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Tytuł:
Synthesis and biochemical evaluation of 17-N-beta-aminoalkyl-4,5α-epoxynormorphinans.
Autorzy:
Ötvös F; Institute of Biochemistry, HUN-REN Biological Research Centre, Temesvári Krt. 62, 6726, Szeged, Hungary. .
Szűcs E; Institute of Biochemistry, HUN-REN Biological Research Centre, Temesvári Krt. 62, 6726, Szeged, Hungary.
Urai Á; Institute of Pharmaceutical Chemistry, Semmelweis Medical University, Hőgyes Endre Utca 9, 1092, Budapest, Hungary.
Köteles I; Institute of Pharmaceutical Chemistry, Semmelweis Medical University, Hőgyes Endre Utca 9, 1092, Budapest, Hungary.; Department of Chemistry and Molecular Biology, University of Gothenburg, Medicinaregatan 19, 41390, Göteborg, Sweden.
Szabó PT; Research Centre for Natural Sciences, MS Metabolomics Research Laboratory, Magyar Tudósok Krt. 2, 1117, Budapest, Hungary.
Varga ZK; Institute of Biochemistry, HUN-REN Biological Research Centre, Temesvári Krt. 62, 6726, Szeged, Hungary.; Theoretical Medical Doctoral School, Faculty of Medicine, University of Szeged, 6726, Szeged, Hungary.
Gombos D; Institute of Biochemistry, HUN-REN Biological Research Centre, Temesvári Krt. 62, 6726, Szeged, Hungary.; Theoretical Medical Doctoral School, Faculty of Medicine, University of Szeged, 6726, Szeged, Hungary.
Hosztafi S; Institute of Pharmaceutical Chemistry, Semmelweis Medical University, Hőgyes Endre Utca 9, 1092, Budapest, Hungary.
Benyhe S; Institute of Biochemistry, HUN-REN Biological Research Centre, Temesvári Krt. 62, 6726, Szeged, Hungary. .
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Źródło:
Scientific reports [Sci Rep] 2023 Nov 20; Vol. 13 (1), pp. 20305. Date of Electronic Publication: 2023 Nov 20.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid, mu*/metabolism
Receptors, Opioid*/metabolism
Molecular Docking Simulation ; Binding, Competitive ; Structure-Activity Relationship ; Receptors, Opioid, kappa/metabolism
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Discovery of 7-Azanorbornane-Based Dual Agonists for the Delta and Kappa Opioid Receptors through an In Situ Screening Protocol.
Autorzy:
Karaki F; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Takamori T; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Kawakami K; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Sakurai S; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Hidaka K; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Ishii K; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Oki T; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Sato N; Analytical Unit for Organic Chemistry, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Atsumi N; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Ashizawa K; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Taguchi A; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Ura A; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Naruse T; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Hirayama S; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Nonaka M; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Miyano K; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Uezono Y; Department of Pain Control Research, Jikei University School of Medicine, 3-25-8, Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Fujii H; Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.; Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Oct 03; Vol. 28 (19). Date of Electronic Publication: 2023 Oct 03.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid, kappa*/metabolism
Copper*
Ligands ; Membrane Proteins ; Receptors, Opioid, mu/metabolism ; Analgesics, Opioid/chemistry
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Optimization of a Nucleophilic Two-Step Radiosynthesis of 6- O -(2-[ F]FE-DPN) for PET Imaging of Brain Opioid Receptors.
Autorzy:
Németh E; Division of Nuclear Medicine and Translational Imaging, Department of Medical Imaging, Faculty of Medicine, University of Debrecen, Nagyerdei Krt. 98, H-4032 Debrecen, Hungary.
Gyuricza B; Division of Nuclear Medicine and Translational Imaging, Department of Medical Imaging, Faculty of Medicine, University of Debrecen, Nagyerdei Krt. 98, H-4032 Debrecen, Hungary.
Forgács V; Division of Nuclear Medicine and Translational Imaging, Department of Medical Imaging, Faculty of Medicine, University of Debrecen, Nagyerdei Krt. 98, H-4032 Debrecen, Hungary.
