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Wyszukujesz frazę ""Receptor, Serotonin, 5-HT1A"" wg kryterium: Temat


Tytuł:
Transcriptional Regulation of the Human 5-HT1A Receptor Gene by Lithium: Role of Deaf1 and GSK3β.
Autorzy:
Harkin EF; Ottawa Hospital Research Institute (Neuroscience), University of Ottawa, 451 Smyth Road, Ottawa, ON K1H-8M5, Canada.
Nasrallah G; Ottawa Hospital Research Institute (Neuroscience), University of Ottawa, 451 Smyth Road, Ottawa, ON K1H-8M5, Canada.
Le François B; Ottawa Hospital Research Institute (Neuroscience), University of Ottawa, 451 Smyth Road, Ottawa, ON K1H-8M5, Canada.
Albert PR; Ottawa Hospital Research Institute (Neuroscience), University of Ottawa, 451 Smyth Road, Ottawa, ON K1H-8M5, Canada.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Oct 26; Vol. 24 (21). Date of Electronic Publication: 2023 Oct 26.
Typ publikacji:
Journal Article
MeSH Terms:
Glycogen Synthase Kinase 3 beta*/genetics
Lithium*/pharmacology
Receptor, Serotonin, 5-HT1A*/genetics
Serotonin*/pharmacology
Humans ; Antidepressive Agents ; HEK293 Cells
Czasopismo naukowe
Tytuł:
Cannabidiol Exerts Anticonvulsant Effects Alone and in Combination with Δ -THC through the 5-HT1A Receptor in the Neocortex of Mice.
Autorzy:
Javadzadeh Y; Krembil Research Institute, University Health Network, Toronto, ON M5S 0T8, Canada.; Institute of Biomedical Engineering, University of Toronto, Toronto, ON M5S 1A1, Canada.
Santos A; Krembil Research Institute, University Health Network, Toronto, ON M5S 0T8, Canada.
Aquilino MS; Krembil Research Institute, University Health Network, Toronto, ON M5S 0T8, Canada.; Institute of Biomedical Engineering, University of Toronto, Toronto, ON M5S 1A1, Canada.
Mylvaganam S; Krembil Research Institute, University Health Network, Toronto, ON M5S 0T8, Canada.
Urban K; Avicanna Inc., Toronto, ON M5G 1V2, Canada.
Carlen PL; Krembil Research Institute, University Health Network, Toronto, ON M5S 0T8, Canada.; Institute of Biomedical Engineering, University of Toronto, Toronto, ON M5S 1A1, Canada.; Department of Medicine (Neurology), University Health Network, Toronto, ON M5G 2C4, Canada.
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Źródło:
Cells [Cells] 2024 Mar 07; Vol. 13 (6). Date of Electronic Publication: 2024 Mar 07.
Typ publikacji:
Journal Article
MeSH Terms:
Cannabidiol*/pharmacology
Cannabinoids*/therapeutic use
Neocortex*
Mice ; Animals ; Anticonvulsants/therapeutic use ; Dronabinol ; Receptor, Serotonin, 5-HT1A ; Serotonin
Czasopismo naukowe
Tytuł:
Beneficial effects of atypical antipsychotics on object recognition deficits after adolescent toluene exposure in mice: involvement of 5-HT 1A receptors.
Autorzy:
Lee MY; Center for Neuropsychiatric Research, National Health Research Institutes, Zhunan, Taiwan.; Department of Pharmacology and Toxicology, Tzu Chi University, Hualien, Taiwan.
Hsieh CP; Center for Neuropsychiatric Research, National Health Research Institutes, Zhunan, Taiwan.
Chan MH; Institute of Neuroscience, National Chengchi University, Taipei, Taiwan.; Research Center for Mind, Brain, and Learning, National Chengchi University, Taipei, Taiwan.; Department of Medical Research, China Medical University Hospital, Taichung, Taiwan.
Chen HH; Center for Neuropsychiatric Research, National Health Research Institutes, Zhunan, Taiwan.; Department of Pharmacology and Toxicology, Tzu Chi University, Hualien, Taiwan.; Institute of Neuroscience, National Chengchi University, Taipei, Taiwan.
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Źródło:
The American journal of drug and alcohol abuse [Am J Drug Alcohol Abuse] 2022 Nov 02; Vol. 48 (6), pp. 673-683. Date of Electronic Publication: 2022 Sep 22.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptor, Serotonin, 5-HT1A*/metabolism
Toluene*/adverse effects
Antipsychotic Agents*/therapeutic use
Cognition*/drug effects
Animals ; Male ; Mice
Czasopismo naukowe
Tytuł:
Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation.
