pharmaceutical Sciences, Pharmaceutical Chemistry, University of Graz, Schubertstraße 1, A-8010 Graz, Austria.
Seebacher W; Institute of Pharmaceutical Sciences, Pharmaceutical Chemistry, University of Graz, Schubertstraße 1, A-8010 Graz, Austria.
Saf R; Institute for Chemistry and Technology of Materials (ICTM), Graz University of Technology, Stremayrgasse 9, A-8010 Graz, Austria.
Pferschy-Wenzig EM; Institute of Pharmaceutical Sciences, Pharmacognosy, University of Graz, Beethovenstraße 8, A-8010 Graz, Austria.
Kaiser M; Swiss Tropical and Public Health Institute, Kreuzstraße 2, CH-4123 Allschwil, Switzerland.; Faculty of Philosophy and Natural Sciences, University of Basel, Swiss TPH, Petersplatz 1, CH-4003 Basel, Switzerland.
Mäser P; Swiss Tropical and Public Health Institute, Kreuzstraße 2, CH-4123 Allschwil, Switzerland.; Faculty of Philosophy and Natural Sciences, University of Basel, Swiss TPH, Petersplatz 1, CH-4003 Basel, Switzerland.
Weis R; Institute of Pharmaceutical Sciences, Pharmaceutical Chemistry, University of Graz, Schubertstraße 1, A-8010 Graz, Austria.
Pokaż więcej
Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Sep 23; Vol. 24 (19). Date of Electronic Publication: 2023 Sep 23.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/chemistry
Malaria, Falciparum*/drug therapy
Malaria*/drug therapy
Humans ; Chloroquine/pharmacology ; Plasmodium falciparum ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
The impact of anti-malarial markets on artemisinin resistance: perspectives from Burkina Faso.
Autorzy:
Guissou RM; Institut de Recherche en Sciences de la Sante, Centre National de la Recherche Scientifique et Technologique, Ouagadougou, Burkina Faso. .
Amaratunga C; Mahidol Oxford Tropical Medicine Research Unit, Faculty of Tropical Medicine, Mahidol University, Bangkok, Thailand.; Center for Tropical Medicine and Global Health, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
de Haan F; Copernicus Institute of Sustainable Development, Utrecht University, Utrecht, The Netherlands.
Tou F; Institut des Sciences et Techniques, Bobo-Dioulasso, Burkina Faso.
Cheah PY; Mahidol Oxford Tropical Medicine Research Unit, Faculty of Tropical Medicine, Mahidol University, Bangkok, Thailand.; Center for Tropical Medicine and Global Health, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
Yerbanga RS; Institut de Recherche en Sciences de la Sante, Centre National de la Recherche Scientifique et Technologique, Ouagadougou, Burkina Faso.; Institut des Sciences et Techniques, Bobo-Dioulasso, Burkina Faso.
Moors EHM; Copernicus Institute of Sustainable Development, Utrecht University, Utrecht, The Netherlands.
Dhorda M; Mahidol Oxford Tropical Medicine Research Unit, Faculty of Tropical Medicine, Mahidol University, Bangkok, Thailand.; Center for Tropical Medicine and Global Health, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
Tindana P; School of Public Health, College of Health Sciences, University of Ghana, Accra, Ghana.
Boon WPC; Copernicus Institute of Sustainable Development, Utrecht University, Utrecht, The Netherlands.
Dondorp AM; Mahidol Oxford Tropical Medicine Research Unit, Faculty of Tropical Medicine, Mahidol University, Bangkok, Thailand.; Center for Tropical Medicine and Global Health, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
Ouédraogo JB; Institut des Sciences et Techniques, Bobo-Dioulasso, Burkina Faso.
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Sep 13; Vol. 22 (1), pp. 269. Date of Electronic Publication: 2023 Sep 13.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Antimalarials*/pharmacology
Artemisinins*/pharmacology
Humans ; Burkina Faso ; Chloroquine ; Administrative Personnel
Czasopismo naukowe
Tytuł:
Rebound of multiple infections and prevalence of anti-malarial resistance associated markers following malaria upsurges in Dielmo village, Senegal, West Africa.
Autorzy:
Wotodjo AN; VITROME, UMR 257 IRD, Campus UCAD-IRD, Dakar, Senegal. .; Medical Research Council Unit, London School of Hygiene and Tropical Medicine, Fajara, The Gambia. .
