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Wyszukujesz frazę ""Khan, Mohammad Faheem"" wg kryterium: Autor


Wyświetlanie 1-34 z 34
Tytuł:
Antioxidant constituents from Ribes glaciale Wall.: bioassay targeted in-vitro and in-silico evaluation.
Autorzy:
Singh R; Department of Chemistry, Government P.G. College Gopeshwar, Chamoli, Uttarakhand India.
Verma R; Department of Chemistry, Government P.G. College Gopeshwar, Chamoli, Uttarakhand India.
Sati N; Department of Pharmacetical Science, HNB Garhwal University (A Central University) Srinagar Garhwal, Uttarakhand, India.
Ansari WA; Department of Chemistry and Department of Biotechnology, Era University, Sarfarazganj, Hardoi Road, Lucknow, UP, India.
Khan MF; Department of Chemistry and Department of Biotechnology, Era University, Sarfarazganj, Hardoi Road, Lucknow, UP, India.
Źródło:
Natural product research [Nat Prod Res] 2024 Mar 10, pp. 1-4. Date of Electronic Publication: 2024 Mar 10.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Natural product-inspired synthesis of coumarin-chalcone hybrids as potential anti-breast cancer agents.
Autorzy:
Alhakamy NA; Department of Pharmaceutics, Faculty of Pharmacy, King Abdulaziz University, Jeddah, Saudi Arabia.; Mohamed Saeed Tamer Chair for Pharmaceutical Industries, Faculty of Pharmacy, King Abdulaziz University, Jeddah, Saudi Arabia.; Center of Excellence for Drug Research and Pharmaceutical Industries, King Abdulaziz University, Jeddah, Saudi Arabia.
Saquib M; Department of Chemistry, University of Allahabad, Prayagraj, India.
Sanobar; Department of Chemistry, Government Raza Post Graduate College, Rampur, India.; M. J. P. Rohilkhand University, Bareilly, India.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College, Era University, Lucknow, India.
Ansari WA; Department of Biotechnology, Era's Lucknow Medical College, Era University, Lucknow, India.
Arif DO; Mohamed Saeed Tamer Chair for Pharmaceutical Industries, Faculty of Pharmacy, King Abdulaziz University, Jeddah, Saudi Arabia.; Center of Excellence for Drug Research and Pharmaceutical Industries, King Abdulaziz University, Jeddah, Saudi Arabia.; Faculty of Medicine, Ibn Sina National College, Jeddah, Saudi Arabia.
Irfan M; Department of Medicine, Jawaharlal Nehru Medical College and Hospital, Aligarh Muslim University (AMU), Aligarh, India.
Khan MI; Departments of Biochemistry, Faculty of Science, King Abdulaziz University, Jeddah, Saudi Arabia.; Centre of Artificial Intelligence in Precision Medicine, King Abdulaziz University, Jeddah, Saudi Arabia.
Hussain MK; Department of Chemistry, Government Raza Post Graduate College, Rampur, India.; M. J. P. Rohilkhand University, Bareilly, India.
Źródło:
Frontiers in pharmacology [Front Pharmacol] 2023 Sep 06; Vol. 14, pp. 1231450. Date of Electronic Publication: 2023 Sep 06 (Print Publication: 2023).
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Pentafuhalol-B, a Phlorotannin from Brown Algae, Strongly Inhibits the PLK-1 Overexpression in Cancer Cells as Revealed by Computational Analysis.
Autorzy:
Ansari WA; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Sarfarazganj, Hardoi Road, Lucknow 226003, India.; Department of Chemistry, Era University, Sarfarazganj, Hardoi Road, Lucknow 226003, India.
Rab SO; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, King Khalid University, Abha 62529, Saudi Arabia.
Saquib M; Department of Chemistry, University of Allahabad, Prayagraj 211002, India.
Sarfraz A; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Sarfarazganj, Hardoi Road, Lucknow 226003, India.
Hussain MK; Department of Chemistry, Government Raza P.G. College, Rampur, M. J. P. Rohilkhand University, Bareilly 244901, India.
