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Wyszukujesz frazę ""Sévigny, Jean"" wg kryterium: Autor


Wyświetlanie 1-13 z 13
Tytuł:
Tricyclic coumarin sulphonate derivatives with alkaline phosphatase inhibitory effects: in vitro and docking studies.
Autorzy:
Iqbal J; a Centre for Advanced Drug Research , COMSATS Institute of Information Technology , Abbottabad , Pakistan.
El-Gamal MI; b Department of Medicinal Chemistry, College of Pharmacy , University of Sharjah , Sharjah , United Arab Emirates.; c Sharjah Institute for Medical Research , University of Sharjah , Sharjah , United Arab Emirates.; d Department of Medicinal Chemistry , University of Mansoura , Mansoura , Egypt.
Ejaz SA; a Centre for Advanced Drug Research , COMSATS Institute of Information Technology , Abbottabad , Pakistan.
Lecka J; e Département de microbiologie-infectiologie et d'immunologie, Faculté de Médecine , Université Laval , Québec , Canada.; f Centre de Recherche du CHU de Québec , Université Laval , Québec , Canada.
Sévigny J; e Département de microbiologie-infectiologie et d'immunologie, Faculté de Médecine , Université Laval , Québec , Canada.; f Centre de Recherche du CHU de Québec , Université Laval , Québec , Canada.
Oh CH; g Center for Biomaterials , Korea Institute of Science and Technology , Seoul , Republic of Korea.; h Department of Biomolecular Science , University of Science and Technology , Daejeon , Republic of Korea.
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Źródło:
Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2018 Dec; Vol. 33 (1), pp. 479-484.
Typ publikacji:
Journal Article
MeSH Terms:
Molecular Docking Simulation*
Alkaline Phosphatase/*antagonists & inhibitors
Coumarins/*pharmacology
Enzyme Inhibitors/*pharmacology
Sulfonic Acids/*pharmacology
Alkaline Phosphatase/metabolism ; Coumarins/chemical synthesis ; Coumarins/chemistry ; Dose-Response Relationship, Drug ; Enzyme Inhibitors/chemical synthesis ; Enzyme Inhibitors/chemistry ; GPI-Linked Proteins/antagonists & inhibitors ; GPI-Linked Proteins/metabolism ; Humans ; Molecular Structure ; Structure-Activity Relationship ; Sulfonic Acids/chemical synthesis ; Sulfonic Acids/chemistry
Czasopismo naukowe
Tytuł:
Isonicotinohydrazones as inhibitors of alkaline phosphatase and ecto-5'-nucleotidase.
Autorzy:
Channar PA; Department of Chemistry, Quaid-I-Azam University, Islamabad, Pakistan.
Shah SJ; Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan.
Hassan S; Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan.
Nisa ZU; Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan.
Lecka J; Département de microbiologie-infectiologie et d'immunologie, Faculté de Médecine, Université Laval, Québec, QC, Canada.; Centre de Recherche du CHU de Québec - Université Laval, Québec, QC, Canada.
Sévigny J; Département de microbiologie-infectiologie et d'immunologie, Faculté de Médecine, Université Laval, Québec, QC, Canada.; Centre de Recherche du CHU de Québec - Université Laval, Québec, QC, Canada.
Bajorath J; Department of Life Science Informatics, B-IT, LIMES Program Unit Chemical Biology and Medicinal Chemistry, Rheinische Friedrich-Wilhelms-Universität, Bonn, Germany.
Saeed A; Department of Chemistry, Quaid-I-Azam University, Islamabad, Pakistan.
Iqbal J; Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan.
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Źródło:
Chemical biology & drug design [Chem Biol Drug Des] 2017 Mar; Vol. 89 (3), pp. 365-370. Date of Electronic Publication: 2016 Oct 26.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
5'-Nucleotidase/*antagonists & inhibitors
Alkaline Phosphatase/*antagonists & inhibitors
Enzyme Inhibitors/*chemistry
Enzyme Inhibitors/*pharmacology
5'-Nucleotidase/chemistry ; Alkaline Phosphatase/chemistry ; Animals ; Chemistry Techniques, Synthetic ; Drug Evaluation, Preclinical/methods ; Enzyme Inhibitors/chemical synthesis ; GPI-Linked Proteins/antagonists & inhibitors ; GPI-Linked Proteins/chemistry ; Humans ; Isoniazid/chemistry ; Models, Molecular ; Molecular Docking Simulation ; Protein Conformation ; Rats ; Structure-Activity Relationship
Czasopismo naukowe
Tytuł:
Characterization of a monoclonal antibody as the first specific inhibitor of human NTP diphosphohydrolase-3 : partial characterization of the inhibitory epitope and potential applications.
Autorzy:
Munkonda MN; Centre de Recherche en Rhumatologie et Immunologie, Centre Hospitalier Universitaire de Québec, Université Laval, Canada.
Pelletier J
Ivanenkov VV
Fausther M
Tremblay A
Künzli B
Kirley TL
Sévigny J
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Źródło:
The FEBS journal [FEBS J] 2009 Jan; Vol. 276 (2), pp. 479-96.
