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Wyszukujesz frazę ""Kaplancikli ZA"" wg kryterium: Autor


Tytuł:
Synthesis and biological evaluation of novel 1,3,4-thiadiazole derivatives as possible anticancer agents
Autorzy:
Çevik Ulviye Acar
Osmaniye Derya
Levent Serkan
Sağlik Begüm Nurpelin
Çavuşoğlu Betül Kaya
Karaduman Abdullah Burak
Özkay Yusuf
Kaplancikli Zafer Asim
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Temat:
4-thiadiazole
anticancer activity
aromatase inhibitory activity
mtt assay
Pharmaceutical industry
HD9665-9675
Źródło:
Acta Pharmaceutica, Vol 70, Iss 4, Pp 499-513 (2020)
Opis pliku:
electronic resource
Relacje:
https://doaj.org/toc/1846-9558
Dostęp URL:
https://doaj.org/article/0297ca8d7ca049128a13d18cc4e1efe5  Link otwiera się w nowym oknie
Czasopismo naukowe
Tytuł:
The 4-(dimethylaminoalkyl)piperazine inhibitors of α-glucosidase: allosteric enzyme inhibition and identification of interacting chemical groups.
Autorzy:
Ghani U; Clinical Biochemistry Unit, Department of Pathology, College of Medicine, King Saud University, Riyadh, Saudi Arabia.
Ashraf S; Dr. Panjwani Center for Molecular Medicine & Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Ul Haq Z; Dr. Panjwani Center for Molecular Medicine & Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Demirci F; Department of Pharmacognosy, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Afzal S; Biomedical Research Laboratory, College of Medicine, Alfaisal University, Riyadh, Saudi Arabia.
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Źródło:
Turkish journal of chemistry [Turk J Chem] 2022 May 20; Vol. 46 (5), pp. 1484-1492. Date of Electronic Publication: 2022 May 20 (Print Publication: 2022).
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Dithiocarbamate derivatives inhibit α-glucosidase through an apparent allosteric site on the enzyme.
Autorzy:
Ghani U; Clinical Biochemistry Unit, Department of Pathology, College of Medicine, King Saud University, Riyadh, Saudi Arabia.
Ashraf S; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Ul-Haq Z; Dr. Panjwani Center for Molecular Medicine and Drug Research, International Center for Chemical and Biological Sciences, University of Karachi, Karachi, Pakistan.
Mujamammi AH; Clinical Biochemistry Unit, Department of Pathology, College of Medicine, King Saud University, Riyadh, Saudi Arabia.
Özkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
Demirci F; Department of Pharmacognosy, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.; Faculty of Pharmacy, Eastern Mediterranean University, Mersin, Turkey.
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey.
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Źródło:
Chemical biology & drug design [Chem Biol Drug Des] 2021 Aug; Vol. 98 (2), pp. 283-294. Date of Electronic Publication: 2021 Jun 19.
Typ publikacji:
Journal Article
MeSH Terms:
Glycoside Hydrolase Inhibitors/*chemistry
Thiocarbamates/*chemistry
alpha-Glucosidases/*chemistry
Allosteric Site ; Binding Sites ; Catalytic Domain ; Diabetes Mellitus/drug therapy ; Glycoside Hydrolase Inhibitors/metabolism ; Glycoside Hydrolase Inhibitors/therapeutic use ; Humans ; Hypoglycemic Agents/chemistry ; Hypoglycemic Agents/metabolism ; Hypoglycemic Agents/therapeutic use ; Kinetics ; Molecular Docking Simulation ; Structure-Activity Relationship ; Thiocarbamates/metabolism ; alpha-Glucosidases/metabolism
Czasopismo naukowe
Tytuł:
Synthesis and AChE-Inhibitory Activity of New Benzimidazole Derivatives.
Autorzy:
Acar Cevik U; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Saglik BN; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Levent S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Osmaniye D; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Kaya Cavuşoglu B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Ozkay Y; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .; Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26210 Eskişehir, Turkey. .
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2019 Feb 28; Vol. 24 (5). Date of Electronic Publication: 2019 Feb 28.
Typ publikacji:
Journal Article
MeSH Terms:
Acetylcholinesterase*/chemistry
Cholinesterase Inhibitors*/chemical synthesis
Cholinesterase Inhibitors*/chemistry
Molecular Docking Simulation*
Butyrylcholinesterase/*chemistry
GPI-Linked Proteins/antagonists & inhibitors ; GPI-Linked Proteins/chemistry ; Humans ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Novel 1-(2-pyrimidin-2-yl)piperazine derivatives as selective monoamine oxidase (MAO)-A inhibitors.
