Temat: "Propionates" - OpacWWW

Skocz do pozycji: 1.

Tytuł:: Development a novel robust method to enhance the solubility of Oxaprozin as nonsteroidal anti-inflammatory drug based on machine-learning.
Autorzy:: Abdelbasset WK; Department of Health and Rehabilitation Sciences, College of Applied Medical Sciences, Prince Sattam Bin Abdulaziz University, P.O. Box. 173, Al-Kharj, 11942, Saudi Arabia. .; Department of Physical Therapy, Kasr Al-Aini Hospital, Cairo University, Giza, 12613, Egypt. .
Elkholi SM; Department of Rehabilitation Sciences, College of Health and Rehabilitation Sciences, Princess Nourah Bint Abdulrahman University, P.O. Box. 84428, 11671, Riyadh, Saudi Arabia.
Ismail KA; Department of Clinical Laboratory Sciences, College of Applied Medical Sciences, Taif University, P.O.BOX.11099, Taif, 21944, Saudi Arabia.
Alshehri S; Department of Pharmaceutics and Industrial Pharmacy, College of Pharmacy, Taif University, P.O.Box 11099, Taif, 21944, Saudi Arabia.
Alobaida A; Department of Pharmaceutics, College of Pharmacy, University of Hail, Hail, 81442, Saudi Arabia.
Huwaimel B; Department of Pharmaceutical Chemistry, College of Pharmacy, University of Hail, Hail, 81442, Saudi Arabia.
Alatawi AD; Department of Clinical Pharmacy, College of Pharmacy, Jouf University, Sakaka, Al-Jouf, Saudi Arabia.
Alsubaiyel AM; Department of Pharmaceutics, College of Pharmacy, Qassim University, Buraidah, 52571, Saudi Arabia. .
Venkatesan K; Department of Pharmaceutical Chemistry, College of Pharmacy, King Khalid University, Abha, 62529, Kingdom of Saudi Arabia.
Abourehab MAS; Department of Pharmaceutics, College of Pharmacy, Umm Al-Qura University, Makkah, 21955, Saudi Arabia. .; Department of Pharmaceutics and Industrial Pharmacy, Faculty of Pharmacy, Minia University, Minia, 61519, Egypt. .; Pokaż więcej
Źródło:: Scientific reports [Sci Rep] 2022 Jul 30; Vol. 12 (1), pp. 13138. Date of Electronic Publication: 2022 Jul 30.
Typ publikacji:: Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:: Anti-Inflammatory Agents, Non-Steroidal*
Propionates*
Humans ; Machine Learning ; Oxaprozin ; Solubility

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 2.

Tytuł:: Anti-tumor effects of a nonsteroidal anti-inflammatory drug zaltoprofen on chondrosarcoma via activating peroxisome proliferator-activated receptor gamma and suppressing matrix metalloproteinase-2 expression.
Autorzy:: Higuchi T; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Takeuchi A; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Munesue S; Department of Biochemistry and Molecular Vascular Biology, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8640, Japan.
Yamamoto N; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Hayashi K; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Kimura H; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Miwa S; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Inatani H; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Shimozaki S; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Kato T; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Aoki Y; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Abe K; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Taniguchi Y; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Aiba H; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Murakami H; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.
Harashima A; Department of Biochemistry and Molecular Vascular Biology, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8640, Japan.
Yamamoto Y; Department of Biochemistry and Molecular Vascular Biology, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8640, Japan.
Tsuchiya H; Department of Orthopaedic Surgery, Kanazawa University Graduate School of Medical Sciences, 13-1 Takara-machi, Kanazawa, 920-8641, Japan.; Pokaż więcej
Źródło:: Cancer medicine [Cancer Med] 2018 May; Vol. 7 (5), pp. 1944-1954. Date of Electronic Publication: 2018 Mar 23.
Typ publikacji:: Case Reports; Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:: Anti-Inflammatory Agents, Non-Steroidal/*administration & dosage
Benzopyrans/*administration & dosage
Bone Neoplasms/*drug therapy
Chondrosarcoma/*drug therapy
Matrix Metalloproteinase 2/*genetics
PPAR gamma/*genetics
Propionates/*administration & dosage
Adult ; Anti-Inflammatory Agents, Non-Steroidal/pharmacology ; Benzopyrans/pharmacology ; Bone Neoplasms/genetics ; Bone Neoplasms/metabolism ; Bone Neoplasms/surgery ; Cell Line, Tumor ; Cell Movement ; Cell Proliferation/drug effects ; Cell Survival/drug effects ; Chondrosarcoma/genetics ; Chondrosarcoma/metabolism ; Chondrosarcoma/surgery ; Gene Expression Regulation, Neoplastic/drug effects ; Humans ; Male ; Neck ; PPAR gamma/metabolism ; Promoter Regions, Genetic ; Propionates/pharmacology ; Treatment Outcome

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 3.

