Informacja

Drogi użytkowniku, aplikacja do prawidłowego działania wymaga obsługi JavaScript. Proszę włącz obsługę JavaScript w Twojej przeglądarce.

Wyszukujesz frazę ""M3 Muscarinic receptor"" wg kryterium: Wszystkie pola


Tytuł:
Immobilization of M3 Muscarinic Receptor to Rapidly Analyze Drug-Protein Interactions and Bioactive Components in a Natural Plant.
Autorzy:
Fan H; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Huang X; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Zhang Z; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Wang T; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Wang L; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Zhang Y; Key Laboratory of Resource Biology and Biotechnology in Western China, Ministry of Education, College of Life Sciences, Northwest University, Xi'an 710069, China.
Pokaż więcej
Źródło:
International journal of molecular sciences [Int J Mol Sci] 2023 Apr 12; Vol. 24 (8). Date of Electronic Publication: 2023 Apr 12.
Typ publikacji:
Journal Article
MeSH Terms:
Pilocarpine*
Receptor, Muscarinic M3*/metabolism
Scopolamine Derivatives ; Plant Extracts/pharmacology
Czasopismo naukowe
Tytuł:
Two-step structural changes in M3 muscarinic receptor activation rely on the coupled Gq protein cycle
Autorzy:
Yong-Seok Kim
Jun-Hee Yeon
Woori Ko
Byung-Chang Suh
Pokaż więcej
Temat:
Science
Źródło:
Nature Communications, Vol 14, Iss 1, Pp 1-18 (2023)
Opis pliku:
electronic resource
Relacje:
https://doaj.org/toc/2041-1723
Dostęp URL:
https://doaj.org/article/76c3427152204628b71f01a92634b1e7  Link otwiera się w nowym oknie
Czasopismo naukowe
Tytuł:
Acetylcholine acts through M3 muscarinic receptor to activate the EGFR signaling and promotes gastric cancer cell proliferation.
Autorzy:
Yu H; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Xia H; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Tang Q; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Xu H; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Wei G; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Chen Y; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Dai X; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Gong Q; Department of Radiology, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Bi F; Department of Medical Oncology and Laboratory of Molecular Targeted Therapy in Oncology, State Key Laboratory of Biotherapy, West China Hospital, Sichuan University, Chengdu 610041, Sichuan, China.
Pokaż więcej
Źródło:
Scientific reports [Sci Rep] 2017 Jan 19; Vol. 7, pp. 40802. Date of Electronic Publication: 2017 Jan 19.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Signal Transduction*/drug effects
Acetylcholine/*metabolism
ErbB Receptors/*metabolism
Receptor, Muscarinic M3/*metabolism
Stomach Neoplasms/*metabolism
Acetylcholine/pharmacology ; Animals ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Disease Models, Animal ; Drug Resistance, Neoplasm/drug effects ; Extracellular Signal-Regulated MAP Kinases/metabolism ; Heterografts ; Humans ; Mice ; Mitogen-Activated Protein Kinase 3/metabolism ; Phosphorylation ; Proto-Oncogene Proteins c-akt/metabolism ; Receptor, Muscarinic M3/agonists ; Receptor, Muscarinic M3/antagonists & inhibitors ; Stomach Neoplasms/pathology
Czasopismo naukowe
Tytuł:
The insect repellent N,N-diethyl-m-toluamide (DEET) induces angiogenesis via allosteric modulation of the M3 muscarinic receptor in endothelial cells.
Autorzy:
Legeay S; University Bretagne Loire, Université d'Angers, UFR santé, département pharmacie, Angers, France.
Clere N; University Bretagne Loire, Université d'Angers, UFR santé, département pharmacie, Angers, France.
Hilairet G; University Bretagne Loire, Université d'Angers, UFR santé, département pharmacie, Angers, France.
Do QT; GreenPharma S.A.S. 03 allée du titane, 45100 Orléans, France.
Bernard P; GreenPharma S.A.S. 03 allée du titane, 45100 Orléans, France.
Quignard JF; Inserm U1045-Centre de Recherche Cardio-Thoracique de Bordeaux, Université de Bordeaux, France.
Apaire-Marchais V; Laboratoire des Récepteurs et Canaux Ioniques Membranaires (RCIM), UPRES-EA 2647, USC INRA 1330, Angers, France.
Lapied B; Laboratoire des Récepteurs et Canaux Ioniques Membranaires (RCIM), UPRES-EA 2647, USC INRA 1330, Angers, France.
Faure S; University Bretagne Loire, Université d'Angers, UFR santé, département pharmacie, Angers, France.
