Optimizing the Multimerization Properties of Quinoline-Based Allosteric HIV-1 Integrase Inhibitors.
Autorzy:
Sun J; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA. KesslJJ; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA.
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Źródło:
Viruses [Viruses] 2024 Jan 28; Vol. 16 (2). Date of Electronic Publication: 2024 Jan 28.
Multi-Substituted Quinolines as HIV-1 Integrase Allosteric Inhibitors.
Autorzy:
Dinh LP; Department of Chemistry, University of South Alabama, Mobile, AL 36688, USA. Sun J; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA. Glenn CD; Department of Chemistry, University of South Alabama, Mobile, AL 36688, USA. Patel K; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA. Pigza JA; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA. Donahue MG; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA. Yet L; Department of Chemistry, University of South Alabama, Mobile, AL 36688, USA. KesslJJ; Department of Chemistry and Biochemistry, University of Southern Mississippi, Hattiesburg, MS 39406, USA.
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Źródło:
Viruses [Viruses] 2022 Jul 02; Vol. 14 (7). Date of Electronic Publication: 2022 Jul 02.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, N.I.H., Extramural
HIV-1 Integrase-Targeted Short Peptides Derived from a Viral Protein R Sequence.
Autorzy:
Zhao XZ; Chemical Biology Laboratory, Center of Cancer Research, Frederick, MD 21702, USA. . Métifiot M; Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, MD 20892, USA. . Kiselev E; Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, MD 20892, USA. . KesslJJ; College of Pharmacy and Center for Retrovirus Research, The Ohio State University, Columbus, OH 43210, USA. Jacques.Kessl@usm.edu.; Department of Chemistry and Biochemistry, The University of Southern Mississippi, Hattiesburg, MS 39406, USA. Jacques.Kessl@usm.edu. Maddali K; Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, MD 20892, USA. . Marchand C; Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, MD 20892, USA. . Kvaratskhelia M; College of Pharmacy and Center for Retrovirus Research, The Ohio State University, Columbus, OH 43210, USA. .; Division of Infectious Diseases, University of Colorado School of Medicine, Aurora, CO 80045, USA. . Pommier Y; Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, MD 20892, USA. . Burke TR Jr; Chemical Biology Laboratory, Center of Cancer Research, Frederick, MD 21702, USA. .
A new class of multimerization selective inhibitors of HIV-1 integrase.
Autorzy:
Sharma A; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. Slaughter A; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. Jena N; Division of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. Feng L; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. KesslJJ; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. Fadel HJ; Department of Molecular Medicine & Division of Infectious Diseases, Mayo Clinic College of Medicine, Rochester, Minnesota, United States of America. Malani N; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America. Male F; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America. Wu L; Center for Retrovirus Research and Department of Veterinary Biosciences, The Ohio State University, Columbus, Ohio, United States of America. Poeschla E; Department of Molecular Medicine & Division of Infectious Diseases, Mayo Clinic College of Medicine, Rochester, Minnesota, United States of America. Bushman FD; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America. Fuchs JR; Division of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America. Kvaratskhelia M; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
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Źródło:
PLoS pathogens [PLoS Pathog] 2014 May 29; Vol. 10 (5), pp. e1004171. Date of Electronic Publication: 2014 May 29 (Print Publication: 2014).
KesslJJ; Center for Retrovirus Research and Comprehensive Cancer Center, College of Pharmacy, The Ohio State University, Columbus, OH 43210, USA; E-Mails: kessl. (J.J.K.); (C.J.M.); eidahl. (J.O.E.), shkriabai. (N.S.); (A.K.). McKee CJ Eidahl JO Shkriabai N Katz A Kvaratskhelia M
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Źródło:
Viruses [Viruses] 2009 Dec; Vol. 1 (3), pp. 713-36. Date of Electronic Publication: 2009 Nov 05.
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