Oboh MA; Medical Research Council Unit, London School of Hygiene and Tropical Medicine, Fajara, The Gambia.; Department of Biological Sciences, University of Medical Sciences, Ondo, Nigeria.; Department of Biomedical Sciences, Rochester Institute of Technology, Rochester, NY, USA.
Doucoure S; VITROME, UMR 257 IRD, Campus UCAD-IRD, Dakar, Senegal.
Diagne N; VITROME, UMR 257 IRD, Campus UCAD-IRD, Dakar, Senegal.
Diène-Sarr F; Institut Pasteur de Dakar, 36 Avenue Pasteur, 220, Dakar, Senegal.
Niang M; Institut Pasteur de Dakar, 36 Avenue Pasteur, 220, Dakar, Senegal.
Trape JF; UMR MIVEGEC, Laboratoire de Paludologie et Zoologie Médicale, IRD, Dakar, Senegal.
Sokhna C; VITROME, UMR 257 IRD, Campus UCAD-IRD, Dakar, Senegal.
Amambua-Ngwa A; Medical Research Council Unit, London School of Hygiene and Tropical Medicine, Fajara, The Gambia.
D'Alessandro U; Medical Research Council Unit, London School of Hygiene and Tropical Medicine, Fajara, The Gambia.
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Sep 05; Vol. 22 (1), pp. 257. Date of Electronic Publication: 2023 Sep 05.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*
Malaria*
Malaria, Falciparum*
Humans ; Senegal ; Prevalence ; Africa, Western ; Chloroquine ; Membrane Transport Proteins
Czasopismo naukowe
Tytuł:
Therapeutic efficacy of Chloroquine for the treatment of uncomplicated Plasmodium vivax infection in Shewa Robit, Northeast Ethiopia.
Autorzy:
Belay H; Department of Medical Laboratory Science College of Medicine and Health Science, Wolkite University, Wolkite, Ethiopia.
Alemu M; Department of Medical Laboratory Science, College of Medicine and Health Sciences, Bahir Dar University, Bahir Dar, Ethiopia.
Hailu T; Department of Medical Laboratory Science, College of Medicine and Health Sciences, Bahir Dar University, Bahir Dar, Ethiopia.
Mohammed H; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.
Sime H; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.
Hailegeorgies H; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.
Gidey B; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.
Haile M; Ethiopian Ministry of Health, Addis Ababa, Ethiopia.
Assefa G; Ethiopian Ministry of Health, Addis Ababa, Ethiopia.
Bekele W; World Health Organization Addis Ababa, Ethiopia.
Alebachew Reta M; Department of Medical Laboratory Science, College of Medicine and Health Sciences, Wollo University, Dessie, Ethiopia.
Almaw Tamene A; Department of Medical Laboratory Science, College of Health Sciences, Debre Tabor University, Debre Tabor, Ethiopia.
Tasew G; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.
Assefa A; Ethiopian Public Health Institute, Addis Ababa, Ethiopia.; Institute for Global Health and Infectious Disease, University of North Carolina at Chapel Hill, Chapel, North Carolina, United States of America.
Pokaż więcej
Źródło:
PloS one [PLoS One] 2023 Jan 12; Vol. 18 (1), pp. e0277362. Date of Electronic Publication: 2023 Jan 12 (Print Publication: 2023).
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/therapeutic use
Chloroquine*/therapeutic use
Malaria, Vivax*/epidemiology
Humans ; Ethiopia/epidemiology ; Hemoglobins ; Plasmodium vivax ; Prospective Studies ; Treatment Outcome ; Infant ; Child, Preschool ; Child ; Adolescent ; Young Adult ; Adult ; Middle Aged
Czasopismo naukowe
Tytuł:
Transmission-blocking activity of antimalarials for Plasmodium vivax malaria in Anopheles darlingi.
Autorzy:
Andrade AO; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Santos NAC; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.; Programa de Pós-Graduação em Biologia Experimental, Fundação Universidade Federal de Rondônia, FIOCRUZ Rondônia, Porto Velho, Rondônia, Brazil.