Cumming P; Department of Nuclear Medicine, Bern University Hospital, Freiburgstraße 18, CH-3010 Bern, Switzerland.; School of Psychology and Counselling, Queensland University of Technology, Brisbane QLD-4059, Australia.
Henriksen G; Norwegian Medical Cyclotron Centre Ltd., Sognsvannsveien 20, N-0372 Oslo, Norway.; Institute of Basic Medical Sciences, University of Oslo, N-0317 Oslo, Norway.; Institute of Physics, University of Oslo, Sem Sælands Vei 24, N-0371 Oslo, Norway.
Marton J; ABX Advanced Biochemical Compounds Biomedizinische Forschungsreagenzien GmbH, Heinrich-Glaeser-Strasse 10-14, D-01454 Radeberg, Germany.
Bauer B; ABX Advanced Biochemical Compounds Biomedizinische Forschungsreagenzien GmbH, Heinrich-Glaeser-Strasse 10-14, D-01454 Radeberg, Germany.
Mikecz P; Division of Nuclear Medicine and Translational Imaging, Department of Medical Imaging, Faculty of Medicine, University of Debrecen, Nagyerdei Krt. 98, H-4032 Debrecen, Hungary.
Fekete A; Division of Nuclear Medicine and Translational Imaging, Department of Medical Imaging, Faculty of Medicine, University of Debrecen, Nagyerdei Krt. 98, H-4032 Debrecen, Hungary.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Aug 24; Vol. 24 (17). Date of Electronic Publication: 2023 Aug 24.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid*
Brain*/diagnostic imaging
Diprenorphine ; Positron-Emission Tomography ; Receptors, Opioid, mu
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Distinct Profiles of Desensitization of µ-Opioid Receptors Caused by Remifentanil or Fentanyl: In Vitro Assay with Cells and Three-Dimensional Structural Analyses.
Autorzy:
Uezono E; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.
Mizobuchi Y; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.; Department of Anesthesiology and Resuscitology, Okayama University Graduate School of Medicine, Dentistry and Pharmaceutical Sciences, Okayama 700-0194, Japan.
Miyano K; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.; Division of Cancer Pathophysiology, National Cancer Center Research Institute, Tokyo 104-0045, Japan.; Department of Dentistry, National Cancer Center Hospital, Tokyo 104-0045, Japan.
Ohbuchi K; Tsumura Research Laboratories, Tsumura and Co., Ibaraki 300-1192, Japan.
Murata H; Department of Anesthesiology and Intensive Care Medicine, Nagasaki University Graduate School of Biomedical Sciences, Nagasaki 852-8501, Japan.
Komatsu A; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.
Manabe S; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.; Department of Anesthesiology and Resuscitology, Okayama University Graduate School of Medicine, Dentistry and Pharmaceutical Sciences, Okayama 700-0194, Japan.
Nonaka M; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.; Division of Cancer Pathophysiology, National Cancer Center Research Institute, Tokyo 104-0045, Japan.
Hirokawa T; Chemical Biology and In Silico Drug Design, Division of Biomedical Science, Faculty of Medicine, University of Tsukuba, Tsukuba 305-8575, Japan.
Yamaguchi K; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Anesthesiology and Pain Medicine, Juntendo Tokyo Koto Geriatric Medical Center, Tokyo 136-0075, Japan.
Iseki M; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.
Uezono Y; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, Tokyo 105-8461, Japan.; Division of Cancer Pathophysiology, National Cancer Center Research Institute, Tokyo 104-0045, Japan.; Department of Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Supportive and Palliative Care Research Support Office, National Cancer Center Hospital East, Chiba 277-8577, Japan.
Hayashida M; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.
Kawagoe I; Department of Anesthesiology and Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.; Department of Pain Medicine, Juntendo University Graduate School of Medicine, Tokyo 113-8421, Japan.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 May 06; Vol. 24 (9). Date of Electronic Publication: 2023 May 06.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid*/metabolism
Fentanyl*/pharmacology
Remifentanil/pharmacology ; Receptors, Opioid, mu/metabolism ; Analgesics, Opioid/pharmacology ; beta-Arrestins/metabolism ; Morphine
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Three-Dimensional Structural Insights Have Revealed the Distinct Binding Interactions of Agonists, Partial Agonists, and Antagonists with the µ Opioid Receptor.