Pokaż więcej
Źródło:
Scientific reports [Sci Rep] 2016 Jun 27; Vol. 6, pp. 28546. Date of Electronic Publication: 2016 Jun 27.
Typ publikacji:
Journal Article
MeSH Terms:
Allosteric Regulation/*drug effects
DEET/*pharmacology
Endothelial Cells/*drug effects
Insect Repellents/*pharmacology
Neovascularization, Pathologic/*chemically induced
Receptor, Muscarinic M3/*metabolism
Acetylcholine/pharmacology ; Animals ; Biological Availability ; Calcium Signaling/drug effects ; Cell Adhesion/drug effects ; Cell Line ; Cell Line, Tumor ; Cell Movement/drug effects ; Cell Proliferation/drug effects ; Endothelial Cells/metabolism ; HEK293 Cells ; Human Umbilical Vein Endothelial Cells ; Humans ; Male ; Mice ; Mice, Nude ; Neovascularization, Pathologic/metabolism ; Vascular Endothelial Growth Factor A/metabolism
Czasopismo naukowe
Tytuł:
M3 muscarinic receptor in the ventral medial prefrontal cortex modulating the expression of contextual fear conditioning in rats.
Autorzy:
Fedoce AG; Department of Pharmacology, Ribeirao Preto School of Medicine, University of Sao Paulo, Av. Bandeirantes, 3900, CEP: 14049-900, Ribeirao Preto, SP, Brazil.; Center for Interdisciplinary Research on Applied Neurosciences (NAPNA), University of Sao Paulo, Sao Paulo, Brazil.
Ferreira-Junior NC; Department of Pharmacology, Ribeirao Preto School of Medicine, University of Sao Paulo, Av. Bandeirantes, 3900, CEP: 14049-900, Ribeirao Preto, SP, Brazil.; Center for Interdisciplinary Research on Applied Neurosciences (NAPNA), University of Sao Paulo, Sao Paulo, Brazil.
Reis DG; Department of Pharmacology, Ribeirao Preto School of Medicine, University of Sao Paulo, Av. Bandeirantes, 3900, CEP: 14049-900, Ribeirao Preto, SP, Brazil.; Center for Interdisciplinary Research on Applied Neurosciences (NAPNA), University of Sao Paulo, Sao Paulo, Brazil.
Corrêa FM; Department of Pharmacology, Ribeirao Preto School of Medicine, University of Sao Paulo, Av. Bandeirantes, 3900, CEP: 14049-900, Ribeirao Preto, SP, Brazil.
Resstel LB; Department of Pharmacology, Ribeirao Preto School of Medicine, University of Sao Paulo, Av. Bandeirantes, 3900, CEP: 14049-900, Ribeirao Preto, SP, Brazil. .; Center for Interdisciplinary Research on Applied Neurosciences (NAPNA), University of Sao Paulo, Sao Paulo, Brazil. .
Pokaż więcej
Źródło:
Psychopharmacology [Psychopharmacology (Berl)] 2016 Jan; Vol. 233 (2), pp. 267-80. Date of Electronic Publication: 2015 Oct 31.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Conditioning, Psychological*/drug effects
Fear/*psychology
Prefrontal Cortex/*metabolism
Receptor, Muscarinic M3/*metabolism
Animals ; Benzodiazepines/agonists ; Cholinesterase Inhibitors/pharmacology ; Emotions ; Male ; Muscarinic Antagonists/pharmacology ; Parasympathetic Nervous System/drug effects ; Prefrontal Cortex/drug effects ; Rats ; Rats, Wistar ; Receptor, Muscarinic M3/drug effects ; Synaptic Transmission/drug effects
Czasopismo naukowe
Tytuł:
Immobilization of M3 Muscarinic Receptor to Rapidly Analyze Drug—Protein Interactions and Bioactive Components in a Natural Plant
Autorzy:
Hushuai Fan
Xiaomin Huang
Ziru Zhang
Ting Wang
Ludan Wang
Yajun Zhang
Pokaż więcej
Temat:
immobilized receptor
M3 muscarinic receptors
drug–protein interaction
bioactive components
Daturae Flos
Biology (General)
QH301-705.5
Chemistry
QD1-999
Źródło:
International Journal of Molecular Sciences, Vol 24, Iss 8, p 7171 (2023)
Opis pliku:
electronic resource
Relacje:
https://www.mdpi.com/1422-0067/24/8/7171; https://doaj.org/toc/1661-6596; https://doaj.org/toc/1422-0067
Dostęp URL:
https://doaj.org/article/0e0cf5257836485e9678b455680c2377  Link otwiera się w nowym oknie
Czasopismo naukowe
Tytuł:
The M3 muscarinic receptor is required for optimal adaptive immunity to helminth and bacterial infection.