Bastos AS; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Pontual JDC; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Araújo JE; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.; Programa de Pós-Graduação em Biologia Experimental, Fundação Universidade Federal de Rondônia, FIOCRUZ Rondônia, Porto Velho, Rondônia, Brazil.
Silva AMV; Ambulatório de Malária, Centro de Pesquisa em Medicina Tropical, Porto Velho, Rondônia, Brazil.
Martinez LN; Programa de Pós-Graduação em Biologia Experimental, Fundação Universidade Federal de Rondônia, FIOCRUZ Rondônia, Porto Velho, Rondônia, Brazil.; Plataforma de Bioensaios de Malária e Leishmaniose da Fiocruz (PBML), Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Lima AA; Ambulatório de Malária, Centro de Pesquisa em Medicina Tropical, Porto Velho, Rondônia, Brazil.
Aguiar ACC; Universidade Federal de São Paulo, Departamento de Biociência, Santos, São Paulo, Brazil.
G Teles CB; Programa de Pós-Graduação em Biologia Experimental, Fundação Universidade Federal de Rondônia, FIOCRUZ Rondônia, Porto Velho, Rondônia, Brazil.; Plataforma de Bioensaios de Malária e Leishmaniose da Fiocruz (PBML), Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Medeiros JF; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.; Programa de Pós-Graduação em Biologia Experimental, Fundação Universidade Federal de Rondônia, FIOCRUZ Rondônia, Porto Velho, Rondônia, Brazil.
Pereira DB; Ambulatório de Malária, Centro de Pesquisa em Medicina Tropical, Porto Velho, Rondônia, Brazil.
Vinetz JM; Section of Infectious Diseases, Department of Internal Medicine, Yale School of Medicine, New Haven, Connecticut, United States of America.
Gazzinelli RT; Laboratório de Imunopatologia, Instituto René Rachou, Fundação Oswaldo Cruz, Belo Horizonte, Minas Gerais, Brazil.; Department of Medicine, University of Massachusetts Medical School, Worcester, Massachusetts, United States of America.
Araújo MS; Plataforma de Produção e Infecção de Vetores da Malária (PIVEM), Laboratório de Entomologia, Fiocruz Rondônia, Porto Velho, Rondônia, Brazil.
Pokaż więcej
Źródło:
PLoS neglected tropical diseases [PLoS Negl Trop Dis] 2023 Jun 16; Vol. 17 (6), pp. e0011425. Date of Electronic Publication: 2023 Jun 16 (Print Publication: 2023).
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/pharmacology
Antimalarials*/therapeutic use
Malaria, Vivax*/drug therapy
Malaria, Vivax*/parasitology
Anopheles*/parasitology
Malaria*/drug therapy
Animals ; Humans ; Primaquine/pharmacology ; Primaquine/therapeutic use ; Chloroquine/pharmacology ; Chloroquine/therapeutic use ; Plasmodium vivax
Czasopismo naukowe
Tytuł:
PfCRT mutations conferring piperaquine resistance in falciparum malaria shape the kinetics of quinoline drug binding and transport.
Autorzy:
Gomez GM; Center of Infectious Diseases, Parasitology, Universitätsklinikum Heidelberg, Im Neuenheimer Feld, Heidelberg, Germany.
D'Arrigo G; Molecular and Cellular Modelling Group, Heidelberg Institute for Theoretical Studies (HITS), Schloss-Wolfsbrunnenweg, Heidelberg, Germany.
Sanchez CP; Center of Infectious Diseases, Parasitology, Universitätsklinikum Heidelberg, Im Neuenheimer Feld, Heidelberg, Germany.
Berger F; Center of Infectious Diseases, Parasitology, Universitätsklinikum Heidelberg, Im Neuenheimer Feld, Heidelberg, Germany.
Wade RC; Molecular and Cellular Modelling Group, Heidelberg Institute for Theoretical Studies (HITS), Schloss-Wolfsbrunnenweg, Heidelberg, Germany.; Center for Molecular Biology (ZMBH), DKFZ-ZMBH Alliance, Heidelberg University, Im Neuenheimer Feld, Heidelberg, Germany.; Interdisciplinary Center for Scientific Computing (IWR), Heidelberg University, Im Neuenheimer Feld, Heidelberg, Germany.