Autorzy:
Stępnicki P; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University of Lublin, Lublin, Poland.
Wronikowska-Denysiuk O; Independent Laboratory of Behavioral Studies, Chair of Biomedical Sciences, Faculty of Biomedicine, Medical University of Lublin, Lublin, Poland.
Zięba A; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University of Lublin, Lublin, Poland.
Targowska-Duda KM; Department of Biopharmacy, Faculty of Pharmacy, Medical University of Lublin, Lublin, Poland.
Bartyzel A; Department of General and Coordination Chemistry and Crystallography, Institute of Chemical Sciences, Faculty of Chemistry, Maria Curie-Sklodowska University in Lublin, Lublin, Poland.
Wróbel MZ; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, Warsaw, Poland.
Wróbel TM; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University of Lublin, Lublin, Poland.
Szałaj K; Department of Bioanalytics, Faculty of Biomedicine, Medical University of Lublin, Lublin, Poland.
Chodkowski A; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, Warsaw, Poland.
Mirecka K; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, Warsaw, Poland.
Budzyńska B; Independent Laboratory of Behavioral Studies, Chair of Biomedical Sciences, Faculty of Biomedicine, Medical University of Lublin, Lublin, Poland.
Fornal E; Department of Bioanalytics, Faculty of Biomedicine, Medical University of Lublin, Lublin, Poland.
Turło J; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, Warsaw, Poland.
Castro M; Department of Pharmacology, Center for Research in Molecular Medicine and Chronic Diseases (CIMUS), Universidade de Santiago de Compostela, Santiago de Compostela, Spain.; Instituto de Investigación Sanitaria de Santiago de Compostela (IDIS), Santiago de Compostela, Spain.
Kaczor AA; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University of Lublin, Lublin, Poland.; School of Pharmacy, University of Eastern Finland, Kuopio, Finland.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2209828.
Typ publikacji:
Journal Article
MeSH Terms:
Schizophrenia*/drug therapy
Antipsychotic Agents*/pharmacology
Antipsychotic Agents*/chemistry
Humans ; Piperazine/pharmacology ; Dopamine/therapeutic use ; Ligands ; Indazoles ; Serotonin/therapeutic use ; Receptors, Serotonin ; Receptor, Serotonin, 5-HT1A/therapeutic use
Czasopismo naukowe
Tytuł:
Therapeutic Effects of Quetiapine and 5-HT 1A Receptor Agonism on Hyperactivity in Dopamine-Deficient Mice.
Autorzy:
Ochiai Y; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo 156-8506, Japan.; Department of Neurology, Tokyo Metropolitan Neurological Hospital, Tokyo 183-0042, Japan.
Fujita M; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo 156-8506, Japan.
Hagino Y; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo 156-8506, Japan.
Kobayashi K; Department of Molecular Genetics, Institute of Biomedical Sciences, Fukushima Medical University, Fukushima 960-1295, Japan.
Okiyama R; Department of Neurology, Tokyo Metropolitan Neurological Hospital, Tokyo 183-0042, Japan.
Takahashi K; Department of Neurology, Tokyo Metropolitan Neurological Hospital, Tokyo 183-0042, Japan.
Ikeda K; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo 156-8506, Japan.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Jul 04; Vol. 23 (13). Date of Electronic Publication: 2022 Jul 04.
Typ publikacji:
Journal Article
MeSH Terms:
Antipsychotic Agents*/pharmacology
Dopamine*/deficiency
Dopamine*/metabolism
Quetiapine Fumarate*/pharmacology
Receptor, Serotonin, 5-HT1A*/metabolism
Serotonin 5-HT1 Receptor Agonists*/pharmacology
Animals ; Mice ; Serotonin/metabolism ; Serotonin Antagonists/pharmacology
Czasopismo naukowe
Tytuł:
Dopamine D 2 and Serotonin 5-HT 1A Dimeric Receptor-Binding Monomeric Antibody scFv as a Potential Ligand for Carrying Drugs Targeting Selected Areas of the Brain.
Autorzy:
Kowalik A; Department of Physical Biochemistry, Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, 30-387 Krakow, Poland.
Majerek M; Department of Physical Biochemistry, Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, 30-387 Krakow, Poland.
Mrowiec K; Department of Physical Biochemistry, Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, 30-387 Krakow, Poland.
Solich J; Department of Pharmacology, Maj Institute of Pharmacology, Polish Academy of Science, 31-343 Krakow, Poland.
Faron-Górecka A; Department of Pharmacology, Maj Institute of Pharmacology, Polish Academy of Science, 31-343 Krakow, Poland.