Tytuł:: Preparation, optimization, and evaluation of Zaltoprofen-loaded microemulsion and microemulsion-based gel for transdermal delivery.
Autorzy:: Mishra R; a Department of Quality Assurance and.
Prabhavalkar KS; b Department of Pharmacology , SVKM's Dr. Bhanuben Nanavati College of Pharmacy , Mumbai , Maharashtra , India.
Bhatt LK; b Department of Pharmacology , SVKM's Dr. Bhanuben Nanavati College of Pharmacy , Mumbai , Maharashtra , India.; Pokaż więcej
Źródło:: Journal of liposome research [J Liposome Res] 2016 Dec; Vol. 26 (4), pp. 297-306. Date of Electronic Publication: 2016 Jan 19.
Typ publikacji:: Journal Article
MeSH Terms:: Drug Delivery Systems*
Analgesics/*administration & dosage
Anti-Inflammatory Agents, Non-Steroidal/*administration & dosage
Benzopyrans/*administration & dosage
Propionates/*administration & dosage
Administration, Cutaneous ; Analgesics/pharmacokinetics ; Analgesics/pharmacology ; Animals ; Anti-Inflammatory Agents, Non-Steroidal/pharmacokinetics ; Anti-Inflammatory Agents, Non-Steroidal/pharmacology ; Benzopyrans/pharmacokinetics ; Benzopyrans/pharmacology ; Chemistry, Pharmaceutical ; Disease Models, Animal ; Emulsions/administration & dosage ; Emulsions/chemistry ; Emulsions/pharmacokinetics ; Gels/administration & dosage ; Gels/chemistry ; Gels/pharmacokinetics ; Inflammation/drug therapy ; Kinetics ; Pain/drug therapy ; Propionates/pharmacokinetics ; Propionates/pharmacology ; Rats ; Rats, Wistar ; Skin/drug effects ; Skin Absorption/drug effects ; Surface-Active Agents/administration & dosage ; Surface-Active Agents/chemistry ; Surface-Active Agents/pharmacokinetics

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 4.

Tytuł:: In Silico Evaluation of Ibuprofen and Two Benzoylpropionic Acid Derivatives with Potential Anti-Inflammatory Activity.
Autorzy:: Bittencourt JAHM; Graduate Program of Pharmaceutical Innovation, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .
Neto MFA; Laboratory of Molecular Modeling, State University of Feira de Santana, Feira de Santana-BA 44036-900, Brazil. .
Lacerda PS; Laboratory of Bioinformatics and Molecular Modeling, School of Pharmacy, Federal University of Bahia, Barão de Jeremoabo Street, Salvador 40170-115, BA, Brazil. .
Bittencourt RCVS; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .
Silva RC; Computational Laboratory of Pharmaceutical Chemistry, University of Sao Paulo, Av. Prof. do Café, s/n - Monte Alegre, Ribeirão Preto, São Paulo 14040-903, Brazil. .
Lobato CC; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Nucleus of Studies and Selection of Bioactive Molecules, Institute of Health Sciences, Federal University of Pará, Belém-PA 66075-110, Brazil. .
Silva LB; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .
Leite FHA; Laboratory of Molecular Modeling, State University of Feira de Santana, Feira de Santana-BA 44036-900, Brazil. .
Zuliani JP; Laboratory Cellular Immunology Applied to Health, Oswaldo Cruz Foundation, FIOCRUZ Rondônia, Rua da Beira, 7671 BR-364, Porto Velho-RO 78912-000, Brazil. .
Rosa JMC; Department of Pharmaceutical and Organic Chemistry, Faculty of Pharmacy, Institute of Biosanitary Research ibs.GRANADA. University of Granada, 18071 Granada, Spain. .
Borges RS; Graduate Program of Pharmaceutical Innovation, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Nucleus of Studies and Selection of Bioactive Molecules, Institute of Health Sciences, Federal University of Pará, Belém-PA 66075-110, Brazil. .
Santos CBR; Graduate Program of Pharmaceutical Innovation, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Laboratory of Modeling and Computational Chemistry, Department of Biological and Health Sciences, Federal University of Amapá, Macapá-AP 68902-280, Brazil. .; Nucleus of Studies and Selection of Bioactive Molecules, Institute of Health Sciences, Federal University of Pará, Belém-PA 66075-110, Brazil. .; Pokaż więcej
Źródło:: Molecules (Basel, Switzerland) [Molecules] 2019 Apr 15; Vol. 24 (8). Date of Electronic Publication: 2019 Apr 15.
Typ publikacji:: Journal Article
MeSH Terms:: Computer Simulation*
Molecular Docking Simulation*
Anti-Inflammatory Agents, Non-Steroidal/*chemistry
Benzoates/*chemistry
Cyclooxygenase 2/*chemistry
Cyclooxygenase 2 Inhibitors/*chemistry
Ibuprofen/*chemistry
Propionates/*chemistry
Animals ; Humans ; Mice ; Rats

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 5.

