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Wyszukujesz frazę ""Kaplancikli ZA"" wg kryterium: Autor


Tytuł :
Synthesis and biological evaluation of novel 1,3,4-thiadiazole derivatives as possible anticancer agents
Autorzy :
Çevik Ulviye Acar
Osmaniye Derya
Levent Serkan
Sağlik Begüm Nurpelin
Çavuşoğlu Betül Kaya
Karaduman Abdullah Burak
Özkay Yusuf
Kaplancikli Zafer Asim
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Temat :
4-thiadiazole
anticancer activity
aromatase inhibitory activity
mtt assay
Pharmaceutical industry
HD9665-9675
Źródło :
Acta Pharmaceutica, Vol 70, Iss 4, Pp 499-513 (2020)
Opis pliku :
electronic resource
Relacje :
https://doaj.org/toc/1846-9558
Dostęp URL :
https://doaj.org/article/0297ca8d7ca049128a13d18cc4e1efe5
Czasopismo naukowe
Tytuł :
Design, synthesis, in vitro, and in silico studies of 1,2,4-triazole-piperazine hybrid derivatives as potential MAO inhibitors.
Autorzy :
Uslu H; Firat University, Department of Medical Services and Techniques, Vocational School of Health Services, 23119 Elazığ, Turkey. Electronic address: .
Osmaniye D; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 26470 Eskişehir, Turkey; Anadolu University, Faculty of Pharmacy, Doping and Narcotic Compounds Analysis Laboratory, 26470 Eskişehir, Turkey.
Sağlik BN; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 26470 Eskişehir, Turkey; Anadolu University, Faculty of Pharmacy, Doping and Narcotic Compounds Analysis Laboratory, 26470 Eskişehir, Turkey.
Levent S; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 26470 Eskişehir, Turkey; Anadolu University, Faculty of Pharmacy, Doping and Narcotic Compounds Analysis Laboratory, 26470 Eskişehir, Turkey.
Özkay Y; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 26470 Eskişehir, Turkey; Anadolu University, Faculty of Pharmacy, Doping and Narcotic Compounds Analysis Laboratory, 26470 Eskişehir, Turkey.
Benkli K; Badakbas Pharmacy, Altintepe Street Koknarli 6/C Maltepe, 34840 Istanbul, Turkey.
Kaplancikli ZA; Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 26470 Eskişehir, Turkey.
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Źródło :
Bioorganic chemistry [Bioorg Chem] 2021 Dec; Vol. 117, pp. 105430. Date of Electronic Publication: 2021 Oct 16.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Novel Thiosemicarbazone Derivatives: In Vitro and In Silico Evaluation as Potential MAO-B Inhibitors.
Autorzy :
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Kurban B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
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Źródło :
Molecules (Basel, Switzerland) [Molecules] 2021 Nov 02; Vol. 26 (21). Date of Electronic Publication: 2021 Nov 02.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Design, Synthesis and Biological Evaluation of New N-Acyl Hydrazones with a Methyl Sulfonyl Moiety as Selective COX-2 Inhibitors.
Autorzy :
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Research Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Research Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Research Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Research Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
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Źródło :
Chemistry & biodiversity [Chem Biodivers] 2021 Nov; Vol. 18 (11), pp. e2100521. Date of Electronic Publication: 2021 Sep 29.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Novel thiazolyl-hydrazone derivatives including piperazine ring: synthesis, in vitro evaluation, and molecular docking as selective MAO-A inhibitor.
Autorzy :
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
Alaşan R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir26470, Turkey.
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Źródło :
Zeitschrift fur Naturforschung. C, Journal of biosciences [Z Naturforsch C J Biosci] 2021 Oct 21. Date of Electronic Publication: 2021 Oct 21.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Design, synthesis, in vitro and in silico studies of some novel thiazole-dihydrofuran derivatives as aromatase inhibitors.
Autorzy :
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Görgülü Ş; Medicinal Plant, Drug and Scientific Research and Application Center (AUBIBAM), 26470 Eskişehir, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey. Electronic address: .
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Źródło :
Bioorganic chemistry [Bioorg Chem] 2021 Sep; Vol. 114, pp. 105123. Date of Electronic Publication: 2021 Jun 25.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Synthesis of new hydrazone derivatives and evaluation of their monoamine oxidase inhibitory activity.
Autorzy :
Tok F; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Marmara University, Istanbul, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Ilgın S; Department of Pharmaceutical Toxicology, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Koçyiğit-Kaymakçıoğlu B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Marmara University, Istanbul, Turkey. Electronic address: .
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Źródło :
Bioorganic chemistry [Bioorg Chem] 2021 Sep; Vol. 114, pp. 105038. Date of Electronic Publication: 2021 Jun 01.
Typ publikacji :
Journal Article
Czasopismo naukowe
Tytuł :
Dithiocarbamate derivatives inhibit α-glucosidase through an apparent allosteric site on the enzyme.