Woźnicka O; Department of Cell Biology and Imaging, Institute of Zoology and Biomedical Research, Jagiellonian University, 30-387 Krakow, Poland.
Dziedzicka-Wasylewska M; Department of Physical Biochemistry, Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, 30-387 Krakow, Poland.; Department of Pharmacology, Maj Institute of Pharmacology, Polish Academy of Science, 31-343 Krakow, Poland.
Łukasiewicz S; Department of Physical Biochemistry, Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, 30-387 Krakow, Poland.
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Źródło:
Biomolecules [Biomolecules] 2022 May 26; Vol. 12 (6). Date of Electronic Publication: 2022 May 26.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Antipsychotic Agents*/pharmacology
Drug Carriers*
Receptor, Serotonin, 5-HT1A*/metabolism
Receptors, Dopamine D2*/metabolism
Single-Chain Antibodies*
Animals ; Brain/metabolism ; Dopamine/metabolism ; Ligands ; Mice
Czasopismo naukowe
Tytuł:
Antioxioxidant and antiapoptotic effects of Thymosin β4 in Aβ-induced SH-SY5Y cells via the 5-HTR1A/ERK axis.
Autorzy:
Zhang GH; School of Medicine, Xi'an International University, Xi'an, Shaanxi, China.; Faculty of Medicine and Health Sciences, Department of Biomedical Science, Universiti Malaysia Sabah, Kota Kinabalu, Sabah, Malaysia.
Chin KL; Faculty of Medicine and Health Sciences, Department of Biomedical Science, Universiti Malaysia Sabah, Kota Kinabalu, Sabah, Malaysia.
Yan SY; International Innovation Institute of Acupuncture and Moxibustion, Beijing University of Chinese Medicine, Beijing, Hebei, China.
Pare R; Faculty of Medicine and Health Sciences, Department of Biomedical Science, Universiti Malaysia Sabah, Kota Kinabalu, Sabah, Malaysia.
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Źródło:
PloS one [PLoS One] 2023 Oct 03; Vol. 18 (10), pp. e0287817. Date of Electronic Publication: 2023 Oct 03 (Print Publication: 2023).
Typ publikacji:
Journal Article
MeSH Terms:
Alzheimer Disease*/drug therapy
Neuroblastoma*/pathology
Thymosin*/metabolism
Aged ; Humans ; Apoptosis ; Cell Line, Tumor ; Oxidative Stress ; Receptor, Serotonin, 5-HT1A/metabolism ; Signal Transduction ; Neuroprotection
Czasopismo naukowe
Tytuł:
Effects of the 5-HT 1A receptor agonist 8-OH-DPAT on aggressive behavior in juvenile pufferfish, Takifugu rubripes.
Autorzy:
Hu Y; Key Laboratory of Environment Controlled Aquaculture, Ministry of Education, Dalian Ocean University, Dalian, China.
Li H; Key Laboratory of Environment Controlled Aquaculture, Ministry of Education, Dalian Ocean University, Dalian, China.
Zhou C; Key Laboratory of Environment Controlled Aquaculture, Ministry of Education, Dalian Ocean University, Dalian, China.
Liu Y; Key Laboratory of Environment Controlled Aquaculture, Ministry of Education, Dalian Ocean University, Dalian, China.; College of Biosystems Engineering and Food Science, Zhejiang University, Hangzhou, China.
Ma Z; Key Laboratory of Environment Controlled Aquaculture, Ministry of Education, Dalian Ocean University, Dalian, China.
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Źródło:
Aggressive behavior [Aggress Behav] 2022 Mar; Vol. 48 (2), pp. 197-204. Date of Electronic Publication: 2021 Dec 14.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptor, Serotonin, 5-HT1A*
Takifugu*
8-Hydroxy-2-(di-n-propylamino)tetralin/pharmacology ; Aggression/physiology ; Animals ; Humans ; Serotonin Receptor Agonists/pharmacology
Czasopismo naukowe
Tytuł:
Effect of Central Administration of Brain-Derived Neurotrophic Factor (BDNF) on Behavior and Brain Monoamine Metabolism in New Recombinant Mouse Lines Differing by 5-HT 1A Receptor Functionality.
Autorzy:
Bazovkina D; Institute of Cytology and Genetics, Siberian Division of the Russian Academy of Science, 630090 Novosibirsk, Russia.
Naumenko V; Institute of Cytology and Genetics, Siberian Division of the Russian Academy of Science, 630090 Novosibirsk, Russia.
Bazhenova E; Institute of Cytology and Genetics, Siberian Division of the Russian Academy of Science, 630090 Novosibirsk, Russia.