Akhtar MS; Department of Botany, Gandhi Faiz-e-Aam College, Shahjahanpur 242001, India.
Ahmad I; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, King Khalid University, Abha 62529, Saudi Arabia.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Sarfarazganj, Hardoi Road, Lucknow 226003, India.; Department of Chemistry, Era University, Sarfarazganj, Hardoi Road, Lucknow 226003, India.
Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Aug 03; Vol. 28 (15). Date of Electronic Publication: 2023 Aug 03.
Typ publikacji:
Journal Article
MeSH Terms:
Carcinoma, Non-Small-Cell Lung*
Lung Neoplasms*
Antineoplastic Agents*/pharmacology
Antineoplastic Agents*/chemistry
Humans ; Molecular Docking Simulation ; Cell Cycle Proteins/metabolism ; Cell Division
Czasopismo naukowe
Tytuł:
Drug repositioning to discover novel ornithine decarboxylase inhibitors against visceral leishmaniasis.
Autorzy:
Sheikh SY; Department of Chemistry, Integral University, Lucknow, India.
Ansari WA; Department of Biotechnology, Era University, Lucknow, India.
Hassan F; Department of Chemistry, Integral University, Lucknow, India.
Faruqui T; Department of Biosciences, Integral University, Lucknow, India.
Khan MF; Department of Biotechnology, Era University, Lucknow, India.
Akhter Y; Department of Biotechnology, Babasaheb Bhimrao Ambedkar University, Lucknow, India.
Khan AR; Department of Chemistry, Integral University, Lucknow, India.
Siddiqui MA; Chair for DNA Research, Zoology Department, College of Science, King Saud University, Riyadh, Saudi Arabia.
Al-Khedhairy AA; Chair for DNA Research, Zoology Department, College of Science, King Saud University, Riyadh, Saudi Arabia.
Nasibullah M; Department of Chemistry, Integral University, Lucknow, India.
Źródło:
Journal of molecular recognition : JMR [J Mol Recognit] 2023 Jul; Vol. 36 (7), pp. e3021. Date of Electronic Publication: 2023 May 15.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Leishmaniasis, Visceral*
Leishmania donovani*/metabolism
Humans ; Ornithine Decarboxylase Inhibitors/chemistry ; Ornithine Decarboxylase Inhibitors/pharmacology ; Drug Repositioning ; Molecular Docking Simulation ; Ornithine Decarboxylase/chemistry ; Ornithine Decarboxylase/metabolism ; Ornithine Decarboxylase/pharmacology ; Ligands ; Ceftaroline
Czasopismo naukowe
Tytuł:
Immunoinformatics Strategy to Develop a Novel Universal Multiple Epitope-Based COVID-19 Vaccine.
Autorzy:
Khamjan NA; Department of Medical Laboratories Technology, College of Applied Medical Sciences, Jazan University, Jazan 45142, Saudi Arabia.
Lohani M; Department of Emergency Medical Services, College of Applied Medical Sciences, Jazan University, Jazan 45142, Saudi Arabia.; Medical Research Centre, Jazan University, Jazan 45142, Saudi Arabia.
Khan MF; Department of Biotechnology, K.C.M.T., M. J. P. Rohilkhand University, Bareilly 243006, India.
Khan S; Department of Basic Dental and Medical Sciences, College of Dentistry, Hail University, Hail 2440, Saudi Arabia.
Algaissi A; Department of Medical Laboratories Technology, College of Applied Medical Sciences, Jazan University, Jazan 45142, Saudi Arabia.; Medical Research Centre, Jazan University, Jazan 45142, Saudi Arabia.
Źródło:
Vaccines [Vaccines (Basel)] 2023 Jun 12; Vol. 11 (6). Date of Electronic Publication: 2023 Jun 12.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
An ultrasound assisted, ionic liquid-molecular iodine synergy driven efficient green synthesis of pyrrolobenzodiazepine-triazole hybrids as potential anticancer agents.
Autorzy:
Saquib M; Department of Chemistry, University of Allahabad, Prayagraj, Uttar Pradesh, India.
