Informacja

Drogi użytkowniku, aplikacja do prawidłowego działania wymaga obsługi JavaScript. Proszę włącz obsługę JavaScript w Twojej przeglądarce.

Wyszukujesz frazę ""Reinoso RF"" wg kryterium: Autor


Wyświetlanie 1-7 z 7
Tytuł:
EST79232 and EST79376, Two Novel Sigma-1 Receptor Ligands, Exert Neuroprotection on Models of Motoneuron Degeneration.
Autorzy:
Gaja-Capdevila N; Department of Cell Biology, Physiology and Immunology, Institute of Neurosciences, Universitat Autònoma de Barcelona, 01893 Bellaterra, Spain.; Centro de Investigación Biomédica en Red Sobre Enfermedades Neurodegenerativas (CIBERNED), 28031 Madrid, Spain.
Hernández N; Department of Cell Biology, Physiology and Immunology, Institute of Neurosciences, Universitat Autònoma de Barcelona, 01893 Bellaterra, Spain.; Centro de Investigación Biomédica en Red Sobre Enfermedades Neurodegenerativas (CIBERNED), 28031 Madrid, Spain.
Yeste S; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Reinoso RF; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Burgueño J; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Montero A; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Merlos M; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Vela JM; Welab Barcelona, Parc Científic Barcelona, 08028 Barcelona, Spain.
Herrando-Grabulosa M; Department of Cell Biology, Physiology and Immunology, Institute of Neurosciences, Universitat Autònoma de Barcelona, 01893 Bellaterra, Spain.; Centro de Investigación Biomédica en Red Sobre Enfermedades Neurodegenerativas (CIBERNED), 28031 Madrid, Spain.
Navarro X; Department of Cell Biology, Physiology and Immunology, Institute of Neurosciences, Universitat Autònoma de Barcelona, 01893 Bellaterra, Spain.; Centro de Investigación Biomédica en Red Sobre Enfermedades Neurodegenerativas (CIBERNED), 28031 Madrid, Spain.
Pokaż więcej
Źródło:
International journal of molecular sciences [Int J Mol Sci] 2022 Jun 16; Vol. 23 (12). Date of Electronic Publication: 2022 Jun 16.
Typ publikacji:
Journal Article
MeSH Terms:
Amyotrophic Lateral Sclerosis*/metabolism
Animals ; Disease Models, Animal ; Ligands ; Mice ; Mice, Transgenic ; Motor Neurons/metabolism ; Neuroprotection ; Receptors, sigma ; Spinal Cord/metabolism ; Superoxide Dismutase/metabolism ; Superoxide Dismutase-1/metabolism ; Sigma-1 Receptor
Czasopismo naukowe
Tytuł:
Preliminary in vitro approach to evaluate the drug-drug interaction potential of EST73502, a dual µ-opioid receptor partial agonist and σ1 receptor antagonist.
Autorzy:
Ayet E; WELAB, Parc Científic Barcelona, Baldiri Reixac 4-8, Barcelona 08028, Spain.
Yeste S; WELAB, Parc Científic Barcelona, Baldiri Reixac 4-8, Barcelona 08028, Spain.
Reinoso RF; WELAB, Parc Científic Barcelona, Baldiri Reixac 4-8, Barcelona 08028, Spain.
Pretel MJ; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals S.A, Barcelona, Spain.
Balada A; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals S.A, Barcelona, Spain.
Serafini MT; WELAB, Parc Científic Barcelona, Baldiri Reixac 4-8, Barcelona 08028, Spain.
Pokaż więcej
Źródło:
Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2021 May; Vol. 51 (5), pp. 501-512. Date of Electronic Publication: 2021 Feb 23.
Typ publikacji:
Journal Article
MeSH Terms:
Pharmaceutical Preparations*
Receptors, sigma*
Caco-2 Cells ; Drug Interactions ; Humans ; Receptors, Opioid, mu/agonists ; Sigma-1 Receptor
Czasopismo naukowe
Tytuł:
Preliminary in vitro assessment of pharmacokinetic drug-drug interactions of EST64401 and EST64514, two sigma-1 receptor antagonists.
Autorzy:
Reinoso RF; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Yeste S; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Ayet E; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Pretel MJ; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Balada A; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Serafini MT; Early ADME, Drug Discovery and Preclinical Development, ESTEVE Pharmaceuticals, Barcelona, Spain.
Pokaż więcej
Źródło:
Xenobiotica; the fate of foreign compounds in biological systems [Xenobiotica] 2021 Apr; Vol. 51 (4), pp. 373-386. Date of Electronic Publication: 2021 Jan 20.
Typ publikacji:
Journal Article
MeSH Terms:
Cytochrome P-450 Enzyme Inhibitors*
Pharmaceutical Preparations*
ATP Binding Cassette Transporter, Subfamily G, Member 2 ; Caco-2 Cells ; Drug Interactions ; Humans ; Microsomes, Liver ; Neoplasm Proteins ; Receptors, sigma ; Sigma-1 Receptor
Czasopismo naukowe
Tytuł:
Synthesis and pharmacological evaluation of fluorinated benzo[7]annulen-7-amines as GluN2B-selective NMDA receptor antagonists.
Autorzy:
Thum S; Institute of Pharmaceutical and Medicinal Chemistry, Westfälische Wilhelms-Universität Münster, Münster, Germany.
Schepmann D; Institute of Pharmaceutical and Medicinal Chemistry, Westfälische Wilhelms-Universität Münster, Münster, Germany.
Reinoso RF; Esteve Pharmaceuticals, Barcelona, Spain.
Alvarez I; Esteve Pharmaceuticals, Barcelona, Spain.
Ametamey SM; Center for Radiopharmaceutical Science of ETH, PSI, and USZ, ETH-Hönggerberg, Zürich, Switzerland.
Wünsch B; Institute of Pharmaceutical and Medicinal Chemistry, Westfälische Wilhelms-Universität Münster, Münster, Germany.; Cells-in-Motion Cluster of Excellence (EXC 1003-CiM), Westfälische Wilhelms-Universität Münster, Germany.
Pokaż więcej
Źródło:
Journal of labelled compounds & radiopharmaceuticals [J Labelled Comp Radiopharm] 2019 Jun 30; Vol. 62 (8), pp. 354-379.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Halogenation*
Amines/*chemical synthesis
Amines/*pharmacology
Receptors, N-Methyl-D-Aspartate/*antagonists & inhibitors
Amines/chemistry ; Amines/metabolism ; Chemistry Techniques, Synthetic ; Receptors, N-Methyl-D-Aspartate/metabolism ; Substrate Specificity
Czasopismo naukowe
    Wyświetlanie 1-7 z 7

    Ta witryna wykorzystuje pliki cookies do przechowywania informacji na Twoim komputerze. Pliki cookies stosujemy w celu świadczenia usług na najwyższym poziomie, w tym w sposób dostosowany do indywidualnych potrzeb. Korzystanie z witryny bez zmiany ustawień dotyczących cookies oznacza, że będą one zamieszczane w Twoim komputerze. W każdym momencie możesz dokonać zmiany ustawień dotyczących cookies