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Wyszukujesz frazę ""Hydantoins"" wg kryterium: Temat


Tytuł:
[3+2]-Cycloaddition of Nitrile Imines to Parabanic Acid Derivatives-An Approach to Novel Spiroimidazolidinediones.
Autorzy:
Kuznetsova JV; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Tkachenko VT; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Petrovskaya LM; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Filkina ME; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Shybanov DE; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Grishin YK; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Roznyatovsky VA; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Tafeenko VA; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Pestretsova AS; Blokhin National Medical Research Center of Oncology, Ministry of Health of the Russian Federation, 115478 Moscow, Russia.; Occupational Health Risks Lab, Peoples' Friendship University of Russia (RUDN University), 117198 Moscow, Russia.
Yakovleva VA; Department of Biochemistry, People's Friendship University of Russia (RUDN University), 117198 Moscow, Russia.
Pokrovsky VS; Blokhin National Medical Research Center of Oncology, Ministry of Health of the Russian Federation, 115478 Moscow, Russia.; Department of Biochemistry, People's Friendship University of Russia (RUDN University), 117198 Moscow, Russia.; Research Institute of Molecular and Cellular Medicine, People's Friendship University of Russia (RUDN University), 117198 Moscow, Russia.
Kukushkin ME; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Beloglazkina EK; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Dec 19; Vol. 25 (1). Date of Electronic Publication: 2023 Dec 19.
Typ publikacji:
Journal Article
MeSH Terms:
Hydantoins*
Cycloaddition Reaction ; Imines ; Nitriles
Czasopismo naukowe
Tytuł:
Synthesis of Tetracyclic Spirooxindolepyrrolidine-Engrafted Hydantoin Scaffolds: Crystallographic Analysis, Molecular Docking Studies and Evaluation of Their Antimicrobial, Anti-Inflammatory and Analgesic Activities.
Autorzy:
Toumi A; Laboratory of Heterocyclic Chemistry Natural Product and Reactivity (LR11ES39), Department of Chemistry, Faculty of Science of Monastir, University of Monastir, Monastir 5019, Tunisia.
Abdella FIA; Department of Chemistry, College of Science, Ha'il University, Ha'il 81451, Saudi Arabia.
Boudriga S; Laboratory of Heterocyclic Chemistry Natural Product and Reactivity (LR11ES39), Department of Chemistry, Faculty of Science of Monastir, University of Monastir, Monastir 5019, Tunisia.
Alanazi TYA; Department of Chemistry, College of Science, Ha'il University, Ha'il 81451, Saudi Arabia.
Alshamari AK; Department of Chemistry, College of Science, Ha'il University, Ha'il 81451, Saudi Arabia.
Alrashdi AA; Department of Chemistry, College of Science, Ha'il University, Ha'il 81451, Saudi Arabia.
Dbeibia A; Laboratory of Analysis, Treatment and Valorization of Environmental Pollutants and Products, Faculty of Pharmacy, University of Monastir, Monastir 5019, Tunisia.
Hamden K; Laboratory of Bioresources: Integrative Biology and Valorization, Higher Institute of Biotechnology of Monastir, University of Monastir, Monastir 5000, Tunisia.
Daoud I; Department of Matter Sciences, University of Mohamed Khider, BP 145 RP, Biskra 07000, Algeria.; Laboratory of Natural and Bio-Actives Substances, Faculty of Science, Tlemcen University, P.O. Box 119, Tlemcen 13000, Algeria.
Knorr M; Institut UTINAM-UMR CNRS 6213, Université de Franche-Comté, 16 Route de Gray, 25030 Besançon, France.
Kirchhoff JL; Faculty of Chemistry, Inorganic Chemistry, Technical University Dortmund, Otto-Hahn-Strasse 6, 44227 Dortmund, Germany.
Strohmann C; Faculty of Chemistry, Inorganic Chemistry, Technical University Dortmund, Otto-Hahn-Strasse 6, 44227 Dortmund, Germany.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Nov 06; Vol. 28 (21). Date of Electronic Publication: 2023 Nov 06.
