- Tytuł:
- Discovery of highly selective and orally available benzimidazole-based phosphodiesterase 10 inhibitors with improved solubility and pharmacokinetic properties for treatment of pulmonary arterial hypertension
- Autorzy:
- Temat:
-
Phosphodiesterase 10A
Inhibitor
Benzimidazole derivatives
Crystal structure
Metabolic stability
Bioavailability
Therapeutics. Pharmacology
RM1-950 - Źródło:
- Acta Pharmaceutica Sinica B, Vol 10, Iss 12, Pp 2339-2347 (2020)
- Opis pliku:
- electronic resource
- Relacje:
- http://www.sciencedirect.com/science/article/pii/S2211383520305463; https://doaj.org/toc/2211-3835
- Dostęp URL:
- https://doaj.org/article/ccae75c50048476bb23a4e31a9cef74b  Link otwiera się w nowym oknie
Czasopismo naukowe