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Wyszukujesz frazę ""Drug Evaluation, Preclinical"" wg kryterium: Temat


Tytuł:
ACFIS 2.0: an improved web-server for fragment-based drug discovery via a dynamic screening strategy.
Autorzy:
Shi XX; National Key Laboratory of Green Pesticide, Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, Central China Normal University, Wuhan430079, P.R. China.
Wang ZZ; National Key Laboratory of Green Pesticide, Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, Central China Normal University, Wuhan430079, P.R. China.
Wang F; National Key Laboratory of Green Pesticide, Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, Central China Normal University, Wuhan430079, P.R. China.
Hao GF; National Key Laboratory of Green Pesticide, Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, Central China Normal University, Wuhan430079, P.R. China.
Yang GF; National Key Laboratory of Green Pesticide, Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, Central China Normal University, Wuhan430079, P.R. China.
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Źródło:
Nucleic acids research [Nucleic Acids Res] 2023 Jul 05; Vol. 51 (W1), pp. W25-W32.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Discovery*/instrumentation
Drug Discovery*/methods
Data Visualization*
Computer Simulation*
Drug Evaluation, Preclinical*/instrumentation
Drug Evaluation, Preclinical*/methods
Humans ; Depressive Disorder, Major/drug therapy ; Proteins/chemistry ; Neoplasms/drug therapy ; Parkinson Disease/drug therapy ; Internet
Czasopismo naukowe
Tytuł:
Combined Experimental and Computational Study of V-Substituted Lindqvist Polyoxotungstate: Screening by Docking for Potential Antidiabetic Activity.
Autorzy:
Maalaoui A; Laboratory of Materials Chemistry, Faculty of Sciences of Bizerte, 7021 Zarzouna, Bizerte, Tunisia.
Agwamba EC; Department of Chemistry, Covenant University, Idiroko Road, P.M.B, Ota 1023, Ogun State, Nigeria.; Computational and Bio-Simulation Research Group, University of Calabar, P.M.B. 1115, Calabar 540221, Nigeria.
Louis H; Computational and Bio-Simulation Research Group, University of Calabar, P.M.B. 1115, Calabar 540221, Nigeria.; Department of Pure and Applied Chemistry, University of Calabar, P.M.B. 1115, Calabar 540221, Nigeria.
Mathias GE; Computational and Bio-Simulation Research Group, University of Calabar, P.M.B. 1115, Calabar 540221, Nigeria.; Department of Pure and Applied Chemistry, University of Calabar, P.M.B. 1115, Calabar 540221, Nigeria.
Rzaigui M; Laboratory of Materials Chemistry, Faculty of Sciences of Bizerte, 7021 Zarzouna, Bizerte, Tunisia.
Akriche S; Laboratory of Materials Chemistry, Faculty of Sciences of Bizerte, 7021 Zarzouna, Bizerte, Tunisia.
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Źródło:
Inorganic chemistry [Inorg Chem] 2023 Sep 04; Vol. 62 (35), pp. 14279-14290. Date of Electronic Publication: 2023 Aug 24.
Typ publikacji:
Journal Article
MeSH Terms:
Hypoglycemic Agents*/chemistry
Drug Evaluation, Preclinical*/methods
Computer Simulation ; Tungsten Compounds/chemistry ; Polymers/chemistry ; Models, Molecular ; Protein Structure, Tertiary
Czasopismo naukowe
Tytuł:
Breeze 2.0: an interactive web-tool for visual analysis and comparison of drug response data.
Autorzy:
Potdar S; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.
Ianevski F; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.
Ianevski A; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.
Tanoli Z; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.
Wennerberg K; Biotech Research & Innovation Centre (BRIC), University of Copenhagen, Copenhagen, Denmark.
Seashore-Ludlow B; Department of Medical Biochemistry and Biophysics, Chemical Biology Consortium Sweden (CBCS), Science for Life Laboratory, Karolinska Institutet, Stockholm, Sweden.; Department of Oncology-Pathology, Science for Life Laboratory, Karolinska Institutet, Stockholm, Sweden.