Autorzy:
Darby M; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Schnoeller C; Department of Life Sciences, Sir Ernst Chain Building, South Kensington Campus, Imperial College London, London, United Kingdom.
Vira A; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Culley FJ; National Heart and Lung Institute, St.Mary's Campus, Praed Street, Imperial College London, London, United Kingdom.
Bobat S; Medical Research Council Centre for Immune Regulation, School of Immunity and Infection, University of Birmingham, Birmingham, United Kingdom.
Logan E; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Kirstein F; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Wess J; Molecular Signaling Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland, United States of America.
Cunningham AF; Medical Research Council Centre for Immune Regulation, School of Immunity and Infection, University of Birmingham, Birmingham, United Kingdom.
Brombacher F; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Selkirk ME; Department of Life Sciences, Sir Ernst Chain Building, South Kensington Campus, Imperial College London, London, United Kingdom.
Horsnell WG; Institute of Infectious Disease and Molecular Medicine, International Centre for Genetic Engineering and Biotechnology and Division of Immunology, University of Cape Town, Cape Town, South Africa.
Pokaż więcej
Źródło:
PLoS pathogens [PLoS Pathog] 2015 Jan 28; Vol. 11 (1), pp. e1004636. Date of Electronic Publication: 2015 Jan 28 (Print Publication: 2015).
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Adaptive Immunity/*genetics
Nippostrongylus/*immunology
Receptor, Muscarinic M3/*physiology
Salmonella Infections, Animal/*immunology
Salmonella typhimurium/*immunology
Strongylida Infections/*immunology
Animals ; Cells, Cultured ; Lymphocyte Activation/genetics ; Mice ; Mice, Inbred BALB C ; Mice, Knockout ; Salmonella Infections, Animal/genetics ; Signal Transduction/genetics ; Signal Transduction/immunology ; Strongylida Infections/genetics ; Th1 Cells/immunology ; Th2 Cells/immunology
Czasopismo naukowe
Tytuł:
Honokiol blocks store operated calcium entry in CHO cells expressing the M3 muscarinic receptor: honokiol and muscarinic signaling.
Autorzy:
Wang HJ; Department of Biological Sciences, Missouri University of Science & Technology, 400 W, 11th St, Rolla MO 65409, USA.
Martin AG
Chao PK
Reichard RA
Martin AL
Huang YW
Chan MH
Aronstam RS
Pokaż więcej
Źródło:
Journal of biomedical science [J Biomed Sci] 2013 Feb 23; Vol. 20, pp. 11. Date of Electronic Publication: 2013 Feb 23.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Biphenyl Compounds/*administration & dosage
Calcium/*metabolism
Calcium Signaling/*drug effects
Lignans/*administration & dosage
Receptor, Muscarinic M3/*metabolism
Animals ; CHO Cells ; Cricetinae ; Cytoplasm/drug effects ; Cytoplasm/metabolism ; Gene Expression Regulation/drug effects ; Humans ; Inositol 1,4,5-Trisphosphate/metabolism ; Ion Transport/drug effects
Czasopismo naukowe
Tytuł:
M3 muscarinic receptor expression on suburothelial interstitial cells.
Autorzy:
Lamers WH
Pokaż więcej
Źródło:
BJU international [BJU Int] 2009 Nov; Vol. 104 (10), pp. 1538; author reply 1538-9.
Typ publikacji:
Comment; Letter
MeSH Terms:
Receptor, Muscarinic M3/*metabolism
Urinary Bladder/*metabolism
Animals ; Biomarkers/metabolism ; Blotting, Western ; Cell Communication ; Guinea Pigs ; Immunohistochemistry ; Urothelium
Opinia redakcyjna
Tytuł:
In vivo and in vitro pharmacological characterization of SVT-40776, a novel M3 muscarinic receptor antagonist, for the treatment of overactive bladder.
Autorzy:
Salcedo C; Present address: Drug Development & Clinical Research, Palau Pharma S.A. Avinguda Camí Reial 51-57, 08184 Palau Solità i Plegamans, Barcelona, Spain.
Davalillo S
Cabellos J
Lagunas C
Balsa D
Pérez-Del-Pulgar S
Ballarín M
Fernández A
Pokaż więcej
Źródło:
British journal of pharmacology [Br J Pharmacol] 2009 Mar; Vol. 156 (5), pp. 807-17. Date of Electronic Publication: 2009 Feb 16.