Ahamad S; Department of Chemistry, Aligarh Muslim University, Aligarh, Uttar Pradesh, India.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College, Era University, Lucknow, Uttar Pradesh, India.
Khan MI; Department of Biochemistry, Faculty of Science, King Abdulaziz University, Jeddah, Saudi Arabia.; Centre of Artificial Intelligence in Precision Medicine, King Abdulaziz University, Jeddah, Saudi Arabia.
Hussain MK; Department of Chemistry, Govt. Raza P.G. College, Rampur, Uttar Pradesh, India.; M.J.P Rohilkahand University, Bareilly, Uttar Pradesh, India.
Źródło:
Frontiers in pharmacology [Front Pharmacol] 2023 May 05; Vol. 14, pp. 1168566. Date of Electronic Publication: 2023 May 05 (Print Publication: 2023).
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Interaction of Bioactive Compounds of Moringa oleifera Leaves with SARS-CoV-2 Proteins to Combat COVID-19 Pathogenesis: a Phytochemical and In Silico Analysis.
Autorzy:
Siddiqui S; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, 226003, India. .
Upadhyay S; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, 226003, India.
Ahmad R; Department of Biochemistry, Era's Lucknow Medical College and Hospital, Era University, Lucknow, India.
Barkat MA; Department of Pharmaceutics, College of Pharmacy, University of Hafr Al-Batin, Al Jamiah, Hafr Al Batin, 39524, Saudi Arabia.
Jamal A; Health and Basic Science Research Centre, Majmaah University, Majmaah, 11952, Saudi Arabia.; Department of Biology, College of Science, Al-Zulfi, Majmaah University, Majmaah, 11952, Riyadh Region, Saudi Arabia.
Alothaim AS; Department of Biology, College of Science, Al-Zulfi, Majmaah University, Majmaah, 11952, Riyadh Region, Saudi Arabia.
Hassan MZ; Department of Pharmaceutical Chemistry, College of Pharmacy, King Khalid University, Abha, Saudi Arabia.
Rahman MA; Department of Pharmaceutics and Industrial Pharmacy, College of Pharmacy, Taif University, Taif, 21944, Saudi Arabia.
Arshad M; Department of Zoology, Aligarh Muslim University, Aligarh, India.
Ahamad T; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, 226003, India.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, 226003, India.
Shankar H; Research Cell, Era's Lucknow Medical College and Hospital, Lucknow, India.
Ali M; Department of Pharmacognosy, College of Pharmacy, Jazan University, Jazan, Saudi Arabia.
Kaleem S; Avadh Institute of Medical Technologies & Hospital, Lucknow, India.
Ahmad J; Department of Microbiology, Era's Lucknow Medical College and Hospital, Lucknow, India.
Źródło:
Applied biochemistry and biotechnology [Appl Biochem Biotechnol] 2022 Dec; Vol. 194 (12), pp. 5918-5944. Date of Electronic Publication: 2022 Jul 15.
Typ publikacji:
Journal Article
MeSH Terms:
Moringa oleifera*
COVID-19 Drug Treatment*
Humans ; SARS-CoV-2 ; Angiotensin-Converting Enzyme 2 ; beta-Tocopherol ; Phytochemicals/pharmacology ; Plant Leaves ; Molecular Dynamics Simulation ; Plant Extracts/pharmacology ; Protein Binding
Czasopismo naukowe
Tytuł:
Molecular Docking and Dynamics Simulation Revealed Ivermectin as Potential Drug against Schistosoma -Associated Bladder Cancer Targeting Protein Signaling: Computational Drug Repositioning Approach.
Autorzy:
Siddiqui AJ; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College, Era University, Lucknow 226003, India.
Hamadou WS; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.
Goyal M; Molecular Parasitology and Immunology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Jahan S; Department of Medical Laboratory Sciences, College of Applied Medical Sciences, Majmaah University, Al Majmaah 11952, Saudi Arabia.
Jamal A; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.
Ashraf SA; Department of Clinical Nutrition, College of Applied Medial Sciences, University of Hail, Hail 2440, Saudi Arabia.
Sharma P; Molecular Parasitology and Immunology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.; Program in Cellular and Molecular Medicine, Boston Children's Hospital, Boston, MA 02115, USA.