Autorzy:
Li Z; National Center for Toxicological Research, US Food and Drug Administration, Jefferson, AR 72079, USA.
Liu J; National Center for Toxicological Research, US Food and Drug Administration, Jefferson, AR 72079, USA.
Dong F; National Center for Toxicological Research, US Food and Drug Administration, Jefferson, AR 72079, USA.
Chang N; Center for Drug Evaluation and Research, US Food and Drug Administration, Silver Spring, MD 20903, USA.
Huang R; National Center for Advancing Translational Sciences, National Institutes of Health, Bethesda, MD 20892, USA.
Xia M; National Center for Advancing Translational Sciences, National Institutes of Health, Bethesda, MD 20892, USA.
Patterson TA; National Center for Toxicological Research, US Food and Drug Administration, Jefferson, AR 72079, USA.
Hong H; National Center for Toxicological Research, US Food and Drug Administration, Jefferson, AR 72079, USA.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Apr 11; Vol. 24 (8). Date of Electronic Publication: 2023 Apr 11.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Receptors, Opioid*
Analgesics, Opioid*/metabolism
Humans ; Analgesics ; Pain ; Binding Sites ; Receptors, Opioid, mu/metabolism
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Identification of the Putative Binding Site of a Benzimidazole Opioid (Etazene) and Its Metabolites at µ-Opioid Receptor: A Human Liver Microsomal Assay and Systematic Computational Study.
Autorzy:
Chaturvedi K; Department of Chemistry and Biochemistry, University of Mississippi, University, MS 38677, USA.
Hewamanna I; Department of Chemistry and Biochemistry, University of Mississippi, University, MS 38677, USA.
Pandey P; National Center for Natural Products Research, University of Mississippi, University, MS 38677, USA.
Khan W; National Center for Natural Products Research, University of Mississippi, University, MS 38677, USA.
Wang YH; National Center for Natural Products Research, University of Mississippi, University, MS 38677, USA.
Chittiboyina AG; National Center for Natural Products Research, University of Mississippi, University, MS 38677, USA.
Doerksen RJ; Division of Medicinal Chemistry, Department of BioMolecular Sciences, School of Pharmacy, University of Mississippi, University, MS 38677, USA.
Godfrey M; Department of Chemistry and Biochemistry, University of Mississippi, University, MS 38677, USA.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Feb 07; Vol. 28 (4). Date of Electronic Publication: 2023 Feb 07.
Typ publikacji:
Journal Article
MeSH Terms:
Analgesics, Opioid*/chemistry
Receptors, Opioid*
Humans ; Microsomes, Liver/metabolism ; Molecular Docking Simulation ; Receptors, Opioid, mu/metabolism ; Binding Sites ; Liver/metabolism ; Benzimidazoles
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Role of kappa-opioid and mu-opioid receptors in pruritus: Peripheral and central itch circuits.
Autorzy:
Kim BS; Kimberly and Eric J. Waldman Department of Dermatology, Mark Lebwohl Center for Neuroinflammation and Sensation, Marc and Jennifer Lipschultz Precision Immunology Institute, and Friedman Brain Institute, Icahn School of Medicine at Mount Sinai, New York, New York, USA.
Inan S; Center for Substance Abuse Research, Lewis Katz School of Medicine, Temple University, Philadelphia, Pennsylvania, USA.
Ständer S; Department of Dermatology and Center for Chronic Pruritus, University Hospital Műnster, Műnster, Germany.
Sciascia T; Trevi Therapeutics, Inc., New Haven, Connecticut, USA.
Szepietowski JC; Department of Dermatology, Venereology, and Allergology, Wroclaw Medical University, Wroclaw, Poland.
Yosipovitch G; Dr Phillip Frost Department of Dermatology and Cutaneous Surgery, Miami Itch Center, Miller School of Medicine, University of Miami, Miami, Florida, USA.
