- Tytuł:
- Exploring TEAD2 as a drug target for therapeutic intervention of cancer: A multi-computational case study.
- Autorzy:
- Źródło:
- Briefings in bioinformatics [Brief Bioinform] 2021 Sep 02; Vol. 22 (5).
- Typ publikacji:
- Journal Article; Research Support, Non-U.S. Gov't
- MeSH Terms:
-
DNA-Binding Proteins/*antagonists & inhibitors
DNA-Binding Proteins/*metabolism
Drug Discovery/*methodsFlufenamic Acid /*metabolism
Neoplasms/*metabolism
Pharmaceutical Preparations/*metabolism
Transcription Factors/*antagonists & inhibitors
Transcription Factors/*metabolism
Binding Sites ; Crystallization ; DNA-Binding Proteins/chemistry ;Flufenamic Acid /chemistry ; Humans ; Hydrophobic and Hydrophilic Interactions ; Ligands ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Molecular Targeted Therapy/methods ; Neoplasms/drug therapy ; NiflumicAcid /chemistry ; NiflumicAcid /metabolism ; Pharmaceutical Preparations/chemistry ; Protein Binding ; TEA Domain Transcription Factors ; Transcription Factors/chemistry
Czasopismo naukowe