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Wyszukujesz frazę ""Etiocholanolone"" wg kryterium: Temat


Tytuł:
Evaluation of the Anticancer and Biological Activities of Istaroxime via Ex Vivo Analyses, Molecular Docking and Conceptual Density Functional Theory Computations.
Autorzy:
Gok E; Department of Pharmaceutical Biotechnology, Faculty of Pharmacy, Sivas Cumhuriyet University, 58140 Sivas, Turkey.
Unal N; Department of Biochemistry, Faculty of Pharmacy, Yeditepe University, 34755 Istanbul, Turkey.
Gungor B; Department of Biochemistry, Faculty of Pharmacy, Yeditepe University, 34755 Istanbul, Turkey.
Karakus G; Department of Pharmaceutical Basic Sciences, Faculty of Pharmacy, Sivas Cumhuriyet University, 58140 Sivas, Turkey.
Kaya S; Department of Chemistry, Faculty of Science, Sivas Cumhuriyet University, 58140 Sivas, Turkey.
Canturk P; Department of Pharmaceutical Biotechnology, Faculty of Pharmacy, Sivas Cumhuriyet University, 58140 Sivas, Turkey.
Katin KP; Nanoengineering in Electronics, Spintronics and Photonics Institute, National Research Nuclear University MEPhI, 115409 Moscow, Russia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Nov 07; Vol. 28 (22). Date of Electronic Publication: 2023 Nov 07.
Typ publikacji:
Journal Article
MeSH Terms:
Etiocholanolone*/pharmacology
Antineoplastic Agents*/pharmacology
Molecular Docking Simulation ; Density Functional Theory
Czasopismo naukowe
Tytuł:
Selective SERCA2a activator as a candidate for chronic heart failure therapy.
Autorzy:
Arici M; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy.
Hsu SC; CVie Therapeutics Limited, Taipei, 11047, Taiwan.
Ferrandi M; Windtree Therapeutics Inc, Warrington, PA, 18976, USA.
Barassi P; Windtree Therapeutics Inc, Warrington, PA, 18976, USA.
Ronchi C; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy.
Torre E; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy.
Luraghi A; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy.
Chang GJ; Chang Gung University, Tao-Yuan, 333323, Taiwan.
Ferrari P; Windtree Therapeutics Inc, Warrington, PA, 18976, USA.
Bianchi G; Windtree Therapeutics Inc, Warrington, PA, 18976, USA.; Università Vita-Salute San Raffaele, 20132, Milan, Italy.
Peri F; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy.
Zaza A; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy. .
Rocchetti M; Department of Biotechnology and Biosciences, Università Degli Studi di Milano-Bicocca, P.Za Della Scienza 2, 20126, Milan, Italy. .
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Źródło:
Journal of translational medicine [J Transl Med] 2024 Jan 19; Vol. 22 (1), pp. 77. Date of Electronic Publication: 2024 Jan 19.
Typ publikacji:
Journal Article
MeSH Terms:
Heart Failure*/metabolism
Etiocholanolone/*analogs & derivatives
Rats ; Mice ; Animals ; Guinea Pigs ; Chronic Disease ; Enzyme Inhibitors ; Cardiotonic Agents/therapeutic use ; Sarcoplasmic Reticulum Calcium-Transporting ATPases/metabolism ; Myocytes, Cardiac/metabolism ; Calcium/metabolism
Czasopismo naukowe
Tytuł:
Treatment with 24 hour istaroxime infusion in patients hospitalised for acute heart failure: a randomised, placebo-controlled trial.
Autorzy:
Carubelli V; Cardiology, Department of Medical and Surgical Specialties, Radiological Sciences, and Public Health, University and Civil Hospital of Brescia, Brescia, Italy.
Zhang Y; Heart Failure Center, Fuwai Hospital, National Center for Cardiovascular Diseases, Beijing, China.
Metra M; Cardiology, Department of Medical and Surgical Specialties, Radiological Sciences, and Public Health, University and Civil Hospital of Brescia, Brescia, Italy.
Lombardi C; Cardiology, Department of Medical and Surgical Specialties, Radiological Sciences, and Public Health, University and Civil Hospital of Brescia, Brescia, Italy.
Felker GM; Duke University School of Medicine and Duke Clinical Research Institute, Durham, NC, USA.
Filippatos G; National and Kapodistrian University of Athens, Athens, Greece.; Medical School, University of Cyprus, Nicosia, Cyprus.