Typ publikacji:
Journal Article
MeSH Terms:
Hydantoins*
Anti-Infective Agents*/pharmacology
Molecular Docking Simulation ; Anti-Inflammatory Agents, Non-Steroidal/chemistry ; Anti-Inflammatory Agents/chemistry ; Analgesics/chemistry ; Anti-Bacterial Agents/pharmacology ; Anticonvulsants/pharmacology ; Molecular Structure ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
[4+2]-Cycloaddition to 5-Methylidene-Hydantoins and 5-Methylidene-2-Thiohydantoins in the Synthesis of Spiro-2-Chalcogenimidazolones.
Autorzy:
Shybanov DE; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Kukushkin ME; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Hrytseniuk YS; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Grishin YK; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Roznyatovsky VA; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Tafeenko VA; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Skvortsov DA; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Zyk NV; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
Beloglazkina EK; Department of Chemistry, M. V. Lomonosov Moscow State University, 119991 Moscow, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Mar 06; Vol. 24 (5). Date of Electronic Publication: 2023 Mar 06.
Typ publikacji:
Journal Article
MeSH Terms:
Hydantoins*
Humans ; Thiohydantoins ; Cycloaddition Reaction ; Escherichia coli ; HEK293 Cells ; Hydrogen Peroxide ; Cyclopentanes
Czasopismo naukowe
Tytuł:
Benzenesulfonamides Incorporating Hydantoin Moieties Effectively Inhibit Eukaryoticand Human Carbonic Anhydrases.
Autorzy:
Abdoli M; Institute of Technology of Organic Chemistry, Faculty of Materials Science and Applied Chemistry, Riga Technical University, P. Valdenaiela 3, LV-1048 Riga, Latvia.
De Luca V; Department of Biology, Agriculture and Food Sciences, Institute of Biosciences and Bioresources, Via Pietro Castellino 111, 80131 Napoli, Italy.
Capasso C; Department of Biology, Agriculture and Food Sciences, Institute of Biosciences and Bioresources, Via Pietro Castellino 111, 80131 Napoli, Italy.
Supuran CT; NEUROFARBA Department, Pharmaceutical and Nutraceutical Section, University of Florence, Via Ugo Schiff 6, 50019 Florence, Italy.
Žalubovskis R; Institute of Technology of Organic Chemistry, Faculty of Materials Science and Applied Chemistry, Riga Technical University, P. Valdenaiela 3, LV-1048 Riga, Latvia.; Latvian Institute of Organic Synthesis, Aizkraukles 21, LV-1006 Riga, Latvia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Nov 15; Vol. 23 (22). Date of Electronic Publication: 2022 Nov 15.
Typ publikacji:
Journal Article
MeSH Terms:
Carbonic Anhydrase Inhibitors*/pharmacology
Carbonic Anhydrases*/metabolism
Hydantoins*/chemistry
Hydantoins*/pharmacology
Sulfonamides*/chemistry
Sulfonamides*/pharmacology
Humans ; Structure-Activity Relationship ; Benzene Derivatives/chemistry ; Benzene Derivatives/pharmacology ; Eukaryotic Cells/enzymology ; Eukaryotic Cells/metabolism ; Benzenesulfonamides
Czasopismo naukowe
Tytuł:
Regioselective Cycloaddition of Nitrile Imines to 5-Methylidene-3-phenyl-hydantoin: Synthesis and DFT Calculations.
Autorzy:
Filkina ME; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Baray DN; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Beloglazkina EK; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Grishin YK; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Roznyatovsky VA; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
Kukushkin ME; Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory, 1-3, 119991 Moscow, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Jan 09; Vol. 24 (2). Date of Electronic Publication: 2023 Jan 09.
