- Tytuł:
- Novel Imbricatolic acid derivatives as protein tyrosine phosphatase-1B inhibitors: Design, synthesis, biological evaluation and molecular docking.
- Autorzy:
- Źródło:
- Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2016 Apr 15; Vol. 26 (8), pp. 1988-92. Date of Electronic Publication: 2016 Mar 02.
- Typ publikacji:
- Journal Article; Research Support, Non-U.S. Gov't
- MeSH Terms:
-
Drug Design*
Molecular Docking Simulation*
Diterpenes/*pharmacology
Enzyme Inhibitors/*chemical synthesis
Enzyme Inhibitors/*pharmacology
Protein Tyrosine Phosphatase, Non-Receptor Type 1/*antagonists & inhibitors
Cell Line ; Diterpenes/chemical synthesis ; Diterpenes/chemistry ; Dose-Response Relationship, Drug ; Enzyme Inhibitors/chemistry ; Humans ; Molecular Structure ; Protein Tyrosine Phosphatase, Non-Receptor Type 1/metabolism ; Recombinant Proteins/metabolism ; Structure-Activity Relationship
Czasopismo naukowe