Autorzy :
Ghani U; Clinical Biochemistry Unit, Department of Pathology, College of Medicine, King Saud University, Riyadh, Saudi Arabia.
Ashraf S; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Ul-Haq Z; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Mujamammi AH; Clinical Biochemistry Unit, Department of Pathology, College of Medicine, King Saud University, Riyadh, Saudi Arabia.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Demirci F; Department of Pharmacognosy, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Faculty of Pharmacy, Eastern Mediterranean University, Mersin, Turkey.
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
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Źródło :
Chemical biology & drug design [Chem Biol Drug Des] 2021 Aug; Vol. 98 (2), pp. 283-294. Date of Electronic Publication: 2021 Jun 19.
Typ publikacji :
Journal Article
MeSH Terms :
Glycoside Hydrolase Inhibitors/*chemistry
Thiocarbamates/*chemistry
alpha-Glucosidases/*chemistry
Allosteric Site ; Binding Sites ; Catalytic Domain ; Diabetes Mellitus/drug therapy ; Glycoside Hydrolase Inhibitors/metabolism ; Glycoside Hydrolase Inhibitors/therapeutic use ; Humans ; Hypoglycemic Agents/chemistry ; Hypoglycemic Agents/metabolism ; Hypoglycemic Agents/therapeutic use ; Kinetics ; Molecular Docking Simulation ; Structure-Activity Relationship ; Thiocarbamates/metabolism ; alpha-Glucosidases/metabolism
Czasopismo naukowe
Tytuł :
Novel 2,5-disubstituted-1,3,4-oxadiazole derivatives as MAO-B inhibitors: Synthesis, biological evaluation and molecular modeling studies.
Autorzy :
Tok F; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Marmara University, Istanbul, Turkey.
Uğraş Z; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Marmara University, Istanbul, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Koçyiğit-Kaymakçıoğlu B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Marmara University, Istanbul, Turkey. Electronic address: .
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Źródło :
Bioorganic chemistry [Bioorg Chem] 2021 Jul; Vol. 112, pp. 104917. Date of Electronic Publication: 2021 Apr 16.
Typ publikacji :
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms :
Monoamine Oxidase/*metabolism
Monoamine Oxidase Inhibitors/*pharmacology
Oxadiazoles/*pharmacology
Dose-Response Relationship, Drug ; Humans ; Models, Molecular ; Molecular Structure ; Monoamine Oxidase Inhibitors/chemical synthesis ; Monoamine Oxidase Inhibitors/chemistry ; Oxadiazoles/chemical synthesis ; Oxadiazoles/chemistry ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł :
Design, synthesis, biological evaluation, and docking studies of some novel chalcones as selective COX-2 inhibitors.
Autorzy :
Kaya Çavuşoğlu B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Zonguldak Bulent Ecevit University, Zonguldak, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Acar Çevik U; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
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Źródło :
Archiv der Pharmazie [Arch Pharm (Weinheim)] 2021 Mar; Vol. 354 (3), pp. e2000273. Date of Electronic Publication: 2020 Nov 27.
Typ publikacji :
Journal Article
MeSH Terms :
Drug Design*
Molecular Docking Simulation*
Chalcones/*pharmacology
Cyclooxygenase 2/*metabolism
Cyclooxygenase 2 Inhibitors/*pharmacology
Chalcones/chemical synthesis ; Chalcones/chemistry ; Cyclooxygenase 2 Inhibitors/chemical synthesis ; Cyclooxygenase 2 Inhibitors/chemistry ; Dose-Response Relationship, Drug ; Humans ; Molecular Structure ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł :
Synthesis of some new benzoxazole derivatives and investigation of their anticancer activities.
Autorzy :
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Korkut Çelikateş B; Department of Pharmaceutical Toxicology, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Sağlık BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Acar Çevik U; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Kaya Çavuşoğlu B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Bulent Ecevit University, 67600, Zonguldak, Turkey.
Ilgın S; Department of Pharmaceutical Toxicology, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey. Electronic address: .
Kaplancıklı ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470, Eskişehir, Turkey.
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Źródło :
European journal of medicinal chemistry [Eur J Med Chem] 2021 Jan 15; Vol. 210, pp. 112979. Date of Electronic Publication: 2020 Oct 31.
Typ publikacji :
Journal Article
MeSH Terms :
Antineoplastic Agents/*pharmacology
Benzoxazoles/*pharmacology
Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Benzoxazoles/chemical synthesis ; Benzoxazoles/chemistry ; Cell Proliferation/drug effects ; DNA, Neoplasm/antagonists & inhibitors ; DNA, Neoplasm/biosynthesis ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Humans ; Molecular Docking Simulation ; Molecular Structure ; Structure-Activity Relationship ; Tumor Cells, Cultured
Czasopismo naukowe

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