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Wyświetlanie 1-7 z 7
Tytuł:
Cellular and Molecular Effects of Eribulin in Preclinical Models of Hematologic Neoplasms.
Autorzy:
Vicari HP; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulos 05508-000, Brazil.
Lima K; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulos 05508-000, Brazil.; Laboratory of Medical Investigation in Pathogenesis and Targeted Therapy in Onco-Immuno-Hematology (LIM-31), Department of Internal Medicine, Hematology Division, Faculdade de Medicina, University of São Paulo, São Paulo 01246-903, Brazil.
Costa-Lotufo LV; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulos 05508-000, Brazil.
Machado-Neto JA; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulos 05508-000, Brazil.
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Źródło:
Cancers [Cancers (Basel)] 2022 Dec 10; Vol. 14 (24). Date of Electronic Publication: 2022 Dec 10.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Comprehensive analysis of cytoskeleton regulatory genes identifies ezrin as a prognostic marker and molecular target in acute myeloid leukemia.
Autorzy:
Lipreri da Silva JC; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, CEP 05508-900, São Paulo, SP, Brazil.
Coelho-Silva JL; Department of Medical Imaging, Hematology, and Oncology, Ribeirão Preto Medical School, University of São Paulo, Ribeirão Preto, Brazil.
Lima K; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, CEP 05508-900, São Paulo, SP, Brazil.
Vicari HP; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, CEP 05508-900, São Paulo, SP, Brazil.
Lazarini M; Department of Pharmaceutical Sciences, Federal University of São Paulo, Diadema, Brazil.
Costa-Lotufo LV; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, CEP 05508-900, São Paulo, SP, Brazil.
Traina F; Department of Medical Imaging, Hematology, and Oncology, Ribeirão Preto Medical School, University of São Paulo, Ribeirão Preto, Brazil.
Machado-Neto JA; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, CEP 05508-900, São Paulo, SP, Brazil. .
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Źródło:
Cellular oncology (Dordrecht) [Cell Oncol (Dordr)] 2021 Oct; Vol. 44 (5), pp. 1105-1117. Date of Electronic Publication: 2021 Jul 01.
Typ publikacji:
Journal Article
MeSH Terms:
Gene Expression Regulation, Leukemic*
Biomarkers, Tumor/*genetics
Cytoskeletal Proteins/*genetics
Cytoskeleton/*metabolism
Genes, Regulator/*genetics
Leukemia, Myeloid/*genetics
Acute Disease ; Adamantane/analogs & derivatives ; Adamantane/pharmacology ; Adult ; Biomarkers, Tumor/metabolism ; Cell Line, Tumor ; Cell Survival/drug effects ; Cell Survival/genetics ; Cytoskeletal Proteins/antagonists & inhibitors ; Cytoskeletal Proteins/metabolism ; Disease-Free Survival ; Female ; HL-60 Cells ; Humans ; K562 Cells ; Leukemia, Myeloid/diagnosis ; Leukemia, Myeloid/metabolism ; Male ; Phenols/pharmacology ; Prognosis ; Quinolines/pharmacology ; Quinolones/pharmacology ; THP-1 Cells ; U937 Cells
Czasopismo naukowe
Tytuł:
Targeting glioma cells by antineoplastic activity of reversine.
Autorzy:
Hirakata C; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
Lima K; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
De Almeida BO; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
De Miranda LBL; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
Florêncio KGD; Department of Physiology and Pharmacology, Drug Research and Development Center, Federal University of Ceará, Fortaleza, Ceará, CEP 60440-900, Brazil.
Furtado LC; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
Costa-Lotufo LV; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
Machado-Neto JA; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, CEP 05508-900, Brazil.
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Źródło:
Oncology letters [Oncol Lett] 2021 Aug; Vol. 22 (2), pp. 610. Date of Electronic Publication: 2021 Jun 15.
Typ publikacji:
Journal Article
Czasopismo naukowe
Tytuł:
Reversine exerts cytotoxic effects through multiple cell death mechanisms in acute lymphoblastic leukemia.
Autorzy:
Carlos JAEG; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, São Paulo, SP, CEP 05508-900, Brazil.
Lima K; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, São Paulo, SP, CEP 05508-900, Brazil.
Coelho-Silva JL; Department of Medical Images, Hematology and Clinical Oncology, University of São Paulo at Ribeirão Preto Medical School, Ribeirão Preto, São Paulo, SP, Brazil.
de Melo Alves-Paiva R; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, SP, Brazil.
Moreno NC; Department of Microbiology, Institute of Biomedical Sciences, University of São Paulo, São Paulo, SP, Brazil.
Vicari HP; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, São Paulo, SP, CEP 05508-900, Brazil.
de Souza Santos FP; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, SP, Brazil.
Hamerschlak N; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, SP, Brazil.
Costa-Lotufo LV; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, São Paulo, SP, CEP 05508-900, Brazil.
Traina F; Department of Medical Images, Hematology and Clinical Oncology, University of São Paulo at Ribeirão Preto Medical School, Ribeirão Preto, São Paulo, SP, Brazil.
Machado-Neto JA; Department of Pharmacology, Institute of Biomedical Sciences, University of São Paulo, Av. Prof. Lineu Prestes, 1524, São Paulo, SP, CEP 05508-900, Brazil. .