Autorzy:
Kaya B; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
Yurttaş L; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
Sağlik BN; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.; b Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
Levent S; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.; b Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
Özkay Y; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.; b Doping and Narcotic Compounds Analysis Laboratory, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
Kaplancikli ZA; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2017 Dec; Vol. 32 (1), pp. 193-202.
Typ publikacji:
Journal Article
MeSH Terms:
Monoamine Oxidase Inhibitors/*pharmacology
Piperazines/*pharmacology
Kinetics ; Molecular Docking Simulation ; Monoamine Oxidase/metabolism ; Monoamine Oxidase Inhibitors/chemistry ; Piperazines/chemistry ; Spectrum Analysis/methods
Czasopismo naukowe
Tytuł:
Synthesis and biological evaluation of some dibenzofuran-piperazine derivatives.
Autorzy:
Yurttaş L; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
Abu Mohsen U; b Department of Pharmaceutical Chemistry , Faculty of Pharmacy, Al-Azhar University , Gaza , Palestine , and.
Ozkan Y; c Department of Biochemistry , Faculty of Pharmacy, Gazi University , Ankara , Turkey.
Cobanoglu S; c Department of Biochemistry , Faculty of Pharmacy, Gazi University , Ankara , Turkey.
Levent S; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
Kaplancikli ZA; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2016 Dec; Vol. 31 (6), pp. 1177-83. Date of Electronic Publication: 2015 Nov 18.
Typ publikacji:
Journal Article
MeSH Terms:
Benzofurans/*chemistry
Piperazines/*chemical synthesis
Piperazines/*pharmacology
Piperazine ; Piperazines/chemistry ; Platelet Aggregation Inhibitors/pharmacology
Czasopismo naukowe
Tytuł:
Synthesis and evaluation of naphthalene-based thiosemicarbazone derivatives as new anticancer agents against LNCaP prostate cancer cells.
Autorzy:
Altintop MD; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
Sever B; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
Özdemir A; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
Kuş G; b Open Education Faculty , Anadolu University , Eskişehir , Turkey .
Oztopcu-Vatan P; c Department of Biology, Faculty of Arts and Sciences , and.
Kabadere S; d Department of Physiology, Faculty of Medicine , Eskisehir Osmangazi University , Eskişehir , Turkey.
Kaplancikli ZA; a Department of Pharmaceutical Chemistry, Faculty of Pharmacy , Anadolu University , Eskişehir , Turkey .
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2016; Vol. 31 (3), pp. 410-6. Date of Electronic Publication: 2015 Mar 31.
Typ publikacji:
Journal Article
MeSH Terms:
Antineoplastic Agents/*pharmacology
Naphthalenes/*pharmacology
Prostatic Neoplasms/*drug therapy
Prostatic Neoplasms/*pathology
Thiosemicarbazones/*pharmacology
Antineoplastic Agents/chemistry ; Apoptosis/drug effects ; Cell Proliferation/drug effects ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Flow Cytometry ; Humans ; Male ; Molecular Structure ; Naphthalenes/chemistry ; Structure-Activity Relationship ; Thiosemicarbazones/chemical synthesis ; Thiosemicarbazones/chemistry ; Tumor Cells, Cultured
Czasopismo naukowe
Tytuł:
Synthesis and evaluation of new thiadiazole derivatives as potential inhibitors of human carbonic anhydrase isozymes (hCA-I and hCA-II).
Autorzy:
Altintop MD; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Anadolu University , Eskisehir , Turkey .
Ozdemir A
Kucukoglu K
Turan-Zitouni G
Nadaroglu H
Kaplancikli ZA
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2015 Feb; Vol. 30 (1), pp. 32-7. Date of Electronic Publication: 2014 Mar 25.
Typ publikacji:
Journal Article
MeSH Terms:
Acetophenones/*chemistry
Carbonic Anhydrase I/*chemistry
Carbonic Anhydrase II/*chemistry
Carbonic Anhydrase Inhibitors/*chemistry
Thiadiazoles/*chemistry
Acetophenones/chemical synthesis ; Carbonic Anhydrase I/isolation & purification ; Carbonic Anhydrase II/isolation & purification ; Carbonic Anhydrase Inhibitors/chemical synthesis ; Chromatography, Affinity ; Enzyme Assays ; Erythrocytes/chemistry ; Erythrocytes/enzymology ; Humans ; Kinetics ; Structure-Activity Relationship ; Thiadiazoles/chemical synthesis
Czasopismo naukowe
Tytuł:
Synthesis, anticandidal activity and cytotoxicity of some tetrazole derivatives.
Autorzy:
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Graduate School of Health Sciences, Anadolu University , Eskisehir , Turkey .
Yurttaş L
Özdemir A
Turan-Zitouni G
Işcan G
Akalın G
Abu Mohsen U
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2014 Feb; Vol. 29 (1), pp. 43-8. Date of Electronic Publication: 2013 Jan 17.