Sachidanandan M; Department of Oral Radiology, College of Dentistry, University of Hail, Hail 2440, Saudi Arabia.
Badraoui R; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.; Section of Histology-Cytology, Medicine Faculty of Tunis, University of Tunis El Manar, Tunis 1017, Tunisia.
Chaubey KK; Department of Biotechnology, Academic Block VI, GLA University, Mathura 281406, India.
Snoussi M; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.; Laboratory of Genetics, Biodiversity and Valorization of Bio-Resources (LR11ES41), University of Monastir, Higher Institute of Biotechnology of Monastir, Avenue Tahar Haddas BP74, Monastir 5000, Tunisia.
Adnan M; Department of Biology, College of Science, University of Hail, Hail 2440, Saudi Arabia.
Źródło:
Medicina (Kaunas, Lithuania) [Medicina (Kaunas)] 2021 Oct 03; Vol. 57 (10). Date of Electronic Publication: 2021 Oct 03.
Typ publikacji:
Journal Article
MeSH Terms:
Pharmaceutical Preparations*
Urinary Bladder Neoplasms*/drug therapy
Animals ; Drug Repositioning ; Humans ; Ivermectin/pharmacology ; Molecular Docking Simulation ; Schistosoma haematobium ; Vascular Endothelial Growth Factor A
Czasopismo naukowe
Tytuł:
Unmodified household coffee maker assisted extraction and purification of anticancer agents from Dillenia indica fruits.
Autorzy:
Khan MA; Research Unit, Era's Lucknow Medical College & Hospital, Era University, Lucknow, UP, India.
Ahamad T; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, UP, India.
Saquib M; Department of Chemistry, University of Allahabad, Allahabad, UP, India.
Hussain MK; Department of Chemistry, Government Raza Post Graduate College, Rampur, UP, India.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, UP, India.; Department of Chemistry, Era University, Lucknow, UP, India.
Źródło:
Natural product research [Nat Prod Res] 2021 Mar; Vol. 35 (6), pp. 984-987. Date of Electronic Publication: 2019 May 28.
Typ publikacji:
Journal Article
MeSH Terms:
Household Articles*
Antineoplastic Agents/*isolation & purification
Dilleniaceae/*chemistry
Fruit/*chemistry
Antineoplastic Agents/chemistry ; Antineoplastic Agents/pharmacology ; Cell Line, Tumor ; Coffee ; Humans ; Plant Extracts/chemistry
Czasopismo naukowe
Tytuł:
Abatement of neurobehavioral and neurochemical dysfunctions in cerebral ischemia/reperfusion injury by Tetrapleura tetraptera fruit extract.
Autorzy:
Saliu IO; Phytomedicine, Biochemical Pharmacology and Toxicology Research Laboratories, Department of Biochemistry, School of Sciences, The Federal University of Technology, Akure 340001, Nigeria; Department of System Neuroscience, National Brain Research Centre, Manesar 122052, Haryana, India.
Amoo ZA; Phytomedicine, Biochemical Pharmacology and Toxicology Research Laboratories, Department of Biochemistry, School of Sciences, The Federal University of Technology, Akure 340001, Nigeria.
Khan MF; Department of Biotechnology, Era's Lucknow Medical College, Era University, Hardoi Road, Lucknow, 226003, UP, India.
Olaleye MT; Phytomedicine, Biochemical Pharmacology and Toxicology Research Laboratories, Department of Biochemistry, School of Sciences, The Federal University of Technology, Akure 340001, Nigeria.
Rema V; Department of System Neuroscience, National Brain Research Centre, Manesar 122052, Haryana, India.
Akinmoladun AC; Phytomedicine, Biochemical Pharmacology and Toxicology Research Laboratories, Department of Biochemistry, School of Sciences, The Federal University of Technology, Akure 340001, Nigeria. Electronic address: .
Źródło:
Journal of ethnopharmacology [J Ethnopharmacol] 2021 Jan 10; Vol. 264, pp. 113284. Date of Electronic Publication: 2020 Aug 22.