O'Connor CM; Inova Heart and Vascular Institute, Falls Church, VA, USA.
Teerlink JR; Section of Cardiology, San Francisco Veterans Affairs Medical Center, San Francisco, CA, USA.; School of Medicine, University of California, San Francisco, CA, USA.
Simmons P; Windtree Therapeutics, Inc., Warrington, PA, USA.
Segal R; Windtree Therapeutics, Inc., Warrington, PA, USA.
Malfatto G; IRCCS Istituto Auxologico Italiano, Department of Cardiovascular, Neural and Metabolic Sciences, S. Luca Hospital, Milan, Italy.
La Rovere MT; Istituti Clinici Scientifici Maugeri IRCCS, Department of Cardiology, Institute of Montescano, Pavia, Italy.
Li D; Jiangsu Provincial People's Hospital, First Affiliated Hospital of Nanjing Medical University, Nanjing, China.
Han X; The General Hospital of Shenyang Military Region of Chinese People's Liberation Arm, Shenyang, China.
Yuan Z; The First Affiliated Hospital of Xi'An Jiaotong University, Xi'an, China.
Yao Y; The First Hospital of Lanzhou University, Lanzhou, China.
Li B; Lee's Pharmaceutical Limited, Taipei, Taiwan.
Lau LF; CVie Therapeutics Limited, Taipei, Taiwan.
Bianchi G; Windtree Therapeutics, Inc., Warrington, PA, USA.
Zhang J; Heart Failure Center, Fuwai Hospital, National Center for Cardiovascular Diseases, Beijing, China.
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Corporate Authors:
Istaroxime ADHF Trial Group
Źródło:
European journal of heart failure [Eur J Heart Fail] 2020 Sep; Vol. 22 (9), pp. 1684-1693. Date of Electronic Publication: 2020 Jan 23.
Typ publikacji:
Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
MeSH Terms:
Heart Failure*/drug therapy
Etiocholanolone/*analogs & derivatives
Double-Blind Method ; Etiocholanolone/therapeutic use ; Humans ; Stroke Volume ; Ventricular Function, Left
Czasopismo naukowe
Tytuł:
Safety and efficacy of istaroxime in patients with acute heart failure-related pre-cardiogenic shock - a multicentre, randomized, double-blind, placebo-controlled, parallel group study (SEISMiC).
Autorzy:
Metra M; Cardiology Unit, ASST Spedali Civili, Department of Medical and Surgical Specialties, Radiological Sciences, and Public Health, University of Brescia, Brescia, Italy.
Chioncel O; Emergency Institute for Cardiovascular Diseases 'Prof. C.C. Iliescu', Bucharest, Romania.; University of Medicine Carol Davila, Bucharest, Romania.
Cotter G; Momentum Research, Inc, Chapel Hill, NC, USA.; Cardiovascular Markers in Stress Conditions (MASCOT), Université Paris Cité; Inserm UMR-S 942, Paris, France.
Davison B; Momentum Research, Inc, Chapel Hill, NC, USA.; Cardiovascular Markers in Stress Conditions (MASCOT), Université Paris Cité; Inserm UMR-S 942, Paris, France.
Filippatos G; Department of Cardiology, University of Cyprus, School of Medicine & National and Kapodistrian University of Athens, School of Medicine, Attikon University Hospital, Athens, Greece.
Mebazaa A; Cardiovascular Markers in Stress Conditions (MASCOT), Université Paris Cité; Inserm UMR-S 942, Paris, France.; Department of Anesthesiology and Critical Care and Burn Unit, Hôpital Saint-Louis Lariboisière, FHU PROMICE, DMU Parabol, APHP.Nord, Paris, France.
Novosadova M; Momentum Research, Inc, Chapel Hill, NC, USA.
Ponikowski P; Department of Heart Diseases, Wroclaw Medical University, Wrocław, Poland.
Simmons P; Windtree Therapeutics, Inc., Warrington, PA, USA.
Soffer J; Windtree Therapeutics, Inc., Warrington, PA, USA.
Simonson S; Windtree Therapeutics, Inc., Warrington, PA, USA.
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Źródło:
European journal of heart failure [Eur J Heart Fail] 2022 Oct; Vol. 24 (10), pp. 1967-1977. Date of Electronic Publication: 2022 Aug 22.