Typ publikacji:
Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
MeSH Terms:
Antibodies, Monoclonal/*immunology
Enzyme Inhibitors/*immunology
Enzyme Inhibitors/*pharmacology
Epitopes/*immunology
Pyrophosphatases/*antagonists & inhibitors
Pyrophosphatases/*immunology
Amino Acid Substitution ; Animals ; Antibody Formation/immunology ; Antibody Specificity ; Cell Line ; Chlorocebus aethiops ; Humans ; Mice ; Mice, Inbred BALB C ; Models, Molecular ; Pancreas/drug effects ; Pancreas/enzymology ; Pancreas/immunology ; Pancreas/metabolism ; Protein Structure, Tertiary ; Pyrophosphatases/metabolism ; Recombinant Proteins/antagonists & inhibitors ; Recombinant Proteins/genetics ; Recombinant Proteins/immunology ; Recombinant Proteins/metabolism
Czasopismo naukowe
Tytuł:
Inhibition of vascular ectonucleotidase activities by the pro-drugs ticlopidine and clopidogrel favours platelet aggregation.
Autorzy:
Lecka, Joanna
Rana, Manjit Singh
Sévigny, Jean
Sévigny, Jean
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Temat:
ENZYME inhibitors
PRODRUGS
TICLOPIDINE
CLOPIDOGREL
PLATELET aggregation inhibitors
BIOLOGY experiments
NUCLEOTIDES
Źródło:
British Journal of Pharmacology; Nov2010, Vol. 161 Issue 5, p1150-1160, 11p
Czasopismo naukowe
Tytuł:
Investigation of new quinoline derivatives as promising inhibitors of NTPDases: Synthesis, SAR analysis and molecular docking studies.
Autorzy:
Hayat, Komal (AUTHOR)
Afzal, Saira (AUTHOR)
Saeed, Altaf (AUTHOR)
Murtaza, Amna (AUTHOR)
Ur Rahman, Shafiq (AUTHOR)
Khan, Khalid Mohammed (AUTHOR)
Saeed, Aamer (AUTHOR)
Zaib, Sumera (AUTHOR)
Lecka, Joanna (AUTHOR)
Sévigny, Jean (AUTHOR)
Iqbal, Jamshed (AUTHOR)
Hassan, Abbas (AUTHOR)
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Źródło:
Bioorganic Chemistry. Jun2019, Vol. 87, p218-226. 9p.
Czasopismo naukowe
Tytuł:
Hybrid compounds from chalcone and 1,2-benzothiazine pharmacophores as selective inhibitors of alkaline phosphatase isozymes.
Autorzy:
Hartinger, Christian G.
Hanif, Muhammad
Ashraf, Adnan
Siddiqui, Waseeq Ahmad
Ejaz, Syeda Abida
Rahman, Shafiq Ur
Iqbal, Jamshed
Zayed, Mohie E. Moustafa
Arshad, Muhammad Nadeem
Asiri, Abdullah M.
Lecka, Joanna
Sévigny, Jean
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Źródło:
European Journal of Medicinal Chemistry. Nov2018, Vol. 159, p282-291. 10p.
Czasopismo naukowe
Tytuł:
2-Substituted 7-trifluoromethyl-thiadiazolopyrimidones as alkaline phosphatase inhibitors. Synthesis, structure activity relationship and molecular docking study.
Autorzy:
Jafari, Behzad
Ospanov, Meirambek
Ejaz, Syeda Abida
Yelibayeva, Nazym
Khan, Shafi Ullah
Amjad, Sayyeda Tayyeba
Safarov, Sayfidin
Abilov, Zharylkasyn A.
Turmukhanova, Mirgul Zh.
Kalugin, Sergey N.
Ehlers, Peter
Lecka, Joanna
Sévigny, Jean
Iqbal, Jamshed
Langer, Peter
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Źródło:
European Journal of Medicinal Chemistry. Jan2018, Vol. 144, p116-127. 12p.
Czasopismo naukowe
Tytuł:
Structural investigation on thiazolo[5,4-d]pyrimidines to obtain dual-acting blockers of CD73 and adenosine A2A receptor as potential antitumor agents.
Autorzy:
Varano, Flavia (AUTHOR)
Catarzi, Daniela (AUTHOR)
Vincenzi, Fabrizio (AUTHOR)
Pasquini, Silvia (AUTHOR)
Pelletier, Julie (AUTHOR)
Lopes Rangel Fietto, Juliana (AUTHOR)
Espindola Gelsleichter, Nicolly (AUTHOR)
Sarlandie, Marine (AUTHOR)
Guilbaud, Audrey (AUTHOR)
Sévigny, Jean (AUTHOR)
Varani, Katia (AUTHOR)
Colotta, Vittoria (AUTHOR)
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Źródło:
Bioorganic & Medicinal Chemistry Letters. May2020, Vol. 30 Issue 9, pN.PAG-N.PAG. 1p.
Czasopismo naukowe
    Wyświetlanie 1-13 z 13

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