Lanzer M; Center of Infectious Diseases, Parasitology, Universitätsklinikum Heidelberg, Im Neuenheimer Feld, Heidelberg, Germany.
Pokaż więcej
Źródło:
PLoS pathogens [PLoS Pathog] 2023 Jun 07; Vol. 19 (6), pp. e1011436. Date of Electronic Publication: 2023 Jun 07 (Print Publication: 2023).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antimalarials*/chemistry
Malaria, Falciparum*/drug therapy
Plasmodium falciparum*/genetics
Plasmodium falciparum*/metabolism
Quinolines*/pharmacology
Quinolines*/therapeutic use
Humans ; Chloroquine/pharmacology ; Chloroquine/therapeutic use ; Drug Resistance/genetics ; Kinetics ; Mutation ; Protozoan Proteins/metabolism
Czasopismo naukowe
Tytuł:
Clinical isolates of uncomplicated falciparum malaria from high and low malaria transmission areas show distinct pfcrt and pfmdr1 polymorphisms in western Ethiopia.
Autorzy:
Tadele G; Aklilu Lemma Institute of Pathobiology, Addis Ababa University, Addis Ababa, Ethiopia.
Jawara A; Medical Research Council Unit the Gambia, London School of Hygiene and Tropical Medicine, Banjul, Gambia.
Oboh M; Medical Research Council Unit the Gambia, London School of Hygiene and Tropical Medicine, Banjul, Gambia.
Oriero E; Medical Research Council Unit the Gambia, London School of Hygiene and Tropical Medicine, Banjul, Gambia.
Dugassa S; Aklilu Lemma Institute of Pathobiology, Addis Ababa University, Addis Ababa, Ethiopia.
Amambua-Ngwa A; Medical Research Council Unit the Gambia, London School of Hygiene and Tropical Medicine, Banjul, Gambia.
Golassa L; Aklilu Lemma Institute of Pathobiology, Addis Ababa University, Addis Ababa, Ethiopia. .
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Jun 03; Vol. 22 (1), pp. 171. Date of Electronic Publication: 2023 Jun 03.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/pharmacology
Antimalarials*/therapeutic use
Malaria, Falciparum*/parasitology
Malaria*/drug therapy
Humans ; Ethiopia/epidemiology ; Artemether, Lumefantrine Drug Combination/therapeutic use ; Artemether/therapeutic use ; Chloroquine/pharmacology ; Chloroquine/therapeutic use ; Lumefantrine/therapeutic use ; Plasmodium falciparum ; Polymorphism, Single Nucleotide ; Multidrug Resistance-Associated Proteins/genetics ; Protozoan Proteins/genetics ; Protozoan Proteins/therapeutic use ; Drug Resistance/genetics
Czasopismo naukowe
Tytuł:
Development of a human malaria-on-a-chip disease model for drug efficacy and off-target toxicity evaluation.
Autorzy:
Rupar MJ; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Sasserath T; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Smith E; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Comiter B; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Sriram N; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Long CJ; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
McAleer CW; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA.
Hickman JJ; Hesperos, Inc., 12501 Research Parkway, Suite 100, Orlando, FL, 32826, USA. .
Pokaż więcej
Źródło:
Scientific reports [Sci Rep] 2023 Jun 28; Vol. 13 (1), pp. 10509. Date of Electronic Publication: 2023 Jun 28.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antimalarials*/pharmacology
Malaria*/drug therapy
Malaria, Falciparum*/drug therapy
Humans ; Endothelial Cells ; Parasitemia/drug therapy ; Chloroquine/pharmacology ; Lab-On-A-Chip Devices
Czasopismo naukowe
Tytuł:
Characteristics of molecular markers associated with chloroquine resistance in Plasmodium vivax strains from vivax malaria cases in Yunnan Province, China.
Autorzy:
Ding H; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.; Faculty of Life Science and Technology, Kunming University of Science and Technology, Kunming, 650500, China.
Dong Y; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China. .
Deng Y; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Xu Y; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Liu Y; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Wu J; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Chen M; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Zhang C; Yunnan Institute of Parasitic Diseases Control, Yunnan Provincial Key Laboratory, Yunnan Centre of Malaria Research, Pu'er, 665000, China.
Zheng W; Center for Disease Control and Prevention, Baoshan, 678000, China. .