Tytuł:: Dose dependent cytotoxicity of pranoprofen in cultured human corneal endothelial cells by inducing apoptosis.
Autorzy:: Li YH; Laboratory for Corneal Tissue Engineering, College of Marine Life Sciences, Ocean University of China , Qingdao , China and.
Wen Q
Fan TJ
Ge Y
Yu MM
Sun LX
Zhao Y; Pokaż więcej
Źródło:: Drug and chemical toxicology [Drug Chem Toxicol] 2015 Jan; Vol. 38 (1), pp. 16-21. Date of Electronic Publication: 2014 Mar 18.
Typ publikacji:: Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:: Anti-Inflammatory Agents, Non-Steroidal*/administration & dosage
Anti-Inflammatory Agents, Non-Steroidal*/toxicity
Benzopyrans*/administration & dosage
Benzopyrans*/toxicity
Propionates*/administration & dosage
Propionates*/toxicity
Apoptosis/*drug effects
Endothelial Cells/*drug effects
Endothelium, Corneal/*drug effects
Cell Culture Techniques ; Cell Line ; Cell Membrane Permeability/drug effects ; Cell Survival/drug effects ; DNA Fragmentation/drug effects ; Dose-Response Relationship, Drug ; Endothelial Cells/ultrastructure ; Endothelium, Corneal/ultrastructure ; Humans ; Microscopy, Electron, Transmission ; Microscopy, Phase-Contrast ; Time Factors

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 6.

Tytuł:: A comparison of pre and post-operative vedaprofen with ketoprofen for pain control in dogs.
Autorzy:: Fantoni DT; Laboratório de Investigação Médica 8, Anestesiologia, Faculdade de Medicina, Universidade de São Paulo, São Paulo, Brazil, Av. Doutor Arnaldo, 455, 2° andar, sala 2120, Cerqueira César, 01246-903, São Paulo, SP, Brazil. .; Departamento de Cirurgia, Faculdade de Medicina Veterinária e Zootecnia, Universidade de São Paulo, Brazil, Avenida Prof. Orlando Marques Paiva, 87 Cidade Universitária, 05508-270, São Paulo, SP, Brazil. .
Ida KK; Laboratório de Investigação Médica 8, Anestesiologia, Faculdade de Medicina, Universidade de São Paulo, São Paulo, Brazil, Av. Doutor Arnaldo, 455, 2° andar, sala 2120, Cerqueira César, 01246-903, São Paulo, SP, Brazil. .
de Almeida TI; Departamento de Cirurgia, Faculdade de Medicina Veterinária e Zootecnia, Universidade de São Paulo, Brazil, Avenida Prof. Orlando Marques Paiva, 87 Cidade Universitária, 05508-270, São Paulo, SP, Brazil. .
Ambrósio AM; Departamento de Cirurgia, Faculdade de Medicina Veterinária e Zootecnia, Universidade de São Paulo, Brazil, Avenida Prof. Orlando Marques Paiva, 87 Cidade Universitária, 05508-270, São Paulo, SP, Brazil. .; Pokaż więcej
Źródło:: BMC veterinary research [BMC Vet Res] 2015 Feb 07; Vol. 11, pp. 24. Date of Electronic Publication: 2015 Feb 07.
Typ publikacji:: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
MeSH Terms:: Anti-Inflammatory Agents, Non-Steroidal/*therapeutic use
Dog Diseases/*drug therapy
Ketoprofen/*therapeutic use
Naphthalenes/*therapeutic use
Oral Surgical Procedures/*veterinary
Pain, Postoperative/*veterinary
Propionates/*therapeutic use
Animals ; Anti-Inflammatory Agents, Non-Steroidal/administration & dosage ; Dogs ; Hydrocortisone/blood ; Ketoprofen/administration & dosage ; Naphthalenes/administration & dosage ; Oral Surgical Procedures/adverse effects ; Pain, Postoperative/drug therapy ; Pain, Postoperative/etiology ; Propionates/administration & dosage

Czasopismo naukowe

na półce

Pełny tekst Szczegóły

Skocz do pozycji: 7.