Typ publikacji:
Journal Article
MeSH Terms:
Hydantoins*
Cycloaddition Reaction ; Density Functional Theory ; Imines/chemistry ; Nitriles/chemistry ; Anticonvulsants
Czasopismo naukowe
Tytuł:
Biologically Oriented Hybrids of Indole and Hydantoin Derivatives.
Autorzy:
Kochetkov KA; A. N. Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, 28 ul. Vavilova, 119991 Moscow, Russia.
Gorunova ON; A. N. Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, 28 ul. Vavilova, 119991 Moscow, Russia.
Bystrova NA; A. N. Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, 28 ul. Vavilova, 119991 Moscow, Russia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Jan 06; Vol. 28 (2). Date of Electronic Publication: 2023 Jan 06.
Typ publikacji:
Journal Article
MeSH Terms:
Indoles*/pharmacology
Indoles*/chemistry
Hydantoins*/pharmacology
Anticonvulsants ; Indoleacetic Acids
Czasopismo naukowe
Tytuł:
Identification of hydantoin based Decaprenylphosphoryl-β-D-Ribose Oxidase (DprE1) inhibitors as antimycobacterial agents using computational tools.
Autorzy:
Mali SN; Department of Pharmaceutical Sciences and Technology, Birla Institute of Technology, Mesra, 835215, India. .
Pandey A; Department of Pharmaceutical Sciences and Technology, Birla Institute of Technology, Mesra, 835215, India.
Bhandare RR; Department of Pharmaceutical Sciences, College of Pharmacy and Health Sciences, Ajman University, P O Box 346, Ajman, United Arab Emirates. .; Center of Medical and Bio-allied Health Sciences Research, Ajman University, P O Box 346, Ajman, United Arab Emirates. .
Shaik AB; St. Mary's College of Pharmacy, St. Mary's Group of Institutions Guntur, Affiliated to Jawaharlal Nehru Technological University Kakinada, Chebrolu, Guntur, Andhra Pradesh, 522212, India. .
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Źródło:
Scientific reports [Sci Rep] 2022 Sep 30; Vol. 12 (1), pp. 16368. Date of Electronic Publication: 2022 Sep 30.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Hydantoins*
Antitubercular Agents/chemistry ; Antitubercular Agents/pharmacology ; Ethambutol ; Isoniazid ; Ligands ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Oxidoreductases ; Quantitative Structure-Activity Relationship ; Racemases and Epimerases ; Ribose
Czasopismo naukowe
Tytuł:
Evaluation of Two Novel Hydantoin Derivatives Using Reconstructed Human Skin Model Episkin : Perspectives for Application as Potential Sunscreen Agents.
Autorzy:
Słoczyńska K; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Popiół J; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Gunia-Krzyżak A; Department of Bioorganic Chemistry, Chair of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Koczurkiewicz-Adamczyk P; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Żmudzki P; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Pękala E; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Mar 12; Vol. 27 (6). Date of Electronic Publication: 2022 Mar 12.
Typ publikacji:
Journal Article
MeSH Terms:
Hydantoins*/pharmacology
Sunscreening Agents*/metabolism
Sunscreening Agents*/pharmacology
Humans ; Permeability ; Skin/metabolism ; Skin Irritancy Tests
Czasopismo naukowe
Tytuł:
Structure-Activity Relationship Studies of Hydantoin-Cored Ligands for Smoothened Receptor.
Autorzy:
Liu Y; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Zhou F; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Ding K; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Xue D; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Zhu Z; Department of Chemistry, Nanchang University, 999 Xuefu Avenue, Nanchang, 330031, China.
Li C; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.; School of Life Science and Technology, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Li F; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Xu Y; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Xu F; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.; School of Life Science and Technology, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Le Z; Department of Chemistry, Nanchang University, 999 Xuefu Avenue, Nanchang, 330031, China.
Zhao S; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.; School of Life Science and Technology, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
Tao H; iHuman Institute, ShanghaiTech University, 393 Middle Huaxia Road, Shanghai, 201210, China.
