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Wyszukujesz frazę ""Colletier JP"" wg kryterium: Autor


Tytuł:
Time-resolved serial femtosecond crystallography on fatty-acid photodecarboxylase: lessons learned.
Autorzy:
Hadjidemetriou K; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Coquelle N; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Barends TRM; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
De Zitter E; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Schlichting I; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Colletier JP; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Weik M; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
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Źródło:
Acta crystallographica. Section D, Structural biology [Acta Crystallogr D Struct Biol] 2022 Sep 01; Vol. 78 (Pt 9), pp. 1131-1142. Date of Electronic Publication: 2022 Aug 25.
Typ publikacji:
Journal Article
MeSH Terms:
Fatty Acids*
Lasers*
Crystallography ; Crystallography, X-Ray ; Light ; Spectrum Analysis
Czasopismo naukowe
Tytuł:
Xtrapol8 enables automatic elucidation of low-occupancy intermediate-states in crystallographic studies.
Autorzy:
De Zitter E; Univ. Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000, Grenoble, France.
Coquelle N; European Synchrotron Radiation Facility (ESRF), BP 220, 38043, Grenoble, France.
Oeser P; Univ. Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000, Grenoble, France.
Barends TRM; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120, Heidelberg, Germany.
Colletier JP; Univ. Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000, Grenoble, France. colletier@ibs.fr.
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Źródło:
Communications biology [Commun Biol] 2022 Jun 29; Vol. 5 (1), pp. 640. Date of Electronic Publication: 2022 Jun 29.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Crystallography*/methods
Bayes Theorem ; Kinetics ; Ligands
Czasopismo naukowe
Tytuł:
Structural and biochemical characterisation of the Providencia stuartii arginine decarboxylase shows distinct polymerisation and regulation.
Autorzy:
Jessop M; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.; Division of Structural Biology, The Institute of Cancer Research (ICR), London, UK.
Huard K; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Desfosses A; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Tetreau G; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Carriel D; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Bacia-Verloop M; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Mas C; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Mas P; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Fraudeau A; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Colletier JP; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France.
Gutsche I; Institut de Biologie Structurale, Univ Grenoble Alpes, CEA, CNRS, IBS, 71 Avenue des martyrs, F-38044, Grenoble, France. .
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Źródło:
Communications biology [Commun Biol] 2022 Apr 05; Vol. 5 (1), pp. 317. Date of Electronic Publication: 2022 Apr 05.
Typ publikacji:
Journal Article
MeSH Terms:
Carboxy-Lyases*/genetics
Carboxy-Lyases*/metabolism
Providencia*/enzymology
Escherichia coli/metabolism
SCR Organism:
Providencia stuartii
Czasopismo naukowe
Tytuł:
Erratum: Tetreau et al. How Does Bacillus thuringiensis Crystallize Such a Large Diversity of Toxins? Toxins 2021, 13 , 443.
Autorzy:
Tetreau G; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Andreeva EA; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Banneville AS; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
De Zitter E; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Colletier JP; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
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Źródło:
Toxins [Toxins (Basel)] 2021 Aug 27; Vol. 13 (9). Date of Electronic Publication: 2021 Aug 27.
Typ publikacji:
Published Erratum
Tytuł:
How Does Bacillus thuringiensis Crystallize Such a Large Diversity of Toxins?
Autorzy:
Tetreau G; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Andreeva EA; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Banneville AS; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
De Zitter E; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Colletier JP; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
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Źródło:
Toxins [Toxins (Basel)] 2021 Jun 26; Vol. 13 (7). Date of Electronic Publication: 2021 Jun 26.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Bacillus thuringiensis Toxins*/chemistry
Bacillus thuringiensis Toxins*/metabolism
Bacterial Proteins*/chemistry
Bacterial Proteins*/metabolism
Bacillus thuringiensis/*metabolism
Crystallization
Czasopismo naukowe
Tytuł:
Can (We Make) Bacillus thuringiensis Crystallize More Than Its Toxins?
Autorzy:
Tetreau G; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Andreeva EA; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Banneville AS; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
De Zitter E; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
Colletier JP; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, F-38000 Grenoble, France.
