- Tytuł :
- Stabilization Strategies for Linear Minigastrin Analogues: Further Improvements via the Inclusion of Proline into the Peptide Sequence.
- Autorzy :
- Źródło :
- Journal of medicinal chemistry [J Med Chem] 2020 Dec 10; Vol. 63 (23), pp. 14668-14679. Date of Electronic Publication: 2020 Nov 23.
- Typ publikacji :
- Journal Article; Research Support, Non-U.S. Gov't
- MeSH Terms :
-
Gastrins/*metabolism
Heterocyclic Compounds, 1-Ring/*metabolism
Proline/*chemistryRadiopharmaceuticals /*metabolism
Amino Acid Sequence ; Animals ; Cell Line, Tumor ; Drug Stability ; Female ; Gastrins/chemical synthesis ; Gastrins/pharmacokinetics ; Heterocyclic Compounds, 1-Ring/chemical synthesis ; Heterocyclic Compounds, 1-Ring/pharmacokinetics ; Humans ; Indium Radioisotopes/chemistry ; Lutetium/chemistry ; Mice, Inbred BALB C ; Protein Binding ; Radioisotopes/chemistry ;Radiopharmaceuticals /chemical synthesis ;Radiopharmaceuticals /pharmacokinetics ; Rats ; Receptor, Cholecystokinin B/metabolism -
Czasopismo naukowe