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Źródło:
ChemistryOpen [ChemistryOpen] 2021 Oct; Vol. 10 (10), pp. 1028-1032.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Hydantoins*/pharmacology
Binding Sites ; Ligands ; Smoothened Receptor ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Phenylpiperazine 5,5-Dimethylhydantoin Derivatives as First Synthetic Inhibitors of Msr(A) Efflux Pump in Staphylococcus epidermidis .
Autorzy:
Witek K; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.; Department of Pharmaceutical Microbiology, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Latacz G; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Kaczor A; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Czekajewska J; Department of Pharmaceutical Microbiology, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Żesławska E; Institute of Biology, Pedagogical University of Krakow, ul. Podchorążych 2, 30-084 Krakow, Poland.
Chudzik A; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Karczewska E; Department of Pharmaceutical Microbiology, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Nitek W; Faculty of Chemistry, Jagiellonian University, ul. Gronostajowa 2, 30-387 Krakow, Poland.
Kieć-Kononowicz K; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
Handzlik J; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, ul. Medyczna 9, 30-688 Krakow, Poland.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2020 Aug 20; Vol. 25 (17). Date of Electronic Publication: 2020 Aug 20.
Typ publikacji:
Journal Article
MeSH Terms:
Bacterial Proteins*/antagonists & inhibitors
Bacterial Proteins*/chemistry
Bacterial Proteins*/metabolism
Hydantoins*/chemistry
Hydantoins*/pharmacology
Membrane Transport Proteins*/chemistry
Membrane Transport Proteins*/metabolism
Staphylococcus epidermidis*/chemistry
Staphylococcus epidermidis*/metabolism
Crystallography, X-Ray
Czasopismo naukowe
Tytuł:
Self-Assembly and Biorecognition of a Spirohydantoin Derived from α-Tetralone: Interplay between Chirality and Intermolecular Interactions.
Autorzy:
Lazić AM; Innovation Centre of the Faculty of Technology and Metallurgy, Karnegijeva 4, 11120, Belgrade, Serbia.
Đorđević IS; Department of Chemistry - Theoretical chemistry and molecular modeling, Institute of Chemistry, Technology and Metallurgy, National Institute, University of Belgrade, Njegoševa 12, 11000, Belgrade, Serbia.
Radovanović LD; Innovation Centre of the Faculty of Technology and Metallurgy, Karnegijeva 4, 11120, Belgrade, Serbia.
Popović DM; Department of Chemistry - Theoretical chemistry and molecular modeling, Institute of Chemistry, Technology and Metallurgy, National Institute, University of Belgrade, Njegoševa 12, 11000, Belgrade, Serbia.
Rogan JR; Department of General and Inorganic Chemistry, Department of Organic Chemistry, Faculty of Technology and Metallurgy, University of Belgrade Karnegijeva 4, 11120 Belgrade (Serbia).
Janjić GV; Department of Chemistry - Theoretical chemistry and molecular modeling, Institute of Chemistry, Technology and Metallurgy, National Institute, University of Belgrade, Njegoševa 12, 11000, Belgrade, Serbia.
Trišović NP; Department of General and Inorganic Chemistry, Department of Organic Chemistry, Faculty of Technology and Metallurgy, University of Belgrade Karnegijeva 4, 11120 Belgrade (Serbia).
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Źródło:
ChemPlusChem [Chempluschem] 2020 Jun; Vol. 85 (6), pp. 1220-1232.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Hydantoins/*chemistry
Spiro Compounds/*chemistry
Tetrahydronaphthalenes/*chemistry
Crystallography, X-Ray ; Humans ; Hydantoins/metabolism ; Interleukin-1 Receptor-Associated Kinases/metabolism ; Molecular Docking Simulation ; Receptors, Dopamine D3/metabolism ; Spiro Compounds/metabolism ; Stereoisomerism ; Tetrahydronaphthalenes/metabolism
Czasopismo naukowe
Tytuł:
Antitussive and Anti-inflammatory Dual-active Agents Developed from Natural Product Lead Compound 1-Methylhydantoin.