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Źródło:
Toxins [Toxins (Basel)] 2021 Jun 26; Vol. 13 (7). Date of Electronic Publication: 2021 Jun 26.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Bacillus thuringiensis*
Bacillus thuringiensis Toxins/*chemistry
Bacterial Proteins/*chemistry
Crystallization ; Pest Control, Biological
Czasopismo naukowe
Tytuł:
Mechanism and dynamics of fatty acid photodecarboxylase.
Autorzy:
Sorigué D; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Hadjidemetriou K; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Blangy S; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Gotthard G; European Synchrotron Radiation Facility, 38043 Grenoble, France.
Bonvalet A; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Coquelle N; Large-Scale Structures Group, Institut Laue Langevin, 38042 Grenoble Cedex 9, France.
Samire P; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.; Université Paris-Saclay, CEA, CNRS, Institute for Integrative Biology of the Cell (I2BC), 91198 Gif-sur-Yvette, France.
Aleksandrov A; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Antonucci L; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Benachir A; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Boutet S; Linac Coherent Light Source (LCLS), SLAC National Accelerator Laboratory, Menlo Park, CA 94025, USA.
Byrdin M; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Cammarata M; Department of Physics, UMR UR1-CNRS 6251, University of Rennes 1, F-Rennes, France. .
Carbajo S; Linac Coherent Light Source (LCLS), SLAC National Accelerator Laboratory, Menlo Park, CA 94025, USA.
Cuiné S; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Doak RB; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Foucar L; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Gorel A; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Grünbein M; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Hartmann E; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Hienerwadel R; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Hilpert M; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Kloos M; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany. .
Lane TJ; Linac Coherent Light Source (LCLS), SLAC National Accelerator Laboratory, Menlo Park, CA 94025, USA.
Légeret B; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Legrand P; Synchrotron SOLEIL. L'Orme des Merisiers Saint-Aubin, BP 48, 91192 Gif-sur-Yvette, France.
Li-Beisson Y; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Moulin SLY; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Nurizzo D; European Synchrotron Radiation Facility, 38043 Grenoble, France.
Peltier G; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France.
Schirò G; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Shoeman RL; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Sliwa M; Univ. Lille, CNRS, UMR 8516, LASIRE, LAboratoire de Spectroscopie pour les Interactions, la Réactivité et l'Environnement, 59000 Lille, France.
Solinas X; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Zhuang B; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.; Université Paris-Saclay, CEA, CNRS, Institute for Integrative Biology of the Cell (I2BC), 91198 Gif-sur-Yvette, France.
Barends TRM; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany.
Colletier JP; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.
Joffre M; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France.
Royant A; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France.; European Synchrotron Radiation Facility, 38043 Grenoble, France.
Berthomieu C; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France. .
Weik M; Université Grenoble Alpes, CEA, CNRS, Institut de Biologie Structurale, 38000 Grenoble, France. .
Domratcheva T; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany. .; Department of Chemistry, Lomonosov Moscow State University, Moscow 119991, Russia.
Brettel K; Université Paris-Saclay, CEA, CNRS, Institute for Integrative Biology of the Cell (I2BC), 91198 Gif-sur-Yvette, France.
Vos MH; LOB, CNRS, INSERM, Ecole Polytechnique, Institut Polytechnique de Paris, 91128 Palaiseau, France. .
Schlichting I; Max-Planck-Institut für medizinische Forschung, Jahnstrasse 29, 69120 Heidelberg, Germany. .
Arnoux P; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France. .
Müller P; Université Paris-Saclay, CEA, CNRS, Institute for Integrative Biology of the Cell (I2BC), 91198 Gif-sur-Yvette, France. .
Beisson F; Aix-Marseille University, CEA, CNRS, Institute of Biosciences and Biotechnologies, BIAM Cadarache, 13108 Saint-Paul-lez-Durance, France. .