Kallioniemi O; Department of Oncology-Pathology, Science for Life Laboratory, Karolinska Institutet, Stockholm, Sweden.
Östling P; Department of Oncology-Pathology, Science for Life Laboratory, Karolinska Institutet, Stockholm, Sweden.
Aittokallio T; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.; Department of Cancer Genetics, Institute for Cancer Research, Oslo University Hospital, Norway.; Centre for Biostatistics and Epidemiology (OCBE), Faculty of Medicine, University of Oslo, Norway.
Saarela J; Institute for Molecular Medicine Finland (FIMM), HiLIFE, University of Helsinki, Finland.
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Źródło:
Nucleic acids research [Nucleic Acids Res] 2023 Jul 05; Vol. 51 (W1), pp. W57-W61.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Evaluation, Preclinical*
Software*
Computer Graphics ; Reproducibility of Results ; User-Computer Interface ; Internet
Czasopismo naukowe
Tytuł:
Computational approaches streamlining drug discovery.
Autorzy:
Sadybekov AV; Department of Quantitative and Computational Biology, University of Southern California, Los Angeles, CA, USA.; Center for New Technologies in Drug Discovery and Development, Bridge Institute, Michelson Center for Convergent Biosciences, University of Southern California, Los Angeles, CA, USA.
Katritch V; Department of Quantitative and Computational Biology, University of Southern California, Los Angeles, CA, USA. .; Center for New Technologies in Drug Discovery and Development, Bridge Institute, Michelson Center for Convergent Biosciences, University of Southern California, Los Angeles, CA, USA. .; Department of Chemistry, University of Southern California, Los Angeles, CA, USA. .
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Źródło:
Nature [Nature] 2023 Apr; Vol. 616 (7958), pp. 673-685. Date of Electronic Publication: 2023 Apr 26.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Drug Discovery*/instrumentation
Drug Discovery*/methods
Computer Simulation*
Drug Evaluation, Preclinical*/instrumentation
Drug Evaluation, Preclinical*/methods
Ligands ; Humans
Czasopismo naukowe
Tytuł:
Ex-vivo drug screening of surgically resected glioma stem cells to replace murine avatars and provide personalise cancer therapy for glioblastoma patients.
Autorzy:
Gagg H; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
Williams ST; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Neurosurgery, Royal Hallamshire Hospital, Sheffield, S10 2JF, UK.
Conroy S; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Urology, Royal Hallamshire Hospital, Sheffield, S10 2JF, UK.
Myers KN; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
McGarrity-Cottrell C; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
Jones C; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
Helleday T; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Karolinska Institut, Solnavägen, Solna, 171 77, Sweden.
Rantala J; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Misvik Biology Ltd, Karjakatu, Turku, FI-20520, Finland.
Rominiyi O; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Neurosurgery, Royal Hallamshire Hospital, Sheffield, S10 2JF, UK.
Danson SJ; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.; Weston Park Hospital, Sheffield, S10 2SJ, UK.
Collis SJ; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
Wells G; Oncology & Metabolism, The University of Sheffield, Sheffield, England, S10 2RX, UK.
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Źródło:
F1000Research [F1000Res] 2024 Mar 11; Vol. 12, pp. 954. Date of Electronic Publication: 2024 Mar 11 (Print Publication: 2023).
Typ publikacji:
Journal Article
MeSH Terms:
Glioblastoma*/drug therapy
Brain Neoplasms*/drug therapy
Glioma*
Humans ; Animals ; Mice ; Drug Evaluation, Preclinical ; Avatar ; Early Detection of Cancer ; Neoplastic Stem Cells
Czasopismo naukowe
Tytuł:
Construction of luciferase-expressing Neospora caninum and drug screening.
Autorzy:
Wang F; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Xue Y; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Pei Y; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Yin M; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Sun Z; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Zhou Z; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Liu J; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.; Key Laboratory of Animal Epidemiology of the Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China.
Liu Q; National Animal Protozoa Laboratory, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China. .; Key Laboratory of Animal Epidemiology of the Ministry of Agriculture, College of Veterinary Medicine, China Agricultural University, Beijing, 100193, China. .