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Źródło:
Experimental dermatology [Exp Dermatol] 2022 Dec; Vol. 31 (12), pp. 1900-1907. Date of Electronic Publication: 2022 Sep 23.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptors, Opioid, mu*/genetics
Analgesics, Opioid*/pharmacology
Analgesics, Opioid*/therapeutic use
Animals ; Pruritus/drug therapy ; Pruritus/metabolism ; Receptors, Opioid, kappa/metabolism ; Receptors, Opioid, kappa/therapeutic use ; Receptors, Opioid
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Sucrose drinking mimics effects of nucleus accumbens µ-opioid receptor stimulation on fat intake and brain c-Fos-expression.
Autorzy:
Koekkoek LL; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Masís-Vargas A; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Kool T; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Eggels L; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
van der Gun LL; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Lamuadni K; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Slomp M; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Diepenbroek C; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
Kalsbeek A; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Hypothalamic Integration Mechanisms, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
la Fleur SE; Laboratory of Endocrinology, Department of Clinical Chemistry, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Amsterdam Neuroscience, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Department of Endocrinology and Metabolism, Amsterdam University Medical Center, Location AMC, University of Amsterdam, Neuroscience Amsterdam, Amsterdam Gastroenterology, Endocrinology and Metabolism, Amsterdam, The Netherlands.; Metabolism and Reward Group, Netherlands Institute for Neuroscience, Institute of the Royal Netherlands Academy of Arts and Sciences, Amsterdam, The Netherlands.
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Źródło:
Nutritional neuroscience [Nutr Neurosci] 2022 Nov; Vol. 25 (11), pp. 2408-2420. Date of Electronic Publication: 2021 Sep 07.
Typ publikacji:
Journal Article
MeSH Terms:
Nucleus Accumbens*/metabolism
Receptors, Opioid*/metabolism
Animals ; Rats ; Brain/metabolism ; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/pharmacology ; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/metabolism ; Rats, Sprague-Dawley ; Receptors, Opioid, mu/agonists ; Receptors, Opioid, mu/metabolism ; Sucrose ; Water ; Proto-Oncogene Proteins c-fos
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Endometriosis and Opioid Receptors: Are Opioids a Possible/Promising Treatment for Endometriosis?
Autorzy:
Guan Q; Department of Gynecology Charité with Center of Oncological Surgery, Endometriosis Research Center Charité, Campus Virchow-Klinikum, Augustenburger Platz 1, 13353 Berlin, Germany.
Velho RV; Department of Gynecology Charité with Center of Oncological Surgery, Endometriosis Research Center Charité, Campus Virchow-Klinikum, Augustenburger Platz 1, 13353 Berlin, Germany.
Sehouli J; Department of Gynecology Charité with Center of Oncological Surgery, Endometriosis Research Center Charité, Campus Virchow-Klinikum, Augustenburger Platz 1, 13353 Berlin, Germany.
Mechsner S; Department of Gynecology Charité with Center of Oncological Surgery, Endometriosis Research Center Charité, Campus Virchow-Klinikum, Augustenburger Platz 1, 13353 Berlin, Germany.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Jan 13; Vol. 24 (2). Date of Electronic Publication: 2023 Jan 13.
Typ publikacji:
Journal Article; Review
MeSH Terms:
Receptors, Opioid*/agonists
Endometriosis*/drug therapy
Female ; Humans ; Analgesics, Opioid/adverse effects ; Pain/drug therapy ; Analgesics/therapeutic use ; Receptors, Opioid, mu/agonists
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Solving an Old Puzzle: Elucidation and Evaluation of the Binding Mode of Salvinorin A at the Kappa Opioid Receptor.
Autorzy:
Puls K; Department of Biology, Chemistry and Pharmacy, Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, 14195 Berlin, Germany.
Wolber G; Department of Biology, Chemistry and Pharmacy, Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, 14195 Berlin, Germany.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2023 Jan 11; Vol. 28 (2). Date of Electronic Publication: 2023 Jan 11.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid, kappa*/metabolism
Diterpenes, Clerodane*/chemistry
Humans ; Receptors, Opioid ; Analgesics ; Analgesics, Opioid/chemistry
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
Opioid-Modulated Receptor Localization and Erk1/2 Phosphorylation in Cells Coexpressing μ-Opioid and Nociceptin Receptors.