Kondaurova E; Institute of Cytology and Genetics, Siberian Division of the Russian Academy of Science, 630090 Novosibirsk, Russia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2021 Nov 05; Vol. 22 (21). Date of Electronic Publication: 2021 Nov 05.
Typ publikacji:
Journal Article
MeSH Terms:
Aggression/*drug effects
Behavior, Animal/*drug effects
Brain/*metabolism
Brain-Derived Neurotrophic Factor/*pharmacology
Receptor, Serotonin, 5-HT1A/*metabolism
Serotonin/*metabolism
Animals ; Brain/drug effects ; Brain/pathology ; Disease Models, Animal ; Male ; Mice ; Mice, Inbred C57BL ; Mice, Inbred CBA ; Receptor, Serotonin, 5-HT1A/genetics
Czasopismo naukowe
Tytuł:
Evidence for 5-HT 1A receptor-mediated antiallodynic and antihyperalgesic effects of apigenin in mice suffering from mononeuropathy.
Autorzy:
Wu JY; Department of Pharmacology, Ningbo University, School of Medical Science, Ningbo, China.
Li Y; School of Marine Science, Ningbo University, Ningbo, China.
Li BL; School of Mathematics and Statistics, Ningbo University, Ningbo, China.
Wang YG; Department of Geriatrics, Hunan Provincial People's Hospital, Changsha, China.
Cui WG; Department of Pharmacology, Ningbo University, School of Medical Science, Ningbo, China.
Zhou WH; Department of Pharmacology, Ningbo University, School of Medical Science, Ningbo, China.
Zhao X; Department of Pharmacology, Ningbo University, School of Medical Science, Ningbo, China.
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2021 Oct; Vol. 178 (19), pp. 4005-4025. Date of Electronic Publication: 2021 Jun 22.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Mononeuropathies*
Receptor, Serotonin, 5-HT1A*
Animals ; Apigenin/pharmacology ; Disease Models, Animal ; Hyperalgesia/drug therapy ; Male ; Mice ; Mice, Inbred C57BL
Czasopismo naukowe
Tytuł:
The selective 5-HT 1A receptor biased agonists, F15599 and F13714, show antidepressant-like properties after a single administration in the mouse model of unpredictable chronic mild stress.
Autorzy:
Głuch-Lutwin M; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Sałaciak K; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Gawalska A; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Jamrozik M; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Sniecikowska J; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Newman-Tancredi A; Neurolixis SAS, Castres, France.
Kołaczkowski M; Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland.
Pytka K; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, Krakow, Poland. .
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Źródło:
Psychopharmacology [Psychopharmacology (Berl)] 2021 Aug; Vol. 238 (8), pp. 2249-2260. Date of Electronic Publication: 2021 May 10.
Typ publikacji:
Journal Article
MeSH Terms:
Receptor, Serotonin, 5-HT1A*/physiology
Aminopyridines/*administration & dosage
Antidepressive Agents/*administration & dosage
Piperidines/*administration & dosage
Pyrimidines/*administration & dosage
Serotonin 5-HT1 Receptor Agonists/*administration & dosage
Stress, Psychological/*drug therapy
Animals ; Chronic Disease ; Disease Models, Animal ; Dose-Response Relationship, Drug ; Locomotion ; Male ; Mice ; Single-Blind Method ; Stress, Psychological/psychology
Czasopismo naukowe
Tytuł:
Synthesis of Novel Pyrido[1,2- c ]pyrimidine Derivatives with 6-Fluoro-3-(4-piperidynyl)-1,2-benzisoxazole Moiety as Potential SSRI and 5-HT 1A Receptor Ligands.
Autorzy:
Król M; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, 1, Banacha Street, 02-097 Warsaw, Poland.
Ślifirski G; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, 1, Banacha Street, 02-097 Warsaw, Poland.
Kleps J; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, 1, Banacha Street, 02-097 Warsaw, Poland.
Ulenberg S; Department of Pharmaceutical Chemistry, Medical University of Gdańsk, 107, J. Hallera Street, 80-416 Gdańsk, Poland.
Belka M; Department of Pharmaceutical Chemistry, Medical University of Gdańsk, 107, J. Hallera Street, 80-416 Gdańsk, Poland.
Bączek T; Department of Pharmaceutical Chemistry, Medical University of Gdańsk, 107, J. Hallera Street, 80-416 Gdańsk, Poland.
Siwek A; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, 9, Medyczna Street, 30-688 Kraków, Poland.
Stachowicz K; Maj Institute of Pharmacology, Polish Academy of Sciences, 12, Smętna Street, 31-343 Kraków, Poland.