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Źródło:
Cellular oncology (Dordrecht) [Cell Oncol (Dordr)] 2020 Dec; Vol. 43 (6), pp. 1191-1201. Date of Electronic Publication: 2020 Aug 28.
Typ publikacji:
Journal Article
MeSH Terms:
Morpholines/*pharmacology
Precursor Cell Lymphoblastic Leukemia-Lymphoma/*pathology
Purines/*pharmacology
Apoptosis/drug effects ; Aurora Kinase B/metabolism ; Autophagy/drug effects ; Cell Cycle Checkpoints/drug effects ; Cell Death/drug effects ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Clone Cells ; DNA Damage ; Humans ; Precursor Cell Lymphoblastic Leukemia-Lymphoma/enzymology
Czasopismo naukowe
Tytuł:
Reversine exhibits antineoplastic activity in JAK2 -positive myeloproliferative neoplasms.
Autorzy:
Lima K; Department of Pharmacology, Biomedical Sciences Institute, University of São Paulo, São Paulo, Brazil.
Carlos JAEG; Department of Pharmacology, Biomedical Sciences Institute, University of São Paulo, São Paulo, Brazil.
Alves-Paiva RM; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, Brazil.
Vicari HP; Department of Pharmacology, Biomedical Sciences Institute, University of São Paulo, São Paulo, Brazil.
Souza Santos FP; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, Brazil.
Hamerschlak N; Einstein's Teaching and Research Institute, Albert Einstein Hospital, São Paulo, Brazil.
Costa-Lotufo LV; Department of Pharmacology, Biomedical Sciences Institute, University of São Paulo, São Paulo, Brazil.
Traina F; Department of Medical Images, Hematology and Clinical Oncology, University of São Paulo at Ribeirão Preto Medical School, Ribeirão Preto, São Paulo, Brazil.
Machado-Neto JA; Department of Pharmacology, Biomedical Sciences Institute, University of São Paulo, São Paulo, Brazil. .
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Źródło:
Scientific reports [Sci Rep] 2019 Jul 09; Vol. 9 (1), pp. 9895. Date of Electronic Publication: 2019 Jul 09.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Apoptosis*
Mutation*
Biomarkers, Tumor/*metabolism
Gene Expression Regulation, Neoplastic/*drug effects
Janus Kinase 2/*metabolism
Morpholines/*pharmacology
Myeloproliferative Disorders/*pathology
Purines/*pharmacology
Aurora Kinase A/genetics ; Aurora Kinase A/metabolism ; Aurora Kinase B/genetics ; Aurora Kinase B/metabolism ; Biomarkers, Tumor/genetics ; Cell Cycle ; Cell Proliferation ; Humans ; Janus Kinase 2/genetics ; Myeloproliferative Disorders/genetics ; Myeloproliferative Disorders/metabolism ; Protein Kinase Inhibitors ; Tumor Cells, Cultured
Czasopismo naukowe
Tytuł:
Synthesis and biological evaluation of 2,5-bis(alkylamino)-1,4-benzoquinones.
Autorzy:
Barbosa LC; Department of Chemistry, Federal University of Viçosa. Av. P.H. Rolfs, Viçosa, MG, Brazil. />Pereira UA
Maltha CR
Teixeira RR
Moreira Valente VM
Oliveira Ferreira JR
Costa-Lotufo LV
Moraes MO
Pessoa C
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Źródło:
Molecules (Basel, Switzerland) [Molecules] 2010 Aug 13; Vol. 15 (8), pp. 5629-43. Date of Electronic Publication: 2010 Aug 13.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Benzoquinones/*chemical synthesis
Benzoquinones/*pharmacology
Adenosine Triphosphate/metabolism ; Antineoplastic Agents/pharmacology ; Benzoquinones/chemistry ; Biological Assay ; Cell Death/drug effects ; Cell Line, Tumor ; Humans ; Plant Roots/drug effects ; Plant Roots/growth & development
Czasopismo naukowe
Tytuł:
Antitumor activity of two derivatives from 2-acylamine-1, 4-naphthoquinone in mice bearing S180 tumor.
Autorzy:
Bezerra DP; Department of Physiology and Pharmacology, School of Medicine, Federal University of Ceará, P.O. Box 3157, 60430-270 Fortaleza, Ceará, Brazil.
Alves AP
de Alencar NM
Mesquita Rde O
Lima MW
Pessoa C
de Moraes MO
Lopes JN
Lopes NP
Costa-Lotufo LV
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Źródło:
Journal of experimental therapeutics & oncology [J Exp Ther Oncol] 2008; Vol. 7 (2), pp. 113-21.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Anilides/*pharmacology
Antineoplastic Agents/*pharmacology
Naphthoquinones/*pharmacology
Sarcoma 180/*drug therapy
Alanine Transaminase/blood ; Anilides/chemical synthesis ; Anilides/toxicity ; Animals ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/toxicity ; Aspartate Aminotransferases/blood ; Blood Cell Count ; Body Weight/drug effects ; Female ; Kidney/pathology ; Mice ; Naphthoquinones/chemical synthesis ; Naphthoquinones/toxicity ; Neoplasm Transplantation ; Organ Size/drug effects ; Sarcoma 180/pathology ; Urea/blood
Czasopismo naukowe
    Wyświetlanie 1-7 z 7

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