Autorzy:
Zhuo GY; Institute of Translational Medicine and New Drug Development, China Medical University, Taichung 40402, Taiwan.
Chen MC; Institute of Translational Medicine and New Drug Development, China Medical University, Taichung 40402, Taiwan.
Lin TY; Center for Drug Abuse and Addiction, China Medical University Hospital, Taichung 40447, Taiwan.
Lin ST; Integrative Stem Cell Center, China Medical University Hospital, Taichung 40447, Taiwan.
Chen DT; School of Chinese Medicine, China Medical University, Taichung 40402, Taiwan.; Graduate Institute of Biomedical Sciences, China Medical University, Taichung 40402, Taiwan.
Lee CW; Center for Drug Abuse and Addiction, China Medical University Hospital, Taichung 40447, Taiwan.; Graduate Institute of Biomedical Sciences, China Medical University, Taichung 40402, Taiwan.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Jan 05; Vol. 24 (2). Date of Electronic Publication: 2023 Jan 05.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid*/metabolism
Buprenorphine*/pharmacology
Humans ; Nociceptin Receptor ; Analgesics, Opioid/pharmacology ; HEK293 Cells ; Phosphorylation ; Receptors, Opioid, mu/metabolism ; Morphine/pharmacology
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknie Pełny tekstSzczegóły
Tytuł:
-Acetyl β-Endorphin Is an Endogenous Ligand of σ1Rs That Regulates Mu-Opioid Receptor Signaling by Exchanging G Proteins for σ2Rs in σ1R Oligomers.N -Acetyl β-Endorphin Is an Endogenous Ligand of σ1Rs That Regulates Mu-Opioid Receptor Signaling by Exchanging G Proteins for σ2Rs in σ1R Oligomers.
Autorzy:
Garzón-Niño J; Neuropharmacology, Department of Translational Neuroscience, Cajal Institute, CSIC, 28002 Madrid, Spain.
Cortés-Montero E; Neuropharmacology, Department of Translational Neuroscience, Cajal Institute, CSIC, 28002 Madrid, Spain.
Rodríguez-Muñoz M; Neuropharmacology, Department of Translational Neuroscience, Cajal Institute, CSIC, 28002 Madrid, Spain.
Sánchez-Blázquez P; Neuropharmacology, Department of Translational Neuroscience, Cajal Institute, CSIC, 28002 Madrid, Spain.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Dec 29; Vol. 24 (1). Date of Electronic Publication: 2022 Dec 29.
Typ publikacji:
Journal Article
MeSH Terms:
beta-Endorphin*/metabolism
Receptors, Opioid, mu*/metabolism
Receptors, sigma*/metabolism
Animals ; Mice ; GTP-Binding Proteins/metabolism ; Ligands ; Morphine/pharmacology ; Pain ; Receptors, Opioid/metabolism
Czasopismo naukowe
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Tytuł:
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors.
Autorzy:
Wtorek K; Department of Biomolecular Chemistry, Medical University of Lodz, Mazowiecka 6/8, 92-215 Lodz, Poland.
Ghidini A; Department of Chemistry 'G. Ciamician', University of Bologna, Via Selmi 2, 40126 Bologna, Italy.
Gentilucci L; Department of Chemistry 'G. Ciamician', University of Bologna, Via Selmi 2, 40126 Bologna, Italy.
Adamska-Bartłomiejczyk A; Department of Biomolecular Chemistry, Medical University of Lodz, Mazowiecka 6/8, 92-215 Lodz, Poland.
Piekielna-Ciesielska J; Department of Biomolecular Chemistry, Medical University of Lodz, Mazowiecka 6/8, 92-215 Lodz, Poland.
Ruzza C; Department of Neuroscience and Rehabilitation, University of Ferrara, 44121 Ferrara, Italy.
Sturaro C; Department of Neuroscience and Rehabilitation, University of Ferrara, 44121 Ferrara, Italy.
Calò G; Department of Pharmaceutical and Pharmacological Sciences, University of Padova, Largo Meneghetti 2, 35131 Padova, Italy.