Autorzy:
Xu Y; School of Pharmaceutical Sciences, Jilin University, Changchun, Jilin 130021, China.; College of Basic Medical Sciences, Jilin University, Changchun, Jilin 130021, China.; Department of Drug and Food Sciences, Changchun Medical College, Changchun, Jilin 130031, China.
Wang F; College of Basic Medical Sciences, Jilin University, Changchun, Jilin 130021, China.
Guo H; School of Pharmaceutical Sciences, Jilin University, Changchun, Jilin 130021, China.
Wang S; College of Chinese Medicine Materials, Jilin Agricultural University, Changchun 130118, China.
Ni S; School of Pharmaceutical Sciences, Jilin University, Changchun, Jilin 130021, China.
Zhou Y; School of Pharmaceutical Sciences, Jilin University, Changchun, Jilin 130021, China.
Wang Z; Department of Physical Sciences, Eastern New Mexico University, Portales, NM 88130, USA.
Bao H; College of Pharmacy, Changchun University of Chinese Medicine, Changchun, Jilin 130117, China.
Wang Y; School of Pharmaceutical Sciences, Jilin University, Changchun, Jilin 130021, China. .
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2019 Jun 26; Vol. 24 (13). Date of Electronic Publication: 2019 Jun 26.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Inflammatory Agents/*pharmacology
Antitussive Agents/*pharmacology
Biological Products/*pharmacology
Drugs, Chinese Herbal/*pharmacology
Hydantoins/*pharmacology
Animals ; Anti-Inflammatory Agents/chemical synthesis ; Anti-Inflammatory Agents/chemistry ; Antitussive Agents/chemical synthesis ; Antitussive Agents/chemistry ; Biological Products/chemistry ; Cyclooxygenase 1/chemistry ; Cyclooxygenase 1/metabolism ; Cyclooxygenase 2/chemistry ; Cyclooxygenase 2/metabolism ; Drug Design ; Drugs, Chinese Herbal/chemical synthesis ; Drugs, Chinese Herbal/chemistry ; Hydantoins/chemical synthesis ; Hydantoins/chemistry ; Mice ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Molecular Structure ; Protein Binding ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Discovery of Novel UV-Filters with Favorable Safety Profiles in the 5-Arylideneimidazolidine-2,4-dione Derivatives Group.
Autorzy:
Popiół J; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .; Department of Bioorganic Chemistry, Chair of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Gunia-Krzyżak A; Department of Bioorganic Chemistry, Chair of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Piska K; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Żelaszczyk D; Department of Bioorganic Chemistry, Chair of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland.
Koczurkiewicz P; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Słoczyńska K; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Wójcik-Pszczoła K; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Krupa A; Department of Pharmaceutical Technology and Biopharmaceutics, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Kryczyk-Poprawa A; Department of Inorganic and Analytical Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Żesławska E; Department of Chemistry, Institute of Biology, Pedagogical University of Cracow, Podchorążych 2, 30-084 Krakow, Poland. .
Nitek W; Faculty of Chemistry, Jagiellonian University, Gronostajowa 2, 30-387 Krakow, Poland. .
Żmudzki P; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Marona H; Department of Bioorganic Chemistry, Chair of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
Pękala E; Department of Pharmaceutical Biochemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland. .
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2019 Jun 24; Vol. 24 (12). Date of Electronic Publication: 2019 Jun 24.
Typ publikacji:
Journal Article
MeSH Terms:
Ultraviolet Rays*
Hydantoins/*chemistry
Hydantoins/*radiation effects
Radiation-Protective Agents/*chemistry
Radiation-Protective Agents/*radiation effects
Animals ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Cell Proliferation/radiation effects ; Drug Stability ; Humans ; Hydantoins/pharmacology ; Mice ; Models, Molecular ; Molecular Structure ; Radiation-Protective Agents/pharmacology ; Spectrum Analysis ; Structure-Activity Relationship ; Sunscreening Agents/chemistry ; Sunscreening Agents/radiation effects
Czasopismo naukowe
Tytuł:
1,3-Dibromo-5,5-dimethylhydantoin as a Precatalyst for Activation of Carbonyl Functionality.