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Źródło:
Parasites & vectors [Parasit Vectors] 2024 Mar 08; Vol. 17 (1), pp. 118. Date of Electronic Publication: 2024 Mar 08.
Typ publikacji:
Journal Article
MeSH Terms:
Coccidiosis*/drug therapy
Coccidiosis*/veterinary
Coccidiosis*/parasitology
Neospora*/genetics
Cattle Diseases*
Dog Diseases*
Rodent Diseases*
Nitriles*
Pregnancy ; Female ; Animals ; Mice ; Cattle ; Dogs ; Drug Evaluation, Preclinical ; Benzothiazoles/metabolism ; Benzothiazoles/pharmacology ; Benzothiazoles/therapeutic use
Czasopismo naukowe
Tytuł:
A Zebrafish-Based Platform for High-Throughput Epilepsy Modeling and Drug Screening in F0.
Autorzy:
Locubiche S; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.; Faculty of Medicine and Health Sciences, Institute of Neurosciences, University of Barcelona, 08036 Barcelona, Spain.
Ordóñez V; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.
Abad E; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.
Scotto di Mase M; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.
Di Donato V; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.
De Santis F; ZeClinics S.L., Carrer de Laureà Miró, 408-410, 08980 Sant Feliu de Llobregat, Spain.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2024 Mar 04; Vol. 25 (5). Date of Electronic Publication: 2024 Mar 04.
Typ publikacji:
Journal Article
MeSH Terms:
Zebrafish*/genetics
Epilepsy*/genetics
Animals ; Humans ; Drug Evaluation, Preclinical ; Mutation ; CRISPR-Cas Systems
Czasopismo naukowe
Tytuł:
In vitro drug screening models derived from different PC12 cell lines for exploring Parkinson's disease based on electrochemical signals of catecholamine neurotransmitters.
Autorzy:
Zhong Y; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Liu MM; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Li JC; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Lu TC; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Cao X; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Yang YJ; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China.
Lei Y; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China. .
Liu AL; Department of Pharmaceutical Analysis, School of Pharmacy, Fujian Medical University, Fuzhou, 350122, China. .
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Źródło:
Mikrochimica acta [Mikrochim Acta] 2024 Mar 01; Vol. 191 (3), pp. 170. Date of Electronic Publication: 2024 Mar 01.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Parkinson Disease*
Adrenal Gland Neoplasms*
Fluorocarbon Polymers*
Rats ; Animals ; Catecholamines/metabolism ; PC12 Cells ; Nerve Growth Factor ; Drug Evaluation, Preclinical ; Neurotransmitter Agents
Czasopismo naukowe
Tytuł:
Innovative explorations: unveiling the potential of organoids for investigating environmental pollutant exposure.
Autorzy:
Zhang Y; School of Environment, Nanjing Normal University, Nanjing, 210023, China.
Liu K; School of Environment, Nanjing Normal University, Nanjing, 210023, China.
He H; School of Environment, Nanjing Normal University, Nanjing, 210023, China.; Jiangsu Province Engineering Research Center of Environmental Risk Prevention and Emergency Response Technology, Nanjing, 210023, China.
Xiao H; School of Environment, Nanjing Normal University, Nanjing, 210023, China.
Fang Z; School of Environment, Nanjing Normal University, Nanjing, 210023, China.
Chen X; School of Environment, Nanjing Normal University, Nanjing, 210023, China.
Li H; School of Environment, Nanjing Normal University, Nanjing, 210023, China. .; Jiangsu Province Engineering Research Center of Environmental Risk Prevention and Emergency Response Technology, Nanjing, 210023, China. .
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Źródło:
Environmental science and pollution research international [Environ Sci Pollut Res Int] 2024 Mar; Vol. 31 (11), pp. 16256-16273. Date of Electronic Publication: 2024 Feb 12.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Environmental Pollutants*/metabolism
Liver Neoplasms*
Animals ; Humans ; Organoids/metabolism ; Cell Culture Techniques ; Drug Evaluation, Preclinical ; Mammals
Czasopismo naukowe
Tytuł:
Repurposing sodium stibogluconate as an uracil DNA glycosylase inhibitor against prostate cancer using a time-resolved oligonucleotide-based drug screening platform.