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Źródło:
Science (New York, N.Y.) [Science] 2021 Apr 09; Vol. 372 (6538).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Carboxy-Lyases/*chemistry
Carboxy-Lyases/*metabolism
Chlorella/*enzymology
Fatty Acids/*metabolism
Algal Proteins/chemistry ; Algal Proteins/metabolism ; Alkanes/metabolism ; Amino Acid Substitution ; Amino Acids/metabolism ; Bicarbonates/metabolism ; Biocatalysis ; Carbon Dioxide/metabolism ; Catalytic Domain ; Crystallography, X-Ray ; Decarboxylation ; Electron Transport ; Flavin-Adenine Dinucleotide/chemistry ; Hydrogen Bonding ; Light ; Models, Molecular ; Mutant Proteins/chemistry ; Mutant Proteins/metabolism ; Oxidation-Reduction ; Photons ; Protein Conformation ; Temperature
Czasopismo naukowe
Tytuł:
Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probes.
Autorzy:
Pajk S; Faculty of Pharmacy, University of Ljubljana, Ljubljana, Slovenia.
Knez D; Faculty of Pharmacy, University of Ljubljana, Ljubljana, Slovenia.
Košak U; Faculty of Pharmacy, University of Ljubljana, Ljubljana, Slovenia.
Zorović M; Faculty of Medicine, Institute of Pathological Physiology, University of Ljubljana, Ljubljana, Slovenia.
Brazzolotto X; Département de Toxicologie et Risques Chimiques, Institut de Recherche Biomédicale des Armées, Brétigny sur Orge, France.
Coquelle N; Institut Laue Langvein, Grenoble, France.
Nachon F; Département de Toxicologie et Risques Chimiques, Institut de Recherche Biomédicale des Armées, Brétigny sur Orge, France.
Colletier JP; CNRS, CEA, IBS, Université Grenoble Alpes, Grenoble, France.
Živin M; Faculty of Medicine, Institute of Pathological Physiology, University of Ljubljana, Ljubljana, Slovenia.
Stojan J; Faculty of Medicine, Institute of Biochemistry, University of Ljubljana, Ljubljana, Slovenia.
Gobec S; Faculty of Pharmacy, University of Ljubljana, Ljubljana, Slovenia.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2020 Dec; Vol. 35 (1), pp. 498-505.
Typ publikacji:
Journal Article
MeSH Terms:
Amides/*pharmacology
Butyrylcholinesterase/*metabolism
Cholinesterase Inhibitors/*pharmacology
Fluorescent Dyes/*pharmacology
Amides/chemical synthesis ; Amides/chemistry ; Animals ; Butyrylcholinesterase/isolation & purification ; Cholinesterase Inhibitors/chemical synthesis ; Cholinesterase Inhibitors/chemistry ; Crystallography, X-Ray ; Fluorescent Dyes/chemical synthesis ; Fluorescent Dyes/chemistry ; Humans ; Mice ; Models, Molecular ; Molecular Structure
Czasopismo naukowe
Tytuł:
The C. elegans GATA transcription factor elt-2 mediates distinct transcriptional responses and opposite infection outcomes towards different Bacillus thuringiensis strains.
Autorzy:
Zárate-Potes A; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Yang W; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Pees B; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Schalkowski R; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Segler P; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Andresen B; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Haase D; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Nakad R; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Rosenstiel P; Institute for Clinical Molecular Biology (IKMB), Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
Tetreau G; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, Grenoble, France.
Colletier JP; Univ. Grenoble Alpes, CNRS, CEA, Institut de Biologie Structurale, Grenoble, France.
Schulenburg H; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.; Max Planck Institute for Evolutionary Biology, Ploen, Germany.
Dierking K; Department of Evolutionary Ecology and Genetics, Christian-Albrechts-Universität zu Kiel, Kiel, Germany.
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Źródło:
PLoS pathogens [PLoS Pathog] 2020 Sep 24; Vol. 16 (9), pp. e1008826. Date of Electronic Publication: 2020 Sep 24 (Print Publication: 2020).
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
MAP Kinase Signaling System*
Transcription, Genetic*
Bacillus thuringiensis/*metabolism
Bacterial Infections/*metabolism
Caenorhabditis elegans/*metabolism
Caenorhabditis elegans Proteins/*metabolism
GATA Transcription Factors/*metabolism
Animals ; Bacillus thuringiensis/pathogenicity ; Bacterial Infections/genetics ; Bacterial Infections/microbiology ; Caenorhabditis elegans/genetics ; Caenorhabditis elegans/microbiology ; Caenorhabditis elegans Proteins/genetics ; GATA Transcription Factors/genetics
Czasopismo naukowe
Tytuł:
Increasing Polarity in Tacrine and Huprine Derivatives: Potent Anticholinesterase Agents for the Treatment of Myasthenia Gravis.