Typ publikacji:
Randomized Controlled Trial; Multicenter Study; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Heart Failure*/complications
Heart Failure*/drug therapy
Humans ; Shock, Cardiogenic/drug therapy ; Shock, Cardiogenic/etiology ; Cardiotonic Agents/therapeutic use ; Etiocholanolone/therapeutic use ; Double-Blind Method
Czasopismo naukowe
Tytuł:
Activation of the α1β2γ2L GABA A Receptor by Physiological Agonists.
Autorzy:
Pierce SR; Department of Anesthesiology, The Taylor Family Institute for Innovative Psychiatric Research, Washington University School of Medicine, St. Louis, MO 63110, USA.
Germann AL; Department of Anesthesiology, The Taylor Family Institute for Innovative Psychiatric Research, Washington University School of Medicine, St. Louis, MO 63110, USA.
Akk G; Department of Anesthesiology, The Taylor Family Institute for Innovative Psychiatric Research, Washington University School of Medicine, St. Louis, MO 63110, USA.
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Źródło:
Biomolecules [Biomolecules] 2021 Dec 11; Vol. 11 (12). Date of Electronic Publication: 2021 Dec 11.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
GABA-A Receptor Agonists/*pharmacology
Receptors, GABA-A/*metabolism
Taurine/*pharmacology
beta-Alanine/*pharmacology
Allosteric Regulation ; Animals ; Computer Simulation ; Etiocholanolone/pharmacology ; Humans ; Pregnanolone/pharmacology
Czasopismo naukowe
Tytuł:
Istaroxime in acute heart failure: the holy grail is at HORIZON?
Autorzy:
Chioncel O; Emergency Institute for Cardiovascular Diseases 'Prof. C.C. Iliescu', University of Medicine Carol Davila, Bucharest, Romania.
Collins SP; Department of Emergency Medicine, Vanderbilt University School of Medicine, Nashville, TN, USA.
Butler J; Department of Medicine, University of Mississippi Medical Center, Jackson, MS, USA.
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Źródło:
European journal of heart failure [Eur J Heart Fail] 2020 Sep; Vol. 22 (9), pp. 1694-1697. Date of Electronic Publication: 2020 May 06.
Typ publikacji:
Editorial; Comment
MeSH Terms:
Heart Failure*/drug therapy
Cardiotonic Agents/therapeutic use ; Etiocholanolone/analogs & derivatives ; Humans
Opinia redakcyjna
Tytuł:
Anticonvulsant potencies of the enantiomers of the neurosteroids androsterone and etiocholanolone exceed those of the natural forms.
Autorzy:
Zolkowska D; Department of Neurology, University of California, Davis School of Medicine, Sacramento, CA, 20817, USA.
Dhir A
Krishnan K
Covey DF
Rogawski MA
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Źródło:
Psychopharmacology [Psychopharmacology (Berl)] 2014 Sep; Vol. 231 (17), pp. 3325-32. Date of Electronic Publication: 2014 Apr 05.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural
MeSH Terms:
Androsterone/*pharmacology
Anticonvulsants/*pharmacology
Etiocholanolone/*pharmacology
Neurotransmitter Agents/*pharmacology
Androsterone/chemistry ; Animals ; Behavior, Animal/drug effects ; Convulsants/pharmacology ; Dose-Response Relationship, Drug ; Dyskinesia, Drug-Induced/psychology ; Electroshock ; Etiocholanolone/chemistry ; Male ; Mice ; Neurotransmitter Agents/chemistry ; Pentylenetetrazole/antagonists & inhibitors ; Stereoisomerism ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Validation of a Fecal Glucocorticoid Assay to Assess Adrenocortical Activity in Meerkats Using Physiological and Biological Stimuli.
Autorzy:
Braga Goncalves I; Department of Evolutionary Biology and Environmental Studies, Animal Behaviour, University of Zurich, Winterthurerstrasse 190, 8057, Zürich, Switzerland.
Heistermann M; Endocrinology Laboratory, German Primate Center, Kellnerweg 4, D-37077, Göttingen, Germany.
Santema P; Department of Zoology, University of Cambridge, Cambridge, CB2 3EJ, United Kingdom.
Dantzer B; Department of Zoology, University of Cambridge, Cambridge, CB2 3EJ, United Kingdom.
Mausbach J; Department of Evolutionary Biology and Environmental Studies, Animal Behaviour, University of Zurich, Winterthurerstrasse 190, 8057, Zürich, Switzerland.
Ganswindt A; Endocrine Research Laboratory, Department of Anatomy and Physiology, University of Pretoria, 0110, Onderstepoort, South Africa.