Autorzy:
Nao SC; State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China.
Huang LS; State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China.
Shiu-Hin Chan D; Department of Chemistry, City University of Hong Kong, Hong Kong, China.
Wang X; Institute of Medical Research, Northwestern Polytechnical University, Xi'an, Shaanxi 710072, China; Research & Development Institute of Northwestern Polytechnical University in Shenzhen, 45 South Gaoxin Road, Shenzhen 518057, China.
Li GD; State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China.
Wu J; State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China.
Wong CY; Department of Chemistry, City University of Hong Kong, Hong Kong, China. Electronic address: .
Wang W; Institute of Medical Research, Northwestern Polytechnical University, Xi'an, Shaanxi 710072, China; Research & Development Institute of Northwestern Polytechnical University in Shenzhen, 45 South Gaoxin Road, Shenzhen 518057, China. Electronic address: .
Leung CH; State Key Laboratory of Quality Research in Chinese Medicine, Institute of Chinese Medical Sciences, University of Macau, Taipa, Macau 999078, China; Department of Biomedical Sciences, Faculty of Health Sciences, University of Macau, Taipa, Macau, China; Macao Centre for Research and Development in Chinese Medicine, University of Macau, Taipa, Macau, China; MoE Frontiers Science Centre for Precision Oncology, University of Macau, Taipa, Macau, China. Electronic address: .
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Źródło:
Bioorganic chemistry [Bioorg Chem] 2024 Mar; Vol. 144, pp. 107176. Date of Electronic Publication: 2024 Feb 04.
Typ publikacji:
Journal Article
MeSH Terms:
Uracil-DNA Glycosidase*/chemistry
Prostatic Neoplasms*
Humans ; Male ; Oligonucleotides ; Antimony Sodium Gluconate ; Drug Evaluation, Preclinical ; Drug Repositioning ; Early Detection of Cancer
Czasopismo naukowe
Tytuł:
Nanoplasmonic biosensors for multicolor visual analysis of acetylcholinesterase activity and drug inhibitor screening in point-of-care testing.
Autorzy:
Li Y; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Chen L; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Li CY; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Zhang J; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Zhao Y; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Yang YH; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China.
Yang T; College of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, 650500, Yunnan Province, PR China. Electronic address: .
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Źródło:
Biosensors & bioelectronics [Biosens Bioelectron] 2024 Mar 01; Vol. 247, pp. 115912. Date of Electronic Publication: 2023 Dec 08.
Typ publikacji:
Journal Article
MeSH Terms:
Biosensing Techniques*/methods
Metal Nanoparticles*
Acetylcholinesterase ; Hydrogen Peroxide ; Drug Evaluation, Preclinical/methods ; Cholinesterase Inhibitors/pharmacology ; Cholinesterase Inhibitors/analysis ; Point-of-Care Testing
Czasopismo naukowe
Tytuł:
Heart-on-a-chip systems: disease modeling and drug screening applications.
Autorzy:
Butler D; Microsystems and Nanotechnology Division, National Institute of Standards and Technology, Gaithersburg, MD 20899, USA. .
Reyes DR; Microsystems and Nanotechnology Division, National Institute of Standards and Technology, Gaithersburg, MD 20899, USA. .
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Źródło:
Lab on a chip [Lab Chip] 2024 Feb 27; Vol. 24 (5), pp. 1494-1528. Date of Electronic Publication: 2024 Feb 27.
Typ publikacji:
Journal Article; Review; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug-Related Side Effects and Adverse Reactions*
Cardiovascular Diseases*/drug therapy
Animals ; Humans ; Drug Evaluation, Preclinical ; Microfluidics ; Tissue Engineering ; Lab-On-A-Chip Devices
Czasopismo naukowe
Tytuł:
High-throughput microfluidic systems accelerated by artificial intelligence for biomedical applications.