Typ publikacji:
Journal Article
MeSH Terms:
Candida/*drug effects
Tetrazoles/*chemical synthesis
Tetrazoles/*pharmacology
Animals ; Magnetic Resonance Spectroscopy ; Mice ; Microbial Sensitivity Tests ; NIH 3T3 Cells ; Spectrometry, Mass, Fast Atom Bombardment
Czasopismo naukowe
Tytuł:
Synthesis and biological evaluation of some thiazole derivatives as new cholinesterase inhibitors.
Autorzy:
Turan-Zitouni G; Department of Pharmaceutical Chemistry, Anadolu University, Faculty of Pharmacy, Eskişehir, Turkey.
Ozdemir A
Kaplancikli ZA
Altintop MD
Temel HE
Çiftçi GA
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2013 Jun; Vol. 28 (3), pp. 509-14. Date of Electronic Publication: 2012 Feb 03.
Typ publikacji:
Journal Article
MeSH Terms:
Cholinesterase Inhibitors/*chemical synthesis
Cholinesterase Inhibitors/*pharmacology
Thiazoles/*chemistry
Acetylcholinesterase/metabolism ; Animals ; Butyrylcholinesterase/metabolism ; Chemistry Techniques, Synthetic ; Cholinesterase Inhibitors/chemistry ; Dose-Response Relationship, Drug ; Drug Evaluation, Preclinical/methods ; Magnetic Resonance Spectroscopy ; Mice ; Molecular Structure ; NIH 3T3 Cells/drug effects ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Synthesis and analgesic activity of some acetamide derivatives.
Autorzy:
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey. />Altintop MD
Turan-Zitouni G
Ozdemir A
Can OD
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2012 Apr; Vol. 27 (2), pp. 275-80. Date of Electronic Publication: 2011 Jun 10.
Typ publikacji:
Journal Article
MeSH Terms:
Acetamides/*chemical synthesis
Acetamides/*pharmacology
Analgesics/*chemical synthesis
Analgesics/*pharmacology
Pain/*drug therapy
Pain Measurement/*drug effects
Acetic Acid/toxicity ; Animals ; Magnetic Resonance Spectroscopy ; Male ; Mass Spectrometry ; Mice ; Molecular Structure ; Pain/chemically induced ; Spectrophotometry, Infrared ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Synthesis, antimicrobial activity and cytotoxicity of novel oxadiazole derivatives.
Autorzy:
Kaplancikli ZA; Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Anadolu University, Eskişehir, Turkey. />Altintop MD
Turan-Zitouni G
Ozdemir A
Ozic R
Akalin G
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2012 Feb; Vol. 27 (1), pp. 51-7. Date of Electronic Publication: 2011 May 03.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Bacterial Agents/*pharmacology
Bacteria/*drug effects
Oxadiazoles/*pharmacology
Animals ; Anti-Bacterial Agents/chemical synthesis ; Anti-Bacterial Agents/chemistry ; Cell Proliferation/drug effects ; Cells, Cultured ; Dose-Response Relationship, Drug ; Mice ; Microbial Sensitivity Tests ; Molecular Structure ; NIH 3T3 Cells ; Oxadiazoles/chemical synthesis ; Oxadiazoles/chemistry ; Stereoisomerism ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Synthesis of some oxadiazole derivatives as new anticandidal agents.
Autorzy:
Kaplancikli ZA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, 26470 Eskişehir, Turkey.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2011 Sep 07; Vol. 16 (9), pp. 7662-71. Date of Electronic Publication: 2011 Sep 07.
Typ publikacji:
Journal Article
MeSH Terms:
Antifungal Agents/*chemical synthesis
Candida albicans/*drug effects
Oxadiazoles/*chemical synthesis
Pyrimidines/*chemical synthesis
Antifungal Agents/pharmacology ; Microbial Sensitivity Tests ; Oxadiazoles/pharmacology ; Pyrimidines/chemistry ; Pyrimidines/pharmacology ; Sulfides/chemistry
Czasopismo naukowe
Tytuł:
Preparation of some pyrazoline derivatives and evaluation of their antifungal activities.
Autorzy:
Ozdemir A; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Anadolu University, Eskişehir, Turkey. />Turan-Zitouni G
Kaplancikli ZA
Revial G
Demirci F
Işcan G
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2010 Aug; Vol. 25 (4), pp. 565-71.
Typ publikacji:
Journal Article
MeSH Terms:
Antifungal Agents/*chemical synthesis
Pyrazoles/*chemical synthesis
Antifungal Agents/pharmacology ; Fungi/drug effects ; Magnetic Resonance Spectroscopy ; Mass Spectrometry ; Microbial Sensitivity Tests ; Molecular Structure ; Pyrazoles/pharmacology ; Structure-Activity Relationship
Czasopismo naukowe

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