- Tytuł :
-
Synthesis and Characterization of Fluorine-18-Labeled N -(4-Chloro-3-((fluoromethyl- d
2 )thio)phenyl)picolinamide for Imaging of mGluR4 in Brain. - Autorzy :
- Źródło :
- Journal of medicinal chemistry [J Med Chem] 2020 Mar 26; Vol. 63 (6), pp. 3381-3389. Date of Electronic Publication: 2020 Mar 04.
- Typ publikacji :
- Journal Article; Research Support, N.I.H., Extramural
- MeSH Terms :
-
Picolines /*pharmacology
Radiopharmaceuticals/*pharmacology
Receptors, Metabotropic Glutamate/*analysis
Animals ; Brain/metabolism ; Drug Stability ; Fluorine Radioisotopes/chemistry ; Ligands ; Male ; Microsomes, Liver/metabolism ;Picolines /chemical synthesis ;Picolines /pharmacokinetics ; Positron-Emission Tomography ; Radiopharmaceuticals/chemical synthesis ; Radiopharmaceuticals/pharmacokinetics ; Rats, Sprague-Dawley ; Receptors, Metabotropic Glutamate/agonists ; Receptors, Metabotropic Glutamate/metabolism -
Czasopismo naukowe