Pieretti S; Istituto Superiore di Sanità, National Center for Drug Research and Evaluation, 00161 Rome, Italy.
Kluczyk A; Faculty of Chemistry, University of Wroclaw, 50-383 Wroclaw, Poland.
McDonald J; Department of Cardiovascular Sciences, University of Leicester, Anaesthesia, Critical Care and Pain Management, Leicester Royal Infirmary, Leicester LE2 7LX, UK.
Lambert DG; Department of Cardiovascular Sciences, University of Leicester, Anaesthesia, Critical Care and Pain Management, Leicester Royal Infirmary, Leicester LE2 7LX, UK.
Janecka A; Department of Biomolecular Chemistry, Medical University of Lodz, Mazowiecka 6/8, 92-215 Lodz, Poland.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Oct 21; Vol. 23 (20). Date of Electronic Publication: 2022 Oct 21.
Typ publikacji:
Journal Article
MeSH Terms:
Analgesics, Opioid*/therapeutic use
Receptors, Opioid*/agonists
Animals ; Mice ; Receptors, Opioid, kappa ; Narcotic Antagonists/pharmacology ; Receptors, Opioid, mu/agonists ; Molecular Docking Simulation ; Ligands ; Dose-Response Relationship, Drug ; Naloxone ; Analgesics/pharmacology ; Peptides/pharmacology ; Chimera ; Peptides, Cyclic
Czasopismo naukowe
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Tytuł:
Opioid receptor μ, not δ and κ, modulate food intake induced by ghrelin in laying chickens.
Autorzy:
Baghaeikia S; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
Fallah H; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
Khodadadi M; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
Yousefvand S; Basic Sciences Department, Faculty of the Veterinary Medicine, Ferdowsi University of Mashhad, Mashhad, 9177948974, Iran.
Mahdavi K; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
Zendehdel M; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
Rahmani B; Basic Sciences Department, Faculty of the Veterinary Medicine, University of Tehran, Tehran, 1419963111, Iran.
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Źródło:
Canadian journal of physiology and pharmacology [Can J Physiol Pharmacol] 2022 Oct 01; Vol. 100 (10), pp. 983-992. Date of Electronic Publication: 2022 Jul 12.
Typ publikacji:
Journal Article
MeSH Terms:
Ghrelin*/metabolism
Ghrelin*/pharmacology
Receptors, Opioid*/metabolism
Analgesics, Opioid/metabolism ; Animals ; Chickens/metabolism ; Eating ; Receptors, Opioid, kappa/metabolism ; Receptors, Opioid, mu/metabolism
Czasopismo naukowe
Pełny tekst  Link otwiera się w nowym oknieSzczegóły
Tytuł:
OPRM1 Gene Polymorphism in Women with Alcohol Use Disorder.
Autorzy:
Boroń A; Department of Clinical and Molecular Biochemistry, Pomeranian Medical University in Szczecin, Powstańców Wielkopolskich 72 St., 70-111 Szczecin, Poland.
Suchanecka A; Independent Laboratory of Health Promotion, Pomeranian Medical University in Szczecin, Powstańców Wielkopolskich 72 St., 70-111 Szczecin, Poland.
Chmielowiec K; Department of Hygiene and Epidemiology, Collegium Medicum, University of Zielona Góra, 28 Zyty St., 65-045 Zielona Góra, Poland.
Śmiarowska M; Individual Specialized Medical Practice, Swarożyca 3/6 St., 71-601 Szczecin, Poland.
Chmielowiec J; Department of Hygiene and Epidemiology, Collegium Medicum, University of Zielona Góra, 28 Zyty St., 65-045 Zielona Góra, Poland.
Strońska-Pluta A; Independent Laboratory of Health Promotion, Pomeranian Medical University in Szczecin, Powstańców Wielkopolskich 72 St., 70-111 Szczecin, Poland.
Recław R; Foundation Strong in the Spirit, 60 Sienkiewicza St., 90-058 Łódź, Poland.
Grzywacz A; Independent Laboratory of Health Promotion, Pomeranian Medical University in Szczecin, Powstańców Wielkopolskich 72 St., 70-111 Szczecin, Poland.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2024 Mar 06; Vol. 25 (5). Date of Electronic Publication: 2024 Mar 06.