Typ publikacji:
Journal Article
MeSH Terms:
Fruit*
Tetrapleura*
Brain Ischemia/*drug therapy
Open Field Test/*drug effects
Plant Extracts/*therapeutic use
Reperfusion Injury/*drug therapy
Animals ; Brain Ischemia/metabolism ; Brain Ischemia/psychology ; Dose-Response Relationship, Drug ; Male ; Open Field Test/physiology ; Plant Extracts/isolation & purification ; Plant Extracts/pharmacology ; Rats ; Rats, Wistar ; Reperfusion Injury/metabolism ; Reperfusion Injury/psychology ; Water-Electrolyte Balance/drug effects ; Water-Electrolyte Balance/physiology
Czasopismo naukowe
Tytuł:
Specioside (SS) & verminoside (VS) (Iridoid glycosides): isolation, characterization and comparable quantum chemical studies using density functional theory (DFT).
Autorzy:
Saini M; Department of Chemistry, University of Lucknow, Lucknow, 226007, Uttar Pradesh, India.
Sangwan R; Department of Chemistry, University of Lucknow, Lucknow, 226007, Uttar Pradesh, India.
Khan MF; Department of Biotechnology, Era Medical College, Era University, Lucknow, 226003, Uttar Pradesh, India.
Kumar A; Department of Chemistry, University of Lucknow, Lucknow, 226007, Uttar Pradesh, India.
Verma R; Department of Chemistry, University of Lucknow, Lucknow, 226007, Uttar Pradesh, India.
Jain S; Department of Chemistry, University of Lucknow, Lucknow, 226007, Uttar Pradesh, India.
Źródło:
Heliyon [Heliyon] 2019 Jan 11; Vol. 5 (1), pp. e01118. Date of Electronic Publication: 2019 Jan 11 (Print Publication: 2019).
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
In vitro and in vivo antidiabetic effect of extracts of Melia azedarach, Zanthoxylum alatum , and Tanacetum nubigenum .
Autorzy:
Khan MF; Department of Biotechnology, Era's Lucknow Medical College & Hospital, Era University, Lucknow, India.
Rawat AK; Biochemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow, India.
Khatoon S; Department of Botany, D. N. (P.G.) College, Meerut, India.
Hussain MK; Department of Chemistry Govt. Raza Post Graduate College, Rampur, India.
Mishra A; Biochemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow, India.
Negi DS; Department of Chemistry, HNB Garhwal University, Srinagar, India.
Źródło:
Integrative medicine research [Integr Med Res] 2018 Jun; Vol. 7 (2), pp. 176-183. Date of Electronic Publication: 2018 Mar 27.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Novel Imbricatolic acid derivatives as protein tyrosine phosphatase-1B inhibitors: Design, synthesis, biological evaluation and molecular docking.
Autorzy:
Khan MF; Department of Chemistry, University of Lucknow, Lucknow 226007, Uttar Pradesh, India.
Azad CS; 'Hygeia', Center of Excellences in Pharmaceutical Sciences (CEPS), Guru Govind Singh Indraprastha University, Sec 16-C, Dwarka, New Delhi 110078, India.
Kumar A; Department of Chemistry, University of Lucknow, Lucknow 226007, Uttar Pradesh, India.
Saini M; Department of Chemistry, University of Lucknow, Lucknow 226007, Uttar Pradesh, India.
Narula AK; 'Hygeia', Center of Excellences in Pharmaceutical Sciences (CEPS), Guru Govind Singh Indraprastha University, Sec 16-C, Dwarka, New Delhi 110078, India.
Jain S; Department of Chemistry, University of Lucknow, Lucknow 226007, Uttar Pradesh, India. Electronic address: .
