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Wyświetlanie 1-8 z 8
Tytuł:
A rationally designed monomeric peptide triagonist corrects obesity and diabetes in rodents.
Autorzy:
Finan B; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany. [3] Department of Chemistry, Indiana University, Bloomington, Indiana, USA.
Yang B; 1] Department of Chemistry, Indiana University, Bloomington, Indiana, USA. [2] Marcadia Biotech, Carmel, Indiana, USA.
Ottaway N; Metabolic Diseases Institute, Division of Endocrinology, Department of Internal Medicine, University of Cincinnati College of Medicine, Cincinnati, Ohio, USA.
Smiley DL; Department of Chemistry, Indiana University, Bloomington, Indiana, USA.
Ma T; 1] Department of Chemistry, Indiana University, Bloomington, Indiana, USA. [2] Research Center, Beijing Hanmi Pharm., Beijing, China.
Clemmensen C; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany.
Chabenne J; 1] Department of Chemistry, Indiana University, Bloomington, Indiana, USA. [2] AIT Laboratories, Indianapolis, Indiana, USA.
Zhang L; Marcadia Biotech, Carmel, Indiana, USA.
Habegger KM; Comprehensive Diabetes Center, Department of Medicine, Division of Endocrinology, Diabetes and Metabolism, University of Alabama at Birmingham, Birmingham, Alabama, USA.
Fischer K; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany.
Campbell JE; Department of Medicine, Lunenfeld Tanenbaum Research Institute, Mt. Sinai Hospital, University of Toronto, Toronto, Ontario, Canada.
Sandoval D; Metabolic Diseases Institute, Division of Endocrinology, Department of Internal Medicine, University of Cincinnati College of Medicine, Cincinnati, Ohio, USA.
Seeley RJ; Metabolic Diseases Institute, Division of Endocrinology, Department of Internal Medicine, University of Cincinnati College of Medicine, Cincinnati, Ohio, USA.
Bleicher K; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Uhles S; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Riboulet W; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Funk J; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Hertel C; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Belli S; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Sebokova E; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Conde-Knape K; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Konkar A; Pharmaceutical Research and Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Basel, Switzerland.
Drucker DJ; Department of Medicine, Lunenfeld Tanenbaum Research Institute, Mt. Sinai Hospital, University of Toronto, Toronto, Ontario, Canada.
Gelfanov V; Department of Chemistry, Indiana University, Bloomington, Indiana, USA.
Pfluger PT; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany.
Müller TD; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany.
Perez-Tilve D; Metabolic Diseases Institute, Division of Endocrinology, Department of Internal Medicine, University of Cincinnati College of Medicine, Cincinnati, Ohio, USA.
DiMarchi RD; Department of Chemistry, Indiana University, Bloomington, Indiana, USA.
Tschöp MH; 1] Institute for Diabetes and Obesity, Helmholtz Zentrum München, German Research Center for Environmental Health, Neuherberg, Germany. [2] Department of Medicine, Division of Metabolic Diseases,Technische Universität München, Munich, Germany.
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Źródło:
Nature medicine [Nat Med] 2015 Jan; Vol. 21 (1), pp. 27-36. Date of Electronic Publication: 2014 Dec 08.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Diabetes Complications/*metabolism
Diabetes Mellitus, Type 2/*metabolism
Obesity/*metabolism
Peptides/*administration & dosage
Animals ; Blood Glucose/drug effects ; Body Weight/genetics ; Diabetes Complications/drug therapy ; Diabetes Complications/genetics ; Diabetes Mellitus, Type 2/drug therapy ; Diabetes Mellitus, Type 2/genetics ; Glucagon-Like Peptide 1/agonists ; Glucagon-Like Peptide 1/metabolism ; HEK293 Cells ; Humans ; Insulin/biosynthesis ; Insulin/metabolism ; Mice ; Obesity/drug therapy ; Obesity/genetics ; Peptides/chemical synthesis ; Peptides/metabolism ; Rats ; Receptors, Gastrointestinal Hormone/agonists ; Receptors, Gastrointestinal Hormone/metabolism ; Receptors, Glucagon/agonists ; Receptors, Glucagon/metabolism ; Rodentia
Czasopismo naukowe
Tytuł:
Metabolic disease puts up a fight: are diet and exercise helpful for the heart?
Autorzy:
Lovshin JA; Department of Medicine, Lunenfeld Tanenbaum Research Institute, Mt. Sinai Hospital, University of Toronto, Toronto, Ontario, Canada.
Drucker DJ
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Źródło:
Nature medicine [Nat Med] 2013 Oct; Vol. 19 (10), pp. 1216-7.