Typ publikacji:
Journal Article
MeSH Terms:
Carbamates/*pharmacology
Quinuclidines/*pharmacology
Receptor, Muscarinic M3/*antagonists & inhibitors
Animals ; Atrial Function/drug effects ; Benzhydryl Compounds/pharmacology ; Benzofurans/pharmacology ; Cresols/pharmacology ; Guinea Pigs ; In Vitro Techniques ; Male ; Mice ; Muscle Contraction/drug effects ; Muscle, Smooth/drug effects ; Muscle, Smooth/physiology ; Myocardial Contraction/drug effects ; Phenylpropanolamine/pharmacology ; Pyrrolidines/pharmacology ; Solifenacin Succinate ; Tetrahydroisoquinolines/pharmacology ; Tolterodine Tartrate ; Urinary Bladder/drug effects ; Urinary Bladder/physiology
Czasopismo naukowe
Tytuł:
Molecular characterization of M2 and M3 muscarinic receptor expression in bladder from women with refractory idiopathic detrusor overactivity.
Autorzy:
Mansfield KJ; Department of Physiology and Pharmacology, School of Medical Sciences, University of New South Wales, Sydney, Australia.
Liu L
Moore KH
Vaux KJ
Millard RJ
Burcher E
Pokaż więcej
Źródło:
BJU international [BJU Int] 2007 Jun; Vol. 99 (6), pp. 1433-8.
Typ publikacji:
Journal Article; Research Support, Non-U.S. Gov't
MeSH Terms:
Muscarinic Antagonists/*pharmacology
Receptor, Muscarinic M2/*metabolism
Receptor, Muscarinic M3/*metabolism
Urinary Bladder, Overactive/*metabolism
Actins/metabolism ; Adult ; Aged ; Aged, 80 and over ; Biopsy/methods ; Case-Control Studies ; Female ; Humans ; Middle Aged ; Mucous Membrane/metabolism ; Reverse Transcriptase Polymerase Chain Reaction ; Urinary Bladder/metabolism ; Urinary Bladder/pathology ; Urinary Bladder, Overactive/drug therapy ; Urinary Bladder, Overactive/etiology ; Urinary Bladder, Overactive/pathology
Czasopismo naukowe
Tytuł:
The M3 muscarinic receptor i3 domain confers oxidative stress protection on calcium regulation in transfected COS-7 cells.
Autorzy:
Joseph JA; USDA-HNRC, Tufts University, Boston, MA 02111, USA. />Fisher DR
Carey A
Szprengiel A
Pokaż więcej
Źródło:
Aging cell [Aging Cell] 2004 Oct; Vol. 3 (5), pp. 263-71.
Typ publikacji:
Journal Article
MeSH Terms:
Calcium/*metabolism
Oxidative Stress/*physiology
Receptor, Muscarinic M3/*metabolism
Receptors, Muscarinic/*metabolism
Amino Acid Sequence ; Animals ; COS Cells ; Chlorocebus aethiops ; Dopamine/pharmacology ; Molecular Sequence Data ; Oxidative Stress/drug effects ; Oxotremorine/pharmacology ; Protein Structure, Tertiary
Czasopismo naukowe
Tytuł:
Overexpression of M3 Muscarinic Receptor Suppressed Adverse Electrical Remodeling in Hypertrophic Myocardium Via Increasing Repolarizing K+ Currents
Autorzy:
Xue Chen
Yan Bai
Hanqi Sun
Zhenli Su
Jing Guo
Chuan Sun
Zhimin Du
Pokaż więcej
Temat:
Muscarinic acetylcholine receptor
Potassium currents
Electrical remodeling
Cardiomyocytes
Action potential duration
Physiology
QP1-981
Biochemistry
QD415-436
Źródło:
Cellular Physiology and Biochemistry, Vol 43, Iss 3, Pp 915-925 (2017)
Opis pliku:
electronic resource
Relacje:
https://www.karger.com/Article/FullText/481642; https://doaj.org/toc/1015-8987; https://doaj.org/toc/1421-9778
Dostęp URL:
https://doaj.org/article/22ab0fad7a6d4ac7b7fb53cc1b2a8e11  Link otwiera się w nowym oknie
Czasopismo naukowe

Ta witryna wykorzystuje pliki cookies do przechowywania informacji na Twoim komputerze. Pliki cookies stosujemy w celu świadczenia usług na najwyższym poziomie, w tym w sposób dostosowany do indywidualnych potrzeb. Korzystanie z witryny bez zmiany ustawień dotyczących cookies oznacza, że będą one zamieszczane w Twoim komputerze. W każdym momencie możesz dokonać zmiany ustawień dotyczących cookies