Autorzy:
Zhou J; School of Biomedical Engineering, Shenzhen Campus of Sun Yat-sen University, Shenzhen 518107, China. .; Key Laboratory of Sensing Technology and Biomedical Instruments of Guangdong Province, School of Biomedical Engineering, Sun Yat-sen University, Shenzhen 518107, China.
Dong J; School of Biomedical Engineering, Shenzhen Campus of Sun Yat-sen University, Shenzhen 518107, China. .; Key Laboratory of Sensing Technology and Biomedical Instruments of Guangdong Province, School of Biomedical Engineering, Sun Yat-sen University, Shenzhen 518107, China.
Hou H; Beijing Life Science Academy, Beijing 102209, China.
Huang L; School of Biomedical Engineering, Shenzhen Campus of Sun Yat-sen University, Shenzhen 518107, China. .; Key Laboratory of Sensing Technology and Biomedical Instruments of Guangdong Province, School of Biomedical Engineering, Sun Yat-sen University, Shenzhen 518107, China.
Li J; Department of Chemistry, Center for BioAnalytical Chemistry, Key Laboratory of Bioorganic Phosphorus Chemistry & Chemical Biology, Tsinghua University, Beijing 100084, China. .; New Cornerstone Science Laboratory, Shenzhen 518054, China.; Beijing Life Science Academy, Beijing 102209, China.; Center for BioAnalytical Chemistry, Hefei National Laboratory of Physical Science at Microscale, University of Science and Technology of China, Hefei 230026, China.
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Źródło:
Lab on a chip [Lab Chip] 2024 Feb 27; Vol. 24 (5), pp. 1307-1326. Date of Electronic Publication: 2024 Feb 27.
Typ publikacji:
Journal Article; Review; Research Support, Non-U.S. Gov't
MeSH Terms:
Artificial Intelligence*
Microfluidics*
Automation ; Drug Evaluation, Preclinical
Czasopismo naukowe
Tytuł:
Metabolic Dysfunction-Associated Steatotic Liver Disease in a Dish: Human Precision-Cut Liver Slices as a Platform for Drug Screening and Interventions.
Autorzy:
Li M; Department of Pharmaceutical Technology and Biopharmacy, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
Larsen FT; Department of Biochemistry and Molecular Biology, University of Southern Denmark, 5230 Odense M, Denmark.
van den Heuvel MC; Department of Pathology and Medical Biology, Pathology Section, University Medical Center Groningen, 9700 RB Groningen, The Netherlands.
Gier K; Department of Pharmaceutical Technology and Biopharmacy, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
Gorter AR; Department of Pharmaceutical Technology and Biopharmacy, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
Oosterhuis D; Department of Pharmaceutical Technology and Biopharmacy, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
Bijzet J; Amyloidosis Center of Expertise, University Medical Center Groningen, 9713 GZ Groningen, The Netherlands.; Department of Laboratory Medicine, Division of Medical Immunology, University Medical Center Groningen, 9713 GZ Groningen, The Netherlands.
de Meijer VE; Department of Surgery, Division of Hepato-Pancreato-Biliary Surgery and Liver Transplantation, University Medical Center Groningen, 9713 AV Groningen, The Netherlands.
Ravnskjaer K; Department of Biochemistry and Molecular Biology, University of Southern Denmark, 5230 Odense M, Denmark.
Nagelkerke A; Department of Pharmaceutical Analysis, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
Olinga P; Department of Pharmaceutical Technology and Biopharmacy, Groningen Research Institute of Pharmacy, University of Groningen, 9713 AV Groningen, The Netherlands.
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Źródło:
Nutrients [Nutrients] 2024 Feb 23; Vol. 16 (5). Date of Electronic Publication: 2024 Feb 23.
Typ publikacji:
Journal Article
MeSH Terms:
Fatty Liver*
Metabolic Diseases*
Humans ; Drug Evaluation, Preclinical ; Tissue Inhibitor of Metalloproteinase-1 ; Inflammation
Czasopismo naukowe
Tytuł:
Drosophila expressing mutant human KCNT1 transgenes make an effective tool for targeted drug screening in a whole animal model of KCNT1-epilepsy.