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Jun 11; Vol. 22 (1), pp. 181. Date of Electronic Publication: 2023 Jun 11.
Typ publikacji:
Journal Article
MeSH Terms:
Malaria, Vivax*
Antimalarials*/pharmacology
Humans ; Plasmodium vivax/genetics ; Chloroquine/pharmacology ; China/epidemiology ; Biomarkers
Czasopismo naukowe
Tytuł:
Favorable Preclinical Pharmacological Profile of a Novel Antimalarial Pyrrolizidinylmethyl Derivative of 4-amino-7-chloroquinoline with Potent In Vitro and In Vivo Activities.
Autorzy:
Basilico N; Dipartimento di Scienze Biomediche, Chirurgiche e Odontoiatriche (DiSBIOC), Università Degli Studi di Milano, Via Pascal 36, 20133 Milan, Italy.
Parapini S; Dipartimento di Scienze Biomediche per la Salute, Università Degli Studi di Milano, Via Pascal 36, 20133 Milan, Italy.
D'Alessandro S; Dipartimento di Scienze Farmacologiche e Biomolecolari (DISFEB), Università Degli Studi di Milano, Via Pascal 36, 20133 Milan, Italy.
Misiano P; Dipartimento di Scienze Farmacologiche e Biomolecolari (DISFEB), Università Degli Studi di Milano, Via Pascal 36, 20133 Milan, Italy.
Romeo S; Dipartimento di Scienze Farmaceutiche (DISFARM), Università Degli Studi di Milano, Via Mangiagalli 25, 20133 Milan, Italy.
Dondio G; Aphad Srl, Via della Resistenza 65, Buccinasco, 20090 Milan, Italy.
Yardley V; Department of Immunology Biology, Faculty of Infectious and Tropical Diseases, London School of Hygiene and Tropical Medicine (LSHTM), Keppel Street, London WC1E 7HT, UK.
Vivas L; Department of Immunology Biology, Faculty of Infectious and Tropical Diseases, London School of Hygiene and Tropical Medicine (LSHTM), Keppel Street, London WC1E 7HT, UK.
Nasser S; Department of Immunology Biology, Faculty of Infectious and Tropical Diseases, London School of Hygiene and Tropical Medicine (LSHTM), Keppel Street, London WC1E 7HT, UK.
Rénia L; Lee Kong Chian School of Medicine, Nanyang Technological University, Singapore 308232, Singapore.; A*STAR Infectious Diseases Labs, Agency for Science, Technology, and Research, Singapore 138648, Singapore.
Russell BM; Department of Microbiology and Immunology, University of Otago, Dunedin 9054, New Zealand.
Suwanarusk R; Department of Microbiology and Immunology, University of Otago, Dunedin 9054, New Zealand.
Nosten F; Shoklo Malaria Research Unit, Mahidol-Oxford Research Unit, Faculty of Tropical Medicine, Mahidol University, Mae Sot 63110, Thailand.; Centre for Tropical Medicine and Global Health, Nuffield Department of Medicine, University of Oxford, Oxford OX3 7BN, UK.
Sparatore A; Dipartimento di Scienze Farmaceutiche (DISFARM), Università Degli Studi di Milano, Via Mangiagalli 25, 20133 Milan, Italy.
Taramelli D; Dipartimento di Scienze Farmacologiche e Biomolecolari (DISFEB), Università Degli Studi di Milano, Via Pascal 36, 20133 Milan, Italy.
Pokaż więcej
Źródło:
Biomolecules [Biomolecules] 2023 May 14; Vol. 13 (5). Date of Electronic Publication: 2023 May 14.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antimalarials*/therapeutic use
Quinolines*/pharmacology
Malaria*/drug therapy
Malaria*/parasitology
Malaria, Falciparum*/drug therapy
Artemisinins*/pharmacology
Rats ; Animals ; Dogs ; Plasmodium falciparum ; Chloroquine/pharmacology
Czasopismo naukowe
Tytuł:
Molecular epidemiology of potential candidate markers for chloroquine resistance in imported Plasmodium vivax malaria cases in Iran.
Autorzy:
Pirahmadi S; Malaria and Vector Research Group (MVRG), Biotechnology Research Center (BRC), Pasteur Institute of Iran, Tehran, Iran.
