- Tytuł:
-
Discovery of new acetylcholinesterase
inhibitors for Alzheimer's disease: virtual screening and in vitro characterisation. - Autorzy:
- Źródło:
- Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2021 Dec; Vol. 36 (1), pp. 491-496.
- Typ publikacji:
- Journal Article
- MeSH Terms:
-
Drug Discovery*
Acetylcholinesterase/*metabolism
Alzheimer Disease/*drug therapyCholinesterase Inhibitors /*pharmacologyDonepezil /*pharmacology
Physostigmine/*pharmacology
Alzheimer Disease/metabolism ; Animals ;Cholinesterase Inhibitors /chemistry ;Donepezil /chemistry ; Dose-Response Relationship, Drug ; Drug Evaluation, Preclinical ; Electrophorus ; Molecular Docking Simulation ; Molecular Structure ; Physostigmine/chemistry ; Structure-Activity Relationship
Czasopismo naukowe