Manser MB; Department of Evolutionary Biology and Environmental Studies, Animal Behaviour, University of Zurich, Winterthurerstrasse 190, 8057, Zürich, Switzerland.
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Źródło:
PloS one [PLoS One] 2016 Apr 14; Vol. 11 (4), pp. e0153161. Date of Electronic Publication: 2016 Apr 14 (Print Publication: 2016).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't; Validation Study
MeSH Terms:
Feces/*chemistry
Glucocorticoids/*analysis
Herpestidae/*physiology
Hypothalamo-Hypophyseal System/*physiology
Pituitary-Adrenal System/*physiology
Adrenocorticotropic Hormone/pharmacology ; Androsterone/analogs & derivatives ; Androsterone/analysis ; Animals ; Biological Phenomena ; Chromatography, High Pressure Liquid ; Corticosterone/analysis ; Etiocholanolone/analysis ; Female ; Hypothalamo-Hypophyseal System/drug effects ; Immunoassay ; Male ; Physiological Phenomena ; Pituitary-Adrenal System/drug effects ; Reproducibility of Results ; Soil/chemistry ; Time Factors
Czasopismo naukowe
Tytuł:
SERCA2a stimulation by istaroxime: a novel mechanism of action with translational implications.
Autorzy:
Huang CL; Physiological Laboratory, University of Cambridge, Cambridge, UK.
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2013 Oct; Vol. 170 (3), pp. 486-8.
Typ publikacji:
Journal Article; Comment
MeSH Terms:
Calcium/*metabolism
Calcium-Binding Proteins/*antagonists & inhibitors
Etiocholanolone/*analogs & derivatives
Heart Failure/*drug therapy
Heart Failure/*metabolism
Sarcoplasmic Reticulum/*metabolism
Sarcoplasmic Reticulum Calcium-Transporting ATPases/*pharmacokinetics
Animals ; Humans ; Male
Czasopismo naukowe
Tytuł:
Combination of carbon isotope ratio with hydrogen isotope ratio determinations in sports drug testing.
Autorzy:
Piper T; Center for Preventive Doping Research-Institute of Biochemistry, German Sport University Cologne, Am Sportpark Müngersdorf 6, 50933 Köln, Germany. />Emery C
Thomas A
Saugy M
Thevis M
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Źródło:
Analytical and bioanalytical chemistry [Anal Bioanal Chem] 2013 Jun; Vol. 405 (16), pp. 5455-66. Date of Electronic Publication: 2013 Apr 09.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Carbon Isotopes/*analysis
Doping in Sports/*prevention & control
Gas Chromatography-Mass Spectrometry/*methods
Hydrogen/*analysis
Steroids/*urine
Administration, Oral ; Adult ; Androstane-3,17-diol/urine ; Dehydroepiandrosterone/urine ; Etiocholanolone/urine ; Female ; Gas Chromatography-Mass Spectrometry/instrumentation ; Humans ; Male ; Middle Aged ; Reference Values ; Reproducibility of Results ; Sports ; Testosterone/administration & dosage ; Testosterone/analysis ; Testosterone/pharmacology
Czasopismo naukowe
Tytuł:
Validation of noninvasive monitoring of adrenocortical endocrine activity in ground-feeding aardwolves (Proteles cristata): exemplifying the influence of consumption of inorganic material for fecal steroid analysis.
Autorzy:
Ganswindt A; Mammal Research Institute, Department of Zoology and Entomology, University of Pretoria, Pretoria 0002, South Africa.
Muilwijk C
Engelkes M
Muenscher S
Bertschinger H
Paris M
Palme R
Cameron EZ
Bennett NC
Dalerum F
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Źródło:
Physiological and biochemical zoology : PBZ [Physiol Biochem Zool] 2012 Mar-Apr; Vol. 85 (2), pp. 194-9. Date of Electronic Publication: 2012 Feb 01.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't; Validation Study
MeSH Terms:
Adrenal Cortex/*metabolism
Adrenocorticotropic Hormone/*metabolism
Feces/*chemistry
Glucocorticoids/*analysis
Hyaenidae/*metabolism
Immunoenzyme Techniques/*methods
Animals ; Diet ; Etiocholanolone/analogs & derivatives ; Etiocholanolone/immunology ; Feeding Behavior ; Female ; Hydrocortisone/immunology ; Male ; Soil
Czasopismo naukowe
Tytuł:
Metformin-Treatment Option for Social Impairment? An Open Clinical Trial to Elucidate the Effects of Metformin Treatment on Steroid Hormones and Social Behavior
Autorzy:
Benedikt Gasser
Johann Kurz
Samuel Buerki
Markus Mohaupt
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Temat:
GC–MS
urine analysis
androgens
social behavior
androsterone
etiocholanolone
Science
Źródło:
Life, Vol 12, Iss 998, p 998 (2022)
Opis pliku:
electronic resource
Relacje:
https://www.mdpi.com/2075-1729/12/7/998; https://doaj.org/toc/2075-1729
Dostęp URL:
https://doaj.org/article/c15b2b07bf9e401284959ec6ccff228c  Link otwiera się w nowym oknie
Czasopismo naukowe
Tytuł:
Glucocorticoid metabolites inhibit the metabolism of androstenedione in red blood cells of ruminants.