Autorzy:
Hussain R; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.
Lim CX; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.; Pharmacy, School of Health and Biomedical Sciences, RMIT University, Bundoora, VIC, 3083, Australia.
Shaukat Z; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.
Islam A; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.; College of Medicine and Public Health, Flinders University, Bedford Park, SA, 5042, Australia.
Caseley EA; School of Biomedical Sciences, Faculty of Biological Sciences, University of Leeds, Leeds, LS2 9JT, UK.
Lippiat JD; School of Biomedical Sciences, Faculty of Biological Sciences, University of Leeds, Leeds, LS2 9JT, UK.
Rychkov GY; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.; School of Biomedicine, University of Adelaide, Adelaide, SA, 5005, Australia.; South Australian Health and Medical Research Institute, Adelaide, SA, 5005, Australia.
Ricos MG; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia.
Dibbens LM; Epilepsy Research Group, Clinical and Health Sciences, Australian Centre for Precision Health, University of South Australia, Adelaide, SA, 5000, Australia. .
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Źródło:
Scientific reports [Sci Rep] 2024 Feb 09; Vol. 14 (1), pp. 3357. Date of Electronic Publication: 2024 Feb 09.
Typ publikacji:
Journal Article
MeSH Terms:
Drosophila*/genetics
Epilepsy*/drug therapy
Epilepsy*/genetics
Potassium Channels, Sodium-Activated*/genetics
Animals ; Humans ; Drosophila melanogaster/genetics ; Drug Evaluation, Preclinical ; Models, Animal ; Mutation ; Nerve Tissue Proteins/genetics ; Seizures/drug therapy ; Seizures/genetics ; Transgenes
Czasopismo naukowe
Tytuł:
Microfluidics and Organ-on-a-Chip for Disease Modeling and Drug Screening.
Autorzy:
Nasiri R; Science for Life Laboratory, Division of Nanobiotechnology, Department of Protein Science, KTH Royal Institute of Technology, 17165 Solna, Sweden.
Zhu Y; Terasaki Institute for Biomedical Innovation, Los Angeles, CA 91367, USA.
de Barros NR; Terasaki Institute for Biomedical Innovation, Los Angeles, CA 91367, USA.
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Źródło:
Biosensors [Biosensors (Basel)] 2024 Feb 04; Vol. 14 (2). Date of Electronic Publication: 2024 Feb 04.
Typ publikacji:
Editorial
MeSH Terms:
Microfluidics*
Tissue Engineering*
Microphysiological Systems ; Drug Evaluation, Preclinical ; Lab-On-A-Chip Devices
Opinia redakcyjna
Tytuł:
Integrating cfDNA liquid biopsy and organoid-based drug screening reveals PI3K signaling as a promising therapeutic target in colorectal cancer.
Autorzy:
Yang H; Department of Gastrointestinal Surgery, The First Affiliated Hospital of Sun Yat-Sen University, Guangzhou, Guangdong, China.; Guangdong Provincial Key Laboratory of Digestive Cancer Research, Shenzhen, Guangdong, China.
Xiao X; Guangdong Provincial Key Laboratory of Digestive Cancer Research, Shenzhen, Guangdong, China.
Zeng L; Department of Biobank, The Seventh Affiliated Hospital of Sun Yat-Sen University, Shenzhen, Guangdong, China.
Zeng H; Guangdong Provincial Key Laboratory of Digestive Cancer Research, Shenzhen, Guangdong, China.
Zheng Y; Clinical Big Data Research Center, Scientific Research Center, The Seventh Affiliated Hospital of Sun Yat-Sen University, Shenzhen, China.
Wang J; Department of Oncology, Sun Yat-Sen Memorial Hospital, Sun Yat-Sen University, Guangzhou, Guangdong, China.
Li G; Department of Gastrointestinal Surgery, The First Affiliated Hospital of Sun Yat-Sen University, Guangzhou, Guangdong, China.
Dai W; Department of Gastrointestinal Surgery, The First Affiliated Hospital of Sun Yat-Sen University, Guangzhou, Guangdong, China.