Autorzy:
Galdeano C; Laboratory of Pharmaceutical Chemistry (CSIC Associated Unit), Faculty of Pharmacy and Food Sciences, and Institute of Biomedicine (IBUB), University of Barcelona, Av. Joan XXIII 27-31, E-08028 Barcelona, Spain. .
Coquelle N; Institut de Biologie Structurale, Université Grenoble Alpes, Centre National de la Recherche Scientifique (CNRS)-Commissariat à l'Énergie Atomique (CEA) (UMR 5075), F-38054 Grenoble, France. .; Large-Scale Structures Group, Institut Laue-Langevin, 71 Avenue des Martyrs, 38000 Grenoble, France. .
Cieslikiewicz-Bouet M; Laboratory COBRA (UMR 6014), Normandie Université, UNIROUEN, Institut National des Sciences Appliquées (INSA) Rouen, CNRS, 76000 Rouen, France. .
Bartolini M; Department of Pharmacy and Biotechnology, Alma Mater Studiorum University of Bologna, Via Belmeloro 6, I-40126 Bologna, Italy. .
Pérez B; Department of Pharmacology, Therapeutics and Toxicology, Neuroscience Institute, Autonomous University of Barcelona, E-08193 Barcelona, Spain. .
Clos MV; Department of Pharmacology, Therapeutics and Toxicology, Neuroscience Institute, Autonomous University of Barcelona, E-08193 Barcelona, Spain. .
Silman I; Department of Neurobiology, Weizmann Institute of Science, 76100 Rehovot, Israel. .
Jean L; Laboratory COBRA (UMR 6014), Normandie Université, UNIROUEN, Institut National des Sciences Appliquées (INSA) Rouen, CNRS, 76000 Rouen, France. .
Colletier JP; Institut de Biologie Structurale, Université Grenoble Alpes, Centre National de la Recherche Scientifique (CNRS)-Commissariat à l'Énergie Atomique (CEA) (UMR 5075), F-38054 Grenoble, France. colletier@ibs.fr.
Renard PY; Laboratory COBRA (UMR 6014), Normandie Université, UNIROUEN, Institut National des Sciences Appliquées (INSA) Rouen, CNRS, 76000 Rouen, France. .
Muñoz-Torrero D; Laboratory of Pharmaceutical Chemistry (CSIC Associated Unit), Faculty of Pharmacy and Food Sciences, and Institute of Biomedicine (IBUB), University of Barcelona, Av. Joan XXIII 27-31, E-08028 Barcelona, Spain. .
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2018 Mar 11; Vol. 23 (3). Date of Electronic Publication: 2018 Mar 11.
Typ publikacji:
Journal Article
MeSH Terms:
Acetylcholinesterase/*metabolism
Aminoacridines/*chemical synthesis
Aminoquinolines/*chemical synthesis
Cholinesterase Inhibitors/*chemical synthesis
Acetylcholinesterase/chemistry ; Aminoacridines/chemistry ; Aminoacridines/pharmacology ; Aminoquinolines/chemistry ; Aminoquinolines/pharmacology ; Butyrylcholinesterase/chemistry ; Butyrylcholinesterase/metabolism ; Cholinesterase Inhibitors/chemistry ; Cholinesterase Inhibitors/pharmacology ; Down-Regulation ; GPI-Linked Proteins/chemistry ; GPI-Linked Proteins/metabolism ; Heterocyclic Compounds, 4 or More Rings/chemistry ; Humans ; Models, Molecular ; Molecular Structure ; Myasthenia Gravis/drug therapy ; Myasthenia Gravis/enzymology ; Structure-Activity Relationship ; Tacrine/chemistry
Czasopismo naukowe
Tytuł:
Providencia stuartii form biofilms and floating communities of cells that display high resistance to environmental insults.