Typ publikacji:
Journal Article
MeSH Terms:
Diet*
Exercise*
Diabetes Mellitus, Type 2/*physiopathology
Heart/*physiopathology
Diabetes Mellitus, Type 2/diet therapy ; Diabetes Mellitus, Type 2/drug therapy ; Humans ; Hypoglycemic Agents/therapeutic use ; Weight Loss
Czasopismo naukowe
Tytuł:
Liraglutide.
Autorzy:
Drucker DJ; Samuel Lunenfeld Research Institute, Mount Sinai Hospital, 600 University Avenue, Toronto, Ontario, Canada. d.drucker@utoronto.ca
Dritselis A
Kirkpatrick P
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Źródło:
Nature reviews. Drug discovery [Nat Rev Drug Discov] 2010 Apr; Vol. 9 (4), pp. 267-8.
Typ publikacji:
Journal Article
MeSH Terms:
Diabetes Mellitus, Type 2/*drug therapy
Glucagon-Like Peptide 1/*analogs & derivatives
Hypoglycemic Agents/*therapeutic use
Adult ; Drug Approval ; Glucagon-Like Peptide 1/pharmacology ; Glucagon-Like Peptide 1/therapeutic use ; Humans ; Hypoglycemic Agents/pharmacology ; Liraglutide ; Randomized Controlled Trials as Topic ; United States ; United States Food and Drug Administration
Czasopismo naukowe
Tytuł:
Normalization of obesity-associated insulin resistance through immunotherapy.
Autorzy:
Winer S; Department of Pediatrics & Immunology, Research Institute, The Hospital for Sick Children, University of Toronto, Toronto, Ontario, Canada.
Chan Y
Paltser G
Truong D
Tsui H
Bahrami J
Dorfman R
Wang Y
Zielenski J
Mastronardi F
Maezawa Y
Drucker DJ
Engleman E
Winer D
Dosch HM
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Źródło:
Nature medicine [Nat Med] 2009 Aug; Vol. 15 (8), pp. 921-9. Date of Electronic Publication: 2009 Jul 26.
Typ publikacji:
Evaluation Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Insulin Resistance/*immunology
Obesity/*complications
Obesity/*therapy
Adipose Tissue/immunology ; Adipose Tissue/metabolism ; Adipose Tissue/pathology ; Animals ; CD4-Positive T-Lymphocytes/immunology ; CD4-Positive T-Lymphocytes/pathology ; CD4-Positive T-Lymphocytes/physiology ; Cell Separation ; Glucose/metabolism ; Homeodomain Proteins/genetics ; Homeostasis/immunology ; Immunotherapy/methods ; Mice ; Mice, Inbred C57BL ; Mice, Knockout ; Mice, Obese ; Obesity/immunology ; Obesity/pathology
Czasopismo naukowe
Tytuł:
The incretin system: glucagon-like peptide-1 receptor agonists and dipeptidyl peptidase-4 inhibitors in type 2 diabetes.
Autorzy:
Drucker DJ; Samuel Lunenfeld Research Institute, Mount Sinai Hospital, University of Toronto, Toronto, Ontario, Canada. d.drucker@utoronto.ca
Nauck MA
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Źródło:
Lancet (London, England) [Lancet] 2006 Nov 11; Vol. 368 (9548), pp. 1696-705.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't; Review
MeSH Terms:
Adenosine Deaminase Inhibitors*
Dipeptidyl-Peptidase IV Inhibitors*
Hypoglycemic Agents*/administration & dosage
Hypoglycemic Agents*/adverse effects
Hypoglycemic Agents*/therapeutic use
Adamantane/*analogs & derivatives
Diabetes Mellitus, Type 2/*drug therapy
Glucagon-Like Peptide 1/*analogs & derivatives
Glucagon-Like Peptide 1/*physiology
Glycoproteins/*antagonists & inhibitors
Peptides/*therapeutic use
Pyrazines/*therapeutic use
Receptors, Glucagon/*agonists
Triazoles/*therapeutic use
Venoms/*therapeutic use
Adamantane/administration & dosage ; Adamantane/adverse effects ; Adamantane/therapeutic use ; Clinical Trials as Topic ; Dipeptidyl Peptidase 4 ; Drug Administration Schedule ; Exenatide ; Glucagon-Like Peptide 1/administration & dosage ; Glucagon-Like Peptide 1/adverse effects ; Glucagon-Like Peptide 1/biosynthesis ; Glucagon-Like Peptide 1/classification ; Glucagon-Like Peptide 1/therapeutic use ; Glucagon-Like Peptide-1 Receptor ; Humans ; Liraglutide ; Nitriles ; Peptides/administration & dosage ; Peptides/adverse effects ; Pyrazines/administration & dosage ; Pyrazines/adverse effects ; Pyrrolidines ; Sitagliptin Phosphate ; Triazoles/administration & dosage ; Triazoles/adverse effects ; Venoms/administration & dosage ; Venoms/adverse effects ; Vildagliptin
Czasopismo naukowe
    Wyświetlanie 1-8 z 8

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