- Tytuł:
- Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis.
- Autorzy:
- Źródło:
- Nature medicine [Nat Med] 2013 Sep; Vol. 19 (9), pp. 1157-60. Date of Electronic Publication: 2013 Aug 04.
- Typ publikacji:
- Journal Article; Research Support, Non-U.S. Gov't
- MeSH Terms:
-
Adenosine Triphosphate/*biosynthesis
Electron Transport Complex III/*antagonists & inhibitors
Extensively Drug-Resistant Tuberculosis/*drug therapy
Imidazoles/*pharmacology
Mycobacterium tuberculosis/*drug effects
Piperidines/*pharmacology
Pyridines/*pharmacology
Animals ; Cell Proliferation/drug effects ; Disease Models, Animal ; Drug Evaluation, Preclinical ; Electron Transport Complex III/genetics ; Imidazoles/pharmacokinetics ; Mice ; Mice, Inbred BALB C ; Piperidines/pharmacokinetics ; Pyridines/pharmacokinetics ; Rats ; Rats, Sprague-Dawley
Czasopismo naukowe