Autorzy:
Čebular K; Department of Physical and Organic Chemistry, Jožef Stefan Institute, Jamova 39, 1000 Ljubljana, Slovenia.; Jožef Stefan International Postgraduate School, Jamova 39, 1000 Ljubljana, Slovenia.
Božić BĐ; Department of Physical and Organic Chemistry, Jožef Stefan Institute, Jamova 39, 1000 Ljubljana, Slovenia.; Institute of Physiology and Biochemistry, Faculty of Biology, University of Belgrade, Studentski trg 16, 11000 Belgrade, Serbia.
Stavber S; Department of Physical and Organic Chemistry, Jožef Stefan Institute, Jamova 39, 1000 Ljubljana, Slovenia. .; Jožef Stefan International Postgraduate School, Jamova 39, 1000 Ljubljana, Slovenia. .
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2019 Jul 17; Vol. 24 (14). Date of Electronic Publication: 2019 Jul 17.
Typ publikacji:
Journal Article
MeSH Terms:
Catalysis*
Acids/*chemistry
Hydantoins/*chemistry
Esterification ; Hydantoins/chemical synthesis ; Indicators and Reagents/chemistry
Czasopismo naukowe
Tytuł:
In the search for a lead structure among series of potent and selective hydantoin 5-HT 7 R agents: The drug-likeness in vitro study.
Autorzy:
Latacz G; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Lubelska A; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Jastrzębska-Więsek M; Department of Clinical Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Partyka A; Department of Clinical Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Sobiło A; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Olejarz A; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Kucwaj-Brysz K; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Satała G; Department of Medicinal Chemistry Institute of Pharmacology, Polish Academy of Sciences, Kraków, Poland.
Bojarski AJ; Department of Medicinal Chemistry Institute of Pharmacology, Polish Academy of Sciences, Kraków, Poland.
Wesołowska A; Department of Clinical Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Kieć-Kononowicz K; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
Handzlik J; Department of Technology and Biotechnology of Drugs, Jagiellonian University, Medical College, Kraków, Poland.
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Źródło:
Chemical biology & drug design [Chem Biol Drug Des] 2017 Dec; Vol. 90 (6), pp. 1295-1306. Date of Electronic Publication: 2017 Oct 03.
Typ publikacji:
Journal Article
MeSH Terms:
Antidepressive Agents/*chemistry
Hydantoins/*chemistry
Receptors, Serotonin/*metabolism
Animals ; Antidepressive Agents/metabolism ; Antidepressive Agents/pharmacology ; Cell Survival/drug effects ; Cytochrome P-450 Enzyme System/metabolism ; Drug Interactions ; HEK293 Cells ; Hep G2 Cells ; Humans ; Hydantoins/metabolism ; Hydantoins/pharmacology ; Kinetics ; Ligands ; Locomotion/drug effects ; Male ; Maze Learning/drug effects ; Mice ; Microsomes, Liver/metabolism ; Permeability/drug effects ; Receptor, Serotonin, 5-HT1A/chemistry ; Receptor, Serotonin, 5-HT1A/metabolism ; Receptors, Serotonin/chemistry ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Tyrosine-derived novel antimicrobial hydantoin polymers: synthesis and evaluation of anti-bacterial activities.
Autorzy:
Ravichandran V; a Biomaterials Laboratory, Department of Biotechnology, Bhupat and Jyoti Mehta School of Biosciences , Indian Institute of Technology Madras , Chennai , India.
Rai RK; a Biomaterials Laboratory, Department of Biotechnology, Bhupat and Jyoti Mehta School of Biosciences , Indian Institute of Technology Madras , Chennai , India.