Szewczyk B; Maj Institute of Pharmacology, Polish Academy of Sciences, 12, Smętna Street, 31-343 Kraków, Poland.
Nowak G; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, 9, Medyczna Street, 30-688 Kraków, Poland.; Maj Institute of Pharmacology, Polish Academy of Sciences, 12, Smętna Street, 31-343 Kraków, Poland.
Duszyńska B; Maj Institute of Pharmacology, Polish Academy of Sciences, 12, Smętna Street, 31-343 Kraków, Poland.
Herold F; Department of Drug Technology and Pharmaceutical Biotechnology, Faculty of Pharmacy, Medical University of Warsaw, 1, Banacha Street, 02-097 Warsaw, Poland.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2021 Feb 26; Vol. 22 (5). Date of Electronic Publication: 2021 Feb 26.
Typ publikacji:
Journal Article
MeSH Terms:
Pyridines*/chemical synthesis
Pyridines*/chemistry
Pyridines*/pharmacology
Receptor, Serotonin, 5-HT1A*/chemistry
Receptor, Serotonin, 5-HT1A*/metabolism
Serotonin 5-HT1 Receptor Agonists*/chemical synthesis
Serotonin 5-HT1 Receptor Agonists*/chemistry
Serotonin 5-HT1 Receptor Agonists*/pharmacology
Animals ; CHO Cells ; Cricetulus ; Humans
Czasopismo naukowe
Tytuł:
Knockout of NPFFR2 Prevents LPS-Induced Depressive-Like Responses in Mice.
Autorzy:
Yu Z; Department of Medicine, Chang Gung University, Taoyuan 333, Taiwan.
Lin YT; Department of Physiology and Pharmacology, Graduate Institute of Biomedical Sciences, Chang Gung University, Taoyuan 333, Taiwan.; Healthy Aging Research Center, Chang Gung University, Taoyuan 333, Taiwan.
Chen JC; Department of Physiology and Pharmacology, Graduate Institute of Biomedical Sciences, Chang Gung University, Taoyuan 333, Taiwan.; Healthy Aging Research Center, Chang Gung University, Taoyuan 333, Taiwan.; Neuroscience Research Center, Chang Gung Memorial Hospital, Taoyuan 333, Taiwan.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2021 Jul 16; Vol. 22 (14). Date of Electronic Publication: 2021 Jul 16.
Typ publikacji:
Journal Article
MeSH Terms:
Depression/*genetics
Receptor, Serotonin, 5-HT1A/*metabolism
Receptors, Neuropeptide/*genetics
Animals ; Behavior, Animal/physiology ; Depression/metabolism ; Disease Models, Animal ; Female ; Hippocampus/metabolism ; Lipopolysaccharides/adverse effects ; Lipopolysaccharides/pharmacology ; Mice ; Mice, Inbred C57BL ; Mice, Knockout ; Motor Activity/drug effects ; Receptor, Serotonin, 5-HT1A/genetics ; Receptors, Neuropeptide/metabolism ; Toll-Like Receptor 4/metabolism ; Tumor Necrosis Factor-alpha/metabolism
Czasopismo naukowe
Tytuł:
Cardamonin Modulates Neuropathic Pain through the Possible Involvement of Serotonergic 5-HT1A Receptor Pathway in CCI-Induced Neuropathic Pain Mice Model.
Autorzy:
Kaswan NK; Department of Biomedical Science, Faculty of Medicine and Health Sciences, Universiti Putra Malaysia (UPM), Serdang 43400, Selangor, Malaysia.
Mohammed Izham NAB; Department of Biomedical Science, Faculty of Medicine and Health Sciences, Universiti Putra Malaysia (UPM), Serdang 43400, Selangor, Malaysia.
Tengku Mohamad TAS; Department of Biomedical Science, Faculty of Medicine and Health Sciences, Universiti Putra Malaysia (UPM), Serdang 43400, Selangor, Malaysia.
Sulaiman MR; Department of Biomedical Science, Faculty of Medicine and Health Sciences, Universiti Putra Malaysia (UPM), Serdang 43400, Selangor, Malaysia.
Perimal EK; Department of Biomedical Science, Faculty of Medicine and Health Sciences, Universiti Putra Malaysia (UPM), Serdang 43400, Selangor, Malaysia.; Centre of Excellence for Nanoscale BioPhotonics, Australian Research Council, University of Adelaide, Adelaide, SA 5005, Australia.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2021 Jun 16; Vol. 26 (12). Date of Electronic Publication: 2021 Jun 16.