Autorzy:
El Khatib M; Institut de Biologie Structurale, Université Grenoble Alpes - Commissariat à l'Énergie Atomique - Centre National de la Recherche Scientifique, Grenoble, France.
Tran QT; School of Biophysics, Jacobs University of Bremen, Bremen, Germany.
Nasrallah C; Institut de Biologie Structurale, Université Grenoble Alpes - Commissariat à l'Énergie Atomique - Centre National de la Recherche Scientifique, Grenoble, France.
Lopes J; Institut de Biologie Structurale, Université Grenoble Alpes - Commissariat à l'Énergie Atomique - Centre National de la Recherche Scientifique, Grenoble, France.
Bolla JM; Équipe Transporteurs Membranaires, Chimiorésistance et Drug-Design, Université Aix-Marseille - Institut de Recherche Biomédicale des Armées, Marseille, France.
Vivaudou M; Institut de Biologie Structurale, Université Grenoble Alpes - Commissariat à l'Énergie Atomique - Centre National de la Recherche Scientifique, Grenoble, France.
Pagès JM; Équipe Transporteurs Membranaires, Chimiorésistance et Drug-Design, Université Aix-Marseille - Institut de Recherche Biomédicale des Armées, Marseille, France.
Colletier JP; Institut de Biologie Structurale, Université Grenoble Alpes - Commissariat à l'Énergie Atomique - Centre National de la Recherche Scientifique, Grenoble, France.
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Źródło:
PloS one [PLoS One] 2017 Mar 23; Vol. 12 (3), pp. e0174213. Date of Electronic Publication: 2017 Mar 23 (Print Publication: 2017).
Typ publikacji:
Journal Article
MeSH Terms:
Biofilms/*growth & development
Providencia/*physiology
Biofilms/drug effects ; Calcium/pharmacology ; Environment ; Gene Knockdown Techniques ; Hydrogen-Ion Concentration ; Magnesium/pharmacology ; Providencia/drug effects ; Providencia/growth & development ; Urea/pharmacology
Czasopismo naukowe
Tytuł:
The cytotoxic Staphylococcus aureus PSMα3 reveals a cross-α amyloid-like fibril.
Autorzy:
Tayeb-Fligelman E; Department of Biology, Technion-Israel Institute of Technology, Haifa 3200003, Israel.
Tabachnikov O; Department of Biology, Technion-Israel Institute of Technology, Haifa 3200003, Israel.
Moshe A; Department of Biology, Technion-Israel Institute of Technology, Haifa 3200003, Israel.
Goldshmidt-Tran O; Department of Biology, Technion-Israel Institute of Technology, Haifa 3200003, Israel.
Sawaya MR; Department of Biological Chemistry, Department of Chemistry and Biochemistry, and Howard Hughes Medical Institute, University of California at Los Angeles, Los Angeles, CA 90095, USA.
Coquelle N; Institut de Biologie Structurale (IBS), Université Grenoble Alpes-CEA-CNRS UMR 5075, Grenoble 38044, France.
Colletier JP; Institut de Biologie Structurale (IBS), Université Grenoble Alpes-CEA-CNRS UMR 5075, Grenoble 38044, France.
Landau M; Department of Biology, Technion-Israel Institute of Technology, Haifa 3200003, Israel. .
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Źródło:
Science (New York, N.Y.) [Science] 2017 Feb 24; Vol. 355 (6327), pp. 831-833.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Amyloid/*chemistry
Amyloid/*metabolism
Bacterial Toxins/*chemistry
Bacterial Toxins/*metabolism
Staphylococcus aureus/*metabolism
Staphylococcus aureus/*pathogenicity
Cells, Cultured ; Crystallography, X-Ray ; Humans ; Protein Conformation ; T-Lymphocytes/microbiology
Czasopismo naukowe
Tytuł:
Development of an in-vivo active reversible butyrylcholinesterase inhibitor.
Autorzy:
Košak U; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Brus B; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Knez D; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Šink R; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Žakelj S; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Trontelj J; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Pišlar A; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Šlenc J; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Gobec M; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Živin M; Institute of Pathological Physiology, Faculty of Medicine, University of Ljubljana, Vrazov trg 2, 1000 Ljubljana, Slovenia.