Afzali S; Malaria and Vector Research Group (MVRG), Biotechnology Research Center (BRC), Pasteur Institute of Iran, Tehran, Iran.
Mehrizi AA; Malaria and Vector Research Group (MVRG), Biotechnology Research Center (BRC), Pasteur Institute of Iran, Tehran, Iran. .
Raz A; Malaria and Vector Research Group (MVRG), Biotechnology Research Center (BRC), Pasteur Institute of Iran, Tehran, Iran. .
Raeisi A; National Programme Manager for Malaria Control, Ministry of Health and Medical Education, Tehran, Iran.
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Apr 10; Vol. 22 (1), pp. 118. Date of Electronic Publication: 2023 Apr 10.
Typ publikacji:
Journal Article
MeSH Terms:
Malaria, Vivax*/epidemiology
Malaria, Vivax*/drug therapy
Antimalarials*/pharmacology
Antimalarials*/therapeutic use
Humans ; Chloroquine/pharmacology ; Chloroquine/therapeutic use ; Iran/epidemiology ; Molecular Epidemiology ; Multidrug Resistance-Associated Proteins/genetics ; Plasmodium vivax ; Drug Resistance/genetics ; Protozoan Proteins/genetics ; Protozoan Proteins/therapeutic use
Czasopismo naukowe
Tytuł:
Treatment of uncomplicated Plasmodium vivax with chloroquine plus radical cure with primaquine without G6PDd testing is safe in Arba Minch, Ethiopia: assessment of clinical and parasitological response.
Autorzy:
Mekonnen DA; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia. .; Institute of Biotechnology, Addis Ababa University, 1176, Addis Ababa, Ethiopia. .
Abadura GS; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia.
Behaksra SW; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia.
Taffese HS; National Malaria Control Program/Federal Ministry of Health, Addis Ababa, Ethiopia.
Bayissa GA; National Malaria Control Program/Federal Ministry of Health, Addis Ababa, Ethiopia.
Bulto MG; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia.
Tessema TS; Institute of Biotechnology, Addis Ababa University, 1176, Addis Ababa, Ethiopia.
Tadesse FG; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia.
Gadisa E; Malaria and Neglected Tropical Diseases Directorate, Armauer Hansen Research Institute, 1005, Addis Ababa, Ethiopia.
Pokaż więcej
Źródło:
Malaria journal [Malar J] 2023 Apr 25; Vol. 22 (1), pp. 135. Date of Electronic Publication: 2023 Apr 25.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/pharmacology
Malaria, Vivax*/drug therapy
Malaria, Vivax*/prevention & control
Humans ; Primaquine ; Chloroquine/pharmacology ; Plasmodium vivax ; Ethiopia ; Parasitemia/drug therapy
Czasopismo naukowe
Tytuł:
Antileishmanial and Antiplasmodial Activities of Secondary Metabolites from the Root of Antrocaryon klaineanum Pierre (Anacardiaceae).
Autorzy:
Amang À Ngnoung GA; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.; Laboratory of Phytochemistry, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.
Sidjui LS; Laboratory of Phytochemistry, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.; Bioorganic and Medicinal Chemistry Laboratory, Department of Organic Chemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.
Leutcha PB; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.; Natural Product and Environmental Chemistry Group (NAPEC), Department of Chemistry, Higher Teachers' Training College, University of Maroua, Maroua P.O. Box 55, Cameroon.
Nganso Ditchou YO; Department of Chemistry, Faculty of Science, University of Maroua, Maroua P.O. Box 814, Cameroon.; Laboratory of Medicinal Chemistry & Pharmacognosy, Department of Organic Chemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.
Tchokouaha LRY; Laboratory of Pharmacology and Drugs Discovery, IMPM, Yaoundé P.O. Box 13033, Cameroon.
Herbette G; Aix-Marseille Univ, CNRS, Centrale Marseille, FSCM, Spectropole, Campus de St Jérôme-Service 511, 13397 Marseille, France.
Baghdikian B; Aix Marseille Univ, CNRS 7263, IRD 237, Avignon Université, IMBE, 27 Blvd Jean Moulin, Service of Pharmacognosy, Faculty of Pharmacy, 13385 Marseille, France.
Kowa TK; Laboratory of Phytochemistry, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.