Typ publikacji:
Journal Article
MeSH Terms:
Chalcones/*pharmacology
Neuralgia/*drug therapy
Receptor, Serotonin, 5-HT1A/*drug effects
Analgesics/pharmacology ; Animals ; Chalcones/metabolism ; Disease Models, Animal ; Hyperalgesia/drug therapy ; Male ; Mice ; Mice, Inbred ICR ; Receptor, Serotonin, 5-HT1A/metabolism ; Serotonergic Neurons/drug effects ; Serotonergic Neurons/metabolism ; Serotonin/metabolism ; Spinal Cord/drug effects
Czasopismo naukowe
Tytuł:
The effect of 5-HT 1A receptor agonists on the entopeduncular nucleus is modified in 6-hydroxydopamine-lesioned rats.
Autorzy:
Vegas-Suárez S; Department of Pharmacology, Faculty of Medicine and Nursing, University of the Basque Country (UPV/EHU), Leioa, Spain.; Autonomic and Movement Disorders Unit, Neurodegenerative Diseases, Biocruces Health Research Institute, Barakaldo, Spain.
Aristieta A; Department of Biological Sciences, Carnegie Mellon University, Pittsburgh, PA, USA.; Center for the Neural Basis of Cognition, Carnegie Mellon University, Pittsburgh, PA, USA.
Requejo C; LaNCE, Department of Neuroscience, University of the Basque Country (UPV/EHU), Leioa, Spain.
Bengoetxea H; LaNCE, Department of Neuroscience, University of the Basque Country (UPV/EHU), Leioa, Spain.
Lafuente JV; LaNCE, Department of Neuroscience, University of the Basque Country (UPV/EHU), Leioa, Spain.
Miguelez C; Department of Pharmacology, Faculty of Medicine and Nursing, University of the Basque Country (UPV/EHU), Leioa, Spain.; Autonomic and Movement Disorders Unit, Neurodegenerative Diseases, Biocruces Health Research Institute, Barakaldo, Spain.
Ugedo L; Department of Pharmacology, Faculty of Medicine and Nursing, University of the Basque Country (UPV/EHU), Leioa, Spain.; Autonomic and Movement Disorders Unit, Neurodegenerative Diseases, Biocruces Health Research Institute, Barakaldo, Spain.
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Źródło:
British journal of pharmacology [Br J Pharmacol] 2021 Jun; Vol. 178 (12), pp. 2516-2532. Date of Electronic Publication: 2021 May 06.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Entopeduncular Nucleus*
Receptor, Serotonin, 5-HT1A*
8-Hydroxy-2-(di-n-propylamino)tetralin/pharmacology ; Animals ; Buspirone/pharmacology ; Levodopa/pharmacology ; Oxidopamine/toxicity ; Rats ; Rats, Sprague-Dawley
Czasopismo naukowe
Tytuł:
Expression Patterns of Serotonin Receptors 5-HT1A, 5-HT2A, and 5-HT3A during Human Fetal Lung Development.
Autorzy:
Nikolić J; Laboratory for Experimental Neurocardiology, Department of Anatomy, Histology and Embryology, University of Split School of Medicine, Šoltanska 2, 21000 Split, Croatia.; Mediterranean Institute for Life Sciences (MedILS), Meštrovićevo Šetalište 45, 21000 Split, Croatia.
Vukojević K; Laboratory for Early Human Development, Department of Anatomy, Histology and Embryology, University of Split School of Medicine, Šoltanska 2, 21000 Split, Croatia.; Faculty of Health Studies, University of Mostar, 88000 Mostar, Bosnia and Herzegovina.
Šoljić V; Faculty of Health Studies, University of Mostar, 88000 Mostar, Bosnia and Herzegovina.
Mišković J; Department of Anatomy, School of Medicine, University of Mostar, 88000 Mostar, Bosnia and Herzegovina.
Orlović Vlaho M; Faculty of Health Studies, University of Mostar, 88000 Mostar, Bosnia and Herzegovina.
Saraga-Babić M; Laboratory for Early Human Development, Department of Anatomy, Histology and Embryology, University of Split School of Medicine, Šoltanska 2, 21000 Split, Croatia.
Filipović N; Laboratory for Experimental Neurocardiology, Department of Anatomy, Histology and Embryology, University of Split School of Medicine, Šoltanska 2, 21000 Split, Croatia.; Laboratory for Early Human Development, Department of Anatomy, Histology and Embryology, University of Split School of Medicine, Šoltanska 2, 21000 Split, Croatia.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Feb 03; Vol. 24 (3). Date of Electronic Publication: 2023 Feb 03.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Serotonin*/genetics
Receptors, Serotonin*/metabolism
Lung*/metabolism
Infant, Newborn ; Humans ; Fetus/metabolism ; Epithelium/metabolism ; Serotonin/metabolism ; Receptor, Serotonin, 5-HT2A/genetics ; Receptor, Serotonin, 5-HT2A/metabolism ; Receptor, Serotonin, 5-HT1A/genetics ; Receptor, Serotonin, 5-HT1A/metabolism
Czasopismo naukowe
Tytuł:
Dual actions of 5-MeO-DIPT at the serotonin transporter and serotonin 5-HT 1A receptor in the mouse striatum and prefrontal cortex.