Tratnjek L; Institute of Pathological Physiology, Faculty of Medicine, University of Ljubljana, Vrazov trg 2, 1000 Ljubljana, Slovenia.
Perše M; Institute of Pathology, Faculty of Medicine, University of Ljubljana, Korytkova 2, 1000 Ljubljana, Slovenia.
Sałat K; Faculty of Pharmacy, Jagiellonian University, Medyczna 9 St., 30-688 Krakow, Poland.
Podkowa A; Faculty of Pharmacy, Jagiellonian University, Medyczna 9 St., 30-688 Krakow, Poland.
Filipek B; Faculty of Pharmacy, Jagiellonian University, Medyczna 9 St., 30-688 Krakow, Poland.
Nachon F; Institut de Recherche Biomédicale des Armées, 91223 Brétigny sur Orge, France.
Brazzolotto X; Institut de Recherche Biomédicale des Armées, 91223 Brétigny sur Orge, France.
Więckowska A; Faculty of Pharmacy, Jagiellonian University, Medyczna 9 St., 30-688 Krakow, Poland.
Malawska B; Faculty of Pharmacy, Jagiellonian University, Medyczna 9 St., 30-688 Krakow, Poland.
Stojan J; Institute of Biochemistry, Faculty of Medicine, University of Ljubljana, Vrazov trg 2, 1000 Ljubljana, Slovenia.
Raščan IM; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Kos J; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
Coquelle N; University Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Colletier JP; University Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Gobec S; Faculty of Pharmacy, University of Ljubljana, Aškerčeva 7, 1000 Ljubljana, Slovenia.
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Źródło:
Scientific reports [Sci Rep] 2016 Dec 21; Vol. 6, pp. 39495. Date of Electronic Publication: 2016 Dec 21.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Design*
Alzheimer Disease/*drug therapy
Cholinesterase Inhibitors/*pharmacology
Animals ; Blood-Brain Barrier ; Brain/pathology ; Butyrylcholinesterase ; Catalytic Domain ; Chromatography, High Pressure Liquid ; Disease Progression ; Drug Evaluation, Preclinical ; Female ; Humans ; Learning ; Male ; Mice ; Mice, Inbred C57BL ; Mice, Knockout ; Protein Conformation ; Rats ; Rats, Wistar
Czasopismo naukowe
Tytuł:
Rational design of ultrastable and reversibly photoswitchable fluorescent proteins for super-resolution imaging of the bacterial periplasm.
Autorzy:
El Khatib M; Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Martins A; Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Bourgeois D; Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Colletier JP; Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
Adam V; Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France.; CNRS, IBS, F-38044 Grenoble, France.; CEA, IBS, F-38044 Grenoble, France.
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Źródło:
Scientific reports [Sci Rep] 2016 Jan 06; Vol. 6, pp. 18459. Date of Electronic Publication: 2016 Jan 06.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Models, Molecular*
Luminescent Proteins/*chemistry
Luminescent Proteins/*metabolism
Periplasm/*metabolism
Escherichia coli/genetics ; Escherichia coli/metabolism ; Gene Expression ; Hydrogen Bonding ; Luminescent Proteins/genetics ; Microscopy, Fluorescence ; Molecular Imaging ; Mutation ; Protein Conformation ; Quantitative Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Varied Probability of Staying Collapsed/Extended at the Conformational Equilibrium of Monomeric Aβ40 and Aβ42.
Autorzy:
Song W; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Center, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai 201203, China.
Wang Y; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Center, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai 201203, China.
Colletier JP; 1] Univ. Grenoble Alpes, IBS, F-38044 Grenoble, France [2] CNRS, IBS, F-38044 Grenoble, France [3] CEA, IBS, F-38044 Grenoble, France.
Yang H; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Center, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai 201203, China.
Xu Y; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Center, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai 201203, China.
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Źródło:
Scientific reports [Sci Rep] 2015 Jun 05; Vol. 5, pp. 11024. Date of Electronic Publication: 2015 Jun 05.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Amyloid beta-Peptides/*chemistry
Peptide Fragments/*chemistry
Amyloid beta-Peptides/metabolism ; Cluster Analysis ; Hydrophobic and Hydrophilic Interactions ; Magnetic Resonance Spectroscopy ; Molecular Dynamics Simulation ; Peptide Fragments/metabolism ; Protein Structure, Secondary ; Protein Structure, Tertiary
Czasopismo naukowe
Tytuł:
Understanding Voltage Gating of Providencia stuartii Porins at Atomic Level.