Źródło:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2016 Apr 15; Vol. 26 (8), pp. 1988-92. Date of Electronic Publication: 2016 Mar 02.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Design*
Molecular Docking Simulation*
Diterpenes/*pharmacology
Enzyme Inhibitors/*chemical synthesis
Enzyme Inhibitors/*pharmacology
Protein Tyrosine Phosphatase, Non-Receptor Type 1/*antagonists & inhibitors
Cell Line ; Diterpenes/chemical synthesis ; Diterpenes/chemistry ; Dose-Response Relationship, Drug ; Enzyme Inhibitors/chemistry ; Humans ; Molecular Structure ; Protein Tyrosine Phosphatase, Non-Receptor Type 1/metabolism ; Recombinant Proteins/metabolism ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Osteogenic activity of natural diterpenoids isolated from Cupressus sempervirens fruits in calvarial derived osteoblast cells via differentiation and mineralization.
Autorzy:
Khan MF; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Dev K; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Lahiri S; Endocrinology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Dixit M; Endocrinology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Trivedi R; Endocrinology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Singh D; Endocrinology Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Maurya R; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India. Electronic address: .
Źródło:
Phytomedicine : international journal of phytotherapy and phytopharmacology [Phytomedicine] 2014 Dec 15; Vol. 21 (14), pp. 1794-800. Date of Electronic Publication: 2014 Nov 06.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Cupressus/*chemistry
Diterpenes/*pharmacology
Osteoblasts/*drug effects
Osteogenesis/*drug effects
Animals ; Bone Morphogenetic Protein 2/metabolism ; Calcification, Physiologic/drug effects ; Cell Differentiation/drug effects ; Cells, Cultured ; Core Binding Factor Alpha 1 Subunit/metabolism ; Female ; Fruit/chemistry ; Mice ; Mice, Inbred BALB C ; Molecular Structure ; Ovariectomy ; Skull/cytology
Czasopismo naukowe
Tytuł:
Bioactivity-guided chemical analysis of Melia azedarach L. (Meliaceae), displaying antidiabetic activity.
Autorzy:
Khan MF; Department of Chemistry, HNB Garhwal University, Srinagar (Garhwal) 246174, Uttarakhand, India.
Rawat AK; Biochemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow 226031, India.
Pawar B; Department of Chemistry, HNB Garhwal University, Srinagar (Garhwal) 246174, Uttarakhand, India.
Gautam S; Biochemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow 226031, India.
Srivastava AK; Biochemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow 226031, India.
Negi DS; Department of Chemistry, HNB Garhwal University, Srinagar (Garhwal) 246174, Uttarakhand, India. Electronic address: devendra_.
Źródło:
Fitoterapia [Fitoterapia] 2014 Oct; Vol. 98, pp. 98-103. Date of Electronic Publication: 2014 Jul 22.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Hypoglycemic Agents/*chemistry
Melia azedarach/*chemistry
Protein Tyrosine Phosphatase, Non-Receptor Type 1/*antagonists & inhibitors
Triterpenes/*chemistry
Animals ; Cell Line ; Enzyme Inhibitors/chemistry ; Enzyme Inhibitors/isolation & purification ; Fruit/chemistry ; Humans ; Mice ; Molecular Structure ; Plant Leaves/chemistry ; Triterpenes/isolation & purification
Czasopismo naukowe
Tytuł:
Design and synthesis of lupeol analogues and their glucose uptake stimulatory effect in L6 skeletal muscle cells.
Autorzy:
Khan MF; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Maurya CK; Biochemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Dev K; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India; Academy of Scientific and Innovative Research, New Delhi 110001, India.
Arha D; Biochemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India; Academy of Scientific and Innovative Research, New Delhi 110001, India.
Rai AK; Biochemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India.
Tamrakar AK; Biochemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India; Academy of Scientific and Innovative Research, New Delhi 110001, India.
Maurya R; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226031, India; Academy of Scientific and Innovative Research, New Delhi 110001, India. Electronic address: .
Źródło:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2014 Jun 15; Vol. 24 (12), pp. 2674-9. Date of Electronic Publication: 2014 Apr 24.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Drug Design*
Hypoglycemic Agents/*chemical synthesis
Hypoglycemic Agents/*pharmacology
Muscle, Skeletal/*drug effects
Pentacyclic Triterpenes/*chemical synthesis
Pentacyclic Triterpenes/*pharmacology
Biological Transport ; Carbohydrate Metabolism/genetics ; Cells, Cultured ; Dose-Response Relationship, Drug ; Glucose/metabolism ; Humans ; Hypoglycemic Agents/chemistry ; Molecular Structure ; Pentacyclic Triterpenes/chemistry ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Synthesis of novel imbricatolic acid analogues via insertion of N-substituted piperazine at C-15/C-19 positions, displaying glucose uptake stimulation in L6 skeletal muscle cells.