Typ publikacji:
Journal Article
MeSH Terms:
Alcoholism*/genetics
Alcoholism*/psychology
Genetic Predisposition to Disease*
Receptors, Opioid, mu*/genetics
Personality*
Female ; Humans ; Ethanol ; Genotype ; Polymorphism, Single Nucleotide
Czasopismo naukowe
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Tytuł:
Evaluation of the Intracellular Signaling Activities of κ-Opioid Receptor Agonists, Nalfurafine Analogs; Focusing on the Selectivity of G-Protein- and β-Arrestin-Mediated Pathways.
Autorzy:
Yamaguchi M; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.; Medical Affairs, Pfizer Japan Inc., 3-22-7 Yoyogi, Shibuya-ku, Tokyo 151-0053, Japan.
Miyano K; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.; Division of Cancer Pathophysiology, National Cancer Center Research Institute, 5-1-1 Tsukiji, Chuo-ku, Tokyo 104-0045, Japan.
Hirayama S; Laboratory of Medicinal Chemistry and Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1 Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Karasawa Y; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.; Medical Affairs, Viatris Pharmaceuticals Japan Inc., 5-11-2 Toranomon, Minato-ku, Tokyo 105-0001, Japan.
Ohshima K; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Uezono E; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.
Komatsu A; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.
Nonaka M; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.
Fujii H; Laboratory of Medicinal Chemistry and Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1 Shirokane, Minato-ku, Tokyo 108-8641, Japan.
Yamaguchi K; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.
Iseki M; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.
Hayashida M; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.
Uezono Y; Department of Pain Medicine, Juntendo University Graduate School of Medicine, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Department of Pain Control Research, The Jikei University School of Medicine, 3-25-8 Nishi-Shimbashi, Minato-ku, Tokyo 105-8461, Japan.; Department of Anesthesiology and Pain Medicine, Faculty of Medicine, Juntendo University, 2-1-1 Hongo, Bunkyo-ku, Tokyo 113-8421, Japan.; Supportive and Palliative Care Research Support Office, National Cancer Center Hospital East, 6-5-1 Kashiwanoha, Kashiwa-shi, Chiba 277-8577, Japan.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Oct 19; Vol. 27 (20). Date of Electronic Publication: 2022 Oct 19.
Typ publikacji:
Journal Article
MeSH Terms:
Analgesics, Opioid*/pharmacology
Receptors, Opioid, kappa*/agonists
Analgesics ; beta-Arrestins/metabolism ; GTP-Binding Proteins/metabolism ; Receptors, Opioid, mu/metabolism
Czasopismo naukowe
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Tytuł:
Opioid receptor activation modulates the calcium current in the cochlear outer hair cells of the rat.
Autorzy:
Vega R; Instituto de Fisiología, Benemérita Universidad Autónoma de Puebla, Puebla, Mexico.
García-Garibay O; Instituto de Fisiología, Benemérita Universidad Autónoma de Puebla, Puebla, Mexico.
Soto E; Instituto de Fisiología, Benemérita Universidad Autónoma de Puebla, Puebla, Mexico.
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Źródło:
The European journal of neuroscience [Eur J Neurosci] 2022 Jul; Vol. 56 (1), pp. 3543-3552. Date of Electronic Publication: 2022 May 10.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Receptors, Opioid*
Receptors, Opioid, kappa*
3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer/pharmacology ; Analgesics, Opioid ; Animals ; Calcium/metabolism ; Enkephalin, Ala(2)-MePhe(4)-Gly(5)- ; Hair Cells, Auditory, Outer/metabolism ; Opioid Peptides ; Rats ; Receptors, Opioid, mu/agonists
Czasopismo naukowe
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Tytuł:
Mu and Delta Opioid Receptor Targeting Reduces Connexin 43-Based Heterocellular Coupling during Neuropathic Pain.
Autorzy:
Vicario N; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Denaro S; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Turnaturi R; Section of Medicinal Chemistry, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.
Longhitano L; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.; Section of Biochemistry, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Spitale FM; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Spoto S; Section of Pharmacology and Toxicology, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.
