- Tytuł:
- Pyrrolidine-based 3-deoxysphingosylphosphorylcholine analogs as possible candidates against neglected tropical diseases (NTDs): identification of hit compounds towards development of potential treatment of Leishmania donovani .
- Autorzy:
- Źródło:
- Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2021 Dec; Vol. 36 (1), pp. 1922-1930.
- Typ publikacji:
- Journal Article
- MeSH Terms:
-
Antiprotozoal Agents/*chemistry
Leishmania donovani/*drug effects
Phosphorylcholine/*chemistry
Pyrrolidines/*chemistry
Amide Synthases/metabolism ; Antiprotozoal Agents/pharmacology ; Drug Evaluation, Preclinical ; Humans ; Molecular Conformation ; Molecular Docking Simulation ; Palmitates/chemistry ; Pyrrolidines/pharmacology ; Sphingomyelins/chemistry ; Structure-Activity Relationship
Czasopismo naukowe