Autorzy:
Hagino Y; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo, Japan.
Hall FS; Department of Pharmacology and Experimental Therapeutics, College of Pharmacy and Pharmaceutical Sciences, The University of Toledo, Toledo, OH, USA.
Uhl GR; Neurology and Research Services, New Mexico VA Healthcare System, Albuquerque, NM, USA.
Sora I; Department of Psychiatry, Kobe University Graduate School of Medicine, Kobe, Japan.
Ikeda K; Addictive Substance Project, Tokyo Metropolitan Institute of Medical Science, Tokyo, Japan.
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Źródło:
Neuropsychopharmacology reports [Neuropsychopharmacol Rep] 2021 Mar; Vol. 41 (1), pp. 91-101. Date of Electronic Publication: 2021 Feb 06.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
5-Methoxytryptamine/*analogs & derivatives
Corpus Striatum/*drug effects
Prefrontal Cortex/*drug effects
Receptor, Serotonin, 5-HT1A/*drug effects
Serotonin 5-HT1 Receptor Agonists/*pharmacology
Serotonin 5-HT1 Receptor Antagonists/*pharmacology
Serotonin Plasma Membrane Transport Proteins/*drug effects
5-Methoxytryptamine/pharmacology ; 8-Hydroxy-2-(di-n-propylamino)tetralin/pharmacology ; Animals ; Corpus Striatum/metabolism ; Female ; Male ; Mice ; Mice, Knockout ; Microdialysis ; Piperazines/pharmacology ; Prefrontal Cortex/metabolism ; Pyridines/pharmacology ; Receptor, Serotonin, 5-HT1A/metabolism ; Serotonin Plasma Membrane Transport Proteins/metabolism
Czasopismo naukowe
Tytuł:
Anxiolytic-like Effects and Quantitative EEG Profile of Palmitone Induces Responses Like Buspirone Rather Than Diazepam as Clinical Drugs.
Autorzy:
Onofre-Campos D; Laboratorio de Neurofarmacología de Productos Naturales, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.; Biología Experimental, Universidad Autónoma Metropolitana, Ciudad de México 09340, Mexico.
González-Trujano ME; Laboratorio de Neurofarmacología de Productos Naturales, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.
Moreno-Pérez GF; Laboratorio de Neurofarmacología de Productos Naturales, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.
Narváez-González F; ISSSTE Hospital Regional General Ignacio Zaragoza, Calz. Ignacio Zaragoza 1840, Juan Escutia, Iztapalapa, Ciudad de México 09100, Mexico.
González-Gómez JD; Laboratorio de Neurofisiología del Control y la Regulación, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.
Villasana-Salazar B; Laboratorio de Neurofisiología del Control y la Regulación, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.
Martínez-Vargas D; Laboratorio de Neurofisiología del Control y la Regulación, Dirección de Investigaciones en Neurociencias, Instituto Nacional de Psiquiatría Ramón de la Fuente Muñiz, Calz. México-Xochimilco 101, Col. San Lorenzo Huipulco, Tlalpan, Ciudad de México 14370, Mexico.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Apr 24; Vol. 28 (9). Date of Electronic Publication: 2023 Apr 24.
Typ publikacji:
Journal Article
MeSH Terms:
Anti-Anxiety Agents*/pharmacology
Anti-Anxiety Agents*/therapeutic use
COVID-19*
Mice ; Animals ; Buspirone/pharmacology ; Diazepam/pharmacology ; Receptor, Serotonin, 5-HT1A ; 8-Hydroxy-2-(di-n-propylamino)tetralin/pharmacology ; SARS-CoV-2 ; Serotonin Receptor Agonists/pharmacology ; Electroencephalography
Czasopismo naukowe
Tytuł:
HTR1A, TPH2, and 5-HTTLPR Polymorphisms and Their Impact on the Severity of Depressive Symptoms and on the Concentration of Tryptophan Catabolites during Hepatitis C Treatment with Pegylated Interferon-α2a and Oral Ribavirin (PEG-IFN-α2a/RBV).
Autorzy:
Pawlowski T; Department of Psychiatry, Wrocław Medical University, 50-367 Wrocław, Poland.