Autorzy:
Khan MF; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, CSIR, Lucknow 226001, India.
Kumar P
Pandey J
Srivastava AK
Tamrakar AK
Maurya R
Źródło:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2012 Jul 15; Vol. 22 (14), pp. 4636-9. Date of Electronic Publication: 2012 Jun 05.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Diterpenes/*chemistry
Glucose/*metabolism
Muscle Cells/*drug effects
Muscle, Skeletal/*drug effects
Piperazines/*chemistry
Animals ; Cell Line ; Diterpenes/pharmacology ; Molecular Structure ; Muscle Cells/metabolism ; Muscle, Skeletal/metabolism ; Piperazine ; Rats ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Chemical constituents of Kigelia pinnata twigs and their GLUT4 translocation modulatory effect in skeletal muscle cells.
Autorzy:
Khan MF; Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow 226 001, India.
Dixit P
Jaiswal N
Tamrakar AK
Srivastava AK
Maurya R
Źródło:
Fitoterapia [Fitoterapia] 2012 Jan; Vol. 83 (1), pp. 125-9. Date of Electronic Publication: 2011 Oct 15.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Bignoniaceae/*chemistry
Glucose Transporter Type 4/*metabolism
Muscle, Skeletal/*drug effects
Muscle, Skeletal/*metabolism
Plant Extracts/*chemistry
Plant Extracts/*pharmacology
Animals ; Glucose Transporter Type 4/genetics ; Molecular Structure ; Muscle Fibers, Skeletal/drug effects ; Protein Transport ; Rats
Czasopismo naukowe
Tytuł:
Aza-annulation on the 16-dehydropregnenolone, via tandem intermolecular aldol process and intramolecular Michael addition.
Autorzy:
Kumar M; Medicinal and Process Chemistry Division, Central Drug Research Institute, CSIR, Lucknow 226 001, India.
Rawat P
Khan MF
Rawat AK
Srivastava AK
Maurya R
Źródło:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2011 Apr 15; Vol. 21 (8), pp. 2232-7. Date of Electronic Publication: 2011 Mar 04.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Aldehydes/*chemistry
Aza Compounds/*chemistry
Dipeptidyl Peptidase 4/*chemistry
Dipeptidyl-Peptidase IV Inhibitors/*chemistry
Pregnenolone/*analogs & derivatives
Amines/chemistry ; Cyclization ; Dipeptidyl Peptidase 4/metabolism ; Dipeptidyl-Peptidase IV Inhibitors/chemical synthesis ; Dipeptidyl-Peptidase IV Inhibitors/pharmacology ; Pregnenolone/chemical synthesis ; Pregnenolone/chemistry ; Pregnenolone/pharmacology
Czasopismo naukowe
Tytuł:
Phenolic glycosides from Dodecadenia grandiflora and their glucose-6-phosphatase inhibitory activity.
Autorzy:
Kumar M; Medicinal and Process Chemistry Division, Central Drug Research Institute, CSIR, Lucknow 226 001, India.
Rawat P
Khan MF
Tamarkar AK
Srivastava AK
Arya KR
Maurya R
Źródło:
Fitoterapia [Fitoterapia] 2010 Sep; Vol. 81 (6), pp. 475-9. Date of Electronic Publication: 2010 Jan 15.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Glucose-6-Phosphatase/*antagonists & inhibitors
Glycosides/*isolation & purification
Lauraceae/*chemistry
Phenols/*isolation & purification
Enzyme Inhibitors/chemistry ; Enzyme Inhibitors/isolation & purification ; Glycosides/chemistry ; Inhibitory Concentration 50 ; Molecular Structure ; Phenols/chemistry ; Plant Leaves/chemistry
Czasopismo naukowe
    Wyświetlanie 1-34 z 34

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