Marrazzo A; Section of Medicinal Chemistry, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.
Zappalà A; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Tibullo D; Section of Biochemistry, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Li Volti G; Section of Biochemistry, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Chiechio S; Section of Pharmacology and Toxicology, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.; Oasi Research Institute-IRCCS, 94018 Troina, Italy.
Pasquinucci L; Section of Medicinal Chemistry, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.
Parenti R; Section of Physiology, Department of Biomedical and Biotechnological Sciences, University of Catania, 95123 Catania, Italy.
Parenti C; Section of Pharmacology and Toxicology, Department of Drug and Health Sciences, University of Catania, 95123 Catania, Italy.
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Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 May 24; Vol. 23 (11). Date of Electronic Publication: 2022 May 24.
Typ publikacji:
Journal Article
MeSH Terms:
Neuralgia*/drug therapy
Receptors, Opioid, delta*
Analgesics, Opioid/pharmacology ; Connexin 43/therapeutic use ; Humans ; Hyperalgesia/drug therapy ; Receptors, Opioid ; Receptors, Opioid, mu ; Spinal Cord
Czasopismo naukowe
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Tytuł:
Novel 1-(1-Arylimiazolin-2-Yl)-3-Arylalkilurea Derivatives with Modulatory Activity on Opioid MOP Receptors.
Autorzy:
Straszak D; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University, Chodzki 4A, 20-093 Lublin, Poland.
Woźniak S; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University, Chodzki 4A, 20-093 Lublin, Poland.
Siwek A; Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
Głuch-Lutwin M; Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
Kołaczkowski M; Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
Pietrzak A; Department of Dermatology, Venereology, and Paediatric Dermatology, Faculty of Medicine, Medical University, Staszica 11, 20-080 Lublin, Poland.
Drop B; Department of Medical Informatics and Statistics, Medical University, Jaczewskiego 4, 20-090 Lublin, Poland.
Matosiuk D; Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy, Medical University, Chodzki 4A, 20-093 Lublin, Poland.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2024 Jan 24; Vol. 29 (3). Date of Electronic Publication: 2024 Jan 24.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid*/metabolism
Receptors, Opioid, mu*/metabolism
Humans ; Analgesics, Opioid/adverse effects ; Analgesics/pharmacology ; beta-Arrestins/metabolism
Czasopismo naukowe
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Tytuł:
Computational Methods for Understanding the Selectivity and Signal Transduction Mechanism of Aminomethyl Tetrahydronaphthalene to Opioid Receptors.
Autorzy:
Xie P; School of Pharmacy, Fudan University, Shanghai 201301, China.; Novel Technology Center of Chemical Pharmaceutics, Shanghai Institute of Pharmaceutical Industry Co., Ltd., China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai 201203, China.
Zhang J; School of Pharmacy, Fudan University, Shanghai 201301, China.
Chen B; School of Pharmacy, Fudan University, Shanghai 201301, China.
Li X; School of Pharmacy, Fudan University, Shanghai 201301, China.
Zhang W; Novel Technology Center of Chemical Pharmaceutics, Shanghai Institute of Pharmaceutical Industry Co., Ltd., China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai 201203, China.
Zhu M; School of Pharmacy, Fudan University, Shanghai 201301, China.
Li W; School of Pharmacy, Fudan University, Shanghai 201301, China.
Li J; Novel Technology Center of Chemical Pharmaceutics, Shanghai Institute of Pharmaceutical Industry Co., Ltd., China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai 201203, China.
Fu W; School of Pharmacy, Fudan University, Shanghai 201301, China.
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2022 Mar 28; Vol. 27 (7). Date of Electronic Publication: 2022 Mar 28.
Typ publikacji:
Journal Article
MeSH Terms:
Receptors, Opioid*/metabolism
Receptors, Opioid, delta*/metabolism
Molecular Dynamics Simulation ; Receptors, Opioid, mu/metabolism ; Signal Transduction ; Structure-Activity Relationship ; Tetrahydronaphthalenes
Czasopismo naukowe
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Wyświetlanie 1-20 z 2081

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