Soh D; Laboratory of Medicinal Chemistry & Pharmacognosy, Department of Organic Chemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.; Department of Chemistry, Higher Teacher Training College Bambili, The University of Bamenda, Bambili, Bamenda P.O. Box 39, Cameroon.
Kemzeu R; Antimicrobial and Biocontrol Agents Unit, Laboratory for Phytobiochemistry and Medicinal Plants Studies, Department of Biochemistry, Faculty of Science, University of Yaounde 1, Yaounde P.O. Box 812, Cameroon.
Poka M; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Demana PH; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Siwe Noundou X; Department of Pharmaceutical Sciences, School of Pharmacy, Sefako Makgatho Health Sciences University, Pretoria 0204, South Africa.
Tchinda AT; Laboratory of Phytochemistry, Centre for Research on Medicinal Plants and Traditional Medicine, Institute of Medical Research and Medicinal Plants Studies, Yaoundé P.O. Box 13033, Cameroon.
Fekam Boyom F; Antimicrobial and Biocontrol Agents Unit, Laboratory for Phytobiochemistry and Medicinal Plants Studies, Department of Biochemistry, Faculty of Science, University of Yaounde 1, Yaounde P.O. Box 812, Cameroon.
Lannang AM; Natural Product and Environmental Chemistry Group (NAPEC), Department of Chemistry, Higher Teachers' Training College, University of Maroua, Maroua P.O. Box 55, Cameroon.; Department of Chemical Engineering, School of Chemical Engineering and Mineral Industries, University of Ngaoundere, Ngaoundere P.O. Box 454, Cameroon.
Nyassé B; Laboratory of Medicinal Chemistry & Pharmacognosy, Department of Organic Chemistry, Faculty of Science, University of Yaoundé I, Yaoundé P.O. Box 812, Cameroon.
Pokaż więcej
Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Mar 17; Vol. 28 (6). Date of Electronic Publication: 2023 Mar 17.
Typ publikacji:
Journal Article
MeSH Terms:
Antimalarials*/pharmacology
Antimalarials*/chemistry
Anacardiaceae*/chemistry
Antiprotozoal Agents*/pharmacology
Plant Extracts/chemistry ; Chloroquine ; Plasmodium falciparum
Czasopismo naukowe
Tytuł:
Identifying inhibitors of β-haematin formation with activity against chloroquine-resistant Plasmodium falciparum malaria parasites via virtual screening approaches.
Autorzy:
Amod L; Department of Chemistry, University of Cape Town, Rondebosch, 7701, South Africa.
Mohunlal R; Department of Chemistry, University of Cape Town, Rondebosch, 7701, South Africa.
Teixeira N; Department of Chemistry, University of Cape Town, Rondebosch, 7701, South Africa.
Egan TJ; Department of Chemistry, University of Cape Town, Rondebosch, 7701, South Africa.; Institute of Infectious Diseases and Molecular Medicine, University of Cape Town, Rondebosch, 7701, South Africa.
Wicht KJ; Department of Chemistry, University of Cape Town, Rondebosch, 7701, South Africa. .; Drug Discovery and Development Centre (H3D), University of Cape Town, Rondebosch, 7701, South Africa. .; Institute of Infectious Diseases and Molecular Medicine, University of Cape Town, Rondebosch, 7701, South Africa. .
Pokaż więcej
Źródło:
Scientific reports [Sci Rep] 2023 Feb 14; Vol. 13 (1), pp. 2648. Date of Electronic Publication: 2023 Feb 14.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural
MeSH Terms:
Antimalarials*/therapeutic use
Malaria, Falciparum*/drug therapy
Malaria, Falciparum*/parasitology
Humans ; Bayes Theorem ; Chloroquine/therapeutic use ; Molecular Docking Simulation ; Plasmodium falciparum
Czasopismo naukowe

Ta witryna wykorzystuje pliki cookies do przechowywania informacji na Twoim komputerze. Pliki cookies stosujemy w celu świadczenia usług na najwyższym poziomie, w tym w sposób dostosowany do indywidualnych potrzeb. Korzystanie z witryny bez zmiany ustawień dotyczących cookies oznacza, że będą one zamieszczane w Twoim komputerze. W każdym momencie możesz dokonać zmiany ustawień dotyczących cookies