Autorzy:
El-Bahr SM; Institute of Biochemistry, University of Veterinary Medicine, Veterinärplatz 1, A-1210 Vienna, Austria.
Möstl E
Palme R
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Źródło:
Journal of veterinary medicine. A, Physiology, pathology, clinical medicine [J Vet Med A Physiol Pathol Clin Med] 2003 Mar; Vol. 50 (2), pp. 98-102.
Typ publikacji:
Journal Article
MeSH Terms:
Androstenedione/*pharmacokinetics
Erythrocytes/*metabolism
Etiocholanolone/*analogs & derivatives
Etiocholanolone/*pharmacology
Animals ; Cattle ; Chromatography, High Pressure Liquid ; Female ; Goats ; Male ; Sheep
Czasopismo naukowe
Tytuł:
How Is CYP17A1 Activity Altered in Autism? A Pilot Study to Identify Potential Pharmacological Targets
Autorzy:
Benedikt Andreas Gasser
Johann Kurz
Bernhard Dick
Markus Georg Mohaupt
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Temat:
DHEA
androsterone
etiocholanolone
tetrahydrocorticosterone
Science
Źródło:
Life, Vol 12, Iss 6, p 867 (2022)
Opis pliku:
electronic resource
Relacje:
https://www.mdpi.com/2075-1729/12/6/867; https://doaj.org/toc/2075-1729
Dostęp URL:
https://doaj.org/article/8ae6aad3d94b41e59d9ccb60ccc0b204  Link otwiera się w nowym oknie
Czasopismo naukowe
Tytuł:
Suppression of adrenal function by low-dose prednisone: assessment with 24-hour urinary steroid hormone profiles--a review of five cases.
Autorzy:
Friel PN; Washington State Toxicology Laboratory, 2203 Airport Way South, Seattle, WA 98134, USA. />Alexander T
Wright JV
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Źródło:
Alternative medicine review : a journal of clinical therapeutic [Altern Med Rev] 2006 Mar; Vol. 11 (1), pp. 40-6.
Typ publikacji:
Journal Article
MeSH Terms:
Adrenal Glands/*drug effects
Adrenal Insufficiency/*chemically induced
Anti-Inflammatory Agents/*adverse effects
Prednisone/*adverse effects
Adrenal Glands/metabolism ; Adrenal Insufficiency/urine ; Adult ; Aldosterone/urine ; Androsterone/urine ; Anti-Inflammatory Agents/administration & dosage ; Cortisone/urine ; Dehydroepiandrosterone/urine ; Etiocholanolone/urine ; Female ; Humans ; Hydrocortisone/urine ; Middle Aged ; Prednisone/administration & dosage
Czasopismo naukowe
Tytuł:
Molecular cloning, expression and characterization of a monkey steroid UDP-glucuronosyltransferase, UGT2B19, that conjugates testosterone.
Autorzy:
Bélanger G; Medical Research Council Group in Molecular Endocrinology, CHUL Research Center, Laveal University, Quebec, Canada.
Barbier O
Hum DW
Bélanger A
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Źródło:
European journal of biochemistry [Eur J Biochem] 1999 Mar; Vol. 260 (3), pp. 701-8.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Glucuronosyltransferase/*genetics
Testosterone/*metabolism
Amino Acid Sequence ; Androstane-3,17-diol/metabolism ; Animals ; Base Sequence ; Cells, Cultured ; Cloning, Molecular ; Etiocholanolone/metabolism ; Glucuronosyltransferase/metabolism ; Humans ; Macaca fascicularis ; Molecular Sequence Data ; Phylogeny ; RNA, Messenger/metabolism
Czasopismo naukowe

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