He Y; Guangdong Provincial Key Laboratory of Digestive Cancer Research, Shenzhen, Guangdong, China.; Department of Gastrointestinal Surgery, The Seventh Affiliated Hospital of Sun Yat-Sen University, Shenzhen, Guangdong, China.
Wang S; School of Laboratory Medicine and Biotechnology, Southern Medical University, Guangzhou, Guangdong, China. .
Peng J; Department of Gastrointestinal Surgery, The First Affiliated Hospital of Sun Yat-Sen University, Guangzhou, Guangdong, China. .
Chen W; Guangdong Provincial Key Laboratory of Digestive Cancer Research, Shenzhen, Guangdong, China. .; Department of Gastrointestinal Surgery, The Seventh Affiliated Hospital of Sun Yat-Sen University, Shenzhen, Guangdong, China. .
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Źródło:
Journal of translational medicine [J Transl Med] 2024 Feb 03; Vol. 22 (1), pp. 132. Date of Electronic Publication: 2024 Feb 03.
Typ publikacji:
Journal Article
MeSH Terms:
Colorectal Neoplasms*/drug therapy
Colorectal Neoplasms*/genetics
Colorectal Neoplasms*/diagnosis
Cell-Free Nucleic Acids*
Humans ; Phosphatidylinositol 3-Kinases/genetics ; Drug Evaluation, Preclinical ; Proto-Oncogene Proteins p21(ras)/genetics ; Early Detection of Cancer ; Liquid Biopsy ; Phosphoinositide-3 Kinase Inhibitors ; Biomarkers ; Class I Phosphatidylinositol 3-Kinases/genetics ; Mutation/genetics
Czasopismo naukowe
Tytuł:
Review: Human stem cell-based 3D in vitro angiogenesis models for preclinical drug screening applications.
Autorzy:
Esparza A; Department of Metallurgical, Materials, and Biomedical Engineering (MMBME), The University of Texas at El Paso (UTEP), El Paso, TX, USA.; 3D Printed Microphysiological Systems Laboratory, The University of Texas at El Paso, El Paso, TX, USA.
Jimenez N; Department of Metallurgical, Materials, and Biomedical Engineering (MMBME), The University of Texas at El Paso (UTEP), El Paso, TX, USA.; 3D Printed Microphysiological Systems Laboratory, The University of Texas at El Paso, El Paso, TX, USA.
Borrego EA; Department of Metallurgical, Materials, and Biomedical Engineering (MMBME), The University of Texas at El Paso (UTEP), El Paso, TX, USA.; 3D Printed Microphysiological Systems Laboratory, The University of Texas at El Paso, El Paso, TX, USA.
Browne S; Department of Anatomy and Regenerative Medicine, Tissue Engineering Research Group, Royal College of Surgeons, Dublin, Ireland.; CÚRAM, Centre for Research in Medical Devices, University of Galway, Galway, H91 W2TY, Ireland.
Natividad-Diaz SL; Department of Metallurgical, Materials, and Biomedical Engineering (MMBME), The University of Texas at El Paso (UTEP), El Paso, TX, USA. .; 3D Printed Microphysiological Systems Laboratory, The University of Texas at El Paso, El Paso, TX, USA. .; Border Biomedical Research Center, University of Texas at El Paso, El Paso, TX, USA. .
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Źródło:
Molecular biology reports [Mol Biol Rep] 2024 Feb 01; Vol. 51 (1), pp. 260. Date of Electronic Publication: 2024 Feb 01.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Endothelial Cells*
Pluripotent Stem Cells*
Animals ; Humans ; Drug Evaluation, Preclinical ; Angiogenesis ; Neovascularization, Physiologic ; Cell Differentiation
Czasopismo naukowe
Tytuł:
Association of random and observed urine drug screening with long-term retention in opioid treatment programs.
Autorzy:
Michener PS; Clinical and Population Health Research Program, Graduate School of Biomedical Sciences University of Massachusetts Chan Medical School, 55 N Lake Ave, Worcester, MA 01655, USA. Electronic address: .