Autorzy:
Song W; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Centre, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai, China.
Bajaj H; School of Engineering and Sciences, Jacobs University Bremen, Bremen, Germany.
Nasrallah C; University Grenoble Alpes, Institut de Biologie Structurale (IBS), Grenoble, France; CNRS, Institut de Biologie Structurale (IBS), Grenoble, France; CEA, Institut de Biologie Structurale (IBS), Grenoble, France.
Jiang H; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Centre, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai, China.
Winterhalter M; School of Engineering and Sciences, Jacobs University Bremen, Bremen, Germany.
Colletier JP; University Grenoble Alpes, Institut de Biologie Structurale (IBS), Grenoble, France; CNRS, Institut de Biologie Structurale (IBS), Grenoble, France; CEA, Institut de Biologie Structurale (IBS), Grenoble, France.
Xu Y; CAS Key Laboratory of Receptor Research, Drug Discovery and Design Centre, Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CAS), Shanghai, China.
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Źródło:
PLoS computational biology [PLoS Comput Biol] 2015 May 08; Vol. 11 (5), pp. e1004255. Date of Electronic Publication: 2015 May 08 (Print Publication: 2015).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Bacterial Proteins/*chemistry
Bacterial Proteins/*metabolism
Porins/*chemistry
Porins/*metabolism
Providencia/*metabolism
Bacterial Outer Membrane Proteins/chemistry ; Bacterial Outer Membrane Proteins/metabolism ; Binding Sites ; Computational Biology ; Computer Simulation ; Hydrogen Bonding ; Ion Channel Gating ; Models, Biological ; Models, Molecular ; Molecular Dynamics Simulation ; Static Electricity
Czasopismo naukowe
Tytuł:
Structure-guided simulations illuminate the mechanism of ATP transport through VDAC1.
Autorzy:
Choudhary OP; 1] Joint Carnegie Mellon University-University of Pittsburgh PhD Program in Computational Biology, Pittsburgh, Pennsylvania, USA. [2].
Paz A; 1] Department of Physiology, David Geffen School of Medicine, University of California, Los Angeles, Los Angeles, California, USA. [2].
Adelman JL; 1] Department of Biological Sciences, University of Pittsburgh, Pittsburgh, Pennsylvania, USA. [2].
Colletier JP; 1] Université Grenoble Alpes, Institut de Biologie Structurale, Grenoble, France. [2] Centre National de la Recherche Scientifique, Institut de Biologie Structurale, Grenoble, France. [3] Commissariat à l'Énergie Atomique et aux Énergies Alternatives, Direction des Sciences du Vivant, Institut de Biologie Structurale, Grenoble, France. [4].
Abramson J; 1] Department of Physiology, David Geffen School of Medicine, University of California, Los Angeles, Los Angeles, California, USA. [2] Institute for Stem Cell Biology and Regenerative Medicine, National Centre for Biological Sciences-Tata Institute of Fundamental Research, Bangalore, India.
Grabe M; 1] Department of Biological Sciences, University of Pittsburgh, Pittsburgh, Pennsylvania, USA. [2] Cardiovascular Research Institute, Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California, USA.
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Źródło:
Nature structural & molecular biology [Nat Struct Mol Biol] 2014 Jul; Vol. 21 (7), pp. 626-32. Date of Electronic Publication: 2014 Jun 08.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
MeSH Terms:
Adenosine Triphosphate/*metabolism
Voltage-Dependent Anion Channel 1/*chemistry
Adenosine Triphosphate/chemistry ; Animals ; Binding Sites ; Computer Simulation ; Crystallography, X-Ray ; Markov Chains ; Mice ; Mitochondrial Membranes/metabolism ; Models, Molecular ; Protein Structure, Tertiary ; Voltage-Dependent Anion Channel 1/metabolism ; Voltage-Dependent Anion Channel 1/physiology
Czasopismo naukowe

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