Kesavan V; a Biomaterials Laboratory, Department of Biotechnology, Bhupat and Jyoti Mehta School of Biosciences , Indian Institute of Technology Madras , Chennai , India.
Jayakrishnan A; a Biomaterials Laboratory, Department of Biotechnology, Bhupat and Jyoti Mehta School of Biosciences , Indian Institute of Technology Madras , Chennai , India.
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Źródło:
Journal of biomaterials science. Polymer edition [J Biomater Sci Polym Ed] 2017 Dec; Vol. 28 (18), pp. 2131-2142. Date of Electronic Publication: 2017 Sep 19.
Typ publikacji:
Journal Article
MeSH Terms:
Polymerization*
Anti-Bacterial Agents/*chemistry
Anti-Bacterial Agents/*pharmacology
Hydantoins/*chemistry
Hydantoins/*pharmacology
Tyrosine/*chemistry
Anti-Bacterial Agents/chemical synthesis ; Chemistry Techniques, Synthetic ; Escherichia coli/drug effects ; Hydantoins/chemical synthesis ; Microbial Sensitivity Tests ; Staphylococcus aureus/drug effects
Czasopismo naukowe
Tytuł:
The Bucherer-Bergs Multicomponent Synthesis of Hydantoins-Excellence in Simplicity.
Autorzy:
Kalník M; Institute of Chemistry, Center for Glycomics, Slovak Academy of Sciences, Dúbravská cesta 9, SK-845 38 Bratislava, Slovakia.
Gabko P; Institute of Chemistry, Center for Glycomics, Slovak Academy of Sciences, Dúbravská cesta 9, SK-845 38 Bratislava, Slovakia.
Bella M; Institute of Chemistry, Center for Glycomics, Slovak Academy of Sciences, Dúbravská cesta 9, SK-845 38 Bratislava, Slovakia.
Koóš M; Institute of Chemistry, Center for Glycomics, Slovak Academy of Sciences, Dúbravská cesta 9, SK-845 38 Bratislava, Slovakia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2021 Jun 30; Vol. 26 (13). Date of Electronic Publication: 2021 Jun 30.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Chemistry Techniques, Synthetic*
Agrochemicals/*chemical synthesis
Agrochemicals/*chemistry
Hydantoins/*chemical synthesis
Hydantoins/*chemistry
Molecular Structure
Czasopismo naukowe
Tytuł:
Wide distribution of resistance to the fungicides fludioxonil and iprodione in Penicillium species.
Autorzy:
Oiki S; Faculty of Life and Environmental Sciences, University of Tsukuba, Tsukuba, Japan.
Yaguchi T; Medical Mycology Research Center, Chiba University, Chiba, Japan.
Urayama SI; Faculty of Life and Environmental Sciences, University of Tsukuba, Tsukuba, Japan.; Microbiology Research Center for Sustainability, University of Tsukuba, Tsukuba, Japan.
Hagiwara D; Faculty of Life and Environmental Sciences, University of Tsukuba, Tsukuba, Japan.; Microbiology Research Center for Sustainability, University of Tsukuba, Tsukuba, Japan.
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Źródło:
PloS one [PLoS One] 2022 Jan 31; Vol. 17 (1), pp. e0262521. Date of Electronic Publication: 2022 Jan 31 (Print Publication: 2022).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Resistance, Fungal*
Polymorphism, Single Nucleotide*
Aminoimidazole Carboxamide/*analogs & derivatives
Dioxoles/*pharmacology
Fungal Proteins/*genetics
Hydantoins/*pharmacology
Mycoses/*drug therapy
Penicillium/*isolation & purification
Pyrroles/*pharmacology
Aminoimidazole Carboxamide/pharmacology ; Cadaver ; Crops, Agricultural/microbiology ; Food Analysis ; Fungicides, Industrial/pharmacology ; Humans ; Mycoses/genetics ; Mycoses/microbiology ; Penicillium/drug effects ; Penicillium/genetics
Czasopismo naukowe

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