Knee A; Dept. of Medicine, UMass Chan Medical School - Baystate, 759 Chestnut St, Springfield, MA 01199, USA; Epidemiology/Biostatistics Research Core - Baystate Medical Center, Office of Research, 3601 Main Street, Third Floor, Springfield, MA 01199, USA.
Wilson D; Dept. of Medicine, UMass Chan Medical School - Baystate, 759 Chestnut St, Springfield, MA 01199, USA; Epidemiology/Biostatistics Research Core - Baystate Medical Center, Office of Research, 3601 Main Street, Third Floor, Springfield, MA 01199, USA.
Boama-Nyarko E; Clinical and Population Health Research Program, Graduate School of Biomedical Sciences University of Massachusetts Chan Medical School, 55 N Lake Ave, Worcester, MA 01655, USA.
Friedmann PD; Dept. of Medicine, UMass Chan Medical School - Baystate, 759 Chestnut St, Springfield, MA 01199, USA.
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Źródło:
Drug and alcohol dependence [Drug Alcohol Depend] 2024 Feb 01; Vol. 255, pp. 111067. Date of Electronic Publication: 2023 Dec 24.
Typ publikacji:
Journal Article
MeSH Terms:
Analgesics, Opioid*/therapeutic use
Opioid-Related Disorders*/drug therapy
Opioid-Related Disorders*/rehabilitation
Humans ; Cross-Sectional Studies ; Drug Evaluation, Preclinical ; Opiate Substitution Treatment/methods ; Methadone/therapeutic use ; Surveys and Questionnaires
Czasopismo naukowe
Tytuł:
Engineering of novel hemagglutinin biosensors for rapid detection and drug screening of Influenza A H7N9 virus.
Autorzy:
Chen X; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Huang Y; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Gao P; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Wu F; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Han Y; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Zhang C; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China.
Hu Z; The Fifth Affiliated Hospital, Southern Medical University, Guangzhou, Guangdong 510070, China.
Zhao F; National Clinical Research Centre for Infectious Diseases, the Third People's Hospital of Shenzhen and the Second Affiliated Hospital of Southern University of Science and Technology, Shenzhen 518112, Guangdong Province, China.
Shcherbakov DN; State Research Center of Virology and Biotechnology VECTOR, Koltsovo 630559, Russia; Department of Physical-Chemistry Biology and Biotechnology, Altai State University, Barnaul 656049, Russia.
Pan W; State Key Laboratory of Respiratory Disease, National Clinical Research Center for Respiratory Disease, Guangzhou Institute of Respiratory Health, the First Affiliated Hospital of Guangzhou Medical University, Guangzhou, Guangdong 510120, China.
Niu X; State Key Laboratory of Respiratory Disease, National Clinical Research Center for Respiratory Disease, Guangzhou Institute of Respiratory Health, the First Affiliated Hospital of Guangzhou Medical University, Guangzhou, Guangdong 510120, China.
Li X; The Fifth Affiliated Hospital, Southern Medical University, Guangzhou, Guangdong 510070, China. Electronic address: .
Liu S; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China; State Key Laboratory of Organ Failure Research, Guangdong Provincial Institute of Nephrology, Southern Medical University, Guangzhou 510515, China. Electronic address: .
Xu W; Guangdong Provincial Key Laboratory of New Drug Screening, School of Pharmaceutical Sciences, Southern Medical University, Guangzhou, Guangdong 510515, China; Key Laboratory of Infectious Diseases Research in South China, Ministry of Education, Southern Medical University, Guangzhou, Guangdong 510515, China. Electronic address: .
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Źródło:
International journal of biological macromolecules [Int J Biol Macromol] 2024 Feb; Vol. 258 (Pt 2), pp. 129126. Date of Electronic Publication: 2023 Dec 30.
Typ publikacji:
Journal Article
MeSH Terms:
Influenza, Human*
Influenza A Virus, H7N9 Subtype*
Biosensing Techniques*
Humans ; Hemagglutinins ; Drug Evaluation, Preclinical ; Hemagglutinin Glycoproteins, Influenza Virus ; Antiviral Agents
Czasopismo naukowe

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