Tytuł:: Effect of textured eye drop bottles on the photostability of pranoprofen 0.1% ophthalmic solution.
Autorzy:: Iwatsuka K; a Senju Pharmaceutical Co., Ltd , Nishiku Kobe, Hyogo , Japan.
Inada K
Ueoka H
Otsuka T
Maeda M
Yamaguchi M
Yasueda S; Pokaż więcej
Źródło:: Drug development and industrial pharmacy [Drug Dev Ind Pharm] 2015; Vol. 41 (9), pp. 1526-31. Date of Electronic Publication: 2015 Jul 21.
Typ publikacji:: Journal Article
MeSH Terms:: Drug Packaging*
Photochemical Processes*
Anti-Inflammatory Agents, Non-Steroidal/*administration & dosage
Benzopyrans/*administration & dosage
Propionates/*administration & dosage
Anti-Inflammatory Agents, Non-Steroidal/chemistry ; Benzopyrans/chemistry ; Chromatography, High Pressure Liquid ; Drug Stability ; Ophthalmic Solutions ; Propionates/chemistry

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 8.

Tytuł:: Evaluation of anti-inflammatory drug-conjugated silicon quantum dots: their cytotoxicity and biological effect.
Autorzy:: Hanada S; Vice Director-General's Lab, Research Institute, National Center for Global Health and Medicine, Tokyo 162-8655, Japan. .
Fujioka K
Futamura Y
Manabe N
Hoshino A
Yamamoto K; Pokaż więcej
Źródło:: International journal of molecular sciences [Int J Mol Sci] 2013 Jan 10; Vol. 14 (1), pp. 1323-34. Date of Electronic Publication: 2013 Jan 10.
Typ publikacji:: Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:: Quantum Dots*
Anti-Inflammatory Agents, Non-Steroidal/*chemistry
Propionates/*chemistry
Silicon/*chemistry
Anti-Inflammatory Agents, Non-Steroidal/pharmacology ; Arachidonic Acid/metabolism ; Biocatalysis/drug effects ; Cell Survival/drug effects ; Cyclooxygenase 2/metabolism ; Cyclooxygenase 2 Inhibitors/chemistry ; Cyclooxygenase 2 Inhibitors/pharmacology ; Dinoprost/metabolism ; Drug Evaluation, Preclinical ; Enzyme-Linked Immunosorbent Assay ; Hep G2 Cells ; Humans ; Kinetics ; Microscopy, Electron, Transmission ; Propionates/pharmacology ; Proton Magnetic Resonance Spectroscopy ; Spectroscopy, Fourier Transform Infrared

Czasopismo naukowe

na półce

Pełny tekst Szczegóły

Skocz do pozycji: 9.

Tytuł:: Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of new 2-(4-isobutylphenyl)propanoic acid derivatives.
Autorzy:: Raval JP; Department of Pharmaceutical Chemistry, Ashok & Rita Patel Institute of Integrated Study and Research in Biotechnology and Allied Sciences(ARIBAS) , New Vallabh Vidyanagar, Gujarat, India. />Gandhi AN
Akhaja TN
Myangar KN
Patel NH; Pokaż więcej
Źródło:: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2012 Feb; Vol. 27 (1), pp. 110-6. Date of Electronic Publication: 2011 May 25.
Typ publikacji:: Journal Article; Retracted Publication
MeSH Terms:: Analgesics/*pharmacology
Anti-Inflammatory Agents, Non-Steroidal/*pharmacology
Anti-Ulcer Agents/*pharmacology
Propionates/*pharmacology
Stomach Ulcer/*drug therapy
Acute Disease ; Analgesics/chemical synthesis ; Analgesics/chemistry ; Animals ; Anti-Inflammatory Agents, Non-Steroidal/chemical synthesis ; Anti-Inflammatory Agents, Non-Steroidal/chemistry ; Anti-Ulcer Agents/chemical synthesis ; Anti-Ulcer Agents/chemistry ; Disease Models, Animal ; Dose-Response Relationship, Drug ; Drug Evaluation, Preclinical ; Ibuprofen ; Lipid Peroxidation/drug effects ; Male ; Mice ; Propionates/chemical synthesis ; Propionates/chemistry ; Rats ; Rats, Wistar

Czasopismo naukowe

na półce

Pełny tekst Pełny tekst Szczegóły

Skocz do pozycji: 10.

Tytuł:: A new method for production of chiral 2-aryl-2-fluoropropanoic acids using an effective kinetic resolution of racemic 2-aryl-2-fluoropropanoic acids.
Autorzy:: Tengeiji A; Department of Applied Chemistry, Faculty of Science, Tokyo University of Science, 1-3 Kagurazaka, Shinjuku-ku, Tokyo 162-8601, Japan.
Shiina I; Pokaż więcej
Źródło:: Molecules (Basel, Switzerland) [Molecules] 2012 Jun 14; Vol. 17 (6), pp. 7356-78. Date of Electronic Publication: 2012 Jun 14.
Typ publikacji:: Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:: Anti-Inflammatory Agents, Non-Steroidal/*chemical synthesis
Propionates/*chemical synthesis
Catalysis ; Kinetics ; Nuclear Magnetic Resonance, Biomolecular ; Propionates/chemistry ; Solvents/chemistry ; Stereoisomerism