Malyszczak K; Department of Psychiatry, Wrocław Medical University, 50-367 Wrocław, Poland.
Pawlak D; Department of Pharmacodynamics, Medical University of Bialystok, 15-089 Białystok, Poland.
Inglot M; Department of Infectious Diseases, Liver Diseases and Acquired Immune Deficiency, Wroclaw Medical University, 50-367 Wrocław, Poland.
Zalewska M; Department of Infectious Diseases, Liver Diseases and Acquired Immune Deficiency, Wroclaw Medical University, 50-367 Wrocław, Poland.
Grzywacz A; Independent Laboratory of Health Promotion, Pomeranian Medical University in Szczecin, 70-111 Szczecin, Poland.
Radkowski M; Department of Immunopathology of Infectious and Parasitic Diseases, Medical University of Warsaw, 02-091 Warsaw, Poland.
Laskus T; Department of Adult Infectious Diseases, Medical University of Warsaw, 02-091 Warsaw, Poland.
Janocha-Litwin J; Department of Infectious Diseases and Hepatology, Wroclaw Medical University, 50-367 Wroclaw, Poland.
Frydecka D; Department of Psychiatry, Wrocław Medical University, 50-367 Wrocław, Poland.
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Źródło:
Cells [Cells] 2023 Mar 22; Vol. 12 (6). Date of Electronic Publication: 2023 Mar 22.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Depression*/genetics
Depression*/metabolism
Hepatitis C, Chronic*/complications
Hepatitis C, Chronic*/drug therapy
Hepatitis C, Chronic*/genetics
Interferon alpha-2*/adverse effects
Interferon alpha-2*/pharmacology
Interferon alpha-2*/therapeutic use
Tryptophan*/drug effects
Tryptophan*/metabolism
Adult ; Humans ; Antiviral Agents/therapeutic use ; Kynurenine ; Polyethylene Glycols/pharmacology ; Polymorphism, Genetic ; Prospective Studies ; Receptor, Serotonin, 5-HT1A/genetics ; Ribavirin/adverse effects ; Ribavirin/pharmacology ; Ribavirin/therapeutic use ; Tryptophan Hydroxylase/genetics ; Tryptophan Oxygenase/genetics
Czasopismo naukowe
Tytuł:
Ginsenoside Re attenuates 8-OH-DPAT-induced serotonergic behaviors in mice via interactive modulation between PKCδ gene and Nrf2.
Autorzy:
Shin EJ; Neuropsychopharmacology and Toxicology Program, College of Pharmacy, Kangwon National University, Chuncheon, South Korea.
Jeong JH; Department of Global Innovative Drugs, College of Medicine, Graduate School of Chung-Ang University, Chung-Ang University, Seoul, Republic of Korea.
Nguyen BT; Neuropsychopharmacology and Toxicology Program, College of Pharmacy, Kangwon National University, Chuncheon, South Korea.
Sharma N; Neuropsychopharmacology and Toxicology Program, College of Pharmacy, Kangwon National University, Chuncheon, South Korea.; Department of Global Innovative Drugs, College of Medicine, Graduate School of Chung-Ang University, Chung-Ang University, Seoul, Republic of Korea.
Tran CNK; Neuropsychopharmacology and Toxicology Program, College of Pharmacy, Kangwon National University, Chuncheon, South Korea.
Nah SY; Ginsentology Research Laboratory and Department of Physiology, College of Veterinary Medicine and Bio/Molecular Informatics Center, Konkuk University, Seoul, Republic of Korea.
Lee Y; Department of Industrial Plant Science & Technology, Chungbuk National University, Chungju, Republic of Korea.
Byun JK; Korea Society of Forest Environmental Research, Namyangju, Republic of Korea.
Ko SK; Department of Oriental Medical Food and Nutrition, Semyung University, Jecheon, Republic of Korea.
Kim HC; Neuropsychopharmacology and Toxicology Program, College of Pharmacy, Kangwon National University, Chuncheon, South Korea.
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Źródło:
Drug and chemical toxicology [Drug Chem Toxicol] 2023 Mar; Vol. 46 (2), pp. 281-296. Date of Electronic Publication: 2022 Jun 16.
Typ publikacji:
Journal Article
MeSH Terms:
Ginsenosides*/pharmacology
Mice ; Animals ; 8-Hydroxy-2-(di-n-propylamino)tetralin/pharmacology ; NF-E2-Related Factor 2/genetics ; NF-E2-Related Factor 2/metabolism ; Receptor, Serotonin, 5-HT1A/genetics ; Glutathione ; Glutathione Disulfide ; Serotonin Antagonists ; Ligases
Czasopismo naukowe

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